Page last updated: 2024-08-16

sulpiride and thiophenes

sulpiride has been researched along with thiophenes in 16 studies

Research

Studies (16)

TimeframeStudies, this research(%)All Research%
pre-19904 (25.00)18.7374
1990's10 (62.50)18.2507
2000's0 (0.00)29.6817
2010's1 (6.25)24.3611
2020's1 (6.25)2.80

Authors

AuthorsStudies
Fibiger, HC; Nomikos, GG; Tanaka, T; Vincent, SR1
De Vries, JB; Santiago, M; Westerink, BH1
Santiago, M; Westerink, BH3
Johnson, KM; Yi, SJ1
De Boer, P; De Vries, JB; Timmerman, W; Westerink, BH1
Damsma, G; de Boer, P; de Vries, JB; Fibiger, HC; Timmerman, W; Westerink, BH1
Farooqui, T; Harrold, MW; Miller, DD; Uretsky, N; Wallace, LJ; Wallace, RA1
De Vries, JB; Horn, AS; Tepper, PG; Timmerman, W; Westerink, BH1
Budai, D; Duckles, SP; Friedman, DJ; Krause, DN1
Plantjé, JF; Schipper, J; Stoof, JC; Verheijden, PF1
Harley, EA; Middlemiss, DN; Ragan, CI1
Cusack, NJ; Kelly, M; Martin, PL1
Feng, Z; Hou, T; Li, Y1
Johnson, SW; Munhall, AC; Yang, W1

Other Studies

16 other study(ies) available for sulpiride and thiophenes

ArticleYear
Effect of quinine on autoreceptor-regulated dopamine release in the rat striatum.
    Journal of neurochemistry, 1992, Volume: 59, Issue:5

    Topics: Animals; Calcium; Corpus Striatum; Dopamine; Dopamine Agents; Ergolines; Homeostasis; Male; Quinine; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D2; Sulpiride; Tetrahydronaphthalenes; Tetrodotoxin; Thiophenes

1992
In vivo evidence for a concordant response of terminal and dendritic dopamine release during intranigral infusion of drugs.
    Naunyn-Schmiedeberg's archives of pharmacology, 1992, Volume: 346, Issue:6

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Bicuculline; Brain; Dopamine; Dopamine Agents; Male; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Sulpiride; Tetrahydronaphthalenes; Thiophenes

1992
Characterization and pharmacological responsiveness of dopamine release recorded by microdialysis in the substantia nigra of conscious rats.
    Journal of neurochemistry, 1991, Volume: 57, Issue:3

    Topics: 3,4-Dihydroxyphenylacetic Acid; 4-Butyrolactone; Animals; Consciousness; Corpus Striatum; Dialysis; Dopamine; Dopamine Agents; Injections, Intraperitoneal; Male; Microchemistry; Nomifensine; Perfusion; Rats; Rats, Inbred Strains; Receptors, Dopamine; Substantia Nigra; Sulpiride; Tetrahydronaphthalenes; Tetrodotoxin; Thiophenes

1991
The regulation of dopamine release from nigrostriatal neurons in conscious rats: the role of somatodendritic autoreceptors.
    European journal of pharmacology, 1991, Oct-29, Volume: 204, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3,4-Dihydroxyphenylacetic Acid; Animals; Benzazepines; Consciousness; Corpus Striatum; Dendrites; Dopamine; Dopamine Agents; Dopamine Antagonists; Ergolines; Male; Neurons; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Substantia Nigra; Sulpiride; Tetrahydronaphthalenes; Thiophenes

1991
Role of adenylate cyclase in the modulation of the release of dopamine: a microdialysis study in the striatum of the rat.
    Journal of neurochemistry, 1990, Volume: 55, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; 3,4-Dihydroxyphenylacetic Acid; 8-Bromo Cyclic Adenosine Monophosphate; Adenylyl Cyclases; Animals; Corpus Striatum; Dialysis; Dopamine; Dopamine Agents; Homovanillic Acid; Hydroxyindoleacetic Acid; Male; Rats; Rats, Inbred Strains; Stereoisomerism; Sulpiride; Tetrahydronaphthalenes; Thiophenes

1990
Chronic cocaine treatment impairs the regulation of synaptosomal 3H-DA release by D2 autoreceptors.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 36, Issue:3

    Topics: Animals; Behavior, Animal; Calcium; Cocaine; Corpus Striatum; Dopamine; Dopamine Agents; Female; Nucleus Accumbens; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Sulpiride; Synaptosomes; Tetrahydronaphthalenes; Thiophenes

1990
In vivo evidence for the existence of autoreceptors on dopaminergic, serotonergic, and cholinergic neurons in the brain.
    Annals of the New York Academy of Sciences, 1990, Volume: 604

    Topics: Acetylcholine; Animals; Brain; Dialysis; Dopamine; Dopamine Agents; Homeostasis; Male; Neostigmine; Neurons; Parasympathetic Nervous System; Parasympathomimetics; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Serotonin; Stereoisomerism; Sulpiride; Tetrahydronaphthalenes; Thiophenes

1990
Dopaminergic-cholinergic interactions in the striatum: the critical significance of calcium concentrations in brain microdialysis.
    Naunyn-Schmiedeberg's archives of pharmacology, 1990, Volume: 342, Issue:5

    Topics: Acetylcholine; Animals; Apomorphine; Atropine; Calcium; Corpus Striatum; Dextroamphetamine; Dialysis Solutions; Dopamine; Haloperidol; Interneurons; Male; Neostigmine; Nomifensine; Perfusion; Rats; Rats, Inbred Strains; Sodium Chloride; Sulpiride; Tetrahydronaphthalenes; Thiophenes

1990
Synthesis and D2 dopaminergic activity of pyrrolidinium, tetrahydrothiophenium, and tetrahydrothiophene analogues of sulpiride.
    Journal of medicinal chemistry, 1989, Volume: 32, Issue:4

    Topics: Acetylcholine; Animals; Apomorphine; Cell Membrane; Chemical Phenomena; Chemistry; Corpus Striatum; Dopamine Antagonists; Potassium; Pyrrolidines; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Structure-Activity Relationship; Sulpiride; Thiophenes

1989
Microdialysis and striatal dopamine release: stereoselective actions of the enantiomers of N-0437.
    European journal of pharmacology, 1989, Mar-14, Volume: 162, Issue:1

    Topics: 3,4-Dihydroxyphenylacetic Acid; Administration, Cutaneous; Administration, Oral; Animals; Brain Chemistry; Corpus Striatum; Dialysis; Dopamine; Dopamine Agents; Injections, Intraperitoneal; Kainic Acid; Male; Naphthalenes; Rats; Rats, Inbred Strains; Stereoisomerism; Sulpiride; Tetrahydronaphthalenes; Thiophenes

1989
Prejunctional inhibitory effect of a dopamine D-2 agonist, N-0437, on vascular adrenergic responses.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 250, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Arteries; Benzazepines; Dopamine; Dopamine Antagonists; Electric Stimulation; In Vitro Techniques; Naphthalenes; Norepinephrine; Rabbits; Rats; Receptors, Dopamine; Sulpiride; Tetrahydronaphthalenes; Thiophenes; Vasoconstriction; Vasomotor System

1989
D2-dopamine receptors regulate the release of [3H]dopamine in rat basal hypothalamus and neurointermediate lobe of the pituitary gland.
    Brain research, 1987, Jun-16, Volume: 413, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Calcium; Dopamine; Electric Stimulation; Ergolines; Hypothalamus; Male; Norepinephrine; Pituitary Gland; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Sulpiride; Tetrahydronaphthalenes; Thiophenes

1987
Relationship between inhibition of cyclic AMP production in Chinese hamster ovary cells expressing the rat D2(444) receptor and antagonist/agonist binding ratios.
    British journal of pharmacology, 1995, Volume: 115, Issue:7

    Topics: Animals; CHO Cells; Cloning, Molecular; Cricetinae; Cyclic AMP; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Radioligand Assay; Rats; Receptors, Dopamine D2; Sulpiride; Tetrahydronaphthalenes; Thiophenes; Transfection

1995
(-)-2-(N-propyl-N-2-thienylethylamino)-5-hydroxytetralin (N-0923), a selective D2 dopamine receptor agonist demonstrates the presence of D2 dopamine receptors in the mouse vas deferens but not in the rat vas deferens.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 267, Issue:3

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Dopamine Agents; Idazoxan; Male; Mice; Rats; Receptors, Dopamine D2; Species Specificity; Sulpiride; Tetrahydronaphthalenes; Thiophenes; Vas Deferens

1993
Structure-based drug design for dopamine D3 receptor.
    Combinatorial chemistry & high throughput screening, 2012, Volume: 15, Issue:10

    Topics: Animals; Combinatorial Chemistry Techniques; Drug Design; Haloperidol; Humans; Indoles; Mice; Models, Molecular; Molecular Structure; Piperazines; Piperidines; Pyrazoles; Pyridines; Receptors, Dopamine D3; Spiperone; Structure-Activity Relationship; Sulpiride; Thiophenes

2012
Dopamine Evokes a Trace Amine Receptor-dependent Inward Current that is Regulated by AMP Kinase in Substantia Nigra Dopamine Neurons.
    Neuroscience, 2020, 02-10, Volume: 427

    Topics: AMP-Activated Protein Kinases; Animals; Benzamides; Benzazepines; Benzimidazoles; Biphenyl Compounds; Dopamine; Dopamine D2 Receptor Antagonists; Dopamine Plasma Membrane Transport Proteins; Dopaminergic Neurons; Naphthalimides; Pars Compacta; Patch-Clamp Techniques; Piperazines; Pyrazoles; Pyrimidines; Pyrones; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Sulpiride; Thiophenes

2020