Page last updated: 2024-08-16

suramin and diminazene

suramin has been researched along with diminazene in 36 studies

Research

Studies (36)

TimeframeStudies, this research(%)All Research%
pre-199015 (41.67)18.7374
1990's12 (33.33)18.2507
2000's4 (11.11)29.6817
2010's4 (11.11)24.3611
2020's1 (2.78)2.80

Authors

AuthorsStudies
Caffrey, CR; Connelly, M; Greenbaum, D; Guy, RK; Harbut, M; Kosinski, A; Mallari, JP; McKerrow, JH; Obrien, T; Shelat, AA1
Anbazhagan, M; Boykin, DW; Brun, R; Gillingwater, K; Kumar, A; Tidwell, RR1
Brun, R; Fotie, J; Gershkovich, P; He, S; Liu, Q; Patrick, DA; Premalatha, K; Reid, CS; Tidwell, RR; Wang, MZ; Wasan, KM; Wenzler, T; Werbovetz, KA1
Williamson, J1
James, DM1
Hawking, F; Worms, MJ1
Goodwin, LG; Tierney, ED1
Kaminsky, R; Zweygarth, E1
Baltz, T; Giroud, C; Zhang, ZQ2
Kaminsky, R; Webster, P; Zweygarth, E1
Brun, R; Kunz, C1
Jefferies, D; Jenni, L1
Brown, HC; Holmes, PH; Jennings, FW; Waitumbi, JN1
Clarkson, AB; Rosenberg, C; Williams, DE1
Balber, AE; Frommel, TO1
Dieleman, EF1
Borowy, NK; Hirumi, H; Mkoji, G; Waithaka, HK1
Dukes, P1
Jennings, FW; Urquhart, GM1
Emerole, GO; Thabrew, MI1
Jara, A; Monzón, CM; Nantulya, VM1
Kinabo, LD1
Kaminsky, R; Moloo, SK; Zweygarth, E1
Brun, R; Lun, ZR1
Milord, F; Pépin, J1
Bacchi, CJ; Clarkson, AB; Goldberg, B; McCann, PP; Nathan, HC; Saric, M; Sjoerdsma, A; Yarlett, N1
Anene, BM; Anika, SM; Chukwu, CC; Ross, CA1
Coetzer, TH; Jones, R; Lonsdale-Eccles, JD; Morty, RE; Nickel, P; Pike, RN; Troeberg, L1
KILLICK-KENDRICK, R1
Rudenko, G; Sheader, K; te Vruchte, D1
Kaboya, JS; Kibona, SN; Lubega, GW; Matemba, L1
Arafa, RK; Boykin, DW; Brun, R; Gillingwater, K; Ismail, MA; Kumar, A; Stephens, CE; Tidwell, RR1
Bockstal, V; Cnops, J; De Trez, C; Magez, S; Miquel, MC; Radwanska, M1
Birhanu, H; Büscher, P; Gebrehiwot, T; Goddeeris, BM; Van Reet, N1
Auma, JE; Chemuliti, JK; Gitonga, PK; Kurgat, RK; Mdachi, RE; Murilla, GA; Ndung'u, K; Ngae, GN; Thuita, JK; Thungu, DK1

Reviews

3 review(s) available for suramin and diminazene

ArticleYear
Trypanosomiasis in Indonesia. A review of research, 1900-1983.
    The veterinary quarterly, 1986, Volume: 8, Issue:3

    Topics: Animals; Arthropod Vectors; Diminazene; Phenanthridines; Suramin; Trypanosomiasis

1986
Pharmacology of existing drugs for animal trypanosomiasis.
    Acta tropica, 1993, Volume: 54, Issue:3-4

    Topics: Animals; Arsenicals; Diminazene; Ethidium; Phenanthridines; Quinolinium Compounds; Suramin; Trypanocidal Agents; Trypanosomiasis, African

1993
The treatment of human African trypanosomiasis.
    Advances in parasitology, 1994, Volume: 33

    Topics: Animals; Diminazene; Eflornithine; Humans; Melarsoprol; Nifurtimox; Pentamidine; Suramin; Trypanocidal Agents; Trypanosoma brucei gambiense; Trypanosoma brucei rhodesiense; Trypanosomiasis, African

1994

Other Studies

33 other study(ies) available for suramin and diminazene

ArticleYear
Development of potent purine-derived nitrile inhibitors of the trypanosomal protease TbcatB.
    Journal of medicinal chemistry, 2008, Feb-14, Volume: 51, Issue:3

    Topics: Animals; Cathepsin B; Cell Line; Cell Line, Tumor; Humans; Models, Molecular; Nitriles; Purines; Static Electricity; Structure-Activity Relationship; Trypanocidal Agents; Trypanosoma brucei brucei

2008
In vivo investigations of selected diamidine compounds against Trypanosoma evansi using a mouse model.
    Antimicrobial agents and chemotherapy, 2009, Volume: 53, Issue:12

    Topics: Animals; Disease Models, Animal; Female; Mice; Parasitic Sensitivity Tests; Pentamidine; Trypanocidal Agents; Trypanosoma; Trypanosomiasis

2009
Synthesis and antitrypanosomal evaluation of derivatives of N-benzyl-1,2-dihydroquinolin-6-ols: Effect of core substitutions and salt formation.
    Bioorganic & medicinal chemistry, 2011, Jan-01, Volume: 19, Issue:1

    Topics: Animals; Cyclization; Mice; Quinolines; Salts; Structure-Activity Relationship; Trypanocidal Agents

2011
Chemotherapy of African trypanosomiasis.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1976, Volume: 70, Issue:2

    Topics: Arsenicals; Diminazene; Humans; Suramin; Triazines; Trypanocidal Agents; Trypanosomiasis, African

1976
Prophylactic activity in rodents of trypanocides complexed with dextran.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1978, Volume: 72, Issue:5

    Topics: Animals; Benzamidines; Dextrans; Diminazene; Dose-Response Relationship, Drug; Drug Combinations; Mice; Phenanthridines; Pyridinium Compounds; Quinolinium Compounds; Rats; Suramin; Trypanocidal Agents; Trypanosomiasis

1978
Homidium bromide as a macrofilaricide.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1978, Volume: 72, Issue:5

    Topics: Animals; Benzamidines; Diminazene; Ethidium; Female; Filariasis; Male; Phenanthridines; Quinolinium Compounds; Rats; Suramin; Trypanocidal Agents

1978
Trypanocidal activity of blood and tissue fluid from normal and infected rabbits treated with curative drugs.
    Parasitology, 1977, Volume: 74, Issue:1

    Topics: Animals; Benzamidines; Body Fluids; Diminazene; Ethidium; Male; Melarsoprol; Mice; Phenanthridines; Rabbits; Suramin; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis

1977
Evaluation of DL-alpha-difluoromethylornithine against susceptible and drug-resistant Trypanosoma brucei brucei.
    Acta tropica, 1991, Volume: 48, Issue:3

    Topics: Animals; Arsenicals; Culture Media; Diminazene; Drug Antagonism; Drug Synergism; Drug Therapy, Combination; Eflornithine; Female; Humans; Immune Sera; Male; Mice; Phenanthridines; Suramin; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African

1991
In vivo and in vitro sensitivity of Trypanosoma evansi and T. equiperdum to diminazene, suramin, MelCy, quinapyramine and isometamidium.
    Acta tropica, 1991, Volume: 50, Issue:2

    Topics: Animals; Arsenicals; Diminazene; Female; Mice; Phenanthridines; Quinolinium Compounds; Suramin; Trypanocidal Agents; Trypanosoma; Trypanosomiasis

1991
Trypanosoma brucei evansi: dyskinetoplasia and loss of infectivity after long-term in vitro cultivation.
    Acta tropica, 1990, Volume: 48, Issue:2

    Topics: Animals; Diminazene; DNA, Circular; DNA, Kinetoplast; Female; Male; Mice; Microscopy, Electron; Phenanthridines; Quinolinium Compounds; Suramin; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African

1990
In vitro drug sensitivity test for Trypanosoma brucei subgroup bloodstream trypomastigotes.
    Acta tropica, 1989, Volume: 46, Issue:5-6

    Topics: Animals; Arsenicals; Diminazene; Hypoxanthine; Hypoxanthines; Leucine; Pentamidine; Phenanthridines; Suramin; Thymidine; Trypanocidal Agents; Trypanosoma brucei brucei

1989
The effect of trypanocidal drugs on the transmission of Trypanosoma brucei brucei by Glossina morsitans centralis.
    Acta tropica, 1987, Volume: 44, Issue:1

    Topics: Animals; Diminazene; Pentamidine; Phenanthridines; Suramin; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African; Tsetse Flies

1987
The relapse of Trypanosoma brucei brucei infections after chemotherapy in rabbits.
    Acta tropica, 1988, Volume: 45, Issue:1

    Topics: Amidines; Animals; Diminazene; Female; Male; Mice; Rabbits; Recurrence; Suramin; Trypanosoma brucei brucei; Trypanosomiasis, African

1988
Efficacy of DL-alpha-difluoromethylornithine in a rat model of Pneumocystis carinii pneumonia.
    Antimicrobial agents and chemotherapy, 1988, Volume: 32, Issue:8

    Topics: Amphotericin B; Animals; Antiprotozoal Agents; Dapsone; Diminazene; Disease Models, Animal; Drug Combinations; Eflornithine; Female; Immunosuppression Therapy; Pneumonia, Pneumocystis; Random Allocation; Rats; Rats, Inbred Strains; Sulfamethoxazole; Suramin; Trimethoprim; Trimethoprim, Sulfamethoxazole Drug Combination

1988
Flow cytofluorimetric analysis of drug accumulation by multidrug-resistant Trypanosoma brucei brucei and T. b. rhodesiense.
    Molecular and biochemical parasitology, 1987, Volume: 26, Issue:1-2

    Topics: Acriflavine; Animals; Benzimidazoles; Diminazene; Drug Resistance; Ethidium; Flow Cytometry; Fluorescent Dyes; Humans; Indoles; Melarsoprol; Mice; Pentamidine; Suramin; Trypanocidal Agents; Trypanosoma brucei brucei

1987
An assay for screening drugs against animal-infective bloodstream forms of Trypanosoma brucei brucei in vitro.
    Drugs under experimental and clinical research, 1985, Volume: 11, Issue:3

    Topics: Animals; Diminazene; Mice; Parasitology; Quinolinium Compounds; Suramin; Trypanocidal Agents; Trypanosoma brucei brucei

1985
Arsenic and old taxa: subspeciation and drug sensitivity in Trypanosoma brucei.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1984, Volume: 78, Issue:6

    Topics: Animals; Arsenicals; Diminazene; Dose-Response Relationship, Drug; Drug Resistance, Microbial; Isoenzymes; Male; Melarsoprol; Mice; Pentamidine; Suramin; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African

1984
The use of the 2 substituted 5-nitroimidazole, Fexinidazole (Hoe 239) in the treatment of chronic T. brucei infections in mice.
    Zeitschrift fur Parasitenkunde (Berlin, Germany), 1983, Volume: 69, Issue:5

    Topics: Animals; Antiprotozoal Agents; Chronic Disease; Diminazene; Drug Therapy, Combination; Female; Mice; Mice, Inbred Strains; Nitroimidazoles; Suramin; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African

1983
Response of the rat's hepatic drug-metabolizing enzyme system to chemotherapy of Trypanosoma b. brucei infections with Berenil and Suramin.
    Enzyme, 1984, Volume: 31, Issue:3

    Topics: Amidines; Aminopyrine N-Demethylase; Aniline Hydroxylase; Animals; Diminazene; Female; Glutamate Dehydrogenase; Kinetics; L-Lactate Dehydrogenase; Liver; Microsomes, Liver; Phospholipids; Rats; Suramin; Trypanosoma brucei brucei; Trypanosomiasis, African

1984
Sensitivity of antigen ELISA test for detecting Trypanosoma evansi antigen in horses in the subtropical area of Argentina.
    The Journal of parasitology, 1995, Volume: 81, Issue:5

    Topics: Animals; Antigens, Protozoan; Argentina; Diminazene; Disease Outbreaks; Enzyme-Linked Immunosorbent Assay; Equidae; Horse Diseases; Horses; Sensitivity and Specificity; Suramin; Trypanocidal Agents; Trypanosoma; Trypanosomiasis

1995
Trypanosoma simiae: in vitro studies on drug susceptibility.
    Acta tropica, 1993, Volume: 54, Issue:3-4

    Topics: Animals; Arsenicals; Diminazene; Drug Resistance; Eflornithine; Parasitology; Quinolinium Compounds; Species Specificity; Suramin; Trypanocidal Agents; Trypanosoma

1993
Drug sensitivity of Chinese Trypanosoma evansi and Trypanosoma equiperdum isolates.
    Veterinary parasitology, 1994, Volume: 52, Issue:1-2

    Topics: Animals; Buffaloes; China; Diminazene; Drug Resistance; Female; Horses; Hypoxanthine; Hypoxanthines; Melarsoprol; Mice; Mice, Inbred ICR; Perissodactyla; Phenanthridines; Suramin; Trypanocidal Agents; Trypanosoma

1994
Combination chemotherapy of drug-resistant Trypanosoma brucei rhodesiense infections in mice using DL-alpha-difluoromethylornithine and standard trypanocides.
    Antimicrobial agents and chemotherapy, 1994, Volume: 38, Issue:3

    Topics: Animals; Arsenicals; Diminazene; Drug Interactions; Drug Resistance; Drug Therapy, Combination; Eflornithine; Female; Mice; Suramin; Trypanocidal Agents; Trypanosoma brucei rhodesiense; Trypanosomiasis, African

1994
Trypanosoma evansi: in vivo and in vitro determination of trypanocide resistance profiles.
    Experimental parasitology, 1993, Volume: 77, Issue:4

    Topics: Animals; Arsenicals; Diminazene; Drug Resistance; Phenanthridines; Quinolinium Compounds; Suramin; Trypanocidal Agents; Trypanosoma

1993
Trypanocidal resistance in Trypanosoma evansi in vitro: effects of verapamil, cyproheptidine, desipramine and chlorpromazine alone and in combination with trypanocides.
    Veterinary parasitology, 1996, Volume: 62, Issue:1-2

    Topics: Animals; Calcium Channel Blockers; Chlorpromazine; Cyproheptadine; Desipramine; Diminazene; Dose-Response Relationship, Drug; Drug Interactions; Drug Resistance, Multiple; Melarsoprol; Suramin; Trypanocidal Agents; Trypanosoma; Verapamil

1996
A trypanosome oligopeptidase as a target for the trypanocidal agents pentamidine, diminazene and suramin.
    FEBS letters, 1998, Aug-21, Volume: 433, Issue:3

    Topics: Animals; Diminazene; Pentamidine; Serine Endopeptidases; Serine Proteinase Inhibitors; Structure-Activity Relationship; Suramin; Trypanocidal Agents; Trypanosoma

1998
THE APPARENT LOSS OF THE KINETOPLAST OF TRYPANOSOMA EVANSI AFTER TREATMENT OF AN EXPERIMENTALLY INFECTED HORSE WITH BERENIL.
    Annals of tropical medicine and parasitology, 1964, Volume: 58

    Topics: Amidines; Animals; Blood; Blood Proteins; Cell Nucleus; Diminazene; Erythrocytes; Hemoglobins; Horses; Pharmacology; Rabbits; Rats; Research; Suramin; Triazines; Trypanosoma; Trypanosomiasis

1964
Bloodstream form-specific up-regulation of silent vsg expression sites and procyclin in Trypanosoma brucei after inhibition of DNA synthesis or DNA damage.
    The Journal of biological chemistry, 2004, Apr-02, Volume: 279, Issue:14

    Topics: Animals; Antiprotozoal Agents; Aphidicolin; Blood; Diminazene; DNA Damage; Enzyme Inhibitors; Gene Silencing; Genes, Reporter; Green Fluorescent Proteins; Luminescent Proteins; Membrane Glycoproteins; Pentamidine; Protozoan Proteins; RNA Polymerase I; S Phase; Suramin; Transcription, Genetic; Trypanocidal Agents; Trypanosoma brucei brucei; Up-Regulation; Variant Surface Glycoproteins, Trypanosoma

2004
Drug-resistance of Trypanosoma b. rhodesiense isolates from Tanzania.
    Tropical medicine & international health : TM & IH, 2006, Volume: 11, Issue:2

    Topics: Animals; Diminazene; Drug Resistance; Humans; Mass Screening; Melarsoprol; Phenanthridines; Recurrence; Suramin; Tanzania; Trypanocidal Agents; Trypanosoma brucei rhodesiense; Trypanosomiasis, African

2006
In vitro activity and preliminary toxicity of various diamidine compounds against Trypanosoma evansi.
    Veterinary parasitology, 2010, May-11, Volume: 169, Issue:3-4

    Topics: Amidines; Animals; Arsenicals; Cells, Cultured; Diminazene; Drug Resistance; Female; Inhibitory Concentration 50; Mice; Pentamidine; Quinolinium Compounds; Rats; Suramin; Trypanocidal Agents; Trypanosoma; Trypanosomiasis

2010
Curative drug treatment of trypanosomosis leads to the restoration of B-cell lymphopoiesis and splenic B-cell compartments.
    Parasite immunology, 2015, Volume: 37, Issue:9

    Topics: Animals; B-Lymphocyte Subsets; Bone Marrow; Diminazene; Female; Lymphopoiesis; Mice; Mice, Inbred C57BL; Spleen; Suramin; Trypanocidal Agents; Trypanosomiasis; Trypanosomiasis, African

2015
New Trypanosoma evansi Type B Isolates from Ethiopian Dromedary Camels.
    PLoS neglected tropical diseases, 2016, Volume: 10, Issue:4

    Topics: Animals; Arsenicals; Camelus; Diminazene; DNA, Kinetoplast; DNA, Protozoan; Ethiopia; Genotype; Mice; Phenanthridines; Phenotype; Phylogeny; Polymerase Chain Reaction; Proton-Translocating ATPases; Suramin; Triazines; Trypanocidal Agents; Trypanosoma; Trypanosomiasis

2016
Differential virulence of Trypanosoma brucei rhodesiense isolates does not influence the outcome of treatment with anti-trypanosomal drugs in the mouse model.
    PloS one, 2020, Volume: 15, Issue:11

    Topics: Animals; Diminazene; Disease Models, Animal; Drug Resistance; Kenya; Male; Melarsoprol; Mice; Pentamidine; Suramin; Treatment Outcome; Trypanocidal Agents; Trypanosoma brucei rhodesiense; Trypanosomiasis, African; Uganda; Virulence

2020