Page last updated: 2024-08-16

suramin and indomethacin

suramin has been researched along with indomethacin in 24 studies

Research

Studies (24)

TimeframeStudies, this research(%)All Research%
pre-19902 (8.33)18.7374
1990's9 (37.50)18.2507
2000's9 (37.50)29.6817
2010's4 (16.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Schöffel, E; Starke, K; von Kügelgen, I1
Hahn, I; Krieglstein, G; Krieglstein, J; Tschentscher, K1
Giachetti, A; Maggi, CA; Santicioli, P; Zagorodnyuk, V1
Starke, K; Stoffel, D; von Kügelgen, I1
Boarder, MR; Dainty, IA; McKechnie, K; Wilkinson, GF1
Hollingsworth, M; Piper, AS2
Burnstock, G; Knight, GE1
Chiba, S; Matsumoto, T; Nakane, T1
Buda, MD; Hughes, RJ; Insel, PA; Jacobson, JP; Kao, CC; Post, SR; Rump, LC; Zambon, A1
Matsuyama, H; Takewaki, T; Thapaliya, S1
Ralevic, V1
Depoortere, I; Peeters, TL; Thielemans, L; Thijs, T1
Ikomi, F; Kousai, A; Mizuno, R; Ohhashi, T1
Kiss, T1
Boudaka, A; Draid, M; El-Mahmoudy, A; Shiina, T; Shimizu, Y; Takewaki, T1
Pinna, C; Puglisi, L; Sanvito, P1
De Koning, HP; Dogruel, M; Rodgers, J; Sanderson, L; Thomas, SA1
Barajas-López, C; Carbajal, V; Checa, M; Figueroa, A; Flores-Soto, E; García-Hernández, LM; Montaño, LM; Reyes-García, J1
Li, D; Liu, MD; Wang, YB; Xu, LJ; Yuan, WS1

Other Studies

24 other study(ies) available for suramin and indomethacin

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Inhibition by nucleotides acting at presynaptic P2-receptors of sympathetic neuro-effector transmission in the mouse isolated vas deferens.
    Naunyn-Schmiedeberg's archives of pharmacology, 1989, Volume: 340, Issue:5

    Topics: 4-Chloromercuribenzenesulfonate; Animals; Indomethacin; Male; Mice; Muscle, Smooth; Norepinephrine; Protein Synthesis Inhibitors; Purine Nucleosides; Purine Nucleotides; Receptors, Neurotransmitter; Suramin; Sympathetic Nervous System; Triazines; Tritium; Vas Deferens; Yohimbine

1989
Distribution of chlorpromazine in a simplified blood influenced by various drugs.
    Naunyn-Schmiedeberg's archives of pharmacology, 1973, Volume: 278, Issue:1

    Topics: Acetazolamide; Animals; Antidepressive Agents; Benzoates; Binding Sites; Binding, Competitive; Cattle; Chlorothiazide; Chlorpromazine; Coumarins; Deoxycholic Acid; Erythrocytes; Fatty Acids; Indomethacin; Phenylbutazone; Phenytoin; Probenecid; Protein Binding; Quinine; Salicylates; Serum Albumin, Bovine; Solubility; Sulfonamides; Suramin; Tetracycline; Thiopental

1973
Evidence that tachykinin NK1 and NK2 receptors mediate non-adrenergic non-cholinergic excitation and contraction in the circular muscle of guinea-pig duodenum.
    British journal of pharmacology, 1995, Volume: 115, Issue:2

    Topics: Action Potentials; Adenosine Diphosphate; Animals; Apamin; Arginine; Atropine; Dose-Response Relationship, Drug; Duodenum; Electric Stimulation; Guanethidine; Guinea Pigs; Indomethacin; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin-1 Receptor Antagonists; Neuromuscular Junction; Nifedipine; Nitroarginine; Oligopeptides; Peptide Fragments; Peptides, Cyclic; Physalaemin; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Suramin; Thionucleotides

1995
P2-purinoceptor-mediated inhibition of noradrenaline release in rat atria.
    British journal of pharmacology, 1995, Volume: 115, Issue:2

    Topics: Adenosine; Adenosine Diphosphate; Adenosine Triphosphate; Animals; Antihypertensive Agents; Atropine; Desipramine; Dose-Response Relationship, Drug; Electric Stimulation; Heart Atria; Indomethacin; Male; Norepinephrine; Phenethylamines; Protein Synthesis Inhibitors; Purinergic P1 Receptor Antagonists; Purinergic P2 Receptor Antagonists; Rats; Rats, Wistar; Receptors, Purinergic P1; Receptors, Purinergic P2; Suramin; Triazines; Xanthines; Yohimbine

1995
P2Y purinoceptor and nucleotide receptor-induced relaxation of precontracted bovine aortic collateral artery rings: differential sensitivity to suramin and indomethacin.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 268, Issue:2

    Topics: Adenosine Triphosphate; Animals; Aorta; Cattle; Dose-Response Relationship, Drug; In Vitro Techniques; Indomethacin; Nitric Oxide; Receptors, Purinergic P2; Suramin; Uridine Triphosphate; Vasodilation

1994
P2-purinoceptors mediating spasm of the isolated uterus of the non-pregnant guinea-pig.
    British journal of pharmacology, 1996, Volume: 117, Issue:8

    Topics: Adenosine Triphosphate; Animals; Female; Guinea Pigs; Indomethacin; Muscle Contraction; Muscle, Smooth; Platelet Aggregation Inhibitors; Pyridoxal Phosphate; Receptors, Purinergic P1; Receptors, Purinergic P2; Spasm; Suramin; Theophylline; Thioinosine; Thionucleotides; Uridine Triphosphate; Uterus

1996
ATP and beta,gamma-methylene ATP produce relaxation of guinea-pig isolated trachealis muscle via actions at P1 purinoceptors.
    European journal of pharmacology, 1996, Jun-27, Volume: 307, Issue:2

    Topics: Adenosine Triphosphate; Animals; Carbachol; Female; Guinea Pigs; In Vitro Techniques; Indomethacin; Male; Muscle Contraction; Muscle Relaxation; Parasympatholytics; Receptors, Purinergic P1; Receptors, Purinergic P2; Suramin; Theophylline; Thioinosine; Trachea

1996
The effects of purine compounds on the isolated aorta of the frog Rana temporaria.
    British journal of pharmacology, 1996, Volume: 117, Issue:5

    Topics: Adenosine; Adenosine Triphosphate; Animals; Aorta; Dose-Response Relationship, Drug; In Vitro Techniques; Indomethacin; Pyridoxal Phosphate; Rana temporaria; Receptors, Purinergic; Suramin; Uridine Triphosphate; Vasoconstriction; Vasodilation

1996
UTP induces vascular responses in the isolated and perfused canine epicardial coronary artery via UTP-preferring P2Y receptors.
    British journal of pharmacology, 1997, Volume: 122, Issue:8

    Topics: Adenosine Triphosphate; Animals; Anti-Inflammatory Agents, Non-Steroidal; Antinematodal Agents; Coronary Vessels; Diltiazem; Dogs; Female; Hexokinase; Indomethacin; Male; Protein Synthesis Inhibitors; Receptors, Purinergic P2; Saponins; Suramin; Triazines; Uridine Diphosphate; Uridine Triphosphate

1997
ATP activates cAMP production via multiple purinergic receptors in MDCK-D1 epithelial cells. Blockade of an autocrine/paracrine pathway to define receptor preference of an agonist.
    The Journal of biological chemistry, 1998, Sep-04, Volume: 273, Issue:36

    Topics: Adenosine Triphosphate; Animals; Arachidonic Acid; Autocrine Communication; Cyclic AMP; Cyclooxygenase Inhibitors; Dogs; Epithelial Cells; Indomethacin; Paracrine Communication; Prostaglandins; Receptors, Purinergic P2; Receptors, Purinergic P2Y1; Receptors, Purinergic P2Y2; Signal Transduction; Suramin; Thionucleotides; Uridine Triphosphate

1998
ATP released from perivascular nerves hyperpolarizes smooth muscle cells by releasing an endothelium-derived factor in hamster mesenteric arteries.
    The Journal of physiology, 1999, Nov-15, Volume: 521 Pt 1

    Topics: Adenosine Triphosphate; Animals; Cricetinae; Electric Stimulation; Endothelium, Vascular; Excitatory Postsynaptic Potentials; In Vitro Techniques; Indomethacin; Male; Membrane Potentials; Mesenteric Arteries; Mesocricetus; Microelectrodes; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Prazosin; Purinergic P2 Receptor Agonists; Pyridoxal Phosphate; Receptors, Purinergic P2; Suramin; Triazines

1999
Mechanism of prolonged vasorelaxation to ATP in the rat isolated mesenteric arterial bed.
    British journal of pharmacology, 2001, Volume: 132, Issue:3

    Topics: Adenosine Triphosphate; Animals; Capsaicin; Cardiotonic Agents; Cardiovascular Agents; Charybdotoxin; Drug Interactions; Electric Stimulation; Endothelium, Vascular; Glyburide; In Vitro Techniques; Indomethacin; Isotonic Solutions; Male; Mesenteric Arteries; Neurons, Afferent; Ouabain; Pyridoxal Phosphate; Rats; Rats, Wistar; Suramin; Tetraethylammonium; Theophylline; Vasodilation

2001
Mechanisms involved in the loss of excitatory post-stimulus responses by inflammation.
    Naunyn-Schmiedeberg's archives of pharmacology, 2003, Volume: 367, Issue:3

    Topics: Adenosine Triphosphate; Animals; Colitis; Cyclooxygenase Inhibitors; Electric Stimulation; Female; In Vitro Techniques; Indomethacin; Male; Methiothepin; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Piperidines; Purinergic P2 Receptor Antagonists; Quinuclidines; Rabbits; Serotonin Antagonists; Substance P; Suramin; Trinitrobenzenesulfonic Acid

2003
ATP inhibits pump activity of lymph vessels via adenosine A1 receptor-mediated involvement of NO- and ATP-sensitive K+ channels.
    American journal of physiology. Heart and circulatory physiology, 2004, Volume: 287, Issue:6

    Topics: Adenosine Triphosphate; Animals; Anti-Arrhythmia Agents; Antineoplastic Agents; Arginine; Cardiovascular Agents; Endothelium; Enzyme Inhibitors; Glyburide; Indomethacin; Lymphatic System; Male; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Nitric Oxide; Potassium Channels; Rats; Rats, Wistar; Receptor, Adenosine A1; Suramin; Xanthines

2004
G-protein coupled activation of potassium channels by endogenous neuropeptides in snail neurons.
    The European journal of neuroscience, 2005, Volume: 21, Issue:8

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Acetophenones; Animals; Antibodies; Blotting, Western; Cholera Toxin; Codeine; Colforsin; Dose-Response Relationship, Drug; Electric Stimulation; Enzyme Activation; Fishes; GTP-Binding Protein alpha Subunits; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Helix, Snails; Indomethacin; Membrane Potentials; Models, Neurological; Neurons; Neuropeptides; Patch-Clamp Techniques; Pertussis Toxin; Potassium Channels; Signal Transduction; Suramin; Time Factors

2005
Neurally released ATP mediates endothelium-dependent hyperpolarization in the circular smooth muscle cells of chicken anterior mesenteric artery.
    British journal of pharmacology, 2005, Volume: 146, Issue:7

    Topics: Adenosine Triphosphate; Animals; Chickens; Electric Stimulation; Endothelium, Vascular; Female; In Vitro Techniques; Indomethacin; Membrane Potentials; Mesenteric Arteries; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; NG-Nitroarginine Methyl Ester; Nitric Oxide; Prostaglandins I; Pyridoxal Phosphate; Receptors, Purinergic P2; Suramin

2005
Altered neurogenic and mechanical responses to acetylcholine, ATP and substance P in detrusor from rat with outlet obstruction.
    Life sciences, 2006, Aug-22, Volume: 79, Issue:13

    Topics: Acetylcholine; Adenosine Triphosphate; Animals; Atropine; Cholinergic Agonists; Cyclooxygenase Inhibitors; Electric Stimulation; Female; In Vitro Techniques; Indomethacin; Mandelic Acids; Muscarinic Agonists; Muscle Contraction; Muscle, Smooth; Rats; Rats, Sprague-Dawley; Substance P; Suramin; Urethra; Urinary Bladder; Urinary Bladder Neck Obstruction

2006
Pentamidine movement across the murine blood-brain and blood-cerebrospinal fluid barriers: effect of trypanosome infection, combination therapy, P-glycoprotein, and multidrug resistance-associated protein.
    The Journal of pharmacology and experimental therapeutics, 2009, Volume: 329, Issue:3

    Topics: Adenine; Adenosine; Animals; ATP Binding Cassette Transporter, Subfamily B; Biological Transport; Blood-Brain Barrier; Brain; Cerebrospinal Fluid; Disease Models, Animal; Drug Interactions; Eflornithine; Indomethacin; Male; Melarsoprol; Mice; Mice, Inbred BALB C; Mice, Inbred Strains; Mice, Knockout; Multidrug Resistance-Associated Proteins; Nifurtimox; Pentamidine; Perfusion; Suramin; Trypanosoma brucei brucei; Trypanosomiasis, African

2009
In airways ATP refills sarcoplasmic reticulum via P2X smooth muscle receptors and induces contraction through P2Y epithelial receptors.
    Pflugers Archiv : European journal of physiology, 2011, Volume: 461, Issue:2

    Topics: Adenosine Triphosphate; Animals; Calcium; Calcium Signaling; Guinea Pigs; Indomethacin; Male; Muscle Contraction; Muscle, Smooth; Patch-Clamp Techniques; Prostaglandins; Pyridoxal Phosphate; Receptors, Purinergic P2X; Receptors, Purinergic P2Y; Sarcoplasmic Reticulum; Suramin; Trachea; Triazines

2011
[The different contraction between rat gastric longitudinal and circular smooth muscle induced by extracellular nucleotides].
    Zhongguo ying yong sheng li xue za zhi = Zhongguo yingyong shenglixue zazhi = Chinese journal of applied physiology, 2014, Volume: 30, Issue:1

    Topics: Adenosine Triphosphate; Animals; Dinucleoside Phosphates; Indomethacin; Muscle Contraction; Muscle, Smooth; Nucleotides; Rats; Suramin; Uridine Triphosphate

2014