sumatriptan has been researched along with guanosine 5'-o-(3-thiotriphosphate) in 7 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 5 (71.43) | 18.2507 |
2000's | 2 (28.57) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Audinot-Bouchez, V; Chaput, C; Conte, C; Lavielle, G; Lochon, S; Millan, MJ; Newman-Tancredi, A; Verrièle, L | 1 |
Colpaert, FC; Dupuis, DS; Pauwels, PJ | 1 |
Gaster, LM; Hagan, JJ; Ham, P; Joiner, GF; King, FD; Middlemiss, DN; Mulholland, KR; Price, GW; Roberts, C; Routledge, C; Selkirk, J; Slade, PD; Wyman, PA | 1 |
Colpaert, FC; Dupuis, DS; Halazy, S; Pauwels, PJ; Perez, M | 1 |
Grånäs, C; Larhammar, D | 1 |
Boot, JR; Carney, SL; Cohen, ML; Colvin, EM; Conway, RG; Hardy, CH; Lucaites, VL; Nelson, DL; Pullar, IA; Schenck, KW; Tomlinson, R; Wedley, S | 1 |
Ahlgren, C; Eriksson, A; Malmberg, A; Ross, SB; Stenfors, C; Tellefors, P | 1 |
7 other study(ies) available for sumatriptan and guanosine 5'-o-(3-thiotriphosphate)
Article | Year |
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Agonist activity of antimigraine drugs at recombinant human 5-HT1A receptors: potential implications for prophylactic and acute therapy.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Benzopyrans; Binding, Competitive; Cell Membrane; Cricetinae; Dihydroergotamine; Guanosine 5'-O-(3-Thiotriphosphate); Guinea Pigs; Humans; In Vitro Techniques; Indoles; Lisuride; Methysergide; Migraine Disorders; Piperazines; Piperidines; Pizotyline; Propranolol; Propylamines; Protein Binding; Pyridines; Pyrimidines; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Recombinant Proteins; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Tryptamines | 1997 |
G-protein activation at 5-HT1A receptors by the 5-ht1F ligand LY334370 in guinea-pig brain sections and recombinant cell lines.
Topics: Aminopyridines; Animals; Autoradiography; Benzamides; Binding Sites; Binding, Competitive; Brain; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guinea Pigs; HeLa Cells; Hippocampus; Humans; Indoles; Male; Piperazines; Pyridines; Raphe Nuclei; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan | 1998 |
The selective 5-HT1B receptor inverse agonist SB-224289, potently blocks terminal 5-HT autoreceptor function both in vitro and in vivo.
Topics: Animals; Body Temperature Regulation; Cerebral Cortex; CHO Cells; Cricetinae; Dentate Gyrus; Guanosine 5'-O-(3-Thiotriphosphate); Guinea Pigs; Humans; Oxadiazoles; Piperazines; Piperidones; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Recombinant Proteins; Serotonin; Serotonin Antagonists; Spiro Compounds; Sumatriptan; Transfection | 1998 |
Magnitude of 5-HT1B and 5-HT1A receptor activation in guinea-pig and rat brain: evidence from sumatriptan dimer-mediated [35S]GTPgammaS binding responses.
Topics: Animals; Autoradiography; Binding, Competitive; Brain Chemistry; Dimerization; Glioma; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Guinea Pigs; HeLa Cells; Humans; Male; Membrane Proteins; Oxadiazoles; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Receptor Agonists; Sulfur Radioisotopes; Sumatriptan; Tryptamines | 1999 |
Identification of an amino acid residue important for binding of methiothepin and sumatriptan to the human 5-HT(1B) receptor.
Topics: Amino Acid Sequence; Amino Acids; Animals; Benzamides; Binding Sites; Binding, Competitive; CHO Cells; Cricetinae; Dose-Response Relationship, Drug; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Methiothepin; Molecular Sequence Data; Mutation; Protein Binding; Pyridines; Radioligand Assay; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Sequence Homology, Amino Acid; Serotonin Antagonists; Serotonin Receptor Agonists; Sodium; Sumatriptan; Tritium | 1999 |
In vitro activity of LY393558, an inhibitor of the 5-hydroxytryptamine transporter with 5-HT(1B/1D/2) receptor antagonist properties.
Topics: Animals; Binding, Competitive; Carrier Proteins; Cerebral Cortex; Cyclic S-Oxides; Dose-Response Relationship, Drug; Drug Synergism; Guanosine 5'-O-(3-Thiotriphosphate); Humans; In Vitro Techniques; Male; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Nerve Tissue Proteins; Norepinephrine; Potassium; Rabbits; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Saphenous Vein; Serotonin; Serotonin Antagonists; Serotonin Plasma Membrane Transport Proteins; Serotonin Receptor Agonists; Sulfur Radioisotopes; Sumatriptan; Thiadiazines; Tritium; Vasoconstriction | 2001 |
In vitro characterization of AR-A000002, a novel 5-hydroxytryptamine(1B) autoreceptor antagonist.
Topics: Animals; Autoreceptors; Benzamides; Binding, Competitive; Cell Line; Cell Membrane; Cerebral Cortex; Dose-Response Relationship, Drug; Electric Stimulation; Guanosine 5'-O-(3-Thiotriphosphate); Guinea Pigs; Humans; In Vitro Techniques; Indoles; Morpholines; Piperidones; Pyridines; Rabbits; Radioligand Assay; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Saphenous Vein; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Spiro Compounds; Sulfur Radioisotopes; Sumatriptan; Transfection; Tritium; Vasoconstriction; Vasoconstrictor Agents | 2004 |