Page last updated: 2024-09-05

sunepitron and buspirone

sunepitron has been researched along with buspirone in 1 studies

Compound Research Comparison

Studies
(sunepitron)
Trials
(sunepitron)
Recent Studies (post-2010)
(sunepitron)
Studies
(buspirone)
Trials
(buspirone)
Recent Studies (post-2010) (buspirone)
10012,096351382

Protein Interaction Comparison

ProteinTaxonomysunepitron (IC50)buspirone (IC50)
5-hydroxytryptamine receptor 1AHomo sapiens (human)0.025
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)1.75
Angiotensin-converting enzyme Homo sapiens (human)0.024
D(2) dopamine receptorHomo sapiens (human)0.323
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)2.125
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)4.16
DRattus norvegicus (Norway rat)0.12
D(3) dopamine receptorRattus norvegicus (Norway rat)0.12
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.0266
D(2) dopamine receptorBos taurus (cattle)4
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)4.16
Alpha-1D adrenergic receptorHomo sapiens (human)1.077
D(1B) dopamine receptorRattus norvegicus (Norway rat)0.12
5-hydroxytryptamine receptor 2AHomo sapiens (human)2.286
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)0.016
D(4) dopamine receptorRattus norvegicus (Norway rat)0.12
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)2.125
D(3) dopamine receptorHomo sapiens (human)0.044
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.75
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)4.16
D(2) dopamine receptorRattus norvegicus (Norway rat)0.2055
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)3.9811
Alpha-2A adrenergic receptorBos taurus (cattle)0.025
Multidrug and toxin extrusion protein 1Homo sapiens (human)1.7
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.2666
Lysosomal alpha-glucosidaseBos taurus (cattle)0.03

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Becker, OM; Chen, D; Cheruku, S; Dhanoa, DS; Fichman, M; Heifetz, A; Kauffman, M; Marantz, Y; Mohanty, P; Noiman, S; Nudelman, R; Shacham, S; Sharadendu, A1

Other Studies

1 other study(ies) available for sunepitron and buspirone

ArticleYear
An integrated in silico 3D model-driven discovery of a novel, potent, and selective amidosulfonamide 5-HT1A agonist (PRX-00023) for the treatment of anxiety and depression.
    Journal of medicinal chemistry, 2006, Jun-01, Volume: 49, Issue:11

    Topics: Animals; Anti-Anxiety Agents; Antidepressive Agents; Binding, Competitive; Biological Availability; Cell Line; Clinical Trials, Phase I as Topic; Dogs; Drug Design; Half-Life; Humans; In Vitro Techniques; Male; Mice; Microsomes, Liver; Models, Molecular; Patch-Clamp Techniques; Piperazines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Serotonin 5-HT1 Receptor Agonists; Structure-Activity Relationship; Sulfonamides

2006