Page last updated: 2024-08-16

sumatriptan and capsaicin

sumatriptan has been researched along with capsaicin in 32 studies

Research

Studies (32)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's12 (37.50)18.2507
2000's11 (34.38)29.6817
2010's7 (21.88)24.3611
2020's2 (6.25)2.80

Authors

AuthorsStudies
Fisk, L; Greene, N; Naven, RT; Note, RR; Patel, ML; Pelletier, DJ1
Ekins, S; Williams, AJ; Xu, JJ1
Boccalini, P; Moskowitz, MA; Nozaki, K1
Byun, B; Matsubara, T; Moskowitz, MA1
Buzzi, MG; Moskowitz, MA1
Connor, HE; O'Shaughnessy, CT; Waldron, GJ1
Cutrer, FM; Limmroth, V; Moskowitz, MA; Panahian, N; Schoenfeld, D1
Kumar, KL1
Ho, LT; Zochodne, DW1
Byun, B; Huang, Z; Matsubara, T; Moskowitz, MA1
Connor, HE; Feniuk, W; O'Shaughnessy, CT1
Titus, F1
Buckingham, JC; Kennard, C; Rhodes, KF1
Mitsikostas, DD; Moskowitz, MA; Sanchez del Rio, M; Waeber, C1
Longmore, J; Nwagwu, M; Olivar, T; Razzaque, Z1
Mitsikostas, DD; Sanchez del Rio, M; Waeber, C1
Markley, HG1
Cunha-Vaz, JG; Gaspar, MN; Macedo, TR; Ribeiro, CA1
Bigal, ME; Rapoport, AM; Sheftell, FD; Tepper, SJ1
Arulmani, U; Garrelds, IM; Heiligers, JP; Sánchez-López, A; Saxena, PR; Villalón, CM; Willems, EW1
Andrews, PL; Cheng, FH; Moreaux, B; Ngan, MP; Rudd, JA; Sam, TS; Wai, MK; Wan, C1
Centurión, D; Gupta, S; Jiménez-Mena, LR; Lozano-Cuenca, J; MaassenVanDenBrink, A; Mehrotra, S; Muñoz-Islas, E; Sánchez-López, A; Villalón, CM1
Akerman, S; Goadsby, PJ; Gupta, S; Saxena, PR; van den Brink, AM; van den Maagdenberg, AM1
Carmichael, NM; Charlton, MP; Dostrovsky, JO1
Centurión, D; González-Hernández, A; Lozano-Cuenca, J; Maassenvandenbrink, A; Muñoz-Islas, E; Ramírez-Rosas, MB; Sánchez-López, A; Villalón, CM1
Goadsby, PJ; Kavantzas, N; Knight, YE; Lasalandra, M; Mitsikostas, DD1
Durham, PL; Vause, CV1
Chen, PB; Hargreaves, KM; Loyd, DR1
Cheng, X; Disney, KE; Evans, MS; Jeffry, JA; Premkumar, LS1
Jang, IS; Nakamura, M1
Brocardo, PS; Cassol, G; da Silva Fiorin, F; do Espírito Santo, CC; do Nascimento, RS; Fighera, MR; Marques, JLB; Plácido, E; Royes, LFF; Santos, ARS1
Basedau, H; Jürgens, T; May, A; Ortlieb, L; Peng, KP1

Reviews

4 review(s) available for sumatriptan and capsaicin

ArticleYear
Recent advances in the acute management of migraine and cluster headaches.
    Journal of general internal medicine, 1994, Volume: 9, Issue:6

    Topics: Analgesics; Butorphanol; Capsaicin; Cluster Headache; Dihydroergotamine; Humans; Ketorolac; Metoclopramide; Migraine Disorders; Sumatriptan; Tolmetin

1994
[Symptomatic treatment of cluster headache].
    Revista de neurologia, 1995, Volume: 23 Suppl 4

    Topics: Alkaloids; Analgesics; Capsaicin; Cluster Headache; Cocaine; Dihydroergotamine; Ergotamine; Humans; Lidocaine; Methoxyflurane; Narcotics; Oxygen; Sumatriptan; Vasoconstrictor Agents

1995
Topical agents in the treatment of cluster headache.
    Current pain and headache reports, 2003, Volume: 7, Issue:2

    Topics: Administration, Intranasal; Administration, Topical; Capsaicin; Cluster Headache; Cocaine; Dihydroergotamine; Humans; Lidocaine; Oxazolidinones; Serotonin Receptor Agonists; Sumatriptan; Tryptamines; Vasoconstrictor Agents

2003
Intranasal medications for the treatment of migraine and cluster headache.
    CNS drugs, 2004, Volume: 18, Issue:10

    Topics: Administration, Intranasal; Analgesics; Capsaicin; Cluster Headache; Humans; Migraine Disorders; Oxazolidinones; Serotonin Receptor Agonists; Sumatriptan; Tryptamines

2004

Trials

1 trial(s) available for sumatriptan and capsaicin

ArticleYear
Sumatriptan prevents central sensitization specifically in the trigeminal dermatome in humans.
    European journal of pain (London, England), 2022, Volume: 26, Issue:10

    Topics: Capsaicin; Central Nervous System Sensitization; Headache; Humans; Hyperalgesia; Migraine Disorders; Pain; Sumatriptan; Tryptamines

2022

Other Studies

27 other study(ies) available for sumatriptan and capsaicin

ArticleYear
Developing structure-activity relationships for the prediction of hepatotoxicity.
    Chemical research in toxicology, 2010, Jul-19, Volume: 23, Issue:7

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Humans; Structure-Activity Relationship; Tetracyclines; Thiophenes

2010
A predictive ligand-based Bayesian model for human drug-induced liver injury.
    Drug metabolism and disposition: the biological fate of chemicals, 2010, Volume: 38, Issue:12

    Topics: Bayes Theorem; Chemical and Drug Induced Liver Injury; Humans; Ligands

2010
CP-93,129, sumatriptan, dihydroergotamine block c-fos expression within rat trigeminal nucleus caudalis caused by chemical stimulation of the meninges.
    British journal of pharmacology, 1992, Volume: 106, Issue:2

    Topics: Animals; Animals, Newborn; Capsaicin; Carrageenan; Dihydroergotamine; Formaldehyde; Gene Expression Regulation, Neoplastic; Guinea Pigs; Immunohistochemistry; In Vitro Techniques; Indoles; Meninges; Nasal Mucosa; Proto-Oncogene Proteins c-fos; Pyridines; Pyrroles; Rats; Sulfonamides; Sumatriptan

1992
CP-93,129, a potent and selective 5-HT1B receptor agonist blocks neurogenic plasma extravasation within rat but not guinea-pig dura mater.
    British journal of pharmacology, 1991, Volume: 104, Issue:1

    Topics: Animals; Blood Pressure; Capsaicin; Dura Mater; Electric Stimulation; Guinea Pigs; Indoles; Ligands; Male; Plasma; Proteins; Pyridines; Pyrroles; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serum Albumin, Radio-Iodinated; Sulfonamides; Sumatriptan; Trigeminal Ganglion; Vasoconstrictor Agents

1991
The antimigraine drug, sumatriptan (GR43175), selectively blocks neurogenic plasma extravasation from blood vessels in dura mater.
    British journal of pharmacology, 1990, Volume: 99, Issue:1

    Topics: Animals; Blood Pressure; Bradykinin; Capsaicin; Dura Mater; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Indoles; Male; Muscle, Smooth, Vascular; Neuropeptides; Rats; Rats, Inbred Strains; Serotonin; Serum Albumin, Radio-Iodinated; Sulfonamides; Sumatriptan; Tachykinins; Trigeminal Nerve; Vasoconstriction

1990
Lack of effect of sumatriptan and UK-14,304 on capsaicin-induced relaxation of guinea-pig isolated basilar artery.
    British journal of pharmacology, 1993, Volume: 108, Issue:1

    Topics: Animals; Basilar Artery; Brimonidine Tartrate; Calcitonin Gene-Related Peptide; Capsaicin; Dose-Response Relationship, Drug; Guinea Pigs; In Vitro Techniques; Indoles; Male; Quinoxalines; Ruthenium Red; Substance P; Sulfonamides; Sumatriptan; Vasoconstrictor Agents; Vasodilation

1993
Suppression by the sumatriptan analogue, CP-122,288 of c-fos immunoreactivity in trigeminal nucleus caudalis induced by intracisternal capsaicin.
    British journal of pharmacology, 1995, Volume: 114, Issue:5

    Topics: Animals; Aorta, Thoracic; Blood Pressure; Capsaicin; Cisterna Magna; Depression, Chemical; Guinea Pigs; Heart Rate; Immunohistochemistry; In Vitro Techniques; Injections; Male; Nociceptors; Proto-Oncogene Proteins c-fos; Pyrrolidines; Respiratory Mechanics; Sumatriptan; Trigeminal Ganglion

1995
Sumatriptan blocks neurogenic inflammation in the peripheral nerve trunk.
    Neurology, 1994, Volume: 44, Issue:1

    Topics: Animals; Capsaicin; Hyperemia; Male; Microcirculation; Neuritis; Rats; Rats, Sprague-Dawley; Regional Blood Flow; Sciatic Nerve; Sumatriptan; Vascular Resistance

1994
Time-dependent blockade of neurogenic plasma extravasation in dura mater by 5-HT1B/D agonists and endopeptidase 24.11.
    British journal of pharmacology, 1993, Volume: 108, Issue:2

    Topics: Animals; Capsaicin; Disease Models, Animal; Dura Mater; Electric Stimulation; Extravasation of Diagnostic and Therapeutic Materials; Guinea Pigs; Indoles; Male; Neprilysin; Neuropeptides; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Serotonin Receptor Agonists; Sulfonamides; Sumatriptan; Time Factors; Trigeminal Ganglion

1993
Extracellular recordings of membrane potential from guinea-pig isolated trigeminal ganglion: lack of effect of sumatriptan.
    Cephalalgia : an international journal of headache, 1993, Volume: 13, Issue:3

    Topics: Animals; Calcitonin Gene-Related Peptide; Capsaicin; gamma-Aminobutyric Acid; Guinea Pigs; In Vitro Techniques; Indoles; Male; Membrane Potentials; Potassium Chloride; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Sulfonamides; Sumatriptan; Trigeminal Ganglion

1993
The inhibition of nicotine-evoked relaxation of the guinea-pig isolated basilar artery by some analgesic drugs and progesterone.
    British journal of pharmacology, 1999, Volume: 126, Issue:4

    Topics: Analgesics; Animals; Aspirin; Basilar Artery; Capsaicin; Dinoprost; Guinea Pigs; In Vitro Techniques; Indomethacin; Male; Migraine Disorders; NG-Nitroarginine Methyl Ester; Nicotine; Progesterone; Substance P; Sumatriptan; Vasodilation

1999
Both 5-HT1B and 5-HT1F receptors modulate c-fos expression within rat trigeminal nucleus caudalis.
    European journal of pharmacology, 1999, Mar-26, Volume: 369, Issue:3

    Topics: Adrenergic beta-Antagonists; Animals; Capsaicin; Carbazoles; Dose-Response Relationship, Drug; Drug Interactions; Fluorobenzenes; Gene Expression; Genes, fos; Male; Pindolol; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Receptor Agonists; Sumatriptan; Trigeminal Caudal Nucleus

1999
Neurogenic vasodilation in rabbit basilar isolated artery: involvement of calcitonin-gene related peptide.
    European journal of pharmacology, 2000, Apr-21, Volume: 395, Issue:1

    Topics: Animals; Basilar Artery; Calcitonin Gene-Related Peptide; Calcitonin Gene-Related Peptide Receptor Antagonists; Capsaicin; Dose-Response Relationship, Drug; Endothelium, Vascular; Humans; In Vitro Techniques; Male; Oxazoles; Peptide Fragments; Pyrrolidines; Rabbits; Receptors, Vasoactive Intestinal Peptide; Serotonin Receptor Agonists; Sumatriptan; Vasoactive Intestinal Peptide; Vasoconstriction; Vasoconstrictor Agents; Vasodilation

2000
5-Hydroxytryptamine(1B/1D) and 5-hydroxytryptamine1F receptors inhibit capsaicin-induced c-fos immunoreactivity within mouse trigeminal nucleus caudalis.
    Cephalalgia : an international journal of headache, 2002, Volume: 22, Issue:5

    Topics: Anesthetics, General; Animals; Area Postrema; Brain Stem; Capsaicin; Carbazoles; Chloralose; Cisterna Magna; Dose-Response Relationship, Drug; Fluorobenzenes; Gene Expression Regulation; Genes, fos; Hemodynamics; Injections; Male; Mice; Models, Animal; Nerve Tissue Proteins; Pain; Proto-Oncogene Proteins c-fos; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptor, Serotonin, 5-HT1F; Receptors, Serotonin; Serotonin Receptor Agonists; Sumatriptan; Synaptic Transmission; Trigeminal Caudal Nucleus; Urethane; Vasomotor System

2002
Effects of neuropeptides on the sumatriptan-disturbed circulation in the optic nerve head of rabbits.
    Pharmacology, 2004, Volume: 70, Issue:3

    Topics: Animals; Arterioles; Blood-Retinal Barrier; Calcitonin Gene-Related Peptide; Capsaicin; Dose-Response Relationship, Drug; Female; Male; Microinjections; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Neuropeptides; Optic Nerve; Peptide Fragments; Rabbits; Receptors, Calcitonin Gene-Related Peptide; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Retinal Vessels; Substance P; Sumatriptan; Vasodilation

2004
Effects of sumatriptan on capsaicin-induced carotid haemodynamic changes and CGRP release in anaesthetized pigs.
    Cephalalgia : an international journal of headache, 2004, Volume: 24, Issue:9

    Topics: Animals; Calcitonin Gene-Related Peptide; Capsaicin; Carotid Arteries; Dose-Response Relationship, Drug; Female; Hemodynamics; Migraine Disorders; Serotonin Receptor Agonists; Sumatriptan; Sus scrofa; Trigeminal Nerve; Vagotomy; Vasodilation

2004
Evaluation of the anti-emetic potential of anti-migraine drugs to prevent resiniferatoxin-induced emesis in Suncus murinus (house musk shrew).
    European journal of pharmacology, 2005, Jan-31, Volume: 508, Issue:1-3

    Topics: Animals; Antiemetics; Butanols; Capsaicin; Cyclooxygenase Inhibitors; Dihydroergotamine; Diphenhydramine; Diterpenes; Domperidone; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Humans; Indomethacin; Malates; Methysergide; Metoclopramide; Migraine Disorders; Ondansetron; Piperidines; Ruthenium Red; Scopolamine; Serotonin Antagonists; Serotonin Receptor Agonists; Shrews; Sumatriptan; Time Factors; Tropanes; Vomiting

2005
Donitriptan, but not sumatriptan, inhibits capsaicin-induced canine external carotid vasodilatation via 5-HT1B rather than 5-HT1D receptors.
    British journal of pharmacology, 2006, Volume: 149, Issue:1

    Topics: Acetylcholine; Animals; Benzopyrans; Calcitonin Gene-Related Peptide; Capsaicin; Carotid Artery, External; Chromans; Dogs; Dose-Response Relationship, Drug; Hemodynamics; Humans; In Vitro Techniques; Infusions, Intravenous; Nitriles; Phenylephrine; Piperazines; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Serotonin Receptor Agonists; Sumatriptan; Tryptamines; Vasoconstrictor Agents; Vasodilation

2006
Intravital microscopy on a closed cranial window in mice: a model to study trigeminovascular mechanisms involved in migraine.
    Cephalalgia : an international journal of headache, 2006, Volume: 26, Issue:11

    Topics: Animals; Arteries; Calcitonin Gene-Related Peptide; Capsaicin; Disease Models, Animal; Dura Mater; Electric Stimulation; Male; Mice; Mice, Inbred C57BL; Microscopy, Video; Migraine Disorders; Piperazines; Quinazolines; Serotonin Receptor Agonists; Skull; Sumatriptan; Trigeminal Caudal Nucleus; Vasodilation

2006
Activation of the 5-HT1B/D receptor reduces hindlimb neurogenic inflammation caused by sensory nerve stimulation and capsaicin.
    Pain, 2008, Volume: 134, Issue:1-2

    Topics: Animals; Capsaicin; Hindlimb; Male; Neurogenic Inflammation; Neurons, Afferent; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Serotonin 5-HT1 Receptor Agonists; Serotonin Receptor Agonists; Sumatriptan

2008
Spinal sumatriptan inhibits capsaicin-induced canine external carotid vasodilatation via 5-HT1B rather than 5-HT1D receptors.
    European journal of pharmacology, 2009, Aug-01, Volume: 615, Issue:1-3

    Topics: Acetylcholine; Animals; Biphenyl Compounds; Calcitonin Gene-Related Peptide; Capsaicin; Carotid Artery, External; Chromans; Dogs; Dose-Response Relationship, Drug; Heart Rate; Hemodynamics; Infusions, Intravenous; Injections, Spinal; Male; Piperazines; Piperidones; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Spiro Compounds; Sumatriptan; Vasoconstriction; Vasoconstrictor Agents; Vasodilation

2009
Triptans attenuate capsaicin-induced CREB phosphorylation within the trigeminal nucleus caudalis: a mechanism to prevent central sensitization?
    The journal of headache and pain, 2011, Volume: 12, Issue:4

    Topics: Animals; Capsaicin; Cyclic AMP Response Element-Binding Protein; Hyperalgesia; Immunohistochemistry; Male; Pain; Phosphorylation; Piperidines; Rats; Rats, Sprague-Dawley; Sensory System Agents; Sumatriptan; Trigeminal Caudal Nucleus; Tryptamines

2011
Identification of cytokines and signaling proteins differentially regulated by sumatriptan/naproxen.
    Headache, 2012, Volume: 52, Issue:1

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Capsaicin; Cytokines; Drug Combinations; Drug Interactions; Gene Expression Regulation; Male; Naproxen; Protein Array Analysis; Rats; Rats, Sprague-Dawley; Serotonin 5-HT1 Receptor Agonists; Signal Transduction; Sumatriptan; Time Factors; Trigeminal Ganglion; Trigeminal Nucleus, Spinal

2012
Anti-hyperalgesic effects of anti-serotonergic compounds on serotonin- and capsaicin-evoked thermal hyperalgesia in the rat.
    Neuroscience, 2012, Feb-17, Volume: 203

    Topics: Animals; Capsaicin; Female; Hyperalgesia; Ketanserin; Male; Pain Measurement; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan

2012
Sumatriptan inhibits TRPV1 channels in trigeminal neurons.
    Headache, 2012, Volume: 52, Issue:5

    Topics: Action Potentials; Analysis of Variance; Animals; Animals, Newborn; Capsaicin; Carbocyanines; Dura Mater; Electric Stimulation; Excitatory Postsynaptic Potentials; Female; Gene Expression Regulation; In Vitro Techniques; Male; Neurons; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Serotonin 5-HT1 Receptor Agonists; Sumatriptan; Trigeminal Ganglion; TRPV Cation Channels

2012
Characterization of dural afferent neurons innervating cranial blood vessels within the dura in rats.
    Brain research, 2018, 10-01, Volume: 1696

    Topics: Animals; Calcium Channels; Capsaicin; Dura Mater; Female; Ganglia, Spinal; Male; Mechanoreceptors; Migraine Disorders; Nervous System Physiological Phenomena; Neurons, Afferent; Nociceptors; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Sensory Receptor Cells; Sumatriptan; Trigeminal Ganglion

2018
Capsaicin-sensitive fibers mediate periorbital allodynia and activation of inflammatory cells after traumatic brain injury in rats: Involvement of TRPV1 channels in post-traumatic headache.
    Neuropharmacology, 2020, 10-01, Volume: 176

    Topics: Animals; Animals, Newborn; Capsaicin; Headache; Inflammation Mediators; Male; Nerve Fibers; Post-Traumatic Headache; Rats; Rats, Wistar; Sensory System Agents; Sumatriptan; TRPV Cation Channels

2020