Page last updated: 2024-08-16

sumatriptan and ketanserin

sumatriptan has been researched along with ketanserin in 54 studies

Research

Studies (54)

TimeframeStudies, this research(%)All Research%
pre-19903 (5.56)18.7374
1990's34 (62.96)18.2507
2000's12 (22.22)29.6817
2010's5 (9.26)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Buckingham, J; Glen, RC; Hill, AP; Hyde, RM; Martin, GR; Robertson, AD; Salmon, JA; Woollard, PM1
Bull, D; den Daas, I; Foord, S; Goodson, S; Kilpatrick, G; Lee, M; Rees, S1
Adham, N; Bard, JA; Branchek, TA; Vaysse, P; Weinshank, RL; Zgombick, J1
Hamblin, MW; Jose, PA; Metcalf, MA; Monsma, FJ; Shen, Y; Sibley, DR1
Gommeren, W; Haegeman, G; Heylen, L; Lesage, AS; Leysen, JE; Luyten, WH; Schotte, A; Van de Weyer, I; Van Gompel, P; Vanhoenacker, P; Wouters, R1
Chang, DJ; Eglen, RM; Jasper, JR; Kosaka, A; To, ZP1
Beer, MS; Castro, JL; Guiblin, AR; Jelley, RA; Matassa, VG; Russell, MG; Stanton, JA; Sternfeld, F; Street, LJ1
Beer, MS; Broughton, HB; Castro, JL; Hitzel, L; Matassa, VG; Pengilley, RR; Russell, MG; Sohal, B; Stanton, JA; van Niel, MB; Watt, AP1
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Cleves, AE; Jain, AN; Kirshner, D; Langham, JJ; Spitzer, R1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Lepailleur, A; Rochais, C; Thirumaran, SL1
Edvinsson, L; Jansen, I; Mortensen, A; Olesen, J1
Feniuk, W; Saxena, PR; Tadipatri, S; van Heuven-Nolsen, D1
Feniuk, W; Humphrey, PP; Perren, MJ2
Hoyer, D; Sahin-Erdemli, I; Schoeffter, P; Seiler, MP; Stoll, A1
Gaw, AJ; Humphrey, PP; Wadsworth, RM1
Connor, HE; Feniuk, W1
Connor, HE; Feniuk, W; Humphrey, PP1
Hill, RG; Longmore, J; Razzaque, Z1
Clayton, RA; Hillis, SW; MacLean, MR; McIntyre, PD; Peacock, AJ; Templeton, AG1
Martin, GR; Mills, A1
Bax, WA; Bos, E; Renzenbrink, GJ; Saxena, PR; Thijssen, EJ; Van Heuven-Nolsen, D1
Brown, AM; Frenken, M; Kaumann, AJ; Posival, H1
Wallis, DI; Wang, XC; Wu, J1
Bobker, DH1
Edvinsson, L; Jansen, I; Olesen, J1
Bobirnac, I; Schoeffter, P1
Crick, H; Manuel, NA; Wallis, DI1
Frölich, D; Göthert, M; Likungu, J; Molderings, GJ1
Böing, C; Bühlen, M; Fink, K; Göthert, M1
Terrón, JA1
Freudenthaler, S; Kaumann, AJ; Meyer-Dulheuer, F; Verheggen, R1
Ay, I; Ciçek, S; Tatar, H; Tuncer, M; Yildiz, O1
Bodelsson, G; Bodelsson, M; Karlsson, C; Stjernquist, M1
Bard, JA; Branchek, T; Edvinsson, L; Longmore, J; Nilsson, T; Pantev, E; Shaw, D1
Li, XF; Lovren, F; Lytton, J; Triggle, C1
Bult, H; Geerts, IS; Herman, AG; Matthys, KE1
Bischoff, A; Diener, H; Fetscher, C; Limmroth, V; Michel, MC; Wermelskirchen, D1
Ferrari, MD; Maassen Van Den Brink, A; Roon, KI; Saxena, PR1
Akita, H; Inoue, N; Ishida, T; Kawashima, S; Miwa, Y; Sakoda, T; Shimokawa, Y; Shiomi, M; Ueyama, T; Yokoyama, M1
Watts, SW1
Copolov, D; Dean, B; Pavey, G; Scarr, E2
Datté, JY; Offoumou, MA1
Jähnichen, S; Pertz, HH; Radtke, OA1
Gupta, S; Hanff, LM; MaassenVanDenBrink, A; Saxena, PR; Steegers, EA; Visser, W; Vulto, AG2
Jeggo, RD; Jordan, D; Ramage, AG; Wang, Y1
Chen, PB; Hargreaves, KM; Loyd, DR1

Reviews

1 review(s) available for sumatriptan and ketanserin

ArticleYear
Structure-activity relationships of serotonin 5-HT
    European journal of medicinal chemistry, 2019, Dec-01, Volume: 183

    Topics: Animals; Humans; Ligands; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship

2019

Other Studies

53 other study(ies) available for sumatriptan and ketanserin

ArticleYear
Computer-aided design and synthesis of 5-substituted tryptamines and their pharmacology at the 5-HT1D receptor: discovery of compounds with potential anti-migraine properties.
    Journal of medicinal chemistry, 1995, Sep-01, Volume: 38, Issue:18

    Topics: Animals; Aorta; Computer-Aided Design; Drug Design; Haplorhini; In Vitro Techniques; Migraine Disorders; Models, Chemical; Rabbits; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1D; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Saphenous Vein; Serotonin Receptor Agonists; Structure-Activity Relationship; Tryptamines

1995
Cloning and characterisation of the human 5-HT5A serotonin receptor.
    FEBS letters, 1994, Dec-05, Volume: 355, Issue:3

    Topics: Amino Acid Sequence; Animals; Base Sequence; Brain Chemistry; Cloning, Molecular; Genome, Human; GTP-Binding Proteins; Humans; Mice; Molecular Sequence Data; Radioligand Assay; Receptors, Serotonin; Sequence Analysis, DNA; Sequence Homology, Amino Acid; Sequence Homology, Nucleic Acid; Serotonin; Tissue Distribution; Transfection

1994
Cloning of a novel human serotonin receptor (5-HT7) positively linked to adenylate cyclase.
    The Journal of biological chemistry, 1993, Nov-05, Volume: 268, Issue:31

    Topics: Adenylyl Cyclases; Base Sequence; Cloning, Molecular; DNA Primers; Humans; Molecular Sequence Data; Receptors, Serotonin; Sequence Alignment; Sequence Homology, Amino Acid; Serotonin Antagonists; Serotonin Receptor Agonists; Signal Transduction

1993
Molecular cloning and expression of a 5-hydroxytryptamine7 serotonin receptor subtype.
    The Journal of biological chemistry, 1993, Aug-25, Volume: 268, Issue:24

    Topics: Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Cell Line; Cell Membrane; Cloning, Molecular; Cyclic AMP; Gene Expression; Kidney Tubules, Proximal; Lysergic Acid Diethylamide; Molecular Sequence Data; Oligodeoxyribonucleotides; Polymerase Chain Reaction; Radioligand Assay; Rats; Receptors, Serotonin; Recombinant Proteins; Serotonin; Transfection

1993
Alniditan, a new 5-hydroxytryptamine1D agonist and migraine-abortive agent: ligand-binding properties of human 5-hydroxytryptamine1D alpha, human 5-hydroxytryptamine1D beta, and calf 5-hydroxytryptamine1D receptors investigated with [3H]5-hydroxytryptamin
    Molecular pharmacology, 1996, Volume: 50, Issue:6

    Topics: Animals; Benzopyrans; Cattle; Cloning, Molecular; Glioma; HeLa Cells; Humans; Mice; Migraine Disorders; Propylamines; Protein Binding; Pyrimidines; Radioligand Assay; Receptors, Serotonin; Serotonin Receptor Agonists; Signal Transduction; Tritium; Tumor Cells, Cultured; Vasoconstrictor Agents

1996
Cloning, expression and pharmacology of a truncated splice variant of the human 5-HT7 receptor (h5-HT7b).
    British journal of pharmacology, 1997, Volume: 122, Issue:1

    Topics: Alternative Splicing; Amino Acid Sequence; Animals; Base Sequence; Cloning, Molecular; Cyclic AMP; DNA, Complementary; Humans; Molecular Sequence Data; Placenta; Radioligand Assay; Rats; Receptors, Serotonin; RNA, Messenger; Sequence Homology, Amino Acid; Sequence Homology, Nucleic Acid

1997
3-[2-(Pyrrolidin-1-yl)ethyl]indoles and 3-[3-(piperidin-1-yl)propyl]indoles: agonists for the h5-HT1D receptor with high selectivity over the h5-HT1B subtype.
    Journal of medicinal chemistry, 1997, Oct-24, Volume: 40, Issue:22

    Topics: Humans; Piperidines; Protein Binding; Pyrrolidines; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Recombinant Proteins; Serotonin Receptor Agonists

1997
3-[3-(Piperidin-1-yl)propyl]indoles as highly selective h5-HT(1D) receptor agonists.
    Journal of medicinal chemistry, 1999, Dec-02, Volume: 42, Issue:24

    Topics: Animals; Biological Availability; CHO Cells; Computer Simulation; Cricetinae; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Indoles; Male; Models, Molecular; Molecular Structure; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Recombinant Proteins; Serotonin Receptor Agonists; Structure-Activity Relationship; Transfection; Triazoles

1999
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Physical binding pocket induction for affinity prediction.
    Journal of medicinal chemistry, 2009, Oct-08, Volume: 52, Issue:19

    Topics: Binding Sites; Ligands; Models, Molecular; Neural Networks, Computer; Peptide Fragments; Protein Binding; Receptor, Serotonin, 5-HT1A

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Sumatriptan is a potent vasoconstrictor of human dural arteries via a 5-HT1-like receptor.
    Cephalalgia : an international journal of headache, 1992, Volume: 12, Issue:4

    Topics: Cerebral Arteries; Humans; In Vitro Techniques; Indoles; Ketanserin; Meningeal Arteries; Methiothepin; Receptors, Serotonin; Sulfonamides; Sumatriptan; Temporal Arteries; Vasoconstrictor Agents

1992
Analysis of the 5-HT receptors mediating contractions in the rabbit isolated renal artery.
    British journal of pharmacology, 1991, Volume: 104, Issue:4

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Cocaine; In Vitro Techniques; Indoles; Ketanserin; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Oxidopamine; Phentolamine; Prostaglandin Endoperoxides, Synthetic; Rabbits; Receptors, Serotonin; Renal Artery; Serotonin; Serotonin Antagonists; Sulfonamides; Sumatriptan; Sympathectomy; Tetrahydronaphthalenes; Tyramine; Vasoconstrictor Agents; Vasodilation

1991
Vascular 5-HT1-like receptors that mediate contraction of the dog isolated saphenous vein and carotid arterial vasoconstriction in anaesthetized dogs are not of the 5-HT1A or 5-HT1D subtype.
    British journal of pharmacology, 1991, Volume: 102, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Anesthesia; Animals; Atropine; Carotid Arteries; Dogs; Ganglionic Blockers; In Vitro Techniques; Indoles; Ketanserin; Methiothepin; Muscle, Smooth, Vascular; Pyrilamine; Receptors, Serotonin; Saphenous Vein; Spiperone; Sulfonamides; Sumatriptan; Tetrahydronaphthalenes; Vasoconstriction; Vasoconstrictor Agents

1991
5-HT1-like receptors mediate 5-hydroxytryptamine-induced contraction of guinea-pig isolated iliac artery.
    British journal of pharmacology, 1991, Volume: 102, Issue:2

    Topics: Animals; Guinea Pigs; Iliac Artery; In Vitro Techniques; Indoles; Ketanserin; Male; Methiothepin; Receptors, Serotonin; Serotonin; Sulfonamides; Sumatriptan; Tropisetron; Vasoconstriction

1991
Pharmacological characterisation of postjunctional 5-HT receptors in cerebral arteries from the sheep.
    European journal of pharmacology, 1990, Apr-10, Volume: 179, Issue:1-2

    Topics: Animals; Basilar Artery; Cerebral Arteries; Indoles; Ketanserin; Norepinephrine; Receptors, Serotonin; Serotonin; Sheep; Sulfonamides; Sumatriptan; Tropanes; Vasoconstriction

1990
Influence of the endothelium on contractile effects of 5-hydroxytryptamine and selective 5-HT agonists in canine basilar artery.
    British journal of pharmacology, 1989, Volume: 96, Issue:1

    Topics: Animals; Basilar Artery; Detergents; Dogs; Endothelium, Vascular; Female; In Vitro Techniques; Indoles; Ketanserin; Male; Methiothepin; Microscopy, Electron, Scanning; Octoxynol; Polyethylene Glycols; Potassium Chloride; Serotonin; Serotonin Antagonists; Sulfonamides; Sumatriptan

1989
The selective carotid arterial vasoconstrictor action of GR43175 in anaesthetized dogs.
    British journal of pharmacology, 1989, Volume: 96, Issue:1

    Topics: Animals; Barbital; Carotid Arteries; Dogs; Female; Hemodynamics; Indoles; Ketanserin; Male; Methiothepin; Phentolamine; Serotonin Antagonists; Sulfonamides; Sumatriptan; Tropanes; Vasoconstrictor Agents

1989
5-Hydroxytryptamine contracts human coronary arteries predominantly via 5-HT2 receptor activation.
    European journal of pharmacology, 1989, Feb-14, Volume: 161, Issue:1

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adult; Child; Coronary Vessels; Humans; In Vitro Techniques; Indoles; Ketanserin; Male; Middle Aged; Muscle Contraction; Muscle, Smooth, Vascular; Prostaglandin Endoperoxides, Synthetic; Receptors, Serotonin; Serotonin; Sulfonamides; Sumatriptan

1989
Differences in the effects of ketanserin and GR127935 on 5-HT-receptor mediated responses in rabbit saphenous vein and guinea-pig jugular vein.
    European journal of pharmacology, 1995, Sep-05, Volume: 283, Issue:1-3

    Topics: Animals; Dose-Response Relationship, Drug; Guinea Pigs; Jugular Veins; Ketanserin; Male; Myenteric Plexus; Nifedipine; Oxadiazoles; Piperazines; Rabbits; Saphenous Vein; Serotonin; Serotonin Antagonists; Sumatriptan

1995
5-HT1-receptor-mediated vasoconstriction in bovine isolated pulmonary arteries: influences of vascular endothelium and tone.
    Pulmonary pharmacology, 1994, Volume: 7, Issue:1

    Topics: Amino Acid Oxidoreductases; Animals; Arginine; Cattle; Drug Interactions; Endothelium, Vascular; In Vitro Techniques; Ketanserin; Methiothepin; Muscle Contraction; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Pulmonary Artery; Receptors, Serotonin; Sensitivity and Specificity; Serotonin; Serotonin Antagonists; Sumatriptan; Vasoconstriction

1994
Autoradiographic mapping of [3H]sumatriptan binding in cat brain stem and spinal cord.
    European journal of pharmacology, 1995, Jul-04, Volume: 280, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoradiography; Brain Stem; Cats; Ketanserin; Male; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Solitary Nucleus; Spinal Cord; Sumatriptan; Trigeminal Nuclei

1995
5-HT receptors mediating contractions of the isolated human coronary artery.
    European journal of pharmacology, 1993, Aug-03, Volume: 239, Issue:1-3

    Topics: Adolescent; Adult; Arteries; Blood Platelets; Child; Child, Preschool; Coronary Vessels; Dose-Response Relationship, Drug; Ergotamine; Female; Humans; In Vitro Techniques; Infant; Ketanserin; Male; Metergoline; Middle Aged; Muscle Contraction; Muscle, Smooth, Vascular; Pindolol; Potassium; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Substance P; Sumatriptan; Yohimbine

1993
Variable participation of 5-HT1-like receptors and 5-HT2 receptors in serotonin-induced contraction of human isolated coronary arteries. 5-HT1-like receptors resemble cloned 5-HT1D beta receptors.
    Circulation, 1994, Volume: 90, Issue:3

    Topics: Adult; Arteriosclerosis; Binding, Competitive; Cardiomyopathy, Dilated; Cloning, Molecular; Coronary Disease; Coronary Vessels; Female; Humans; In Vitro Techniques; Ketanserin; Male; Middle Aged; Myocardial Ischemia; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sumatriptan; Vasoconstriction

1994
Is 5-hydroxytryptamine mediating descending inhibition in the neonatal rat spinal cord through different receptor subtypes?
    European journal of pharmacology, 1993, Dec-21, Volume: 250, Issue:3

    Topics: Animals; Animals, Newborn; Citalopram; Dioxanes; Dopamine Antagonists; Electric Stimulation; Ketanserin; Lumbar Vertebrae; Methiothepin; Methysergide; Rats; Receptors, Serotonin; Reflex, Monosynaptic; Serotonin; Spinal Cord; Spinal Nerve Roots; Spiperone; Spiro Compounds; Sulpiride; Sumatriptan

1993
A slow excitatory postsynaptic potential mediated by 5-HT2 receptors in nucleus prepositus hypoglossi.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1994, Volume: 14, Issue:4

    Topics: Amphetamines; Animals; Brain Stem; Cyclohexane Monoterpenes; Evoked Potentials; Guinea Pigs; In Vitro Techniques; Ketanserin; Male; Medulla Oblongata; Membrane Potentials; Neurons; Pindolol; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Sumatriptan; Synaptic Transmission

1994
5-Hydroxytryptamine receptor characterization of human cerebral, middle meningeal and temporal arteries: regional differences.
    Acta physiologica Scandinavica, 1993, Volume: 147, Issue:2

    Topics: 5-Methoxytryptamine; Cerebral Arteries; Humans; Indoles; Ketanserin; Meningeal Arteries; Methiothepin; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides; Sumatriptan; Temporal Arteries; Vasoconstriction; Vasoconstrictor Agents

1993
5-Hydroxytryptamine 5-HT1D receptors mediating inhibition of cyclic AMP accumulation in Madin-Darby canine kidney (MDCK) cells.
    Naunyn-Schmiedeberg's archives of pharmacology, 1995, Volume: 352, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Alprostadil; Animals; Cells, Cultured; Cyclic AMP; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Epithelial Cells; Epithelium; Ketanserin; Kidney Cortex; Methiothepin; Oxadiazoles; Pertussis Toxin; Piperazines; Propranolol; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship; Sumatriptan; Virulence Factors, Bordetella; Yohimbine

1995
Ketanserin-sensitive depressant actions of 5-HT receptor agonists in the neonatal rat spinal cord.
    British journal of pharmacology, 1995, Volume: 116, Issue:6

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Animals, Newborn; Depression, Chemical; Dioxanes; Dopamine Antagonists; Drug Interactions; Female; Ketanserin; Male; Motor Neurons; Oxadiazoles; Pindolol; Piperazines; Propranolol; Rats; Rats, Wistar; Receptors, Serotonin; Reflex, Monosynaptic; Serotonin; Serotonin Antagonists; Spinal Cord; Spiro Compounds; Sumatriptan

1995
Inhibition of noradrenaline release via presynaptic 5-HT1D alpha receptors in human atrium.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 353, Issue:3

    Topics: 5-Methoxytryptamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic Uptake Inhibitors; Adult; Aged; Anti-Inflammatory Agents, Non-Steroidal; Cisapride; Corticosterone; Desipramine; Heart Atria; Humans; Indoles; Ketanserin; Male; Middle Aged; Norepinephrine; Oxadiazoles; Piperidines; Receptors, Presynaptic; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Tritium; Tryptamines

1996
Evidence for presynaptic location of inhibitory 5-HT1D beta-like autoreceptors in the guinea-pig brain cortex.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 353, Issue:3

    Topics: Animals; Autoreceptors; Binding, Competitive; Cerebral Cortex; Guinea Pigs; Humans; Indoles; Ketanserin; Male; Methiothepin; Oxadiazoles; Oxymetazoline; Potassium; Radioligand Assay; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship; Sumatriptan; Synaptosomes; Tritium; Tryptamines

1996
GR127935 is a potent antagonist of the 5-HT1-like receptor mediating contraction in the canine coronary artery.
    European journal of pharmacology, 1996, Apr-04, Volume: 300, Issue:1-2

    Topics: Animals; Coronary Vessels; Dogs; Drug Interactions; Ketanserin; Muscle, Smooth, Vascular; Oxadiazoles; Piperazines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sumatriptan; Vasoconstriction

1996
Participation of 5-HT1-like and 5-HT2A receptors in the contraction of human temporal artery by 5-hydroxytryptamine and related drugs.
    British journal of pharmacology, 1996, Volume: 117, Issue:2

    Topics: Adult; Aged; Benzazepines; Collagenases; Endothelium, Vascular; Female; Headache; Humans; In Vitro Techniques; Ketanserin; Male; Middle Aged; Muscle Contraction; Muscle, Smooth, Vascular; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Temporal Arteries

1996
5-HT1-like receptor-mediated contraction in the human internal mammary artery.
    Journal of cardiovascular pharmacology, 1996, Volume: 28, Issue:1

    Topics: Adult; Dose-Response Relationship, Drug; Female; Humans; In Vitro Techniques; Ketanserin; Mammary Arteries; Methiothepin; Middle Aged; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Vasoconstriction; Vasoconstrictor Agents

1996
Characterization of 5-hydroxytryptamine receptors mediating circular smooth muscle contraction in the human umbilical artery.
    Gynecologic and obstetric investigation, 1999, Volume: 47, Issue:2

    Topics: Adolescent; Adult; Female; Humans; Ketanserin; Methiothepin; Muscle Contraction; Muscle, Smooth; Pregnancy; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Tropanes; Umbilical Arteries

1999
Characterisation of 5-HT receptors in human coronary arteries by molecular and pharmacological techniques.
    European journal of pharmacology, 1999, May-07, Volume: 372, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Cardiovascular System; Coronary Vessels; Dose-Response Relationship, Drug; Gene Expression; Humans; Immunohistochemistry; In Vitro Techniques; Ketanserin; Methiothepin; Oxazoles; Oxazolidinones; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Tissue Distribution; Tryptamines; Vasoconstriction

1999
Functional characterization and m-RNA expression of 5-HT receptors mediating contraction in human umbilical artery.
    British journal of pharmacology, 1999, Volume: 127, Issue:5

    Topics: Humans; Ketanserin; Oxadiazoles; Piperazines; Receptors, Serotonin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Serotonin; Sumatriptan; Umbilical Arteries; Vasoconstriction

1999
Involvement of 5-HT1B receptors in collar-induced hypersensitivity to 5-hydroxytryptamine of the rabbit carotid artery.
    British journal of pharmacology, 1999, Volume: 127, Issue:6

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Braces; Carotid Arteries; Dose-Response Relationship, Drug; Hypersensitivity; In Vitro Techniques; Ketanserin; Male; Methysergide; Oxadiazoles; Piperazines; Potassium Chloride; Rabbits; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Sumatriptan; Tryptamines; Vasoconstriction

1999
Effects of alniditan on neurogenic oedema in the rat dura mater and on contraction of rat basilar artery.
    European journal of pharmacology, 1999, Oct-08, Volume: 382, Issue:2

    Topics: Animals; Basilar Artery; Benzopyrans; Brain Edema; Capillary Permeability; Dose-Response Relationship, Drug; Dura Mater; Extravasation of Diagnostic and Therapeutic Materials; In Vitro Techniques; Ketanserin; Male; Oxadiazoles; Piperazines; Propylamines; Pyrimidines; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Agents; Serotonin Antagonists; Substance P; Sumatriptan; Vasoconstriction; Vasoconstrictor Agents

1999
Bovine isolated middle cerebral artery contractions to antimigraine drugs.
    Naunyn-Schmiedeberg's archives of pharmacology, 1999, Volume: 360, Issue:5

    Topics: Animals; Cattle; In Vitro Techniques; Ketanserin; Middle Cerebral Artery; Muscle Contraction; Muscle, Smooth, Vascular; Oxadiazoles; Piperazines; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Vasoconstrictor Agents

1999
Serotonin-induced hypercontraction through 5-hydroxytryptamine 1B receptors in atherosclerotic rabbit coronary arteries.
    Circulation, 2001, Mar-06, Volume: 103, Issue:9

    Topics: Animals; Arteriosclerosis; Calcium; Coronary Vessels; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Ketanserin; Male; Oxadiazoles; Phenylephrine; Piperazines; Rabbits; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; RNA, Messenger; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Vasoconstriction

2001
Serotonin-induced contraction in mesenteric resistance arteries: signaling and changes in deoxycorticosterone acetate-salt hypertension.
    Hypertension (Dallas, Tex. : 1979), 2002, Mar-01, Volume: 39, Issue:3

    Topics: Animals; Carbazoles; Desoxycorticosterone; Dose-Response Relationship, Drug; Fluorobenzenes; Hypertension; In Vitro Techniques; Indoles; Ketanserin; Male; Mesenteric Arteries; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Signal Transduction; Sumatriptan; Thiophenes; Vascular Resistance; Vasoconstriction

2002
Studies on serotonergic markers in the human hippocampus: changes in subjects with bipolar disorder.
    Journal of affective disorders, 2003, Volume: 75, Issue:1

    Topics: Affinity Labels; Binding Sites; Biomarkers; Bipolar Disorder; Carrier Proteins; Cell Count; Citalopram; Culture Techniques; Hippocampus; Humans; Ketanserin; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Serotonin Plasma Membrane Transport Proteins; Serotonin Receptor Agonists; Sumatriptan

2003
Involvement of nitric oxide in fading of 5-hydroxytryptamine-induced vasocontraction in rat isolated vena portae smooth muscle.
    Journal of pharmacy & pharmaceutical sciences : a publication of the Canadian Society for Pharmaceutical Sciences, Societe canadienne des sciences pharmaceutiques, 2004, Jan-23, Volume: 7, Issue:1

    Topics: Animals; Drug Interactions; In Vitro Techniques; Ketanserin; Male; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitric Oxide; Portal Vein; Rats; Rats, Inbred WKY; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptor, Serotonin, 5-HT2B; Serotonin; Serotonin Antagonists; Sumatriptan; Vasoconstriction; Vasoconstrictor Agents

2004
Involvement of 5-HT1B receptors in triptan-induced contractile responses in guinea-pig isolated iliac artery.
    Naunyn-Schmiedeberg's archives of pharmacology, 2004, Volume: 370, Issue:1

    Topics: Animals; Benzamides; Brain; Carbazoles; Dinoprost; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Endothelium, Vascular; Female; Forecasting; Guinea Pigs; Iliac Artery; Indoles; Ketanserin; Male; Muscle Contraction; Muscle, Smooth; Oxadiazoles; Oxazolidinones; Piperazines; Piperidines; Pyrrolidines; Receptor, Serotonin, 5-HT1B; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Sumatriptan; Triazoles; Tryptamines

2004
Hippocampal 5-hydroxytryptamine receptors: abnormalities in postmortem brain from schizophrenic subjects.
    Schizophrenia research, 2004, Dec-01, Volume: 71, Issue:2-3

    Topics: Adult; Aged; Autoradiography; Binding Sites; Female; Hippocampus; Humans; Ketanserin; Male; Middle Aged; Radioligand Assay; Receptors, Serotonin; Schizophrenia; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Tetrahydronaphthalenes

2004
Functional reactivity of 5-HT receptors in human umbilical cord and maternal subcutaneous fat arteries after normotensive or pre-eclamptic pregnancy.
    Journal of hypertension, 2006, Volume: 24, Issue:7

    Topics: Adult; Arteries; Blood Pressure; Data Interpretation, Statistical; Female; Fetus; Humans; Ketanserin; Linear Models; Potassium Chloride; Pre-Eclampsia; Pregnancy; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Subcutaneous Fat; Sumatriptan; Umbilical Arteries; Vasoconstriction

2006
Activation of 5-HT1B and 5-HT1D receptors in the rat nucleus tractus solitarius: opposing action on neurones that receive an excitatory vagal C-fibre afferent input.
    British journal of pharmacology, 2007, Volume: 150, Issue:8

    Topics: Action Potentials; Animals; Benzamides; Drug Synergism; Electric Stimulation; Iontophoresis; Ketanserin; Male; Neural Inhibition; Neurons; Neurons, Afferent; Patch-Clamp Techniques; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Serotonin 5-HT1 Receptor Agonists; Serotonin Antagonists; Serotonin Receptor Agonists; Solitary Nucleus; Sumatriptan; Time Factors; Vagus Nerve

2007
The effect of maternal ketanserin treatment on foetal 5-HT receptor function in umbilical cord artery of pre-eclamptic patients.
    Neonatology, 2007, Volume: 92, Issue:4

    Topics: Adolescent; Adult; Antihypertensive Agents; Benzamides; Case-Control Studies; Dose-Response Relationship, Drug; Female; Humans; Ketanserin; Pre-Eclampsia; Pregnancy; Pyridines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Umbilical Arteries

2007
Anti-hyperalgesic effects of anti-serotonergic compounds on serotonin- and capsaicin-evoked thermal hyperalgesia in the rat.
    Neuroscience, 2012, Feb-17, Volume: 203

    Topics: Animals; Capsaicin; Female; Hyperalgesia; Ketanserin; Male; Pain Measurement; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan

2012