Page last updated: 2024-08-16

sumatriptan and frovatriptan

sumatriptan has been researched along with frovatriptan in 26 studies

Research

Studies (26)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (11.54)18.2507
2000's17 (65.38)29.6817
2010's4 (15.38)24.3611
2020's2 (7.69)2.80

Authors

AuthorsStudies
Adham, N; Audia, JE; Kohlman, DT; Krushinski, J; Liang, SX; Schaus, JM; Walker, C; Xu, YC; Zgombick, JM1
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Brockmöller, J; Dücker, C; Gebauer, L; Jensen, O1
Campbell, CA; Griffiths, R; Hamilton, TC; Hunter, AJ; King, FD; Lewis, VA; Parker, SG; Parsons, AA; Raval, P1
Hunter, J; Kaumann, AJ; King, FD; Parsons, AA; Raval, P; Smith, S; Tilford, N1
Berdeaux, A; Carel, I; Dubois-Rande, JL; Edouard, A; Ghaleh, B; Giudicelli, JF; Parsons, AA1
Marcus, DA1
Rapoport, AM; Tepper, SJ1
Freitag, FG1
Comer, MB1
Géraud, G; Keywood, C; Spierings, EL1
Rapoport, AM; Sheftell, FD; Tepper, SJ1
Csiba, L; Ficzere, A1
Adelman, JU; Lewit, EJ1
Steiner, T; Tfelt-Hansen, P1
Jähnichen, S; Pertz, HH; Radtke, OA1
Balbisi, EA1
Kowa, H; Nakashima, K; Takeshima, T1
Davenport, WJ; Dodick, D; Pringsheim, T1
Tfelt-Hansen, P2
Campbell, JC; Hu, X; MacGregor, EA; Pawsey, SP1
Qi, JZ; Zhang, H; Zhang, ZH1

Reviews

12 review(s) available for sumatriptan and frovatriptan

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Establishing a standard of speed for assessing the efficacy of the serotonin(1B/1D) agonists (triptans).
    Archives of neurology, 2001, Volume: 58, Issue:7

    Topics: Analgesics, Non-Narcotic; Carbazoles; Clinical Trials as Topic; Humans; Indoles; Migraine Disorders; Oxazolidinones; Pain Measurement; Patient Satisfaction; Piperidines; Pyrrolidines; Serotonin Receptor Agonists; Sumatriptan; Time Factors; Treatment Outcome; Triazoles; Tryptamines

2001
Triptans are all different.
    Archives of neurology, 2001, Volume: 58, Issue:9

    Topics: Carbazoles; Headache; Humans; Indoles; Oxazolidinones; Pyrrolidines; Serotonin Receptor Agonists; Sumatriptan; Triazoles; Tryptamines

2001
Acute treatment of migraine and the role of triptans.
    Current neurology and neuroscience reports, 2001, Volume: 1, Issue:2

    Topics: Acute Disease; Blood Flow Velocity; Carbazoles; Clinical Trials as Topic; Drug Administration Routes; Female; Humans; Indoles; Male; Menstruation; Migraine Disorders; Oxazolidinones; Piperidines; Practice Guidelines as Topic; Pyrrolidines; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin Receptor Agonists; Sumatriptan; Treatment Outcome; Triazoles; Tryptamines; Vasoconstriction; Vasoconstrictor Agents

2001
Mechanisms of action of the 5-HT1B/1D receptor agonists.
    Archives of neurology, 2002, Volume: 59, Issue:7

    Topics: Carbazoles; Humans; Indoles; Migraine Disorders; Oxazolidinones; Piperidines; Pyrrolidines; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin Receptor Agonists; Sumatriptan; Triazoles; Tryptamines

2002
[Treatment of migraine in patients with hypertension and ischemic heart disease].
    Ideggyogyaszati szemle, 2002, Jan-20, Volume: 55, Issue:1-2

    Topics: Adjuvants, Pharmaceutic; Analgesics, Non-Narcotic; Anti-Inflammatory Agents, Non-Steroidal; Carbazoles; Contraindications; Dihydroergotamine; Dopamine Agonists; Ergotamine; Humans; Hypertension; Indoles; Migraine Disorders; Myocardial Ischemia; Oxazolidinones; Retrospective Studies; Serotonin Receptor Agonists; Sumatriptan; Triazoles; Tryptamines; Vasoconstrictor Agents

2002
Comparative aspects of triptans in treating migraine.
    Clinical cornerstone, 2001, Volume: 4, Issue:3

    Topics: Carbazoles; Cardiovascular Diseases; Humans; Indoles; Migraine Disorders; Oxazolidinones; Patient Satisfaction; Piperidines; Pyrrolidines; Serotonin Receptor Agonists; Sumatriptan; Treatment Outcome; Triazoles; Tryptamines

2001
Frovatriptan succinate, a 5-HT1B/1D receptor agonist for migraine.
    International journal of clinical practice, 2004, Volume: 58, Issue:7

    Topics: Carbazoles; Dose-Response Relationship, Drug; Double-Blind Method; Female; Humans; Male; Menstruation Disturbances; Migraine Disorders; Multicenter Studies as Topic; Randomized Controlled Trials as Topic; Recurrence; Risk Factors; Serotonin Receptor Agonists; Sumatriptan; Treatment Outcome; Tryptamines

2004
[Meta-analysis of triptan treatment in migraine].
    No to shinkei = Brain and nerve, 2004, Volume: 56, Issue:9

    Topics: Carbazoles; Evidence-Based Medicine; Humans; Indoles; Migraine Disorders; Oxazolidinones; Piperidines; Pyrrolidines; Receptor, Serotonin, 5-HT1D; Serotonin Receptor Agonists; Sumatriptan; Triazoles; Tryptamines

2004
Acute treatment and prevention of menstrually related migraine headache: evidence-based review.
    Neurology, 2008, Apr-22, Volume: 70, Issue:17

    Topics: Anti-Inflammatory Agents, Non-Steroidal; Carbazoles; Double-Blind Method; Estrogens; Evidence-Based Medicine; Female; Humans; Male; Mefenamic Acid; Menstruation; Meta-Analysis as Topic; Migraine Disorders; Randomized Controlled Trials as Topic; Serotonin Receptor Agonists; Sumatriptan; Treatment Outcome; Triazoles; Tryptamines

2008
Safety and tolerability of frovatriptan in the acute treatment of migraine and prevention of menstrual migraine: Results of a new analysis of data from five previously published studies.
    Gender medicine, 2010, Volume: 7, Issue:2

    Topics: Acute Disease; Carbazoles; Cardiovascular Diseases; Clinical Trials, Phase III as Topic; Dose-Response Relationship, Drug; Double-Blind Method; Female; Humans; Logistic Models; Male; Menstruation Disturbances; Migraine Disorders; Multicenter Studies as Topic; Randomized Controlled Trials as Topic; Research Design; Safety; Serotonin Receptor Agonists; Sumatriptan; Treatment Outcome; Tryptamines

2010
Comparative efficacy of different treatments for menstrual migraine: a systematic review and network meta-analysis.
    The journal of headache and pain, 2023, Jul-03, Volume: 24, Issue:1

    Topics: Humans; Migraine Disorders; Network Meta-Analysis; Sumatriptan; Tryptamines

2023

Trials

1 trial(s) available for sumatriptan and frovatriptan

ArticleYear
Tolerability and safety of frovatriptan with short- and long-term use for treatment of migraine and in comparison with sumatriptan.
    Headache, 2002, Volume: 42 Suppl 2

    Topics: Acute Disease; Adult; Carbazoles; Clinical Trials as Topic; Dizziness; Dose-Response Relationship, Drug; Double-Blind Method; Fatigue; Female; Headache; Humans; Male; Middle Aged; Migraine Disorders; Nausea; Paresthesia; Serotonin Receptor Agonists; Sumatriptan; Tryptamines

2002

Other Studies

13 other study(ies) available for sumatriptan and frovatriptan

ArticleYear
N-Methyl-5-tert-butyltryptamine: A novel, highly potent 5-HT1D receptor agonist.
    Journal of medicinal chemistry, 1999, Feb-11, Volume: 42, Issue:3

    Topics: Cell Line; Humans; Magnetic Resonance Spectroscopy; Mass Spectrometry; Radioligand Assay; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin Receptor Agonists; Structure-Activity Relationship; Tryptamines

1999
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Substrates and Inhibitors of the Organic Cation Transporter 3 and Comparison with OCT1 and OCT2.
    Journal of medicinal chemistry, 2022, 09-22, Volume: 65, Issue:18

    Topics: Biological Transport; Cations; Organic Cation Transport Proteins; Organic Cation Transporter 1; Organic Cation Transporter 2

2022
Comparison of the cardiovascular effects of the novel 5-HT(1B/1D) receptor agonist, SB 209509 (VML251), and sumatriptan in dogs.
    Journal of cardiovascular pharmacology, 1997, Volume: 30, Issue:1

    Topics: Animals; Biological Availability; Blood Pressure; Carbazoles; Cardiovascular System; Carotid Arteries; Coronary Circulation; Coronary Vessels; Dogs; Duodenum; Female; Heart Rate; Infusions, Intravenous; Male; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Regional Blood Flow; Serotonin Receptor Agonists; Sumatriptan; Tryptamines; Vascular Resistance

1997
Effects of the novel high-affinity 5-HT(1B/1D)-receptor ligand frovatriptan in human isolated basilar and coronary arteries.
    Journal of cardiovascular pharmacology, 1998, Volume: 32, Issue:2

    Topics: Basilar Artery; Carbazoles; Coronary Circulation; Humans; In Vitro Techniques; Ligands; Muscle Contraction; Muscle, Smooth; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Sumatriptan; Tryptamines; Vasoconstrictor Agents

1998
Comparative effects of frovatriptan and sumatriptan on coronary and internal carotid vascular haemodynamics in conscious dogs.
    British journal of pharmacology, 2001, Volume: 132, Issue:5

    Topics: Animals; Carbazoles; Carotid Artery, Internal; Coronary Vessels; Dogs; Dose-Response Relationship, Drug; Endothelium, Vascular; Hemodynamics; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin Receptor Agonists; Sumatriptan; Tryptamines; Vascular Resistance; Vasoconstriction; Vasodilation

2001
Pharmacology of the selective 5-HT(1B/1D) agonist frovatriptan.
    Headache, 2002, Volume: 42 Suppl 2

    Topics: Animals; Carbazoles; Cerebrovascular Circulation; Guinea Pigs; Humans; In Vitro Techniques; Rabbits; Rats; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin Receptor Agonists; Sumatriptan; Tryptamines; Vasoconstrictor Agents

2002
The truth about frovatriptan.
    Headache, 2003, Volume: 43, Issue:6

    Topics: Carbazoles; Clinical Trials as Topic; Humans; Migraine Disorders; Serotonin Receptor Agonists; Sumatriptan; Tryptamines

2003
Involvement of 5-HT1B receptors in triptan-induced contractile responses in guinea-pig isolated iliac artery.
    Naunyn-Schmiedeberg's archives of pharmacology, 2004, Volume: 370, Issue:1

    Topics: Animals; Benzamides; Brain; Carbazoles; Dinoprost; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Endothelium, Vascular; Female; Forecasting; Guinea Pigs; Iliac Artery; Indoles; Ketanserin; Male; Muscle Contraction; Muscle, Smooth; Oxadiazoles; Oxazolidinones; Piperazines; Piperidines; Pyrrolidines; Receptor, Serotonin, 5-HT1B; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Sumatriptan; Triazoles; Tryptamines

2004
Frovatriptan and data publication.
    Headache, 2008, Volume: 48, Issue:9

    Topics: Carbazoles; Double-Blind Method; Humans; Migraine Disorders; Periodicals as Topic; Randomized Controlled Trials as Topic; Serotonin Receptor Agonists; Sumatriptan; Tryptamines

2008
Effective symptomatic medication should be available in prophylactic trials in cluster headache.
    Headache, 2011, Volume: 51, Issue:2

    Topics: Carbazoles; Cluster Headache; Guidelines as Topic; Humans; Randomized Controlled Trials as Topic; Serotonin Receptor Agonists; Sumatriptan; Treatment Outcome; Tryptamines

2011