Page last updated: 2024-08-16

sumatriptan and methiothepin

sumatriptan has been researched along with methiothepin in 44 studies

Research

Studies (44)

TimeframeStudies, this research(%)All Research%
pre-19904 (9.09)18.7374
1990's36 (81.82)18.2507
2000's3 (6.82)29.6817
2010's1 (2.27)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Beer, MS; Charlesworth, A; Iversen, LL; McAllister, G; Middlemiss, DN; Noble, AJ; Snodin, C; Whiting, P1
Hamblin, MW; Metcalf, MA1
Bull, D; den Daas, I; Foord, S; Goodson, S; Kilpatrick, G; Lee, M; Rees, S1
Adham, N; Bard, JA; Branchek, TA; Vaysse, P; Weinshank, RL; Zgombick, J1
Adham, N; Bard, J; Branchek, TA; Durkin, M; Hartig, PR; Kao, HT; Olsen, M; Schecter, LE; Urquhart, D; Weinshank, RL1
Hamblin, MW; Jose, PA; Metcalf, MA; Monsma, FJ; Shen, Y; Sibley, DR1
Amlaiky, N; Boschert, U; Grailhe, R; Hen, R; Mattei, MG; Matthes, H; Muscatelli, F; Plassat, JL1
Druck, T; Hamblin, MW; Huebner, K; Khan, N; Kohen, R; Lachowicz, JE; Meltzer, HY; Metcalf, MA; Roth, BL; Sibley, DR1
Izzarelli, DG; Lewis-Higgins, L; Palmer, D; Parker, EM; Shapiro, RA1
Gommeren, W; Haegeman, G; Heylen, L; Lesage, AS; Leysen, JE; Luyten, WH; Schotte, A; Van de Weyer, I; Van Gompel, P; Vanhoenacker, P; Wouters, R1
Chang, DJ; Eglen, RM; Jasper, JR; Kosaka, A; To, ZP1
Boess, FG; Monsma, FJ; Sleight, AJ1
Grånäs, C; Larhammar, D1
Audinot, V; Millan, MJ; Moreira, C; Newman-Tancredi, A; Verrièle, L1
Grabtree, GW; Grailhe, R; Hen, R1
Bai, F; Johnstone, EM; Little, SP; Nelson, DL; Su, C; Varga, G; Yin, T1
Lepailleur, A; Rochais, C; Thirumaran, SL1
Connor, HE; Feniuk, W; Humphrey, PP; Stubbs, CM1
Middlemiss, DN; Wilkinson, LO1
Edvinsson, L; Jansen, I; Mortensen, A; Olesen, J1
den Boer, MO; Heiligers, JP; Saxena, PR1
Motevalian, M; Parsons, AA; Whalley, ET1
Feniuk, W; Humphrey, PP; Perren, MJ2
Higgins, GA; Jordan, CC; Skingle, M1
Hoyer, D; Sahin-Erdemli, I; Schoeffter, P; Seiler, MP; Stoll, A1
Connor, HE; Feniuk, W1
Bond, RA; Charlton, KG; Clarke, DE; Craig, DA; Ornstein, AG1
Butina, D; Coates, LH; Connor, HE; Feniuk, W; Humphrey, PP; Oxford, AW; Perren, MJ1
Clayton, RA; Hillis, SW; MacLean, MR; McIntyre, PD; Peacock, AJ; Templeton, AG1
Wallis, DI; Wang, XC; Wu, J1
Edvinsson, L; Jansen, I; Olesen, J1
Drieu la Rochelle, C; O'Connor, SE1
Bobirnac, I; Schoeffter, P1
Castillo, C; Castillo, E; López-Muñoz, FJ; Ramírez-San Juan, E; Terrón, JA; Villalón, CM1
Beattie, DT; Connor, HE; Walsh, DM1
Böing, C; Bühlen, M; Fink, K; Göthert, M1
Burton, M; Jones, BJ; Price, GW; Roberts, C; Watson, J1
Ay, I; Ciçek, S; Tatar, H; Tuncer, M; Yildiz, O1
Choppin, A; O'Connor, SE1
De Vries, P; Heiligers, JP; Saxena, PR; Villalón, CM1
López-Muñoz, FJ; Perusquía, M; Terrón, JA; Villalón, CM1
Bodelsson, G; Bodelsson, M; Karlsson, C; Stjernquist, M1
Bard, JA; Branchek, T; Edvinsson, L; Longmore, J; Nilsson, T; Pantev, E; Shaw, D1

Reviews

1 review(s) available for sumatriptan and methiothepin

ArticleYear
Structure-activity relationships of serotonin 5-HT
    European journal of medicinal chemistry, 2019, Dec-01, Volume: 183

    Topics: Animals; Humans; Ligands; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship

2019

Other Studies

43 other study(ies) available for sumatriptan and methiothepin

ArticleYear
Molecular cloning of a serotonin receptor from human brain (5HT1E): a fifth 5HT1-like subtype.
    Proceedings of the National Academy of Sciences of the United States of America, 1992, Jun-15, Volume: 89, Issue:12

    Topics: Adenylyl Cyclases; Amino Acid Sequence; Base Sequence; Binding, Competitive; Cell Line; Cloning, Molecular; Colforsin; DNA; Frontal Lobe; Gene Library; GTP-Binding Proteins; Hippocampus; Humans; Kinetics; Molecular Sequence Data; Oligodeoxyribonucleotides; Polymerase Chain Reaction; Receptors, Serotonin; Recombinant Proteins; Restriction Mapping; Sequence Homology, Nucleic Acid; Serotonin; Transfection

1992
Primary structure and functional characterization of a human 5-HT1D-type serotonin receptor.
    Molecular pharmacology, 1991, Volume: 40, Issue:2

    Topics: Amino Acid Sequence; Base Sequence; Cloning, Molecular; Cyclic AMP; GTP-Binding Proteins; Humans; Molecular Sequence Data; Pertussis Toxin; Receptors, Serotonin; Virulence Factors, Bordetella

1991
Cloning and characterisation of the human 5-HT5A serotonin receptor.
    FEBS letters, 1994, Dec-05, Volume: 355, Issue:3

    Topics: Amino Acid Sequence; Animals; Base Sequence; Brain Chemistry; Cloning, Molecular; Genome, Human; GTP-Binding Proteins; Humans; Mice; Molecular Sequence Data; Radioligand Assay; Receptors, Serotonin; Sequence Analysis, DNA; Sequence Homology, Amino Acid; Sequence Homology, Nucleic Acid; Serotonin; Tissue Distribution; Transfection

1994
Cloning of a novel human serotonin receptor (5-HT7) positively linked to adenylate cyclase.
    The Journal of biological chemistry, 1993, Nov-05, Volume: 268, Issue:31

    Topics: Adenylyl Cyclases; Base Sequence; Cloning, Molecular; DNA Primers; Humans; Molecular Sequence Data; Receptors, Serotonin; Sequence Alignment; Sequence Homology, Amino Acid; Serotonin Antagonists; Serotonin Receptor Agonists; Signal Transduction

1993
Cloning of another human serotonin receptor (5-HT1F): a fifth 5-HT1 receptor subtype coupled to the inhibition of adenylate cyclase.
    Proceedings of the National Academy of Sciences of the United States of America, 1993, Jan-15, Volume: 90, Issue:2

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Amino Acid Sequence; Animals; Base Sequence; Brain Chemistry; Cloning, Molecular; Colforsin; Dose-Response Relationship, Drug; Gene Library; Guinea Pigs; Humans; Indoles; Lymphocytes; Molecular Sequence Data; Receptors, Serotonin; RNA, Messenger; Sequence Homology, Amino Acid; Serotonin; Serotonin Receptor Agonists; Spiperone; Sulfonamides; Sumatriptan; Tissue Distribution

1993
Molecular cloning and expression of a 5-hydroxytryptamine7 serotonin receptor subtype.
    The Journal of biological chemistry, 1993, Aug-25, Volume: 268, Issue:24

    Topics: Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Cell Line; Cell Membrane; Cloning, Molecular; Cyclic AMP; Gene Expression; Kidney Tubules, Proximal; Lysergic Acid Diethylamide; Molecular Sequence Data; Oligodeoxyribonucleotides; Polymerase Chain Reaction; Radioligand Assay; Rats; Receptors, Serotonin; Recombinant Proteins; Serotonin; Transfection

1993
Mouse 5-hydroxytryptamine5A and 5-hydroxytryptamine5B receptors define a new family of serotonin receptors: cloning, functional expression, and chromosomal localization.
    Molecular pharmacology, 1993, Volume: 43, Issue:3

    Topics: Amino Acid Sequence; Animals; Base Sequence; Brain; Cell Line; Chromosome Mapping; Cloning, Molecular; DNA; Gene Expression; Humans; In Situ Hybridization; Mice; Molecular Sequence Data; Receptors, Serotonin; Serotonin Receptor Agonists

1993
Cloning, characterization, and chromosomal localization of a human 5-HT6 serotonin receptor.
    Journal of neurochemistry, 1996, Volume: 66, Issue:1

    Topics: Adenylyl Cyclases; Amino Acid Sequence; Animals; Antipsychotic Agents; Base Sequence; Brain Chemistry; Cell Line, Transformed; Chlorocebus aethiops; Chromosome Mapping; Chromosomes, Human, Pair 1; Cloning, Molecular; Clozapine; DNA, Complementary; Genes; Humans; Kinetics; Molecular Sequence Data; Open Reading Frames; Protein Conformation; Rats; Receptors, Serotonin; Recombinant Proteins; Sequence Alignment; Sequence Homology, Nucleic Acid; Serotonin Agents; Signal Transduction; Species Specificity

1996
Two amino acid differences in the sixth transmembrane domain are partially responsible for the pharmacological differences between the 5-HT1D beta and 5-HT1E 5-hydroxytryptamine receptors.
    Journal of neurochemistry, 1996, Volume: 67, Issue:5

    Topics: Amino Acid Sequence; Animals; Base Sequence; Binding Sites; Binding, Competitive; Chlorocebus aethiops; Cloning, Molecular; COS Cells; DNA Primers; Ergolines; Glutamic Acid; Humans; Isoleucine; Kinetics; Ligands; Lysine; Models, Structural; Molecular Sequence Data; Point Mutation; Polymerase Chain Reaction; Protein Structure, Secondary; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Recombinant Fusion Proteins; Sequence Homology, Amino Acid; Serine; Serotonin; Transfection

1996
Alniditan, a new 5-hydroxytryptamine1D agonist and migraine-abortive agent: ligand-binding properties of human 5-hydroxytryptamine1D alpha, human 5-hydroxytryptamine1D beta, and calf 5-hydroxytryptamine1D receptors investigated with [3H]5-hydroxytryptamin
    Molecular pharmacology, 1996, Volume: 50, Issue:6

    Topics: Animals; Benzopyrans; Cattle; Cloning, Molecular; Glioma; HeLa Cells; Humans; Mice; Migraine Disorders; Propylamines; Protein Binding; Pyrimidines; Radioligand Assay; Receptors, Serotonin; Serotonin Receptor Agonists; Signal Transduction; Tritium; Tumor Cells, Cultured; Vasoconstrictor Agents

1996
Cloning, expression and pharmacology of a truncated splice variant of the human 5-HT7 receptor (h5-HT7b).
    British journal of pharmacology, 1997, Volume: 122, Issue:1

    Topics: Alternative Splicing; Amino Acid Sequence; Animals; Base Sequence; Cloning, Molecular; Cyclic AMP; DNA, Complementary; Humans; Molecular Sequence Data; Placenta; Radioligand Assay; Rats; Receptors, Serotonin; RNA, Messenger; Sequence Homology, Amino Acid; Sequence Homology, Nucleic Acid

1997
Identification of residues in transmembrane regions III and VI that contribute to the ligand binding site of the serotonin 5-HT6 receptor.
    Journal of neurochemistry, 1998, Volume: 71, Issue:5

    Topics: Adenylyl Cyclases; Amino Acid Substitution; Binding Sites; Binding, Competitive; Cell Line; Cyclic AMP; Humans; Ligands; Lysergic Acid Diethylamide; Mutagenesis, Site-Directed; Mutation; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists

1998
Identification of an amino acid residue important for binding of methiothepin and sumatriptan to the human 5-HT(1B) receptor.
    European journal of pharmacology, 1999, Sep-10, Volume: 380, Issue:2-3

    Topics: Amino Acid Sequence; Amino Acids; Animals; Benzamides; Binding Sites; Binding, Competitive; CHO Cells; Cricetinae; Dose-Response Relationship, Drug; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Methiothepin; Molecular Sequence Data; Mutation; Protein Binding; Pyridines; Radioligand Assay; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Sequence Homology, Amino Acid; Serotonin Antagonists; Serotonin Receptor Agonists; Sodium; Sumatriptan; Tritium

1999
Inverse agonism and constitutive activity as functional correlates of serotonin h5-HT(1B) receptor/G-protein stoichiometry.
    Molecular pharmacology, 2000, Volume: 58, Issue:5

    Topics: Animals; Binding, Competitive; Cell Membrane; CHO Cells; Cricetinae; Dose-Response Relationship, Drug; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Ligands; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin Antagonists; Sulfur Radioisotopes; Tritium

2000
Human 5-HT(5) receptors: the 5-HT(5A) receptor is functional but the 5-HT(5B) receptor was lost during mammalian evolution.
    European journal of pharmacology, 2001, Apr-27, Volume: 418, Issue:3

    Topics: 3T3 Cells; Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Cell Line; COS Cells; DNA; Evolution, Molecular; Gene Expression; Genes; Humans; Membranes; Mice; Molecular Sequence Data; Phylogeny; Radioligand Assay; Receptors, Serotonin; Sequence Alignment; Sequence Analysis, DNA; Sequence Homology, Amino Acid

2001
Molecular cloning and pharmacological characterization of the guinea pig 5-HT1E receptor.
    European journal of pharmacology, 2004, Jan-26, Volume: 484, Issue:2-3

    Topics: Amino Acid Sequence; Animals; Base Sequence; Brain; Chickens; Cloning, Molecular; Cricetinae; Dose-Response Relationship, Drug; Gerbillinae; Guinea Pigs; Haplorhini; Humans; Molecular Sequence Data; Protein Binding; Rabbits; Receptors, Serotonin; Serotonin Agents; Swine

2004
Effect of sumatriptan, a selective 5-HT1-like receptor agonist, on pial vessel diameter in anaesthetised cats.
    Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 1992, Volume: 12, Issue:3

    Topics: Animals; Biological Transport; Cats; Cerebral Arteries; Cerebral Veins; Female; Homeostasis; Indoles; Male; Methiothepin; Pia Mater; Receptors, Serotonin; Sulfonamides; Sumatriptan; Vasoconstriction

1992
Metitepine distinguishes two receptors mediating inhibition of [3H]-5-hydroxytryptamine release in guinea pig hippocampus.
    Naunyn-Schmiedeberg's archives of pharmacology, 1992, Volume: 345, Issue:6

    Topics: Animals; Culture Techniques; Electric Stimulation; Guinea Pigs; Hippocampus; Indoles; Male; Methiothepin; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sulfonamides; Sumatriptan

1992
Sumatriptan is a potent vasoconstrictor of human dural arteries via a 5-HT1-like receptor.
    Cephalalgia : an international journal of headache, 1992, Volume: 12, Issue:4

    Topics: Cerebral Arteries; Humans; In Vitro Techniques; Indoles; Ketanserin; Meningeal Arteries; Methiothepin; Receptors, Serotonin; Sulfonamides; Sumatriptan; Temporal Arteries; Vasoconstrictor Agents

1992
Carotid vascular effects of ergotamine and dihydroergotamine in the pig: no exclusive mediation via 5-HT1-like receptors.
    British journal of pharmacology, 1991, Volume: 104, Issue:1

    Topics: Animals; Arteriovenous Anastomosis; Brain Chemistry; Carotid Arteries; Coronary Circulation; Dihydroergotamine; Dose-Response Relationship, Drug; Ergotamine; Hemodynamics; Indoles; Methiothepin; Muscle, Smooth, Vascular; Oxygen Consumption; Receptors, Serotonin; Sulfonamides; Sumatriptan; Swine; Vasoconstrictor Agents

1991
Contractile effects of 8-hydroxy-2-(di-n-propylamino)tetralin and flesinoxan in human isolated basilar artery.
    European journal of pharmacology, 1991, Sep-04, Volume: 202, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Antihypertensive Agents; Basilar Artery; Humans; In Vitro Techniques; Indoles; Methiothepin; Muscle Contraction; Muscle, Smooth, Vascular; Phentolamine; Piperazines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiperone; Sulfonamides; Sumatriptan; Tetrahydronaphthalenes; Vasoconstrictor Agents

1991
Vascular 5-HT1-like receptors that mediate contraction of the dog isolated saphenous vein and carotid arterial vasoconstriction in anaesthetized dogs are not of the 5-HT1A or 5-HT1D subtype.
    British journal of pharmacology, 1991, Volume: 102, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Anesthesia; Animals; Atropine; Carotid Arteries; Dogs; Ganglionic Blockers; In Vitro Techniques; Indoles; Ketanserin; Methiothepin; Muscle, Smooth, Vascular; Pyrilamine; Receptors, Serotonin; Saphenous Vein; Spiperone; Sulfonamides; Sumatriptan; Tetrahydronaphthalenes; Vasoconstriction; Vasoconstrictor Agents

1991
Evidence that the unilateral activation of 5-HT1D receptors in the substantia nigra of the guinea-pig elicits contralateral rotation.
    British journal of pharmacology, 1991, Volume: 102, Issue:2

    Topics: Animals; Behavior, Animal; Guinea Pigs; Indoles; Male; Methiothepin; Movement; Receptors, Serotonin; Rotation; Serotonin; Substantia Nigra; Sulfonamides; Sumatriptan

1991
5-HT1-like receptors mediate 5-hydroxytryptamine-induced contraction of guinea-pig isolated iliac artery.
    British journal of pharmacology, 1991, Volume: 102, Issue:2

    Topics: Animals; Guinea Pigs; Iliac Artery; In Vitro Techniques; Indoles; Ketanserin; Male; Methiothepin; Receptors, Serotonin; Serotonin; Sulfonamides; Sumatriptan; Tropisetron; Vasoconstriction

1991
Influence of the endothelium on contractile effects of 5-hydroxytryptamine and selective 5-HT agonists in canine basilar artery.
    British journal of pharmacology, 1989, Volume: 96, Issue:1

    Topics: Animals; Basilar Artery; Detergents; Dogs; Endothelium, Vascular; Female; In Vitro Techniques; Indoles; Ketanserin; Male; Methiothepin; Microscopy, Electron, Scanning; Octoxynol; Polyethylene Glycols; Potassium Chloride; Serotonin; Serotonin Antagonists; Sulfonamides; Sumatriptan

1989
The selective carotid arterial vasoconstrictor action of GR43175 in anaesthetized dogs.
    British journal of pharmacology, 1989, Volume: 96, Issue:1

    Topics: Animals; Barbital; Carotid Arteries; Dogs; Female; Hemodynamics; Indoles; Ketanserin; Male; Methiothepin; Phentolamine; Serotonin Antagonists; Sulfonamides; Sumatriptan; Tropanes; Vasoconstrictor Agents

1989
Partial agonistic activity of GR43175 at the inhibitory prejunctional 5-HT1-like receptor in rat kidney.
    Journal of autonomic pharmacology, 1989, Volume: 9, Issue:3

    Topics: Animals; Electric Stimulation; In Vitro Techniques; Indoles; Kidney; Male; Methiothepin; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Sulfonamides; Sumatriptan; Sympathetic Nervous System

1989
GR43175, a selective agonist for the 5-HT1-like receptor in dog isolated saphenous vein.
    British journal of pharmacology, 1988, Volume: 94, Issue:4

    Topics: Animals; Cats; Dogs; Female; In Vitro Techniques; Indoles; Male; Methiothepin; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Pindolol; Rabbits; Rats; Receptors, Serotonin; Saphenous Vein; Serotonin Antagonists; Sulfonamides; Sumatriptan; Swine; Tropanes; Vagus Nerve

1988
5-HT1-receptor-mediated vasoconstriction in bovine isolated pulmonary arteries: influences of vascular endothelium and tone.
    Pulmonary pharmacology, 1994, Volume: 7, Issue:1

    Topics: Amino Acid Oxidoreductases; Animals; Arginine; Cattle; Drug Interactions; Endothelium, Vascular; In Vitro Techniques; Ketanserin; Methiothepin; Muscle Contraction; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Pulmonary Artery; Receptors, Serotonin; Sensitivity and Specificity; Serotonin; Serotonin Antagonists; Sumatriptan; Vasoconstriction

1994
Is 5-hydroxytryptamine mediating descending inhibition in the neonatal rat spinal cord through different receptor subtypes?
    European journal of pharmacology, 1993, Dec-21, Volume: 250, Issue:3

    Topics: Animals; Animals, Newborn; Citalopram; Dioxanes; Dopamine Antagonists; Electric Stimulation; Ketanserin; Lumbar Vertebrae; Methiothepin; Methysergide; Rats; Receptors, Serotonin; Reflex, Monosynaptic; Serotonin; Spinal Cord; Spinal Nerve Roots; Spiperone; Spiro Compounds; Sulpiride; Sumatriptan

1993
5-Hydroxytryptamine receptor characterization of human cerebral, middle meningeal and temporal arteries: regional differences.
    Acta physiologica Scandinavica, 1993, Volume: 147, Issue:2

    Topics: 5-Methoxytryptamine; Cerebral Arteries; Humans; Indoles; Ketanserin; Meningeal Arteries; Methiothepin; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides; Sumatriptan; Temporal Arteries; Vasoconstriction; Vasoconstrictor Agents

1993
Sumatriptan-induced saphenous venoconstriction in the anaesthetized dog through 5-HT1-like receptor activation.
    British journal of pharmacology, 1995, Volume: 116, Issue:4

    Topics: Anesthesia; Animals; Aorta, Thoracic; Brachial Artery; Dogs; Dose-Response Relationship, Drug; Female; Hemodynamics; Male; Methiothepin; Muscle, Smooth, Vascular; Receptors, Serotonin; Saphenous Vein; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Vasoconstriction

1995
5-Hydroxytryptamine 5-HT1D receptors mediating inhibition of cyclic AMP accumulation in Madin-Darby canine kidney (MDCK) cells.
    Naunyn-Schmiedeberg's archives of pharmacology, 1995, Volume: 352, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Alprostadil; Animals; Cells, Cultured; Cyclic AMP; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Epithelial Cells; Epithelium; Ketanserin; Kidney Cortex; Methiothepin; Oxadiazoles; Pertussis Toxin; Piperazines; Propranolol; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship; Sumatriptan; Virulence Factors, Bordetella; Yohimbine

1995
Pharmacological profile of the receptors that mediate external carotid vasoconstriction by 5-HT in vagosympathectomized dogs.
    British journal of pharmacology, 1995, Volume: 116, Issue:6

    Topics: Animals; Carotid Artery, External; Dogs; Dose-Response Relationship, Drug; Female; Hemodynamics; Male; Metergoline; Methiothepin; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Sympathectomy; Vagus Nerve; Vasoconstriction

1995
The activity of 5-HT1D receptor ligands at cloned human 5-HT1D alpha and 5-HT1D beta receptors.
    European journal of pharmacology, 1995, Dec-04, Volume: 287, Issue:1

    Topics: Cyclic AMP; HeLa Cells; Humans; Metergoline; Methiothepin; Oxadiazoles; Piperazines; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan

1995
Evidence for presynaptic location of inhibitory 5-HT1D beta-like autoreceptors in the guinea-pig brain cortex.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 353, Issue:3

    Topics: Animals; Autoreceptors; Binding, Competitive; Cerebral Cortex; Guinea Pigs; Humans; Indoles; Ketanserin; Male; Methiothepin; Oxadiazoles; Oxymetazoline; Potassium; Radioligand Assay; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship; Sumatriptan; Synaptosomes; Tritium; Tryptamines

1996
Functional characterization of the 5-HT terminal autoreceptor in the guinea-pig brain cortex.
    British journal of pharmacology, 1996, Volume: 117, Issue:2

    Topics: Animals; Calcium Channel Blockers; Cerebral Cortex; Guinea Pigs; In Vitro Techniques; Male; Methiothepin; omega-Conotoxins; Peptides; Prefrontal Cortex; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan

1996
5-HT1-like receptor-mediated contraction in the human internal mammary artery.
    Journal of cardiovascular pharmacology, 1996, Volume: 28, Issue:1

    Topics: Adult; Dose-Response Relationship, Drug; Female; Humans; In Vitro Techniques; Ketanserin; Mammary Arteries; Methiothepin; Middle Aged; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Vasoconstriction; Vasoconstrictor Agents

1996
Influence of vascular tone on vasoconstrictor responses to the 5-HT 1-like receptor agonist sumatriptan in anaesthetised rabbits.
    European journal of pharmacology, 1996, May-23, Volume: 304, Issue:1-3

    Topics: Angiotensin II; Animals; Antihypertensive Agents; Blood Pressure; Chlorisondamine; Drug Synergism; Enalapril; Ganglionic Blockers; Heart Rate; Male; Methiothepin; Muscle, Smooth, Vascular; Rabbits; Regional Blood Flow; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Vascular Resistance; Vasoconstriction; Vasoconstrictor Agents

1996
Nature of 5-HT1-like receptors mediating depressor responses in vagosympathectomized rats; close resemblance to the cloned 5-ht7 receptor.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 356, Issue:1

    Topics: 5-Methoxytryptamine; Adrenergic beta-Agonists; Animals; Blood Pressure; Clozapine; Ergolines; Heart Rate; Isoproterenol; Lisuride; Male; Metergoline; Methiothepin; Oxadiazoles; Piperazines; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Sympathectomy

1997
External carotid effects of 2-(2-aminoethyl)-quinoline (D-1997) in vagosympathectomized dogs.
    European journal of pharmacology, 1998, Aug-28, Volume: 356, Issue:1

    Topics: Animals; Carotid Artery, External; Dogs; Dose-Response Relationship, Drug; Female; Hemodynamics; Male; Methiothepin; Quinolines; Regional Blood Flow; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sodium Chloride; Sumatriptan; Sympathectomy; Vagotomy; Vasoconstriction

1998
Characterization of 5-hydroxytryptamine receptors mediating circular smooth muscle contraction in the human umbilical artery.
    Gynecologic and obstetric investigation, 1999, Volume: 47, Issue:2

    Topics: Adolescent; Adult; Female; Humans; Ketanserin; Methiothepin; Muscle Contraction; Muscle, Smooth; Pregnancy; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Tropanes; Umbilical Arteries

1999
Characterisation of 5-HT receptors in human coronary arteries by molecular and pharmacological techniques.
    European journal of pharmacology, 1999, May-07, Volume: 372, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Cardiovascular System; Coronary Vessels; Dose-Response Relationship, Drug; Gene Expression; Humans; Immunohistochemistry; In Vitro Techniques; Ketanserin; Methiothepin; Oxazoles; Oxazolidinones; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Tissue Distribution; Tryptamines; Vasoconstriction

1999