sumatriptan has been researched along with brl 15572 in 11 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 3 (27.27) | 18.2507 |
2000's | 5 (45.45) | 29.6817 |
2010's | 3 (27.27) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Brown, AM; Hundeshagen, AG; Kaumann, AJ; Schindler, M; Verheggen, R | 1 |
Centurión, D; De Vries, P; Heiligers, JP; Sánchez-López, A; Saxena, PR; Villalón, CM | 1 |
De Vries, P; Heiligers, JP; Saxena, PR; Villalón, CM; Willems, EW | 1 |
Centurión, D; Sánchez-López, A; Saxena, PR; Villalón, CM | 1 |
Hopwood, SE; Stamford, JA | 1 |
Crema, A; Crema, F; De Ponti, F; Frigo, G; Moro, E; Nardelli, G | 1 |
Arulmani, U; Centurión, D; Sánchez-López, A; Saxena, PR; Vázquez, E; Villalón, CM | 1 |
Centurión, D; González-Hernández, A; Lozano-Cuenca, J; Maassenvandenbrink, A; Muñoz-Islas, E; Ramírez-Rosas, MB; Sánchez-López, A; Villalón, CM | 1 |
Ribeiro, CA; Silva, SA | 1 |
Argüelles, CF; Godínez-Chaparro, B; Granados-Soto, V; López-Santillán, FJ; Villalón, CM | 1 |
Chan, KY; Danser, AH; de Vries, R; Dirven, C; Garrelds, IM; Labruijere, S; MaassenVanDenBrink, A; Ramírez Rosas, MB; van den Bogaerdt, A; Villalón, CM | 1 |
11 other study(ies) available for sumatriptan and brl 15572
Article | Year |
---|---|
5-HT1B receptor-mediated contractions in human temporal artery: evidence from selective antagonists and 5-HT receptor mRNA expression.
Topics: Adolescent; Adult; Aged; Base Sequence; Biphenyl Compounds; DNA Primers; Female; Humans; In Vitro Techniques; Male; Middle Aged; Muscle Contraction; Piperazines; Piperidones; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; RNA, Messenger; Serotonin Antagonists; Spiro Compounds; Sumatriptan; Temporal Arteries | 1998 |
The canine external carotid vasoconstrictor 5-HT1 receptor: blockade by 5-HT1B (SB224289), but not by 5-HT1D (BRL15572) receptor antagonists.
Topics: Anesthesia; Animals; Biphenyl Compounds; Blood Pressure; Carotid Artery, External; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Ergolines; Heart Rate; Norepinephrine; Piperazines; Piperidones; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiro Compounds; Sumatriptan; Sympathectomy; Vagotomy; Vasoconstriction | 1998 |
Investigation of the role of 5-HT1B and 5-HT1D receptors in the sumatriptan-induced constriction of porcine carotid arteriovenous anastomoses.
Topics: Animals; Arteriovenous Anastomosis; Biphenyl Compounds; Carotid Arteries; Dose-Response Relationship, Drug; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Piperazines; Piperidones; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds; Sumatriptan; Swine; Sympathectomy; Vagotomy; Vasoconstrictor Agents | 1999 |
Unravelling the pharmacological profile of the canine external carotid vasodilator '5-HT1-like' receptors: coexistence of sympatho-inhibitory 5-HT1B and postjunctional 5-HT7 receptors.
Topics: 5-Methoxytryptamine; Acetylcholine; Animals; Biphenyl Compounds; Blood Flow Velocity; Blood Pressure; Carotid Artery, External; Chromans; Dogs; Dose-Response Relationship, Drug; Female; Heart Rate; Hemodynamics; Male; Neuromuscular Junction; Oxadiazoles; Piperazines; Piperidones; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds; Sumatriptan; Sympathetic Nervous System; Vasodilation | 2001 |
Multiple 5-HT(1) autoreceptor subtypes govern serotonin release in dorsal and median raphé nuclei.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoreceptors; Benzamides; Biphenyl Compounds; Drug Synergism; Electric Stimulation; In Vitro Techniques; Male; Oxadiazoles; Piperazines; Protein Isoforms; Pyridines; Pyrroles; Raphe Nuclei; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Time Factors | 2001 |
Role of 5-HT1B/D receptors in canine gastric accommodation: effect of sumatriptan and 5-HT1B/D receptor antagonists.
Topics: Animals; Atropine; Benzamides; Bethanechol; Biphenyl Compounds; Dogs; Enzyme Inhibitors; Female; Gastric Emptying; NG-Nitroarginine Methyl Ester; Oxadiazoles; Parasympatholytics; Parasympathomimetics; Piperazines; Pressure; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Stomach; Sumatriptan; Vagus Nerve | 2003 |
Further characterization of the 5-HT1 receptors mediating cardiac sympatho-inhibition in pithed rats: pharmacological correlation with the 5-HT1B and 5-HT1D subtypes.
Topics: Animals; Biphenyl Compounds; Decerebrate State; Male; Norepinephrine; Oxadiazoles; Piperazines; Piperidones; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Spiro Compounds; Sumatriptan; Sympathomimetics; Tachycardia | 2004 |
Spinal sumatriptan inhibits capsaicin-induced canine external carotid vasodilatation via 5-HT1B rather than 5-HT1D receptors.
Topics: Acetylcholine; Animals; Biphenyl Compounds; Calcitonin Gene-Related Peptide; Capsaicin; Carotid Artery, External; Chromans; Dogs; Dose-Response Relationship, Drug; Heart Rate; Hemodynamics; Infusions, Intravenous; Injections, Spinal; Male; Piperazines; Piperidones; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Spiro Compounds; Sumatriptan; Vasoconstriction; Vasoconstrictor Agents; Vasodilation | 2009 |
Tachyphylaxis to the sumatriptan-induced contractile effect in the human uterine artery but not in human cerebral blood vessels: pharmacological demonstration of the 5-HT(1B) receptor functionality loss.
Topics: Adult; Basilar Artery; Biphenyl Compounds; Dose-Response Relationship, Drug; Drug Interactions; Female; Humans; In Vitro Techniques; Male; Middle Aged; Middle Cerebral Artery; Muscle, Smooth, Vascular; Pindolol; Piperazines; Piperidones; Receptor, Serotonin, 5-HT1B; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Spiro Compounds; Sumatriptan; Tachyphylaxis; Time Factors; Uterine Artery | 2012 |
Role of 5-HT₁B/₁D receptors in the reduction of formalin-induced nociception and secondary allodynia/hyperalgesia produced by antimigraine drugs in rats.
Topics: Acute Pain; Animals; Biphenyl Compounds; Chronic Pain; Dihydroergotamine; Disease Models, Animal; Drug Therapy, Combination; Female; Formaldehyde; Hyperalgesia; Methysergide; Nociceptive Pain; Piperazines; Piperidones; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Serotonin Antagonists; Spiro Compounds; Sumatriptan | 2013 |
Cranioselectivity of sumatriptan revisited: pronounced contractions to sumatriptan in small human isolated coronary artery.
Topics: Adolescent; Adult; Aged; Biphenyl Compounds; Child; Colforsin; Coronary Vessels; Cyclic AMP; Dose-Response Relationship, Drug; Female; Humans; Male; Meningeal Arteries; Middle Aged; Muscle Contraction; Piperazines; Piperidones; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Spiro Compounds; Sumatriptan; Tissue Culture Techniques; Vasoconstrictor Agents; Vasodilator Agents; Young Adult | 2014 |