sumatriptan has been researched along with 5-carboxamidotryptamine in 66 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 4 (6.06) | 18.7374 |
1990's | 52 (78.79) | 18.2507 |
2000's | 10 (15.15) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Branchek, TA; Hartig, PR; Macchi, MJ; Weinshank, RL; Zgombick, JM | 1 |
Beer, MS; Charlesworth, A; Iversen, LL; McAllister, G; Middlemiss, DN; Noble, AJ; Snodin, C; Whiting, P | 1 |
Hamblin, MW; Metcalf, MA | 1 |
Buckingham, J; Glen, RC; Hill, AP; Hyde, RM; Martin, GR; Robertson, AD; Salmon, JA; Woollard, PM | 1 |
Baker, R; Beer, MS; Davey, WB; Guiblin, AR; Jelley, RA; Reeve, AJ; Routledge, H; Sternfeld, F; Street, LJ; Watt, AP | 1 |
Bull, D; den Daas, I; Foord, S; Goodson, S; Kilpatrick, G; Lee, M; Rees, S | 1 |
Adham, N; Bard, JA; Branchek, TA; Vaysse, P; Weinshank, RL; Zgombick, J | 1 |
Adham, N; Bard, J; Branchek, TA; Durkin, M; Hartig, PR; Kao, HT; Olsen, M; Schecter, LE; Urquhart, D; Weinshank, RL | 1 |
Baron, BM; Burns, JE; Craft, CM; Danielson, PE; Erlander, MG; Lovenberg, TW; Racke, M; Siegel, BW; Slone, AL; Sutcliffe, JG | 1 |
Hamblin, MW; Jose, PA; Metcalf, MA; Monsma, FJ; Shen, Y; Sibley, DR | 1 |
Arrang, JM; Diaz, J; Leurs, R; Ruat, M; Schwartz, JC; Tardivel-Lacombe, J; Traiffort, E | 1 |
Amlaiky, N; Boschert, U; Grailhe, R; Hen, R; Mattei, MG; Matthes, H; Muscatelli, F; Plassat, JL | 1 |
Baker, R; Beer, MS; Castro, JL; Chambers, MS; Guiblin, AR; Hobbs, SC; Matassa, VG; Middlemiss, DN; Reeve, AJ; Street, LJ | 1 |
Brown, AM; Gaster, LM; Kaumann, AJ; King, FD; Medhurst, AD; Parker, SG; Parsons, AA; Patch, TL; Raval, P | 1 |
Druck, T; Hamblin, MW; Huebner, K; Khan, N; Kohen, R; Lachowicz, JE; Meltzer, HY; Metcalf, MA; Roth, BL; Sibley, DR | 1 |
Izzarelli, DG; Lewis-Higgins, L; Palmer, D; Parker, EM; Shapiro, RA | 1 |
Gommeren, W; Haegeman, G; Heylen, L; Lesage, AS; Leysen, JE; Luyten, WH; Schotte, A; Van de Weyer, I; Van Gompel, P; Vanhoenacker, P; Wouters, R | 1 |
Chang, DJ; Eglen, RM; Jasper, JR; Kosaka, A; To, ZP | 1 |
Boess, FG; Monsma, FJ; Sleight, AJ | 1 |
Grabtree, GW; Grailhe, R; Hen, R | 1 |
Bai, F; Johnstone, EM; Little, SP; Nelson, DL; Su, C; Varga, G; Yin, T | 1 |
Cleves, AE; Jain, AN; Kirshner, D; Langham, JJ; Spitzer, R | 1 |
Middlemiss, DN; Wilkinson, LO | 1 |
Eison, AS; Freeman, R; Wright, RN | 1 |
Beer, MS; Bevan, Y; Chauhan, NS; Middlemiss, DN; Stanton, JA | 1 |
Kaumann, AJ; Parsons, AA; Raval, P; Stutchbury, C | 1 |
Buzzi, MG; Byun, B; Moskowitz, MA; Peroutka, SJ | 1 |
Peroutka, SJ | 1 |
Feniuk, W; Saxena, PR; Tadipatri, S; van Heuven-Nolsen, D | 1 |
Higgins, GA; Jordan, CC; Skingle, M | 1 |
Hoyer, D; Sahin-Erdemli, I; Schoeffter, P; Seiler, MP; Stoll, A | 1 |
Connor, HE; Feniuk, W | 1 |
Connor, HE; Feniuk, W; Humphrey, PP | 1 |
Parsons, AA; Whalley, ET | 2 |
Cambridge, D; Whiting, MV | 1 |
Choppin, A; O'Connor, SE | 1 |
Baez, M; Cohen, ML; Cushing, DJ; Kursar, JD; Schenck, K | 1 |
Bruinvels, AT; Hoyer, D; Landwehrmeyer, B; Palacios, JM; Probst, A | 1 |
Ormandy, GC | 1 |
Edvinsson, L; Jansen, I; Olesen, J | 1 |
Carter, D; Champney, M; Eglen, RM; Hwang, B | 1 |
Bobirnac, I; Schoeffter, P | 1 |
Crick, H; Manuel, NA; Wallis, DI | 1 |
Castanon, N; Chauveau, J; Chaveau, J; Hen, R; Macor, JE; Moskowitz, MA; Scearce, K; Waeber, C; Yu, XJ | 1 |
Frölich, D; Göthert, M; Likungu, J; Molderings, GJ | 1 |
Böing, C; Bühlen, M; Fink, K; Göthert, M | 1 |
Feuerstein, TJ; Hüring, H; Landwehrmeyer, GB; Lücking, CH; van Velthoven, V | 1 |
Gutierrez, M; Lübbert, H; Schoeffter, P; Ullmer, C; Weitz-Schmidt, G | 1 |
Burton, M; Jones, BJ; Price, GW; Roberts, C; Watson, J | 1 |
Bonnafous, R; John, GW; Valentin, JP | 1 |
Cutrer, FM; Moskowitz, MA; Waeber, C; Yu, XJ | 1 |
De Vries, P; Heiligers, JP; Saxena, PR; Villalón, CM | 1 |
Curtis, MJ; Ellwood, AJ | 1 |
Colpaert, FC; Dupuis, DS; Pauwels, PJ | 1 |
Coupar, IM; Hemedah, M; Mitchelson, FJ | 1 |
Bard, JA; Branchek, T; Edvinsson, L; Longmore, J; Nilsson, T; Pantev, E; Shaw, D | 1 |
Falcón-Neri, A; Terrón, JA | 1 |
Bult, H; Geerts, IS; Herman, AG; Matthys, KE | 1 |
Bravo, G; Centurión, D; De Vries, P; Ortiz, MI; Saxena, PR; Villalón, CM | 1 |
Bax, WA; Maassen VanDenBrink, A; Reekers, M; Saxena, PR | 1 |
Cordi, AA; Ragonnet, C; Vayssettes-Courchay, C; Verbeuren, TJ | 1 |
Centurión, D; Sánchez-López, A; Saxena, PR; Villalón, CM | 1 |
Akita, H; Inoue, N; Ishida, T; Kawashima, S; Miwa, Y; Sakoda, T; Shimokawa, Y; Shiomi, M; Ueyama, T; Yokoyama, M | 1 |
Jähnichen, S; Pertz, HH; Radtke, OA | 1 |
Caparrotta, L; Dorigo, P; Froldi, G; Montopoli, M; Zanetti, M | 1 |
66 other study(ies) available for sumatriptan and 5-carboxamidotryptamine
Article | Year |
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Human serotonin 1D receptor is encoded by a subfamily of two distinct genes: 5-HT1D alpha and 5-HT1D beta.
Topics: Amino Acid Sequence; Animals; Brain; Cattle; Cell Membrane; Cloning, Molecular; DNA Probes; Female; Gene Library; Humans; Kinetics; Molecular Sequence Data; Multigene Family; Placenta; Pregnancy; Receptors, Serotonin; Recombinant Proteins; Sequence Homology, Nucleic Acid | 1992 |
Molecular cloning of a serotonin receptor from human brain (5HT1E): a fifth 5HT1-like subtype.
Topics: Adenylyl Cyclases; Amino Acid Sequence; Base Sequence; Binding, Competitive; Cell Line; Cloning, Molecular; Colforsin; DNA; Frontal Lobe; Gene Library; GTP-Binding Proteins; Hippocampus; Humans; Kinetics; Molecular Sequence Data; Oligodeoxyribonucleotides; Polymerase Chain Reaction; Receptors, Serotonin; Recombinant Proteins; Restriction Mapping; Sequence Homology, Nucleic Acid; Serotonin; Transfection | 1992 |
Primary structure and functional characterization of a human 5-HT1D-type serotonin receptor.
Topics: Amino Acid Sequence; Base Sequence; Cloning, Molecular; Cyclic AMP; GTP-Binding Proteins; Humans; Molecular Sequence Data; Pertussis Toxin; Receptors, Serotonin; Virulence Factors, Bordetella | 1991 |
Computer-aided design and synthesis of 5-substituted tryptamines and their pharmacology at the 5-HT1D receptor: discovery of compounds with potential anti-migraine properties.
Topics: Animals; Aorta; Computer-Aided Design; Drug Design; Haplorhini; In Vitro Techniques; Migraine Disorders; Models, Chemical; Rabbits; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1D; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Saphenous Vein; Serotonin Receptor Agonists; Structure-Activity Relationship; Tryptamines | 1995 |
Synthesis and serotonergic activity of N,N-dimethyl-2-[5-(1,2,4-triazol-1-ylmethyl)-1H-indol-3-yl]ethylamine and analogues: potent agonists for 5-HT1D receptors.
Topics: Animals; Rabbits; Rats; Serotonin Receptor Agonists; Structure-Activity Relationship; Triazoles; Tryptamines | 1995 |
Cloning and characterisation of the human 5-HT5A serotonin receptor.
Topics: Amino Acid Sequence; Animals; Base Sequence; Brain Chemistry; Cloning, Molecular; Genome, Human; GTP-Binding Proteins; Humans; Mice; Molecular Sequence Data; Radioligand Assay; Receptors, Serotonin; Sequence Analysis, DNA; Sequence Homology, Amino Acid; Sequence Homology, Nucleic Acid; Serotonin; Tissue Distribution; Transfection | 1994 |
Cloning of a novel human serotonin receptor (5-HT7) positively linked to adenylate cyclase.
Topics: Adenylyl Cyclases; Base Sequence; Cloning, Molecular; DNA Primers; Humans; Molecular Sequence Data; Receptors, Serotonin; Sequence Alignment; Sequence Homology, Amino Acid; Serotonin Antagonists; Serotonin Receptor Agonists; Signal Transduction | 1993 |
Cloning of another human serotonin receptor (5-HT1F): a fifth 5-HT1 receptor subtype coupled to the inhibition of adenylate cyclase.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Amino Acid Sequence; Animals; Base Sequence; Brain Chemistry; Cloning, Molecular; Colforsin; Dose-Response Relationship, Drug; Gene Library; Guinea Pigs; Humans; Indoles; Lymphocytes; Molecular Sequence Data; Receptors, Serotonin; RNA, Messenger; Sequence Homology, Amino Acid; Serotonin; Serotonin Receptor Agonists; Spiperone; Sulfonamides; Sumatriptan; Tissue Distribution | 1993 |
Molecular cloning and functional expression of 5-HT1E-like rat and human 5-hydroxytryptamine receptor genes.
Topics: Amino Acid Sequence; Animals; Base Sequence; Brain; Cell Line; Cell Membrane; Cloning, Molecular; Cyclic AMP; DNA; Gene Library; GTP-Binding Proteins; Humans; Kinetics; Lysergic Acid Diethylamide; Molecular Sequence Data; Multigene Family; Oligodeoxyribonucleotides; Organ Specificity; Polymerase Chain Reaction; Protein Processing, Post-Translational; Rats; Receptors, Serotonin; RNA, Messenger; Sequence Homology, Amino Acid; Transfection | 1993 |
Molecular cloning and expression of a 5-hydroxytryptamine7 serotonin receptor subtype.
Topics: Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Cell Line; Cell Membrane; Cloning, Molecular; Cyclic AMP; Gene Expression; Kidney Tubules, Proximal; Lysergic Acid Diethylamide; Molecular Sequence Data; Oligodeoxyribonucleotides; Polymerase Chain Reaction; Radioligand Assay; Rats; Receptors, Serotonin; Recombinant Proteins; Serotonin; Transfection | 1993 |
Molecular cloning, characterization, and localization of a high-affinity serotonin receptor (5-HT7) activating cAMP formation.
Topics: Amino Acid Sequence; Animals; Base Sequence; Blotting, Northern; Brain; CHO Cells; Cricetinae; Cyclic AMP; DNA; Genomic Library; Kinetics; Lysergic Acid Diethylamide; Mianserin; Molecular Sequence Data; Multigene Family; Oligodeoxyribonucleotides; Organ Specificity; Rats; Receptors, Serotonin; Restriction Mapping; Serotonin; Serotonin Receptor Agonists; Transfection | 1993 |
Mouse 5-hydroxytryptamine5A and 5-hydroxytryptamine5B receptors define a new family of serotonin receptors: cloning, functional expression, and chromosomal localization.
Topics: Amino Acid Sequence; Animals; Base Sequence; Brain; Cell Line; Chromosome Mapping; Cloning, Molecular; DNA; Gene Expression; Humans; In Situ Hybridization; Mice; Molecular Sequence Data; Receptors, Serotonin; Serotonin Receptor Agonists | 1993 |
Synthesis and serotonergic activity of 5-(oxadiazolyl)tryptamines: potent agonists for 5-HT1D receptors.
Topics: Animals; Binding, Competitive; Brain; In Vitro Techniques; Oxadiazoles; Rabbits; Receptors, Serotonin; Serotonin Receptor Agonists; Structure-Activity Relationship; Swine; Tryptamines; Vasoconstriction | 1993 |
(+/-) 3-Amino-6-carboxamido-1,2,3,4-tetrahydrocarbazole: a conformationally restricted analogue of 5-carboxamidotryptamine with selectivity for the serotonin 5-HT1D receptor.
Topics: Animals; Brain; Carbazoles; Dogs; In Vitro Techniques; Molecular Conformation; Rabbits; Rats; Receptors, Serotonin; Serotonin Receptor Agonists; Swine; Vasoconstriction | 1993 |
Cloning, characterization, and chromosomal localization of a human 5-HT6 serotonin receptor.
Topics: Adenylyl Cyclases; Amino Acid Sequence; Animals; Antipsychotic Agents; Base Sequence; Brain Chemistry; Cell Line, Transformed; Chlorocebus aethiops; Chromosome Mapping; Chromosomes, Human, Pair 1; Cloning, Molecular; Clozapine; DNA, Complementary; Genes; Humans; Kinetics; Molecular Sequence Data; Open Reading Frames; Protein Conformation; Rats; Receptors, Serotonin; Recombinant Proteins; Sequence Alignment; Sequence Homology, Nucleic Acid; Serotonin Agents; Signal Transduction; Species Specificity | 1996 |
Two amino acid differences in the sixth transmembrane domain are partially responsible for the pharmacological differences between the 5-HT1D beta and 5-HT1E 5-hydroxytryptamine receptors.
Topics: Amino Acid Sequence; Animals; Base Sequence; Binding Sites; Binding, Competitive; Chlorocebus aethiops; Cloning, Molecular; COS Cells; DNA Primers; Ergolines; Glutamic Acid; Humans; Isoleucine; Kinetics; Ligands; Lysine; Models, Structural; Molecular Sequence Data; Point Mutation; Polymerase Chain Reaction; Protein Structure, Secondary; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Recombinant Fusion Proteins; Sequence Homology, Amino Acid; Serine; Serotonin; Transfection | 1996 |
Alniditan, a new 5-hydroxytryptamine1D agonist and migraine-abortive agent: ligand-binding properties of human 5-hydroxytryptamine1D alpha, human 5-hydroxytryptamine1D beta, and calf 5-hydroxytryptamine1D receptors investigated with [3H]5-hydroxytryptamin
Topics: Animals; Benzopyrans; Cattle; Cloning, Molecular; Glioma; HeLa Cells; Humans; Mice; Migraine Disorders; Propylamines; Protein Binding; Pyrimidines; Radioligand Assay; Receptors, Serotonin; Serotonin Receptor Agonists; Signal Transduction; Tritium; Tumor Cells, Cultured; Vasoconstrictor Agents | 1996 |
Cloning, expression and pharmacology of a truncated splice variant of the human 5-HT7 receptor (h5-HT7b).
Topics: Alternative Splicing; Amino Acid Sequence; Animals; Base Sequence; Cloning, Molecular; Cyclic AMP; DNA, Complementary; Humans; Molecular Sequence Data; Placenta; Radioligand Assay; Rats; Receptors, Serotonin; RNA, Messenger; Sequence Homology, Amino Acid; Sequence Homology, Nucleic Acid | 1997 |
Identification of residues in transmembrane regions III and VI that contribute to the ligand binding site of the serotonin 5-HT6 receptor.
Topics: Adenylyl Cyclases; Amino Acid Substitution; Binding Sites; Binding, Competitive; Cell Line; Cyclic AMP; Humans; Ligands; Lysergic Acid Diethylamide; Mutagenesis, Site-Directed; Mutation; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists | 1998 |
Human 5-HT(5) receptors: the 5-HT(5A) receptor is functional but the 5-HT(5B) receptor was lost during mammalian evolution.
Topics: 3T3 Cells; Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Cell Line; COS Cells; DNA; Evolution, Molecular; Gene Expression; Genes; Humans; Membranes; Mice; Molecular Sequence Data; Phylogeny; Radioligand Assay; Receptors, Serotonin; Sequence Alignment; Sequence Analysis, DNA; Sequence Homology, Amino Acid | 2001 |
Molecular cloning and pharmacological characterization of the guinea pig 5-HT1E receptor.
Topics: Amino Acid Sequence; Animals; Base Sequence; Brain; Chickens; Cloning, Molecular; Cricetinae; Dose-Response Relationship, Drug; Gerbillinae; Guinea Pigs; Haplorhini; Humans; Molecular Sequence Data; Protein Binding; Rabbits; Receptors, Serotonin; Serotonin Agents; Swine | 2004 |
Physical binding pocket induction for affinity prediction.
Topics: Binding Sites; Ligands; Models, Molecular; Neural Networks, Computer; Peptide Fragments; Protein Binding; Receptor, Serotonin, 5-HT1A | 2009 |
Metitepine distinguishes two receptors mediating inhibition of [3H]-5-hydroxytryptamine release in guinea pig hippocampus.
Topics: Animals; Culture Techniques; Electric Stimulation; Guinea Pigs; Hippocampus; Indoles; Male; Methiothepin; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sulfonamides; Sumatriptan | 1992 |
Peripheral 5-carboxamidotryptamine induces hindlimb scratching by stimulating 5-HT1A receptors in rats.
Topics: 5-Methoxytryptamine; Animals; Behavior, Animal; Hindlimb; Indoles; Male; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Sulfonamides; Sumatriptan; Tryptamines | 1992 |
An investigation of the 5-HT1D receptor binding affinity of 5-hydroxytryptamine, 5-carboxyamidotryptamine and sumatriptan in the central nervous system of seven species.
Topics: Animals; Brain; Cattle; Caudate Nucleus; Cerebral Cortex; Cricetinae; Dogs; Guinea Pigs; Humans; Indoles; Kinetics; Rabbits; Radioligand Assay; Receptors, Serotonin; Serotonin; Species Specificity; Sulfonamides; Sumatriptan; Swine | 1992 |
Sumatriptan contracts large coronary arteries of beagle dogs through 5-HT1-like receptors.
Topics: Animals; Arteries; Coronary Vessels; Dogs; Endothelium, Vascular; Female; In Vitro Techniques; Indoles; Male; Methysergide; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Potassium Chloride; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Sulfonamides; Sumatriptan | 1992 |
Further characterization of the putative 5-HT receptor which mediates blockade of neurogenic plasma extravasation in rat dura mater.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Blood Pressure; Blood Proteins; Conjunctiva; Dura Mater; Ganglia, Sympathetic; Indoles; Inflammation; Male; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sulfonamides; Sumatriptan; Sympathectomy; Tetrahydronaphthalenes; Trigeminal Nerve; Vasoconstrictor Agents | 1991 |
Cortical and striatal variations in drug competition studies with putative 5-hydroxytryptamine1D binding sites.
Topics: Animals; Binding, Competitive; Cattle; Caudate Nucleus; Cerebral Cortex; Guinea Pigs; Humans; Indoles; Kinetics; Receptors, Serotonin; Serotonin; Sulfonamides; Sumatriptan; Swine | 1991 |
Analysis of the 5-HT receptors mediating contractions in the rabbit isolated renal artery.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Cocaine; In Vitro Techniques; Indoles; Ketanserin; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Oxidopamine; Phentolamine; Prostaglandin Endoperoxides, Synthetic; Rabbits; Receptors, Serotonin; Renal Artery; Serotonin; Serotonin Antagonists; Sulfonamides; Sumatriptan; Sympathectomy; Tetrahydronaphthalenes; Tyramine; Vasoconstrictor Agents; Vasodilation | 1991 |
Evidence that the unilateral activation of 5-HT1D receptors in the substantia nigra of the guinea-pig elicits contralateral rotation.
Topics: Animals; Behavior, Animal; Guinea Pigs; Indoles; Male; Methiothepin; Movement; Receptors, Serotonin; Rotation; Serotonin; Substantia Nigra; Sulfonamides; Sumatriptan | 1991 |
5-HT1-like receptors mediate 5-hydroxytryptamine-induced contraction of guinea-pig isolated iliac artery.
Topics: Animals; Guinea Pigs; Iliac Artery; In Vitro Techniques; Indoles; Ketanserin; Male; Methiothepin; Receptors, Serotonin; Serotonin; Sulfonamides; Sumatriptan; Tropisetron; Vasoconstriction | 1991 |
Influence of the endothelium on contractile effects of 5-hydroxytryptamine and selective 5-HT agonists in canine basilar artery.
Topics: Animals; Basilar Artery; Detergents; Dogs; Endothelium, Vascular; Female; In Vitro Techniques; Indoles; Ketanserin; Male; Methiothepin; Microscopy, Electron, Scanning; Octoxynol; Polyethylene Glycols; Potassium Chloride; Serotonin; Serotonin Antagonists; Sulfonamides; Sumatriptan | 1989 |
Characterization of 5-HT receptors mediating contraction of canine and primate basilar artery by use of GR43175, a selective 5-HT1-like receptor agonist.
Topics: Animals; Basilar Artery; Dogs; Female; In Vitro Techniques; Indoles; Macaca fascicularis; Male; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sulfonamides; Sumatriptan; Vasoconstriction | 1989 |
Characterization of the 5-hydroxytryptamine receptor which mediates contraction of the human isolated basilar artery.
Topics: Basilar Artery; Female; Humans; In Vitro Techniques; Indoles; Male; Muscle Contraction; Muscle, Smooth, Vascular; Receptors, Serotonin; Serotonin; Sulfonamides; Sumatriptan | 1989 |
Evidence for the presence of 5-HT1-like receptors in rabbit isolated basilar arteries.
Topics: Animals; Basilar Artery; Dinoprost; Endothelium, Vascular; In Vitro Techniques; Indoles; Male; Muscle Contraction; Muscle Tonus; Muscle, Smooth, Vascular; Rabbits; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sulfonamides; Sumatriptan | 1989 |
Canine renovascular responses to sumatriptan and 5-carboxamidotryptamine: modulation through endothelial 5-HT1-like receptors by endogenous nitric oxide.
Topics: Acetylcholine; Animals; Arginine; Blood Pressure; Dogs; Dose-Response Relationship, Drug; Endothelium, Vascular; Hemodynamics; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Receptors, Serotonin; Renal Artery; Renal Circulation; Serotonin; Serotonin Receptor Agonists; Sumatriptan | 1995 |
Presence of vasoconstrictor 5HT1-like receptors revealed by precontraction of rabbit isolated mesenteric artery.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; In Vitro Techniques; Male; Mesenteric Arteries; Muscle Contraction; Muscle, Smooth, Vascular; Potassium Chloride; Prostaglandin Endoperoxides, Synthetic; Rabbits; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Thromboxane A2; Vasoconstriction; Vasoconstrictor Agents | 1995 |
Serotonin-induced contraction in canine coronary artery and saphenous vein: role of a 5-HT1D-like receptor.
Topics: 5-Methoxytryptamine; Adrenergic alpha-Antagonists; Animals; Base Sequence; Blotting, Southern; Coronary Vessels; Dioxanes; DNA Primers; Dogs; Dose-Response Relationship, Drug; Gene Expression; Idazoxan; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth, Vascular; Piperazines; Polymerase Chain Reaction; Prazosin; Receptors, Serotonin; RNA, Messenger; Saphenous Vein; Serotonin; Serotonin Receptor Agonists; Sumatriptan; Tryptamines | 1994 |
A comparative autoradiographic study of 5-HT1D binding sites in human and guinea-pig brain using different radioligands.
Topics: Aged; Animals; Autoradiography; Binding Sites; Binding, Competitive; Brain; Dipeptides; Female; Guinea Pigs; Humans; Iodine Radioisotopes; Kinetics; Ligands; Male; Organ Specificity; Pyridines; Pyrroles; Receptors, Serotonin; Serotonin; Species Specificity; Sumatriptan; Tritium; Yohimbine | 1994 |
Increased cyclic AMP reduces 5-HT1D receptor-mediated inhibition of [3H]5-hydroxytryptamine release from guinea-pig cortical slices.
Topics: Animals; Bucladesine; Cerebral Cortex; Colforsin; Cyclic AMP; Guinea Pigs; In Vitro Techniques; Indoles; Phosphodiesterase Inhibitors; Potassium; Pyrrolidinones; Receptors, Serotonin; Rolipram; Serotonin; Serotonin Receptor Agonists; Sulfonamides; Sumatriptan | 1993 |
5-Hydroxytryptamine receptor characterization of human cerebral, middle meningeal and temporal arteries: regional differences.
Topics: 5-Methoxytryptamine; Cerebral Arteries; Humans; Indoles; Ketanserin; Meningeal Arteries; Methiothepin; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides; Sumatriptan; Temporal Arteries; Vasoconstriction; Vasoconstrictor Agents | 1993 |
Characterization of a postjunctional 5-HT receptor mediating relaxation of guinea-pig isolated ileum.
Topics: 5-Methoxytryptamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Cloning, Molecular; Drug Interactions; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; N,N-Dimethyltryptamine; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Substance P; Sumatriptan; Tryptamines | 1995 |
5-Hydroxytryptamine 5-HT1D receptors mediating inhibition of cyclic AMP accumulation in Madin-Darby canine kidney (MDCK) cells.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Alprostadil; Animals; Cells, Cultured; Cyclic AMP; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Epithelial Cells; Epithelium; Ketanserin; Kidney Cortex; Methiothepin; Oxadiazoles; Pertussis Toxin; Piperazines; Propranolol; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship; Sumatriptan; Virulence Factors, Bordetella; Yohimbine | 1995 |
Ketanserin-sensitive depressant actions of 5-HT receptor agonists in the neonatal rat spinal cord.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Animals, Newborn; Depression, Chemical; Dioxanes; Dopamine Antagonists; Drug Interactions; Female; Ketanserin; Male; Motor Neurons; Oxadiazoles; Pindolol; Piperazines; Propranolol; Rats; Rats, Wistar; Receptors, Serotonin; Reflex, Monosynaptic; Serotonin; Serotonin Antagonists; Spinal Cord; Spiro Compounds; Sumatriptan | 1995 |
5-Carboxamido-tryptamine, CP-122,288 and dihydroergotamine but not sumatriptan, CP-93,129, and serotonin-5-O-carboxymethyl-glycyl -tyrosinamide block dural plasma protein extravasation in knockout mice that lack 5-hydroxytryptamine1B receptors.
Topics: Animals; Capillary Permeability; Dihydroergotamine; Dipeptides; Mice; Mice, Knockout; Pyridines; Pyrroles; Pyrrolidines; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Sumatriptan; Trigeminal Ganglion | 1996 |
Inhibition of noradrenaline release via presynaptic 5-HT1D alpha receptors in human atrium.
Topics: 5-Methoxytryptamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic Uptake Inhibitors; Adult; Aged; Anti-Inflammatory Agents, Non-Steroidal; Cisapride; Corticosterone; Desipramine; Heart Atria; Humans; Indoles; Ketanserin; Male; Middle Aged; Norepinephrine; Oxadiazoles; Piperidines; Receptors, Presynaptic; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Tritium; Tryptamines | 1996 |
Evidence for presynaptic location of inhibitory 5-HT1D beta-like autoreceptors in the guinea-pig brain cortex.
Topics: Animals; Autoreceptors; Binding, Competitive; Cerebral Cortex; Guinea Pigs; Humans; Indoles; Ketanserin; Male; Methiothepin; Oxadiazoles; Oxymetazoline; Potassium; Radioligand Assay; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship; Sumatriptan; Synaptosomes; Tritium; Tryptamines | 1996 |
5-HT1D-like receptors inhibit the release of endogenously formed [3H]GABA in human, but not in rabbit, neocortex.
Topics: 3-Mercaptopropionic Acid; Adult; Animals; Cerebral Cortex; Electric Stimulation; Female; GABA Agents; GABA Antagonists; gamma-Aminobutyric Acid; Humans; In Vitro Techniques; Male; Middle Aged; Nicotinic Acids; Nipecotic Acids; Oximes; Rabbits; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Species Specificity; Sumatriptan; Tetrodotoxin | 1996 |
Functional serotonin 5-HT1D receptors and 5-HT1D beta receptor mRNA expression in human umbilical vein endothelial cells.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Cells, Cultured; Colforsin; Cyclic AMP; Endothelium, Vascular; Humans; Polymerase Chain Reaction; Receptors, Serotonin; RNA, Messenger; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Umbilical Veins | 1995 |
Functional characterization of the 5-HT terminal autoreceptor in the guinea-pig brain cortex.
Topics: Animals; Calcium Channel Blockers; Cerebral Cortex; Guinea Pigs; In Vitro Techniques; Male; Methiothepin; omega-Conotoxins; Peptides; Prefrontal Cortex; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan | 1996 |
Influence of the endothelium and nitric oxide on the contractile responses evoked by 5-HT1D receptor agonists in the rabbit isolated saphenous vein.
Topics: Animals; Endothelium, Vascular; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Oxadiazoles; Piperazines; Rabbits; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Saphenous Vein; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan | 1996 |
The 5-HT1D receptor antagonist GR-127,935 prevents inhibitory effects of sumatriptan but not CP-122,288 and 5-CT on neurogenic plasma extravasation within guinea pig dura mater.
Topics: Animals; Dose-Response Relationship, Drug; Dura Mater; Electric Stimulation; Female; Guinea Pigs; Male; Oxadiazoles; Pertussis Toxin; Piperazines; Prosencephalon; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sumatriptan; Trigeminal Nerve; Virulence Factors, Bordetella | 1997 |
Nature of 5-HT1-like receptors mediating depressor responses in vagosympathectomized rats; close resemblance to the cloned 5-ht7 receptor.
Topics: 5-Methoxytryptamine; Adrenergic beta-Agonists; Animals; Blood Pressure; Clozapine; Ergolines; Heart Rate; Isoproterenol; Lisuride; Male; Metergoline; Methiothepin; Oxadiazoles; Piperazines; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Sympathectomy | 1997 |
Involvement of 5-HT(1B/1D) and 5-HT2A receptors in 5-HT-induced contraction of endothelium-denuded rabbit epicardial coronary arteries.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Coronary Vessels; Endothelium, Vascular; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Oxadiazoles; Pericardium; Piperazines; Rabbits; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Vasoconstrictor Agents | 1997 |
G-protein activation at 5-HT1A receptors by the 5-ht1F ligand LY334370 in guinea-pig brain sections and recombinant cell lines.
Topics: Aminopyridines; Animals; Autoradiography; Benzamides; Binding Sites; Binding, Competitive; Brain; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guinea Pigs; HeLa Cells; Hippocampus; Humans; Indoles; Male; Piperazines; Pyridines; Raphe Nuclei; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan | 1998 |
[3H]-Mesulergine labels 5-HT7 sites in rat brain and guinea-pig ileum but not rat jejunum.
Topics: 5-Methoxytryptamine; Animals; Binding Sites; Binding, Competitive; Brain; Dose-Response Relationship, Drug; Ergolines; Female; Free Radical Scavengers; Guinea Pigs; Ileum; In Vitro Techniques; Jejunum; Male; Muscle Contraction; Ondansetron; Radioligand Assay; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds; Sulfonamides; Sumatriptan; Tritium | 1999 |
Characterisation of 5-HT receptors in human coronary arteries by molecular and pharmacological techniques.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Cardiovascular System; Coronary Vessels; Dose-Response Relationship, Drug; Gene Expression; Humans; Immunohistochemistry; In Vitro Techniques; Ketanserin; Methiothepin; Oxazoles; Oxazolidinones; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Tissue Distribution; Tryptamines; Vasoconstriction | 1999 |
Pharmacological evidence for the 5-HT7 receptor mediating smooth muscle relaxation in canine cerebral arteries.
Topics: Animals; Basilar Artery; Cerebral Arteries; Dinoprost; Dogs; Endothelium, Vascular; Female; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Spiperone; Sumatriptan | 1999 |
Involvement of 5-HT1B receptors in collar-induced hypersensitivity to 5-hydroxytryptamine of the rabbit carotid artery.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Braces; Carotid Arteries; Dose-Response Relationship, Drug; Hypersensitivity; In Vitro Techniques; Ketanserin; Male; Methysergide; Oxadiazoles; Piperazines; Potassium Chloride; Rabbits; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Sumatriptan; Tryptamines; Vasoconstriction | 1999 |
Further pharmacological analysis of the orphan 5-HT receptors mediating feline vasodepressor responses: close resemblance to the 5-HT7, receptor.
Topics: 5-Methoxytryptamine; Acetylcholine; Animals; Blood Pressure; Cats; Drug Interactions; Female; Heart Rate; Male; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Sympathectomy; Vagotomy | 2000 |
Human isolated coronary artery contraction to sumatriptan characterised by the selective 5-HT1B/1D receptor antagonist GR55562.
Topics: Benzamides; Coronary Vessels; Dinoprost; Dose-Response Relationship, Drug; Drug Interactions; Humans; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Potassium; Pyridines; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Substance P; Sumatriptan; Vasoconstrictor Agents | 2000 |
In vivo analysis of adrenergic and serotoninergic constrictions of the rabbit saphenous vein.
Topics: Adrenergic Agents; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Anesthesia; Animals; Benzazepines; Blood Pressure; Dogs; Dose-Response Relationship, Drug; Ergolines; Imidazoles; Indoles; Injections, Intravenous; Isoindoles; Oxadiazoles; Peripheral Nervous System; Phenylephrine; Piperazines; Prazosin; Rabbits; Receptors, Adrenergic, alpha; Receptors, Serotonin; Saphenous Vein; Serotonin; Serotonin Agents; Serotonin Receptor Agonists; Sumatriptan; Tetrahydronaphthalenes; Time Factors; Ultrasonography, Doppler; Vasoconstrictor Agents | 2000 |
Unravelling the pharmacological profile of the canine external carotid vasodilator '5-HT1-like' receptors: coexistence of sympatho-inhibitory 5-HT1B and postjunctional 5-HT7 receptors.
Topics: 5-Methoxytryptamine; Acetylcholine; Animals; Biphenyl Compounds; Blood Flow Velocity; Blood Pressure; Carotid Artery, External; Chromans; Dogs; Dose-Response Relationship, Drug; Female; Heart Rate; Hemodynamics; Male; Neuromuscular Junction; Oxadiazoles; Piperazines; Piperidones; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds; Sumatriptan; Sympathetic Nervous System; Vasodilation | 2001 |
Serotonin-induced hypercontraction through 5-hydroxytryptamine 1B receptors in atherosclerotic rabbit coronary arteries.
Topics: Animals; Arteriosclerosis; Calcium; Coronary Vessels; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Ketanserin; Male; Oxadiazoles; Phenylephrine; Piperazines; Rabbits; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; RNA, Messenger; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Vasoconstriction | 2001 |
Involvement of 5-HT1B receptors in triptan-induced contractile responses in guinea-pig isolated iliac artery.
Topics: Animals; Benzamides; Brain; Carbazoles; Dinoprost; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Endothelium, Vascular; Female; Forecasting; Guinea Pigs; Iliac Artery; Indoles; Ketanserin; Male; Muscle Contraction; Muscle, Smooth; Oxadiazoles; Oxazolidinones; Piperazines; Piperidines; Pyrrolidines; Receptor, Serotonin, 5-HT1B; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Sumatriptan; Triazoles; Tryptamines | 2004 |
5-HT1B receptor subtype and aging in rat resistance vessels.
Topics: Aging; Animals; Cerebral Arteries; Male; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Reverse Transcriptase Polymerase Chain Reaction; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Serotonin Receptor Agonists; Sumatriptan; Vascular Resistance; Vasoconstriction; Vasoconstrictor Agents; Vasodilator Agents | 2008 |