sulpiride has been researched along with raclopride in 37 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 4 (10.81) | 18.7374 |
1990's | 16 (43.24) | 18.2507 |
2000's | 14 (37.84) | 29.6817 |
2010's | 3 (8.11) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Guo, YZ; Kasliwal, R; Kung, HF; Kung, MP; Mach, RH; Pan, SG | 1 |
Clanton, JA; de Paulis, T; Janowsky, A; Kessler, RM; Smith, HE | 1 |
Topliss, JG; Yoshida, F | 1 |
Fang, X; Hu, Z; Levant, B; Min, J; Varady, J; Wang, S; Wu, X | 1 |
Annand, R; Gozalbes, R; Jacewicz, M; Pineda-Lucena, A; Tsaioun, K | 1 |
Budygin, EA; Gaĭnetdinov, RR; Kovalev, GI; Kudrin, VS; Raevskiĭ, KS | 1 |
Brent, PJ | 1 |
Arrigoni, J; Dement, WC; Guilleminault, C; Mignot, E; Miller, JD; Nishino, S; Valtier, D | 1 |
Ahlenius, S; Briem, S; Hillegaart, V; Magnusson, O | 1 |
Hall, H; Wedel, I | 1 |
Farde, L; Halldin, C; Sedvall, G; Stone-Elander, S | 1 |
Deinum, ME; Schuiling, GA; Timmerman, W; Westerink, BH | 1 |
Andersson, I; Gustafsson, K; Westlind-Danielsson, A | 1 |
Ferré, S; Fuxe, K; O'Connor, WT; Snaprud, P; Ungerstedt, U | 1 |
Skarsfeldt, T | 1 |
Goldman-Rakic, PS; Sawaguchi, T | 1 |
Joppa, MA; Meisel, RL; Rowe, RK | 1 |
Derbiszewska, T; Nowak, JZ; Zawilska, JB | 1 |
Costall, B; Neill, JC; Smith, JK | 1 |
Fosbraey, P; Kitchen, I; Ridd, MJ | 1 |
Handley, SL; McCreary, AC | 1 |
Costall, B; Neill, JC; Smith, AG | 1 |
Carta, G; Gessa, GL; Nava, F | 1 |
Aguilar, MA; Arenas, MC; Miñarro, J; Parra, A; Simón, VM; Vinader-Caerols, C | 1 |
Hillefors, M; von Euler, G | 1 |
Arezzi, A; Drago, F; Virzì, A | 1 |
De Boer, P; De Vries, JB; Geels, C; Kawahara, Y; Kruse, CG; Long, SK; Van Kalkeren, A; Van Vliet, B; Westerink, BH; Wikström, HV | 1 |
Geary, N; Lutz, TA; Mollet, A; Scharrer, E; Tschudy, S | 1 |
Kapur, S; Ko, F; Seeman, P; Sun, WS | 1 |
Basta-Kaim, A; Budziszewska, B; Jaworska-Feil, L; Kubera, M; Lasoń, W; Leśkiewicz, M; Tetich, M | 1 |
Biala, G; Duarte, C; Hamon, M; Le Bihan, C; Thiébot, MH | 1 |
Durand, CJ; Lan, H; Neve, KA; Teeter, MM | 1 |
Bastianetto, S; Danik, M; Mennicken, F; Quirion, R; Williams, S | 1 |
Grasby, PM; Kitamura, Y; Mehta, MA; Montgomery, AJ | 1 |
Baroni, S; Betti, L; Castagna, M; Catena Dell'Osso, M; Consoli, G; Giannaccini, G; Lucacchini, A; Marazziti, D; Masala, I; Palego, L | 1 |
Ekström, J; Godoy, T; Riva, A | 1 |
Bussey, TJ; Heath, CJ; Saksida, LM | 1 |
1 trial(s) available for sulpiride and raclopride
Article | Year |
---|---|
Dopamine D2 receptor occupancy levels of acute sulpiride challenges that produce working memory and learning impairments in healthy volunteers.
Topics: Adult; Affect; Antipsychotic Agents; Carbon Radioisotopes; Corpus Striatum; Dopamine Antagonists; Dose-Response Relationship, Drug; Double-Blind Method; Humans; Male; Memory, Short-Term; Motor Activity; Neuropsychological Tests; Orientation; Pain Measurement; Pattern Recognition, Visual; Positron-Emission Tomography; Probability Learning; Prolactin; Raclopride; Reaction Time; Receptors, Dopamine D2; Serial Learning; Sulpiride | 2008 |
36 other study(ies) available for sulpiride and raclopride
Article | Year |
---|---|
Dopamine D-2 receptor imaging radiopharmaceuticals: synthesis, radiolabeling, and in vitro binding of (R)-(+)- and (S)-(-)-3-iodo-2-hydroxy-6-methoxy-N- [(1-ethyl-2-pyrrolidinyl)methyl]benzamide.
Topics: Animals; Benzamides; Chemical Phenomena; Chemistry; Corpus Striatum; In Vitro Techniques; Iodine Radioisotopes; Male; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Stereoisomerism; Structure-Activity Relationship | 1988 |
(S)-N-[(1-ethyl-2-pyrrolidinyl)methyl]-5-[125I]iodo- 2-methoxybenzamide hydrochloride, a new selective radioligand for dopamine D-2 receptors.
Topics: Animals; Benzamides; Chromatography, High Pressure Liquid; Isomerism; Kinetics; Male; Pyrrolidines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine | 1988 |
QSAR model for drug human oral bioavailability.
Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship | 2000 |
Molecular modeling of the three-dimensional structure of dopamine 3 (D3) subtype receptor: discovery of novel and potent D3 ligands through a hybrid pharmacophore- and structure-based database searching approach.
Topics: Algorithms; Binding Sites; Computational Biology; Crystallography, X-Ray; Databases, Protein; Humans; Kinetics; Ligands; Lipid Bilayers; Models, Molecular; Molecular Conformation; Mutation; Receptors, Dopamine D2; Receptors, Dopamine D3; Reproducibility of Results; Solvents; Structure-Activity Relationship; Tetrahydronaphthalenes; Water | 2003 |
QSAR-based permeability model for drug-like compounds.
Topics: Caco-2 Cells; Cell Membrane Permeability; Drug Discovery; Humans; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship | 2011 |
[Different effects of typical and atypical neuroleptics on K+-stimulated dopamine release from isolated rat striatum].
Topics: Animals; Antipsychotic Agents; Carbolines; Clozapine; Corpus Striatum; Dopamine; Dopamine Antagonists; In Vitro Techniques; Male; Metoclopramide; Potassium; Raclopride; Rats; Rats, Wistar; Remoxipride; Salicylamides; Stimulation, Chemical; Sulpiride; Thioridazine; Tiapamil Hydrochloride; Trifluoperazine | 1992 |
Behavioural effects of selective dopamine D-1 and D-2 agonists and antagonists in guinea-pigs.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Dopamine Antagonists; Dose-Response Relationship, Drug; Ergolines; Female; Guinea Pigs; Male; Motor Activity; Quinpirole; Raclopride; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Salicylamides; Sulpiride | 1991 |
Dopamine D2 mechanisms in canine narcolepsy.
Topics: Animals; Catalepsy; Dogs; Dopamine Antagonists; Ergolines; Motor Activity; Narcolepsy; Quinpirole; Raclopride; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Salicylamides; Sleep, REM; Sulpiride | 1991 |
Diffusion and absorption of (-)sulpiride and raclopride after intracerebral administration in the rat.
Topics: Absorption; Animals; Brain; Chromatography, High Pressure Liquid; Dopamine; Male; Raclopride; Rats; Rats, Inbred Strains; Salicylamides; Sulpiride | 1990 |
Comparisons between the in vitro binding of two substituted benzamides and two butyrophenones to dopamine-D2 receptors in the rat striatum.
Topics: Animals; Benzamides; Butyrophenones; Corpus Striatum; Domperidone; In Vitro Techniques; Ketanserin; Kinetics; Male; Piperidines; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Salicylamides; Spiperone; Sulpiride | 1986 |
PET analysis of human dopamine receptor subtypes using 11C-SCH 23390 and 11C-raclopride.
Topics: Adult; Benzazepines; Brain; Carbon Radioisotopes; Flupenthixol; Humans; Male; Middle Aged; Raclopride; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Salicylamides; Schizophrenia; Sulpiride | 1987 |
Lack of evidence for dopamine autoreceptors in the mediobasal hypothalamus: a microdialysis study in awake rats.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Benzazepines; Consciousness; Dopamine Antagonists; Haloperidol; Hypothalamus, Middle; Male; Microdialysis; Nomifensine; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine; Salicylamides; Sulpiride | 1995 |
Remoxipride shows low propensity to block functional striatal dopamine D2 receptors in vitro.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Action Potentials; Animals; Calcium; Colforsin; Corpus Striatum; Cyclic AMP; Dopamine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Haloperidol; In Vitro Techniques; Male; Pergolide; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Remoxipride; Salicylamides; Structure-Activity Relationship; Sulpiride | 1994 |
Antagonistic interaction between adenosine A2A receptors and dopamine D2 receptors in the ventral striopallidal system. Implications for the treatment of schizophrenia.
Topics: Adenosine; Animals; Antihypertensive Agents; Antipsychotic Agents; Autoradiography; Binding, Competitive; Dopamine D2 Receptor Antagonists; gamma-Aminobutyric Acid; Globus Pallidus; Microdialysis; Neostriatum; Nucleus Accumbens; Phenethylamines; Purinergic P1 Receptor Antagonists; Raclopride; Rats; Rats, Sprague-Dawley; Salicylamides; Schizophrenia; Sulpiride | 1994 |
Comparison of the effect of substituted benzamides on midbrain dopamine neurones after treatment of rats for 21 days.
Topics: Animals; Antipsychotic Agents; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Dopamine; Dopamine D2 Receptor Antagonists; Male; Neurons; Pyrrolidines; Raclopride; Rats; Rats, Wistar; Salicylamides; Substantia Nigra; Sulpiride; Ventral Tegmental Area | 1993 |
The role of D1-dopamine receptor in working memory: local injections of dopamine antagonists into the prefrontal cortex of rhesus monkeys performing an oculomotor delayed-response task.
Topics: Animals; Antipsychotic Agents; Appetitive Behavior; Attention; Benzazepines; Dominance, Cerebral; Dopamine; Dopamine Antagonists; Eye Movements; Fixation, Ocular; Haloperidol; Injections; Ketanserin; Macaca mulatta; Male; Mental Recall; Orientation; Prefrontal Cortex; Raclopride; Reaction Time; Receptors, Dopamine D1; Saccades; Salicylamides; Sulpiride | 1994 |
Dopamine receptor antagonists attenuate conditioned place preference following sexual behavior in female Syrian hamsters.
Topics: Animals; Behavior, Animal; Conditioning, Psychological; Cricetinae; Dopamine Antagonists; Dose-Response Relationship, Drug; Female; Raclopride; Salicylamides; Sexual Behavior, Animal; Sulpiride | 1996 |
Pharmacological modifications in dopaminergic neurotransmission affect the quinpirole-evoked suppression of serotonin N-acetyltransferase activity in chick retina: an impact on dopamine D4-like receptors.
Topics: Animals; Antipsychotic Agents; Arylamine N-Acetyltransferase; Chickens; Circadian Rhythm; Clozapine; Dopamine Agents; Enzyme Inhibitors; Levodopa; Male; Quinpirole; Raclopride; Receptors, Dopamine D2; Receptors, Dopamine D4; Retina; Salicylamides; Sulpiride; Synaptic Transmission | 1996 |
Bidirectional effects of dopamine D2 receptor antagonists on responding for a conditioned reinforcer.
Topics: Amphetamine; Animals; Benzazepines; Conditioning, Operant; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Female; Haloperidol; Motivation; Pimozide; Raclopride; Rats; Reinforcement, Psychology; Reward; Salicylamides; Sulpiride | 1997 |
The effect of acute kainic acid treatment on dopamine D2 receptors in rat brain.
Topics: Animals; Brain; Iodine Radioisotopes; Isotope Labeling; Kainic Acid; Male; Neurons; Protein Binding; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D2; Salicylamides; Spiperone; Sulpiride; Tritium | 1998 |
The thyrotrophin-releasing hormone analogue MK771 induces tic-like behaviours: the effects of dopamine D1 and D2 receptor antagonists.
Topics: Animals; Antidepressive Agents; Behavior, Animal; Behavioral Symptoms; Benzazepines; Blinking; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Male; Mice; Raclopride; Receptors, Dopamine D1; Salicylamides; Sulpiride; Thiazolidines; Thyrotropin-Releasing Hormone; Tic Disorders | 1999 |
The dopamine D3/D2 receptor agonist 7-OH-DPAT induces cognitive impairment in the marmoset.
Topics: Adrenergic alpha-Antagonists; Animals; Callithrix; Cognition; Discrimination Learning; Dopamine Agonists; Dopamine Antagonists; Female; Male; Raclopride; Receptors, Dopamine D2; Receptors, Dopamine D3; Salicylamides; Sulpiride; Tetrahydronaphthalenes; Yohimbine | 1999 |
Dopamine D(2) receptor antagonists prevent delta(9)-tetrahydrocannabinol-induced antinociception in rats.
Topics: Analgesics, Non-Narcotic; Animals; Bromocriptine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dronabinol; Male; Nociceptors; Pain; Piperidines; Pyrazoles; Quinpirole; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Rimonabant; Sulpiride | 1999 |
Predicting how equipotent doses of chlorpromazine, haloperidol, sulpiride, raclopride and clozapine reduce locomotor activity in mice.
Topics: Animals; Antipsychotic Agents; Chlorpromazine; Clozapine; Female; Haloperidol; Male; Mice; Motor Activity; Raclopride; Sulpiride | 2000 |
Pharmacology of [3H]R(+)-7-OH-DPAT binding in the rat caudate-putamen.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Benzopyrans; Binding, Competitive; Caudate Nucleus; Clozapine; Dopamine; Dopamine Agonists; Dopamine Antagonists; Guanidines; Guanosine Triphosphate; Haloperidol; Heterotrimeric GTP-Binding Proteins; Indans; Kinetics; Magnesium; Male; Oxazines; Protein Binding; Putamen; Quinpirole; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Remoxipride; Sodium; Specific Pathogen-Free Organisms; Sulfones; Sulpiride; Tetrahydronaphthalenes | 2001 |
Effects of acute or chronic administration of substituted benzamides in experimental models of depression in rats.
Topics: Animals; Antidepressive Agents; Benzamides; Clomipramine; Depression; Disease Models, Animal; Dose-Response Relationship, Drug; Male; Raclopride; Rats; Rats, Wistar; Sulpiride | 2000 |
Antipsychotic drugs classified by their effects on the release of dopamine and noradrenaline in the prefrontal cortex and striatum.
Topics: Animals; Antipsychotic Agents; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Haloperidol; Male; Norepinephrine; Prefrontal Cortex; Raclopride; Rats; Rats, Wistar; Receptors, Serotonin; Sulpiride | 2001 |
Dopamine D(2) receptors mediate amylin's acute satiety effect.
Topics: Amyloid; Animals; Anorexia; Benzazepines; Circadian Rhythm; Dextroamphetamine; Dopamine Agents; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Eating; Food Deprivation; Injections, Intraperitoneal; Islet Amyloid Polypeptide; Male; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Satiety Response; Sulpiride | 2001 |
Dopamine D2 receptors internalize in their low-affinity state.
Topics: Animals; Binding, Competitive; Brain; Cell Membrane; CHO Cells; Concanavalin A; Cricetinae; Dopamine; Dopamine Antagonists; Endocytosis; Guanine Nucleotides; Neurons; Protein Binding; Protein Transport; Raclopride; Radioligand Assay; Receptors, Dopamine D2; Sucrose; Sulpiride | 2002 |
Chlorpromazine inhibits the glucocorticoid receptor-mediated gene transcription in a calcium-dependent manner.
Topics: Animals; Antipsychotic Agents; Calcimycin; Calcium; Calcium Channel Blockers; Cell Line; Cell Line, Transformed; Chloramphenicol O-Acetyltransferase; Chlorpromazine; Clozapine; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Inhibitors; Estrenes; Fibroblasts; Gene Expression Regulation; Genes, Reporter; Haloperidol; Histamine; Histamine H1 Antagonists; Ionophores; Mammary Tumor Virus, Mouse; Mice; Nifedipine; Phorbol Esters; Phosphodiesterase Inhibitors; Protein Kinase C; Protein Kinase C-alpha; Pyrilamine; Pyrrolidinones; Raclopride; Receptors, Glucocorticoid; Remoxipride; Sulfonamides; Sulpiride; Tetradecanoylphorbol Acetate; Thionucleotides; Transcription, Genetic; Type C Phospholipases | 2002 |
Respective roles of dopamine D2 and D3 receptors in food-seeking behaviour in rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Amisulpride; Analysis of Variance; Animals; Apomorphine; Benzazepines; Benzopyrans; Conditioning, Operant; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Synergism; Feeding Behavior; Haloperidol; Male; Naphthalenes; Pyrroles; Pyrrolidines; Quinolines; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Reinforcement, Psychology; Sulpiride; Tetrahydronaphthalenes | 2003 |
Structural determinants of pharmacological specificity between D(1) and D(2) dopamine receptors.
Topics: Alternative Splicing; Animals; Benzazepines; Cell Line; Dopamine Antagonists; Models, Molecular; Mutation; Protein Conformation; Raclopride; Radioligand Assay; Rats; Receptors, Dopamine D1; Receptors, Dopamine D2; Solvents; Spiperone; Sulpiride | 2006 |
Prototypical antipsychotic drugs protect hippocampal neuronal cultures against cell death induced by growth medium deprivation.
Topics: Animals; Anisoles; Antipsychotic Agents; Benzazepines; Butaclamol; Caspase Inhibitors; Cell Death; Cells, Cultured; Chlorpromazine; Clozapine; Domperidone; Dopamine Antagonists; Excitatory Amino Acid Antagonists; Ginkgo biloba; Haloperidol; Hippocampus; Indans; Isoxazoles; Neurons; Neuroprotective Agents; Peptides; Piperidines; Plant Extracts; Propylamines; Raclopride; Rats; Rats, Sprague-Dawley; Reactive Oxygen Species; Receptors, N-Methyl-D-Aspartate; Remoxipride; Risperidone; Sulpiride | 2006 |
[(3)H]-YM-09151-2 binding sites in human brain postmortem.
Topics: Aged; Benzamides; Binding Sites; Brain Chemistry; Data Interpretation, Statistical; Dopamine Antagonists; Female; Hippocampus; Humans; In Vitro Techniques; Kinetics; Male; Middle Aged; Neostriatum; Postmortem Changes; Prefrontal Cortex; Propylamines; Raclopride; Receptors, Dopamine D4; Receptors, sigma; Sulpiride | 2009 |
Atypical antipsychotics--effects of amisulpride on salivary secretion and on clozapine-induced sialorrhea.
Topics: Amisulpride; Amylases; Animals; Antipsychotic Agents; Autonomic Agents; Bethanechol; Clozapine; Denervation; Female; Isoproterenol; Methacholine Chloride; Parasympathetic Nervous System; Parotid Gland; Raclopride; Rats; Rats, Sprague-Dawley; Saliva; Salivation; Sialorrhea; Submandibular Gland; Substance P; Sulpiride; Sympathetic Nervous System | 2012 |
Motivational assessment of mice using the touchscreen operant testing system: effects of dopaminergic drugs.
Topics: Amphetamine; Animals; Choice Behavior; Cognition; Conditioning, Operant; Dopamine Agents; Male; Mice; Mice, Inbred C57BL; Motivation; Raclopride; Reward; Sulpiride | 2015 |