tacrine and gamma-aminobutyric acid

tacrine has been researched along with gamma-aminobutyric acid in 20 studies

Research

Studies (20)

TimeframeStudies, this research(%)All Research%
pre-19904 (20.00)18.7374
1990's9 (45.00)18.2507
2000's3 (15.00)29.6817
2010's3 (15.00)24.3611
2020's1 (5.00)2.80

Authors

AuthorsStudies
Bellman, K; Knegtel, RM; Settimo, L1
Baĭmanov, TD; Burov, IuV; Maĭsov, NI1
Dawson, RM; Poretski, M1
de Belleroche, J; Gardiner, IM2
Bowen, DM; Lowe, SL; Palmer, AM; Steele, JE2
Jarema, M1
Otomo, E1
Kameyama, T; Nabeshima, T; Yoshida, S1
Borisova, AO; Burov, IuV; Robakidze, TN1
Conlan, A; Finn, M; Mayorga, AJ; Salamone, JD1
Carlier, PR; Han, YF; Hui, KM; Li, CY; Li, ZW; Pang, YP; Wang, H; Xue, H1
Kolbaev, SN; Sharonova, IN; Skrebitskiĭ, VG; Vorob'ev, VS1
Bunce, JG; Chrobak, JJ; Giuliana, D; Sabolek, HR1
Carlier, PR; Clement, EC; Han, Y; Hui, K; Kan, KK; Li, C; Li, M; Li, W; Li, Z; Liu, X; Pang, Y; Ren, H; Wang, H; Xiong, K; Xue, H1
Ai, YX; Han, YF; Li, CY; Li, ZW; Liu, YW; Pang, YP; Peoples, RW; Tian, X; Yang, M; Zhou, L1
Cheong, JH; Cho, YW; Jeon, SJ; Kim, DH; Kim, JM; Ko, KH; Lee, HJ; Moon, JH; Park, SJ; Ryu, JH; Son, KH1
Alves, G; Falcao, A; Matias, M; Silvestre, S1
Andrén, PE; Fridjonsdottir, E; Mantas, I; Nilsson, A; Odell, LR; Schembri, LS; Shariatgorji, R; Svenningsson, P; Vallianatou, T1

Reviews

3 review(s) available for tacrine and gamma-aminobutyric acid

ArticleYear
Tacrine in relation to amino acid transmitters in Alzheimer's disease.
    Advances in neurology, 1990, Volume: 51

    Topics: Alzheimer Disease; Aminoacridines; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Humans; Tacrine

1990
[Progress in the studies of the etiology and treatment of Alzheimer's disease].
    Wiadomosci lekarskie (Warsaw, Poland : 1960), 1988, Jun-01, Volume: 41, Issue:11

    Topics: Acetylcholine; Alzheimer Disease; Brain; Chromosome Aberrations; Chromosomes, Human, 21-22 and Y; Dopamine; gamma-Aminobutyric Acid; Humans; Physostigmine; Tacrine

1988
Recent Highlights on Molecular Hybrids Potentially Useful in Central Nervous System Disorders.
    Mini reviews in medicinal chemistry, 2017, Volume: 17, Issue:6

    Topics: Analgesics; Central Nervous System Diseases; Choline; Donepezil; Epilepsy; gamma-Aminobutyric Acid; Humans; Indans; Opioid Peptides; Pain; Piperidines; Tacrine

2017

Other Studies

17 other study(ies) available for tacrine and gamma-aminobutyric acid

ArticleYear
Comparison of the accuracy of experimental and predicted pKa values of basic and acidic compounds.
    Pharmaceutical research, 2014, Volume: 31, Issue:4

    Topics: Chemistry, Pharmaceutical; Forecasting; Hydrogen-Ion Concentration; Pharmaceutical Preparations; Random Allocation

2014
[Effects of amiridin and tacrine, drugs effective in Alzheimer's disease, on synaptosomal uptake of neuromediators].
    Biulleten' eksperimental'noi biologii i meditsiny, 1992, Volume: 113, Issue:4

    Topics: Alzheimer Disease; Aminoquinolines; Animals; Cholinesterase Inhibitors; Dopamine; Epinephrine; gamma-Aminobutyric Acid; Neurotransmitter Agents; Norepinephrine; Physostigmine; Piracetam; Psychotropic Drugs; Rats; Serotonin; Synaptosomes; Tacrine

1992
The interaction of tacrine with benzodiazepine and GABA binding sites of guinea pig brain.
    Neuroscience letters, 1991, Aug-19, Volume: 129, Issue:2

    Topics: Animals; Bicuculline; Binding, Competitive; Brain Chemistry; Cerebral Cortex; Flunitrazepam; gamma-Aminobutyric Acid; Guinea Pigs; Hippocampus; In Vitro Techniques; Kinetics; Radioligand Assay; Receptors, GABA-A; Tacrine

1991
Modulation of gamma-aminobutyric acid release in cerebral cortex by fluoride, phorbol ester, and phosphodiesterase inhibitors: differential sensitivity of acetylcholine release to fluoride and K+ channel blockers.
    Journal of neurochemistry, 1990, Volume: 54, Issue:4

    Topics: 1-Methyl-3-isobutylxanthine; Acetylcholine; Animals; Cerebral Cortex; gamma-Aminobutyric Acid; Phorbol Esters; Phosphodiesterase Inhibitors; Potassium; Potassium Channels; Rats; Sodium Fluoride; Tacrine; Theophylline

1990
Influence of tetrahydro-9-aminoacridine on excitatory amino acid release.
    Clinical neuropharmacology, 1990, Volume: 13, Issue:1

    Topics: Amino Acids; Aminoacridines; Animals; Aspartic Acid; Brain Chemistry; Cerebral Cortex; Chromatography, High Pressure Liquid; Dialysis; gamma-Aminobutyric Acid; Glutamates; Injections; Injections, Intraperitoneal; Male; Potassium; Rats; Rats, Inbred Strains; Tacrine

1990
Inhibitory effect of 1,2,3,4-tetrahydro-9-aminoacridine on the depolarization-induced release of GABA from cerebral cortex.
    British journal of pharmacology, 1988, Volume: 94, Issue:4

    Topics: Aminoacridines; Animals; Cerebral Cortex; gamma-Aminobutyric Acid; In Vitro Techniques; Neuromuscular Depolarizing Agents; Rats; Tacrine

1988
[Drug therapy of Alzheimer's disease. General concepts on nootropic drugs].
    Nihon rinsho. Japanese journal of clinical medicine, 1988, Volume: 46, Issue:7

    Topics: Aged; Aged, 80 and over; Alzheimer Disease; Amantadine; Aminoacridines; Dementia; gamma-Aminobutyric Acid; Humans; Pantothenic Acid; Tacrine

1988
Effects of the novel compound NIK-247 on impairment of passive avoidance response in mice.
    European journal of pharmacology, 1988, Sep-23, Volume: 154, Issue:3

    Topics: Aminoquinolines; Amnesia; Animals; Avoidance Learning; Choline; Cholinesterase Inhibitors; Cycloheximide; Electroshock; gamma-Aminobutyric Acid; Male; Memory; Mice; Phencyclidine; Picrotoxin; Tacrine

1988
[Effect of amiridine on rat learning in a radial maze].
    Biulleten' eksperimental'noi biologii i meditsiny, 1996, Volume: 121, Issue:5

    Topics: Aminoquinolines; Animals; Cholinesterase Inhibitors; gamma-Aminobutyric Acid; Learning; Male; Memory; Neuroprotective Agents; Nootropic Agents; Piracetam; Rats; Tacrine

1996
Involvement of pallidal and nigral GABA mechanisms in the generation of tremulous jaw movements in rats.
    Neuroscience, 1997, Volume: 80, Issue:2

    Topics: Animals; Cholinesterase Inhibitors; GABA Agonists; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Globus Pallidus; Injections; Jaw; Male; Microinjections; Movement; Muscimol; Muscle, Skeletal; Rats; Rats, Sprague-Dawley; Substantia Nigra; Tacrine

1997
Bis(7)-tacrine, a novel dimeric AChE inhibitor, is a potent GABA(A) receptor antagonist.
    Neuroreport, 1999, Mar-17, Volume: 10, Issue:4

    Topics: Alzheimer Disease; Animals; Cholinesterase Inhibitors; Electric Stimulation; Electrophysiology; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Hippocampus; Membrane Potentials; Mice; Neurons; Patch-Clamp Techniques; Physostigmine; Radioligand Assay; Rats; Receptors, Muscarinic; Tacrine

1999
[Mechanisms of tacrine modulation of the GABA-activated currents in the isolated cerebellar neurons].
    Biulleten' eksperimental'noi biologii i meditsiny, 1999, Volume: 127, Issue:5

    Topics: Animals; Cerebellum; Electrophysiology; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Purkinje Cells; Rats; Receptors, GABA-A; Tacrine

1999
Within-subject memory decline in middle-aged rats: effects of intraseptal tacrine.
    Neurobiology of aging, 2004, Volume: 25, Issue:9

    Topics: Acetylcholine; Aging; Animals; Catheterization; Cholinergic Fibers; Drug Administration Routes; Early Diagnosis; gamma-Aminobutyric Acid; Male; Maze Learning; Memory Disorders; Memory, Short-Term; Nootropic Agents; Rats; Rats, Long-Evans; Septal Nuclei; Septum of Brain; Tacrine; Treatment Failure

2004
Alkylene tether-length dependent gamma-aminobutyric acid type A receptor competitive antagonism by tacrine dimers.
    Neuropharmacology, 2007, Volume: 52, Issue:2

    Topics: Alkylation; Animals; Bicuculline; Dimerization; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Drug Interactions; Electric Stimulation; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Ganglia, Spinal; Inhibitory Concentration 50; Male; Membrane Potentials; Models, Molecular; Neurons; Patch-Clamp Techniques; Radioligand Assay; Rats; Rats, Sprague-Dawley; Structure-Activity Relationship; Tacrine

2007
Mechanism of bis(7)-tacrine inhibition of GABA-activated current in cultured rat hippocampal neurons.
    Neuropharmacology, 2009, Volume: 57, Issue:1

    Topics: Analysis of Variance; Animals; Biophysics; Cells, Cultured; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Embryo, Mammalian; Enzyme Inhibitors; gamma-Aminobutyric Acid; Hippocampus; Membrane Potentials; Neural Inhibition; Neurons; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Tacrine

2009
Cognitive dysfunctions induced by a cholinergic blockade and Aβ 25-35 peptide are attenuated by salvianolic acid B.
    Neuropharmacology, 2011, Volume: 61, Issue:8

    Topics: Amyloid beta-Peptides; Animals; Animals, Newborn; Benzofurans; Cholinergic Antagonists; Cholinesterase Inhibitors; Cognition Disorders; Disease Models, Animal; Dose-Response Relationship, Drug; Female; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Injections, Intraventricular; Male; Maze Learning; Membrane Potentials; Mice; Neurons; Patch-Clamp Techniques; Peptide Fragments; Pregnancy; Rats; Tacrine

2011
Region-Specific and Age-Dependent Multitarget Effects of Acetylcholinesterase Inhibitor Tacrine on Comprehensive Neurotransmitter Systems.
    ACS chemical biology, 2022, 01-21, Volume: 17, Issue:1

    Topics: Aging; Animals; Brain; Brain Mapping; Cholinesterase Inhibitors; Dopaminergic Neurons; gamma-Aminobutyric Acid; Least-Squares Analysis; Mice; Neurotransmitter Agents; Norepinephrine; Serotonin; Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization; Tacrine

2022