Page last updated: 2024-08-16

suramin and sirtinol

suramin has been researched along with sirtinol in 6 studies

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (16.67)29.6817
2010's5 (83.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Berger, SL; Brent, M; Dang, W; Howitz, K; Jackson, B; Marmorstein, R; Sanders, BD; Schreiber, SL; Taylor, AM1
Madsen, AS; Olsen, CA1
Fischer, F; Steegborn, C; Suenkel, B1
Aquilani, L; Belyanskaya, SL; Blum, CA; Chiu, CH; Coppo, F; Cuozzo, JW; Dai, H; Deng, J; Disch, JS; Evindar, G; Graybill, TL; Jin, L; Lavu, S; Lind, KE; Mao, C; Perni, RB; Schuman, E; Vlasuk, GP1
He, W; Jung, M; Maurer, B; Rumpf, T; Scharfe, M; Schmitt, ML; Sippl, W; Stolfa, DA; Verdin, E1
He, B; Huang, W; Li, Y; Xie, T; You, L1

Other Studies

6 other study(ies) available for suramin and sirtinol

ArticleYear
Identification and characterization of novel sirtuin inhibitor scaffolds.
    Bioorganic & medicinal chemistry, 2009, Oct-01, Volume: 17, Issue:19

    Topics: Drug Evaluation, Preclinical; Enzyme Inhibitors; Fibroblast Growth Factor 6; Fungal Proteins; Humans; Inhibitory Concentration 50; Kinetics; Sirtuins; Structure-Activity Relationship

2009
Substrates for efficient fluorometric screening employing the NAD-dependent sirtuin 5 lysine deacylase (KDAC) enzyme.
    Journal of medicinal chemistry, 2012, Jun-14, Volume: 55, Issue:11

    Topics: Benzamides; Coumarins; Enzyme Assays; Fluorometry; Furans; Humans; Isoenzymes; Kinetics; Lysine; Naphthols; Protein Processing, Post-Translational; Quinolines; Recombinant Proteins; Sirtuins; Structure-Activity Relationship; Substrate Specificity; Succinates; Suramin

2012
Inhibition of the human deacylase Sirtuin 5 by the indole GW5074.
    Bioorganic & medicinal chemistry letters, 2013, Jan-01, Volume: 23, Issue:1

    Topics: Humans; Indoles; Phenols; Protein Binding; Sirtuins; Substrate Specificity

2013
Discovery of thieno[3,2-d]pyrimidine-6-carboxamides as potent inhibitors of SIRT1, SIRT2, and SIRT3.
    Journal of medicinal chemistry, 2013, May-09, Volume: 56, Issue:9

    Topics: Drug Discovery; Humans; Models, Molecular; Protein Conformation; Pyrimidines; Sirtuin 1; Sirtuin 2; Sirtuin 3; Sirtuins

2013
Inhibitors of the NAD(+)-Dependent Protein Desuccinylase and Demalonylase Sirt5.
    ACS medicinal chemistry letters, 2012, Dec-13, Volume: 3, Issue:12

    Topics:

2012
A FRET-based assay for screening SIRT5 specific modulators.
    Bioorganic & medicinal chemistry letters, 2015, Apr-15, Volume: 25, Issue:8

    Topics: Amino Acid Sequence; Coumarins; Enzyme Assays; Enzyme Inhibitors; Fluorescence Resonance Energy Transfer; Fluorescent Dyes; Kinetics; Molecular Sequence Data; p-Dimethylaminoazobenzene; Peptides; Sirtuins; Substrate Specificity

2015