Page last updated: 2024-08-16

sumatriptan and pyrroles

sumatriptan has been researched along with pyrroles in 18 studies

Research

Studies (18)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's10 (55.56)18.2507
2000's5 (27.78)29.6817
2010's0 (0.00)24.3611
2020's3 (16.67)2.80

Authors

AuthorsStudies
Boccalini, P; Moskowitz, MA; Nozaki, K1
Byun, B; Matsubara, T; Moskowitz, MA1
Brain, SD; Gupta, P; Kajekar, R; Shepperson, NB1
Bruinvels, AT; Hoyer, D; Landwehrmeyer, B; Palacios, JM; Probst, A1
Byun, B; Huang, Z; Matsubara, T; Moskowitz, MA1
Castanon, N; Chauveau, J; Chaveau, J; Hen, R; Macor, JE; Moskowitz, MA; Scearce, K; Waeber, C; Yu, XJ1
Davidson, C; Stamford, JA2
Hotta, H; Messlinger, K; Pawlak, M; Schmidt, RF1
Anmella, MC; Gardier, AM; Hen, R; Jacquot, C; Malagié, I; Pons, D; Scearce, K; Trillat, AC1
Centurión, D; Rabelo, G; Sánchez-López, A; Villalón, CM1
Hopwood, SE; Stamford, JA1
Blier, P; Hen, R; Richer, M1
Arulmani, U; Centurión, D; Sánchez-López, A; Saxena, PR; Vázquez, E; Villalón, CM1
Jeggo, RD; Jordan, D; Ramage, AG; Wang, Y1
Boinpally, R; Butler, M; Jakate, A; Lu, K; McGeeney, D; Periclou, A1
Banerjee, P; Behravesh, S; Dodick, DW; Navratilova, E; Oyarzo, J; Porreca, F1
Boinpally, R; Butler, M; Jakate, A; Periclou, A1

Trials

2 trial(s) available for sumatriptan and pyrroles

ArticleYear
Evaluation of the Pharmacokinetic Interaction of Ubrogepant Coadministered With Sumatriptan and of the Safety of Ubrogepant With Triptans.
    Headache, 2020, Volume: 60, Issue:7

    Topics: Adult; Calcitonin Gene-Related Peptide Receptor Antagonists; Cross-Over Studies; Drug Interactions; Drug Therapy, Combination; Female; Humans; Male; Migraine Disorders; Pyridines; Pyrroles; Sumatriptan; Tryptamines

2020
Atogepant and sumatriptan: no clinically relevant drug-drug interactions in a randomized, open-label, crossover trial.
    Pain management, 2022, Volume: 12, Issue:4

    Topics: Adult; Area Under Curve; Cross-Over Studies; Drug Interactions; Humans; Piperidines; Pyridines; Pyrroles; Spiro Compounds; Sumatriptan

2022

Other Studies

16 other study(ies) available for sumatriptan and pyrroles

ArticleYear
CP-93,129, sumatriptan, dihydroergotamine block c-fos expression within rat trigeminal nucleus caudalis caused by chemical stimulation of the meninges.
    British journal of pharmacology, 1992, Volume: 106, Issue:2

    Topics: Animals; Animals, Newborn; Capsaicin; Carrageenan; Dihydroergotamine; Formaldehyde; Gene Expression Regulation, Neoplastic; Guinea Pigs; Immunohistochemistry; In Vitro Techniques; Indoles; Meninges; Nasal Mucosa; Proto-Oncogene Proteins c-fos; Pyridines; Pyrroles; Rats; Sulfonamides; Sumatriptan

1992
CP-93,129, a potent and selective 5-HT1B receptor agonist blocks neurogenic plasma extravasation within rat but not guinea-pig dura mater.
    British journal of pharmacology, 1991, Volume: 104, Issue:1

    Topics: Animals; Blood Pressure; Capsaicin; Dura Mater; Electric Stimulation; Guinea Pigs; Indoles; Ligands; Male; Plasma; Proteins; Pyridines; Pyrroles; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serum Albumin, Radio-Iodinated; Sulfonamides; Sumatriptan; Trigeminal Ganglion; Vasoconstrictor Agents

1991
Effect of a 5-HT1 receptor agonist, CP-122,288, on oedema formation induced by stimulation of the rat saphenous nerve.
    British journal of pharmacology, 1995, Volume: 115, Issue:1

    Topics: Analysis of Variance; Animals; Edema; Electric Stimulation; Male; Neuritis; Neurons, Afferent; Pyridines; Pyrroles; Pyrrolidines; Rats; Rats, Wistar; Serotonin Receptor Agonists; Sumatriptan

1995
A comparative autoradiographic study of 5-HT1D binding sites in human and guinea-pig brain using different radioligands.
    Brain research. Molecular brain research, 1994, Volume: 21, Issue:1-2

    Topics: Aged; Animals; Autoradiography; Binding Sites; Binding, Competitive; Brain; Dipeptides; Female; Guinea Pigs; Humans; Iodine Radioisotopes; Kinetics; Ligands; Male; Organ Specificity; Pyridines; Pyrroles; Receptors, Serotonin; Serotonin; Species Specificity; Sumatriptan; Tritium; Yohimbine

1994
Time-dependent blockade of neurogenic plasma extravasation in dura mater by 5-HT1B/D agonists and endopeptidase 24.11.
    British journal of pharmacology, 1993, Volume: 108, Issue:2

    Topics: Animals; Capsaicin; Disease Models, Animal; Dura Mater; Electric Stimulation; Extravasation of Diagnostic and Therapeutic Materials; Guinea Pigs; Indoles; Male; Neprilysin; Neuropeptides; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Serotonin Receptor Agonists; Sulfonamides; Sumatriptan; Time Factors; Trigeminal Ganglion

1993
5-Carboxamido-tryptamine, CP-122,288 and dihydroergotamine but not sumatriptan, CP-93,129, and serotonin-5-O-carboxymethyl-glycyl -tyrosinamide block dural plasma protein extravasation in knockout mice that lack 5-hydroxytryptamine1B receptors.
    Molecular pharmacology, 1996, Volume: 49, Issue:5

    Topics: Animals; Capillary Permeability; Dihydroergotamine; Dipeptides; Mice; Mice, Knockout; Pyridines; Pyrroles; Pyrrolidines; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Sumatriptan; Trigeminal Ganglion

1996
Chronic paroxetine desensitises 5-HT1D but not 5-HT1B autoreceptors in rat lateral geniculate nucleus.
    Brain research, 1997, Jun-20, Volume: 760, Issue:1-2

    Topics: Animals; Autoreceptors; Geniculate Bodies; Male; Paroxetine; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin Receptor Agonists; Sumatriptan; Time Factors

1997
Effects of the 5-HT1 receptor agonists, sumatriptan and CP 93,129, on dural arterial flow in the rat.
    European journal of pharmacology, 1997, Aug-06, Volume: 332, Issue:2

    Topics: Animals; Cerebrovascular Circulation; Dura Mater; Male; Meningeal Arteries; Pyridines; Pyrroles; Rats; Rats, Wistar; Serotonin Receptor Agonists; Sumatriptan; Trigeminal Ganglion

1997
Regulation of serotonin release in the frontal cortex and ventral hippocampus of homozygous mice lacking 5-HT1B receptors: in vivo microdialysis studies.
    Journal of neurochemistry, 1997, Volume: 69, Issue:5

    Topics: Animals; Frontal Lobe; Hippocampus; Homozygote; Male; Mice; Mice, Knockout; Mice, Transgenic; Microdialysis; Nerve Endings; Potassium; Pyridines; Pyrroles; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Sumatriptan

1997
Pharmacological profile of the prejunctional 5-HT1 receptors mediating inhibition of sympathetic vasopressor outflow in the pithed rat.
    Annals of the New York Academy of Sciences, 1998, Dec-15, Volume: 861

    Topics: 5-Methoxytryptamine; Animals; Blood Pressure; Central Nervous System; Oxadiazoles; Pindolol; Piperazines; Pyridines; Pyrroles; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Sympathetic Nervous System

1998
Effect of chronic paroxetine treatment on 5-HT1B and 5-HT1D autoreceptors in rat dorsal raphe nucleus.
    Neurochemistry international, 2000, Volume: 36, Issue:2

    Topics: Animals; Electric Stimulation; Male; Paroxetine; Piperazines; Pyridines; Pyrroles; Raphe Nuclei; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan

2000
Multiple 5-HT(1) autoreceptor subtypes govern serotonin release in dorsal and median raphé nuclei.
    Neuropharmacology, 2001, Volume: 40, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoreceptors; Benzamides; Biphenyl Compounds; Drug Synergism; Electric Stimulation; In Vitro Techniques; Male; Oxadiazoles; Piperazines; Protein Isoforms; Pyridines; Pyrroles; Raphe Nuclei; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Time Factors

2001
Modification of serotonin neuron properties in mice lacking 5-HT1A receptors.
    European journal of pharmacology, 2002, Jan-25, Volume: 435, Issue:2-3

    Topics: Animals; Autoreceptors; Brimonidine Tartrate; Hippocampus; In Vitro Techniques; Male; Mice; Neurons; Norepinephrine; Pyridines; Pyrroles; Quinoxalines; Raphe Nuclei; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Adrenergic, alpha-2; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Receptor Agonists; Sumatriptan; Tritium

2002
Further characterization of the 5-HT1 receptors mediating cardiac sympatho-inhibition in pithed rats: pharmacological correlation with the 5-HT1B and 5-HT1D subtypes.
    Naunyn-Schmiedeberg's archives of pharmacology, 2004, Volume: 369, Issue:2

    Topics: Animals; Biphenyl Compounds; Decerebrate State; Male; Norepinephrine; Oxadiazoles; Piperazines; Piperidones; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Spiro Compounds; Sumatriptan; Sympathomimetics; Tachycardia

2004
Activation of 5-HT1B and 5-HT1D receptors in the rat nucleus tractus solitarius: opposing action on neurones that receive an excitatory vagal C-fibre afferent input.
    British journal of pharmacology, 2007, Volume: 150, Issue:8

    Topics: Action Potentials; Animals; Benzamides; Drug Synergism; Electric Stimulation; Iontophoresis; Ketanserin; Male; Neural Inhibition; Neurons; Neurons, Afferent; Patch-Clamp Techniques; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Serotonin 5-HT1 Receptor Agonists; Serotonin Antagonists; Serotonin Receptor Agonists; Solitary Nucleus; Sumatriptan; Time Factors; Vagus Nerve

2007
Ubrogepant does not induce latent sensitization in a preclinical model of medication overuse headache.
    Cephalalgia : an international journal of headache, 2020, Volume: 40, Issue:9

    Topics: Analgesics; Animals; Central Nervous System Sensitization; Disease Models, Animal; Female; Headache Disorders, Secondary; Hyperalgesia; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Sumatriptan

2020