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suramin and 1-(5-isoquinolinesulfonyl)-2-methylpiperazine

suramin has been researched along with 1-(5-isoquinolinesulfonyl)-2-methylpiperazine in 11 studies

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (9.09)18.2507
2000's7 (63.64)29.6817
2010's3 (27.27)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chen, YH; Fu, WM; Lee, KF; Liou, JC1
Barnard, EA; Chessell, IP; Humphrey, PP; Jones, CA; Michel, AD; Miller, KJ; Simon, J1
Baldelli, P; Carabelli, V; Carbone, E; Hernández-Guijo, JM1
Kimura, J; Matsuoka, I; Watano, T1
Markwardt, F; Schmalzing, G; Seyffert, C1
Brock, JA; Yeoh, M1
Clay, WC; Condreay, JP; Fonfria, E; Goodwin, JA; Levy, DS; Michel, AD; Roman, S; Smith, GD1
Escartin, C; Nagasawa, K; Swanson, RA1
Jin, A; Junger, WG; Liu, J; Yu, T; Yuan, C; Zeng, Y; Zhao, Y; Zheng, X1
Iglesias, RM; Spray, DC1
Kanjanamekanant, K; Luckprom, P; Pavasant, P1

Other Studies

11 other study(ies) available for suramin and 1-(5-isoquinolinesulfonyl)-2-methylpiperazine

ArticleYear
Regulation of quantal transmitter secretion by ATP and protein kinases at developing neuromuscular synapses.
    The European journal of neuroscience, 1997, Volume: 9, Issue:4

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 6-Cyano-7-nitroquinoxaline-2,3-dione; Acetylcholine; Adenosine Triphosphate; Animals; Cells, Cultured; Coculture Techniques; Embryo, Nonmammalian; Enzyme Inhibitors; Evoked Potentials; Kinetics; Muscle, Skeletal; Neuromuscular Junction; Neurons; Protein Kinases; Quantum Theory; Suramin; Synapses; Synaptic Transmission; Theophylline; Triazines; Xenopus laevis

1997
Functional characterization of the P2X(4) receptor orthologues.
    British journal of pharmacology, 2000, Volume: 129, Issue:2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenine Nucleotides; Adenosine Triphosphate; Animals; Axons; Calcium-Calmodulin-Dependent Protein Kinases; Cell Line; Electric Stimulation; Electrophysiology; Enzyme Inhibitors; Humans; Membrane Potentials; Mice; Patch-Clamp Techniques; Purinergic P2 Receptor Agonists; Purinergic P2 Receptor Antagonists; Pyridoxal Phosphate; Rats; Receptors, Purinergic P2; Receptors, Purinergic P2X4; Recombinant Proteins; Suramin

2000
Direct autocrine inhibition and cAMP-dependent potentiation of single L-type Ca2+ channels in bovine chromaffin cells.
    The Journal of physiology, 2001, Apr-01, Volume: 532, Issue:Pt 1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 1-Methyl-3-isobutylxanthine; Adenosine Triphosphate; Animals; Autocrine Communication; Calcium; Calcium Channels, L-Type; Cattle; Cells, Cultured; Chromaffin Cells; Colforsin; Cyclic AMP; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enzyme Inhibitors; GABA Antagonists; Isoquinolines; Kinetics; Naloxone; Narcotic Antagonists; Patch-Clamp Techniques; Picrotoxin; Protein Kinase Inhibitors; Sulfonamides; Suramin

2001
Characteristics of ATP-induced current through P2X7 receptor in NG108-15 cells: unique antagonist sensitivity and lack of pore formation.
    Japanese journal of pharmacology, 2002, Volume: 88, Issue:4

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Triphosphate; Animals; Benzoxazoles; Cations; Cell Membrane Permeability; Fluorescent Dyes; Mice; Patch-Clamp Techniques; Purinergic P2 Receptor Antagonists; Pyridoxal Phosphate; Quinolinium Compounds; Rats; Receptors, Purinergic P2; Receptors, Purinergic P2X7; Suramin; Triazines; Tumor Cells, Cultured

2002
Dissecting individual current components of co-expressed human P2X1 and P2X7 receptors.
    Current topics in medicinal chemistry, 2004, Volume: 4, Issue:16

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Triphosphate; Animals; Benzenesulfonates; Dose-Response Relationship, Drug; Humans; In Vitro Techniques; Kinetics; Magnesium; Oocytes; Patch-Clamp Techniques; Purinergic P2 Receptor Agonists; Purinergic P2 Receptor Antagonists; Receptors, Purinergic P2; Receptors, Purinergic P2X; Receptors, Purinergic P2X7; Suramin; Time Factors; Xenopus laevis

2004
Rho kinase inhibitors reduce neurally evoked contraction of the rat tail artery in vitro.
    British journal of pharmacology, 2005, Volume: 146, Issue:6

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Triphosphate; Adrenergic alpha-Antagonists; Amides; Animals; Arteries; Clonidine; Electric Stimulation; Electrophysiology; Female; Idazoxan; In Vitro Techniques; Indoles; Intracellular Signaling Peptides and Proteins; Phenylephrine; Prazosin; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Purinergic P2 Receptor Antagonists; Pyridines; Rats; Rats, Wistar; rho-Associated Kinases; Suramin; Tail; Vasoconstriction

2005
Cloning and pharmacological characterization of the guinea pig P2X7 receptor orthologue.
    British journal of pharmacology, 2008, Volume: 153, Issue:3

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Triphosphate; Amino Acid Sequence; Animals; Cloning, Molecular; Guinea Pigs; Humans; Mice; Purinergic P2 Receptor Agonists; Purinergic P2 Receptor Antagonists; Rats; Receptors, Purinergic P2; Receptors, Purinergic P2X7; Rosaniline Dyes; Species Specificity; Suramin

2008
Astrocyte cultures exhibit P2X7 receptor channel opening in the absence of exogenous ligands.
    Glia, 2009, Apr-15, Volume: 57, Issue:6

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Triphosphate; Animals; Apyrase; Astrocytes; Benzenesulfonates; Benzoxazoles; Cell Line; Cells, Cultured; Gene Knockdown Techniques; Humans; Ligands; Mice; Phenolsulfonphthalein; Propidium; Purinergic P2 Receptor Antagonists; Quinolinium Compounds; Rats; Rats, Wistar; Receptors, Purinergic P2; Receptors, Purinergic P2X7; RNA, Small Interfering; Suramin

2009
Shockwaves increase T-cell proliferation and IL-2 expression through ATP release, P2X7 receptors, and FAK activation.
    American journal of physiology. Cell physiology, 2010, Volume: 298, Issue:3

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Triphosphate; Apyrase; Cell Proliferation; Cell Survival; Enzyme Activation; Focal Adhesion Kinase 1; High-Energy Shock Waves; Humans; Interleukin-2; Jurkat Cells; Lymphocyte Activation; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Purinergic P2 Receptor Antagonists; Receptors, Purinergic P2; Receptors, Purinergic P2X7; RNA Interference; Signal Transduction; Suramin; T-Lymphocytes

2010
Pannexin1-mediated ATP release provides signal transmission between Neuro2A cells.
    Neurochemical research, 2012, Volume: 37, Issue:6

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Triphosphatases; Adenosine Triphosphate; Animals; Apyrase; Carbenoxolone; Cell Communication; Cell Line, Tumor; Connexins; Gap Junctions; Humans; Membrane Potentials; Mice; Nerve Tissue Proteins; Neuroblastoma; Patch-Clamp Techniques; Purinergic P2X Receptor Antagonists; Signal Transduction; Suramin

2012
Mechanical stress-induced interleukin-1beta expression through adenosine triphosphate/P2X7 receptor activation in human periodontal ligament cells.
    Journal of periodontal research, 2013, Volume: 48, Issue:2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Diphosphate; Adenosine Triphosphate; Apyrase; Benzenesulfonates; Calcium Channel Blockers; Calcium Signaling; Cell Culture Techniques; Cell Survival; Cells, Cultured; Coloring Agents; Dactinomycin; Homeostasis; Humans; Interleukin-1beta; Luminescent Measurements; Periodontal Ligament; Purinergic P2X Receptor Antagonists; Receptors, Purinergic P2X7; RNA, Small Interfering; Signal Transduction; Stress, Mechanical; Suramin; Tetrazolium Salts; Thiazoles; Time Factors; Up-Regulation

2013