Page last updated: 2024-08-16

sumatriptan and colforsin

sumatriptan has been researched along with colforsin in 18 studies

Research

Studies (18)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's14 (77.78)18.2507
2000's2 (11.11)29.6817
2010's2 (11.11)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Feniuk, W; Humphrey, PP; McCormick, JD; Sumner, MJ1
Demchyshyn, L; King, A; Miller, KJ; Niznik, H; Teitler, M1
Bondiolotti, G; Cattaneo, MG; Palazzi, E; Vicentini, LM1
Allgeier, A; Czernilofsky, A; Dumont, JE; Maenhaut, C; Massart, C; Van Sande, J; Vassart, G1
Adham, N; Bard, J; Branchek, TA; Durkin, M; Hartig, PR; Kao, HT; Olsen, M; Schecter, LE; Urquhart, D; Weinshank, RL1
Ormandy, GC1
Colpaert, FC; Pauwels, PJ1
Gutierrez, M; Lübbert, H; Schoeffter, P; Ullmer, C; Weitz-Schmidt, G1
Pauwels, PJ1
Movahedi, H; Purdy, RE1
Durham, PL; Russo, AF; Sharma, RV1
Dickenson, JM; Hill, SJ1
Ehlert, F; Purdy, RE; Yildiz, O1
Durham, PL; Russo, AF1
Beleta, J; Bou, J; Domènech, T; Fernández-Forner, D; Gras, J; Heredia, A; Palacios, JM; Puig, J1
Carruthers, AM; Feniuk, W; Humphrey, PP; Jarvie, EM; Jenkins, DW; Sellers, LA1
Bönisch, H; Haenisch, B1
Chan, KY; Danser, AH; de Vries, R; Dirven, C; Garrelds, IM; Labruijere, S; MaassenVanDenBrink, A; Ramírez Rosas, MB; van den Bogaerdt, A; Villalón, CM1

Other Studies

18 other study(ies) available for sumatriptan and colforsin

ArticleYear
Studies on the mechanism of 5-HT1 receptor-induced smooth muscle contraction in dog saphenous vein.
    British journal of pharmacology, 1992, Volume: 105, Issue:3

    Topics: Adenylyl Cyclase Inhibitors; Animals; Brain Chemistry; Calcium; Colforsin; Cyclic AMP; Dinoprostone; Dogs; Female; In Vitro Techniques; Indoles; Isometric Contraction; Male; Muscle Contraction; Muscle, Smooth, Vascular; Receptors, Serotonin; Saphenous Vein; Serotonin; Serotonin Antagonists; Sulfonamides; Sumatriptan; Vasoconstrictor Agents

1992
Agonist activity of sumatriptan and metergoline at the human 5-HT1D beta receptor: further evidence for a role of the 5-HT1D receptor in the action of sumatriptan.
    European journal of pharmacology, 1992, Sep-01, Volume: 227, Issue:1

    Topics: Cells, Cultured; Colforsin; Cyclic AMP; Humans; Indoles; Metergoline; Radioimmunoassay; Receptors, Serotonin; Serotonin Receptor Agonists; Sulfonamides; Sumatriptan

1992
5-HT1D receptor type is involved in stimulation of cell proliferation by serotonin in human small cell lung carcinoma.
    European journal of pharmacology, 1994, Aug-16, Volume: 268, Issue:3

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Carcinoma, Small Cell; Cell Division; Colforsin; Humans; Lung Neoplasms; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sumatriptan; Thymidine; Tumor Cells, Cultured

1994
The human and dog 5-HT1D receptors can both activate and inhibit adenylate cyclase in transfected cells.
    European journal of pharmacology, 1993, Oct-15, Volume: 247, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Adrenal Glands; Animals; Base Sequence; Cells, Cultured; CHO Cells; Cloning, Molecular; Colforsin; Cricetinae; Cyclic AMP; Dogs; Enzyme Activation; Humans; Molecular Sequence Data; Pertussis Toxin; Proteins; Receptors, Serotonin; Serotonin; Sumatriptan; Transfection; Virulence Factors, Bordetella

1993
Cloning of another human serotonin receptor (5-HT1F): a fifth 5-HT1 receptor subtype coupled to the inhibition of adenylate cyclase.
    Proceedings of the National Academy of Sciences of the United States of America, 1993, Jan-15, Volume: 90, Issue:2

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Amino Acid Sequence; Animals; Base Sequence; Brain Chemistry; Cloning, Molecular; Colforsin; Dose-Response Relationship, Drug; Gene Library; Guinea Pigs; Humans; Indoles; Lymphocytes; Molecular Sequence Data; Receptors, Serotonin; RNA, Messenger; Sequence Homology, Amino Acid; Serotonin; Serotonin Receptor Agonists; Spiperone; Sulfonamides; Sumatriptan; Tissue Distribution

1993
Increased cyclic AMP reduces 5-HT1D receptor-mediated inhibition of [3H]5-hydroxytryptamine release from guinea-pig cortical slices.
    European journal of pharmacology, 1993, Jan-15, Volume: 244, Issue:2

    Topics: Animals; Bucladesine; Cerebral Cortex; Colforsin; Cyclic AMP; Guinea Pigs; In Vitro Techniques; Indoles; Phosphodiesterase Inhibitors; Potassium; Pyrrolidinones; Receptors, Serotonin; Rolipram; Serotonin; Serotonin Receptor Agonists; Sulfonamides; Sumatriptan

1993
Stereoselectivity of 8-OH-DPAT enantiomers at cloned human 5-HT1D receptor sites.
    European journal of pharmacology, 1996, Apr-04, Volume: 300, Issue:1-2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Cell Line; Colforsin; Cyclic AMP; Humans; Neuroglia; Rats; Receptors, Serotonin; Stereoisomerism; Sumatriptan; Transfection

1996
Functional serotonin 5-HT1D receptors and 5-HT1D beta receptor mRNA expression in human umbilical vein endothelial cells.
    Naunyn-Schmiedeberg's archives of pharmacology, 1995, Volume: 352, Issue:5

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Cells, Cultured; Colforsin; Cyclic AMP; Endothelium, Vascular; Humans; Polymerase Chain Reaction; Receptors, Serotonin; RNA, Messenger; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Umbilical Veins

1995
Competitive and silent antagonism of recombinant 5-HT1B receptors by amiloride.
    General pharmacology, 1997, Volume: 29, Issue:5

    Topics: Amiloride; Animals; Binding, Competitive; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Diuretics; Guinea Pigs; Receptors, Serotonin; Serotonin Antagonists; Sumatriptan

1997
Pharmacological characterization of the "silent" 5-hydroxytryptamine1B-like receptors of rabbit ear artery.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 283, Issue:2

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Animals; Calcium; Colforsin; Dose-Response Relationship, Drug; Ear; Male; Pertussis Toxin; Phenylephrine; Rabbits; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin; Sumatriptan; Vasoconstriction; Virulence Factors, Bordetella

1997
Repression of the calcitonin gene-related peptide promoter by 5-HT1 receptor activation.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1997, Dec-15, Volume: 17, Issue:24

    Topics: Animals; Calcitonin Gene-Related Peptide; Calcium; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Enhancer Elements, Genetic; Gene Expression Regulation; Genes, Reporter; Neurons; Promoter Regions, Genetic; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; RNA, Messenger; Serotonin Receptor Agonists; Sumatriptan; Thyroid Neoplasms; Time Factors; Transcription, Genetic; Trigeminal Ganglion; Tumor Cells, Cultured

1997
Human 5-HT1B receptor stimulated inositol phospholipid hydrolysis in CHO cells: synergy with Gq-coupled receptors.
    European journal of pharmacology, 1998, May-08, Volume: 348, Issue:2-3

    Topics: Animals; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; DNA, Complementary; Dose-Response Relationship, Drug; GTP-Binding Proteins; Humans; Hydrolysis; Inositol Phosphates; Muscle Contraction; Muscle, Smooth, Vascular; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Second Messenger Systems; Serotonin Receptor Agonists; Sumatriptan

1998
Characterization of the "silent" 5-HT1B receptors of rabbit iliac artery.
    Annals of the New York Academy of Sciences, 1998, Dec-15, Volume: 861

    Topics: Animals; Colforsin; Iliac Artery; In Vitro Techniques; Isometric Contraction; Muscle, Smooth, Vascular; Phenylephrine; Rabbits; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Sumatriptan; Vasoconstriction; Vasodilation; Virulence Factors, Bordetella

1998
Regulation of calcitonin gene-related peptide secretion by a serotonergic antimigraine drug.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1999, May-01, Volume: 19, Issue:9

    Topics: Animals; Animals, Newborn; Calcitonin Gene-Related Peptide; Cells, Cultured; Colforsin; Cyclic AMP; HeLa Cells; Humans; Inflammation; Kinetics; Models, Neurological; Neurons; Okadaic Acid; Oxadiazoles; Potassium Chloride; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Recombinant Proteins; Serotonin Receptor Agonists; Sumatriptan; Transfection; Trigeminal Ganglion; Tryptamines

1999
Pharmacological characterization of almotriptan: an indolic 5-HT receptor agonist for the treatment of migraine.
    European journal of pharmacology, 2000, Dec-20, Volume: 410, Issue:1

    Topics: Animals; Cattle; Colforsin; Cyclic AMP; Dogs; Dose-Response Relationship, Drug; HeLa Cells; Humans; Indoles; Male; Meningeal Arteries; Migraine Disorders; Muscle, Smooth, Vascular; Rabbits; Rats; Rats, Wistar; Saphenous Vein; Serotonin Receptor Agonists; Sumatriptan; Swine; Transfection; Tryptamines; Vasoconstriction; Vasoconstrictor Agents

2000
Adenosine A(1) receptor-mediated inhibition of protein kinase A-induced calcitonin gene-related peptide release from rat trigeminal neurons.
    Molecular pharmacology, 2001, Volume: 59, Issue:6

    Topics: Adenosine; Analgesics, Opioid; Animals; Calcitonin Gene-Related Peptide; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Cyclic AMP-Dependent Protein Kinases; Drug Interactions; Fentanyl; Male; Neurons; Phenethylamines; Phosphorylation; Purinergic P1 Receptor Agonists; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Purinergic P1; Receptors, Serotonin; Serotonin Receptor Agonists; Sumatriptan; Synaptic Vesicles; Trigeminal Nerve

2001
Pharmacological characterization of tegaserod at the wild type and 124Cys variant of the human 5-HT1B receptor.
    Pharmacogenetics and genomics, 2011, Volume: 21, Issue:7

    Topics: Adenylyl Cyclases; Animals; Cell Line, Tumor; Colforsin; Coronary Vessels; Cyclic AMP; Genetic Variation; Genotype; GTP-Binding Proteins; Humans; Indoles; Rats; Receptor, Serotonin, 5-HT1B; Serotonin 5-HT1 Receptor Agonists; Sumatriptan; Transfection

2011
Cranioselectivity of sumatriptan revisited: pronounced contractions to sumatriptan in small human isolated coronary artery.
    CNS drugs, 2014, Volume: 28, Issue:3

    Topics: Adolescent; Adult; Aged; Biphenyl Compounds; Child; Colforsin; Coronary Vessels; Cyclic AMP; Dose-Response Relationship, Drug; Female; Humans; Male; Meningeal Arteries; Middle Aged; Muscle Contraction; Piperazines; Piperidones; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Spiro Compounds; Sumatriptan; Tissue Culture Techniques; Vasoconstrictor Agents; Vasodilator Agents; Young Adult

2014