tacrine and isoflurophate

tacrine has been researched along with isoflurophate in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19901 (11.11)18.7374
1990's4 (44.44)18.2507
2000's3 (33.33)29.6817
2010's1 (11.11)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Agnusdei, M; Belinskaya, T; Borriello, M; Brindisi, M; Butini, S; Campiani, G; Catalanotti, B; Fattorusso, C; Fiorini, I; Gemma, S; Nacci, V; Novellino, E; Panico, A; Persico, M; Ros, S; Saxena, A1
Galli, A; Gori, I; Lucherini, M; Mori, F1
Galli, A; Mori, F1
Lindmar, R; Löffelholz, K1
Cecchini, L; Galli, A; Lucherini, M; Mazri, A; Mori, F1
Wu, CS; Yang, JT1
Chang, DC; Fu, H; Han, Y; Kan, KK; Lao, Y; Lee, NT; Li, M; Li, W; Li, Z; Luo, J; Pang, Y; Tsang, HW; Tsim, KW1
Boopathy, R; Chitra, L; Layer, PG; Rajesh, RV1
Hasan, MY; Kuča, K; Lorke, DE; Nurulain, SM; Petroianu, GA; Shafiullah, M1

Other Studies

9 other study(ies) available for tacrine and isoflurophate

ArticleYear
Exploiting protein fluctuations at the active-site gorge of human cholinesterases: further optimization of the design strategy to develop extremely potent inhibitors.
    Journal of medicinal chemistry, 2008, Jun-12, Volume: 51, Issue:11

    Topics: Acetylcholinesterase; Binding Sites; Butyrylcholinesterase; Cholinesterase Inhibitors; Computational Biology; Crystallography, X-Ray; Drug Design; Humans; Models, Molecular; Protein Conformation; Structure-Activity Relationship; Tacrine

2008
In vitro protection of acetylcholinesterase and butyrylcholinesterase by tetrahydroaminoacridine. Comparison with physostigmine.
    Biochemical pharmacology, 1992, Jun-09, Volume: 43, Issue:11

    Topics: Acetylcholinesterase; Binding Sites; Butyrylcholinesterase; Cholinesterase Reactivators; Dose-Response Relationship, Drug; Isoflurophate; Neostigmine; Organophosphorus Compounds; Physostigmine; Tacrine

1992
Effectiveness of 1,2,3,4-tetrahydro-9-aminoacridine (THA) as a pretreatment drug for protection of mice from acute diisopropylfluorophosphate (DFP) intoxication.
    Archives of toxicology, 1991, Volume: 65, Issue:4

    Topics: Animals; Brain; Cholinesterase Inhibitors; Diaphragm; Dose-Response Relationship, Drug; Isoflurophate; Male; Mice; Physostigmine; Poisoning; Pyridostigmine Bromide; Tacrine; Time Factors

1991
The effect of tacrine on acetylcholine overflow in the heart.
    European journal of pharmacology, 1990, Nov-06, Volume: 190, Issue:1-2

    Topics: Acetylcholine; Animals; Chickens; Electric Stimulation; Guinea Pigs; Heart; Ileum; In Vitro Techniques; Isoflurophate; Myocardium; Tacrine

1990
Prevention of diisopropylfluorophosphate (DFP)-induced lethality by meptazinol and 9-amino-tetrahydroacridine (THA) in the mouse.
    Acta physiologica Hungarica, 1990, Volume: 75 Suppl

    Topics: Acetylcholinesterase; Aminoacridines; Animals; Atropine; Azepines; Brain; In Vitro Techniques; Isoflurophate; Meptazinol; Mice; Respiratory Muscles; Tacrine

1990
Tacrine protection of acetylcholinesterase from inactivation by diisopropylfluorophosphate: a circular dichroism study.
    Molecular pharmacology, 1989, Volume: 35, Issue:1

    Topics: Acetylcholinesterase; Aminoacridines; Binding Sites; Circular Dichroism; Isoflurophate; Kinetics; Tacrine; Time Factors

1989
Bis(7)-tacrine attenuates beta amyloid-induced neuronal apoptosis by regulating L-type calcium channels.
    Journal of neurochemistry, 2006, Volume: 98, Issue:5

    Topics: Acetylcholinesterase; Amyloid beta-Peptides; Analysis of Variance; Animals; Apoptosis; Calcium; Calcium Channel Blockers; Calcium Channels, L-Type; Cell Survival; Cells, Cultured; Cerebral Cortex; Cholinesterase Inhibitors; Donepezil; Dose-Response Relationship, Drug; Drug Interactions; Embryo, Mammalian; Hippocampus; Indans; Isoflurophate; Membrane Potentials; Neurons; Nimodipine; Patch-Clamp Techniques; Peptide Fragments; Piperidines; Rats; Tacrine; Time Factors

2006
The aryl acylamidase activity is much more sensitive to Alzheimer drugs than the esterase activity of acetylcholinesterase in chicken embryonic brain.
    Biochimie, 2009, Volume: 91, Issue:9

    Topics: Acetylcholinesterase; Amidohydrolases; Animals; Benzenaminium, 4,4'-(3-oxo-1,5-pentanediyl)bis(N,N-dimethyl-N-2-propenyl-), Dibromide; Brain; Chick Embryo; Chickens; Cholinesterase Inhibitors; Donepezil; Enzyme Activation; Esterases; In Vitro Techniques; Indans; Isoflurophate; Piperidines; Tacrine

2009
Pretreatment for acute exposure to diisopropylfluorophosphate: in vivo efficacy of various acetylcholinesterase inhibitors.
    Journal of applied toxicology : JAT, 2011, Volume: 31, Issue:6

    Topics: Amiloride; Animals; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Erythrocytes; Female; Humans; Inhibitory Concentration 50; Isoflurophate; Male; Methylene Blue; Metoclopramide; Oximes; Physostigmine; Proportional Hazards Models; Pyridinium Compounds; Pyridostigmine Bromide; Ranitidine; Rats; Tacrine; Tiapride Hydrochloride

2011