Page last updated: 2024-08-16

sulpiride and piperidines

sulpiride has been researched along with piperidines in 52 studies

Research

Studies (52)

TimeframeStudies, this research(%)All Research%
pre-199017 (32.69)18.7374
1990's15 (28.85)18.2507
2000's12 (23.08)29.6817
2010's6 (11.54)24.3611
2020's2 (3.85)2.80

Authors

AuthorsStudies
Beckett, PR; Nahorski, SR; Roberts, DJ; Salazar, W1
Beckett, PR; Berga, P; Roberts, DJ1
Colombo, M; Llupia, J; Roberts, DJ; Salazar, W1
Ahlenius, S1
Bertolo, C; Forgione, A; Mussini, E; Salomoni, M; Zuccato, E1
Budziszewska, B; Grochmal, A; Przegaliński, E1
Bogdanov, MB; Gaĭnetdinov, RR; Kudrin, VS; Medvedev, OS; Val'dman, AV1
Gerlach, J1
D'Urso, R; Falaschi, P; Melis, GB; Proietti, A; Rocco, A; Rosa, M1
Fink, H; Morgenstern, R; Ott, T; Schremmer, C1
Henderson, G; Kennedy, C1
Duckles, SP; Massamiri, T1
Hatano, K; Hatazawa, J; Ido, T; Ishiwata, K; Itoh, M; Kawashima, K1
Altar, CA; Marshall, JF; O'Neil, S; Walter, RJ1
Andree, TH; Koenig, JI; Meltzer, HY; Mikuni, M; Tong, CY1
Carnoy, P; Puech, AJ; Simon, P; Soubrie, P1
Di Chiara, G; Longoni, R; Spina, L1
Hall, H; Wedel, I1
Bagetta, G; De Sarro, G; Nisticò, G; Priolo, E1
Appel, JB; Callahan, PM; Cunningham, KA2
Kruse, A; Lühdorf, K; Schulz, V1
Broekkamp, CL; Gower, AJ1
Collu, M; Gessa, GL; Serra, G1
Draper, R; Mulder, AH; Schoffelmeer, AN; Sminia, P; Stoof, JC1
Ståhle, L; Ungerstedt, U1
Perrault, G; Sanger, DJ1
Chiodo, LA; Freeman, AS; Zhang, J1
Bailey, MA; Kaiser, C; Karbon, EW; Mathew, RM; Mewshaw, RE; Sherrill, RG1
Akiyama, K; Kuroda, S; Okumura, K; Ujike, H1
Fang, H; Helmeste, DM; Li, M; Tang, SW1
Carta, G; Gessa, GL; Nava, F1
Blanchet, F; Gauchy, C; Glowinski, J; Kemel, ML; Pérez, S; Soubrié, P1
Fushiki, T; Imaizumi, M; Takeda, M1
Battasi, AM; Carta, G; Gessa, GL; Nava, F1
Fu, D; Javitch, JA; Lin, H; Strange, PG; Wilson, J1
Aceves, J; Arias-Montaño, JA; Floran, B; Garcia, M; Young, JM1
Doleviczényi, Z; Halmos, G; Kittel, A; Lendvai, B; Répássy, G; Vizi, ES; Zelles, T1
Kruse, CG; McCreary, AC; Olijslagers, JE; Perlstein, B; Siarey, R; Wadman, WJ; Werkman, TR1
Kreitzer, AC; Malenka, RC1
Bastianetto, S; Danik, M; Mennicken, F; Quirion, R; Williams, S1
Adermark, L; Lovinger, DM; Park, BS; Yin, HH1
Kumar, R; Sachdev, PS1
Haeri-Rohani, A; Nasehi, M; Sahebgharani, M; Zarrindast, MR1
Marti, M; Morari, M; Viaro, R1
Begemann, MJ; Leucht, S; Sommer, IE; Temmerman, A1
Adermark, L1
Feng, Z; Hou, T; Li, Y1
Dulawa, SC; Ho, EV; Klenotich, SJ; McMurray, MS; Server, CH1
Dang, DK; Jang, CG; Jeong, JH; Kim, HC; Ledent, C; Mai, AT; Nabeshima, T; Nah, SY; Onaivi, ES; Shin, EJ; Yamamoto, T1
Fanjul, A; Fothergill, LJ; Furness, JB; Furness, SGB; Pustovit, RV; Ringuet, MT; Syder, AJ; Whitfield, EA; Wykosky, J; Yoo, EJ1
Axelsson, SFA; Horiguchi, N; Horst, NK; Robbins, TW; Roberts, AC1

Reviews

3 review(s) available for sulpiride and piperidines

ArticleYear
New antipsychotics: classification, efficacy, and adverse effects.
    Schizophrenia bulletin, 1991, Volume: 17, Issue:2

    Topics: Antipsychotic Agents; Basal Ganglia Diseases; Benzamides; Humans; Isoxazoles; Piperidines; Receptors, Dopamine; Receptors, Glutamate; Receptors, Neurotransmitter; Receptors, Serotonin; Remoxipride; Risperidone; Schizophrenia; Serotonin Antagonists; Sulpiride

1991
Akathisia and second-generation antipsychotic drugs.
    Current opinion in psychiatry, 2009, Volume: 22, Issue:3

    Topics: Amisulpride; Antipsychotic Agents; Aripiprazole; Benzodiazepines; Clozapine; Dibenzothiazepines; Humans; Isoxazoles; Olanzapine; Piperazines; Piperidines; Prevalence; Psychomotor Agitation; Psychotic Disorders; Quetiapine Fumarate; Quinolones; Risk Factors; Risperidone; Sulpiride; Thiazoles

2009
Pharmacological augmentation strategies for schizophrenia patients with insufficient response to clozapine: a quantitative literature review.
    Schizophrenia bulletin, 2012, Volume: 38, Issue:5

    Topics: Antipsychotic Agents; Brief Psychiatric Rating Scale; Citalopram; Clozapine; Dioxoles; Double-Blind Method; Drug Synergism; Drug Therapy, Combination; Fructose; Humans; Lamotrigine; Piperidines; Psychiatric Status Rating Scales; Psychotropic Drugs; Randomized Controlled Trials as Topic; Schizophrenia; Schizophrenic Psychology; Sulpiride; Topiramate; Treatment Outcome; Triazines

2012

Trials

2 trial(s) available for sulpiride and piperidines

ArticleYear
New antipsychotics: classification, efficacy, and adverse effects.
    Schizophrenia bulletin, 1991, Volume: 17, Issue:2

    Topics: Antipsychotic Agents; Basal Ganglia Diseases; Benzamides; Humans; Isoxazoles; Piperidines; Receptors, Dopamine; Receptors, Glutamate; Receptors, Neurotransmitter; Receptors, Serotonin; Remoxipride; Risperidone; Schizophrenia; Serotonin Antagonists; Sulpiride

1991
Effect of ritanserin, specific 5HT-2 antagonist, on PRL secretion in normal subjects and in different hyperprolactinaemic conditions.
    Clinical endocrinology, 1991, Volume: 34, Issue:6

    Topics: Adenoma; Female; Follicular Phase; Humans; Hyperprolactinemia; Piperidines; Pituitary Neoplasms; Postpartum Period; Pregnancy; Prolactin; Ritanserin; Serotonin Antagonists; Single-Blind Method; Sulpiride

1991

Other Studies

48 other study(ies) available for sulpiride and piperidines

ArticleYear
[Clebopride, a new orthopramide with potent and selective central antidopaminergic properties].
    Archivos de farmacologia y toxicologia, 1978, Volume: 4, Issue:1

    Topics: Alprenolol; Animals; Benzamides; Dihydroergotoxine; Haloperidol; Metoclopramide; Piperidines; Rats; Receptors, Dopamine; Sulpiride

1978
[Antagonism of pre- and postsynaptic dopamine receptors by clebopride and related orthopramides].
    Archivos de farmacologia y toxicologia, 1979, Volume: 5, Issue:3

    Topics: Animals; Apomorphine; Benzamides; Dopamine Antagonists; Drug Interactions; Metoclopramide; Mice; Piperidines; Sulpiride; Synapses

1979
[Comparison of antiapomorphinic activity of metoclopramide, sulpiride and clebopride in the rat and dog].
    Archivos de farmacologia y toxicologia, 1978, Volume: 4, Issue:1

    Topics: Administration, Oral; Animals; Apomorphine; Benzamides; Dogs; Injections, Intravenous; Metoclopramide; Piperidines; Rats; Sulpiride

1978
Effects of the local application of 3-PPP and sulpiride enantiomers into the nucleus accumbens or into the ventral tegmental area on rat locomotor activity: evidence for the functional importance of somatodendritic autoreceptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1992, Volume: 345, Issue:5

    Topics: Animals; Dopamine Agents; Male; Motor Activity; Nucleus Accumbens; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sulpiride; Tegmentum Mesencephali

1992
The effects of S(-) and R(+) sulpiride, metoclopramide, cisapride and domperidone on the small intestine suggest DA2-receptors are involved in the control of small intestinal transit time in rats.
    Pharmacological research, 1992, Volume: 26, Issue:2

    Topics: Animals; Cisapride; Domperidone; Gastrointestinal Transit; Intestine, Small; Male; Metoclopramide; Piperidines; Random Allocation; Rats; Receptors, Dopamine D2; Serotonin Antagonists; Stereoisomerism; Sulpiride

1992
Oxaprotiline enantiomers stimulate ACTH and corticosterone secretion in the rat.
    Journal of neural transmission. General section, 1991, Volume: 85, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenocorticotropic Hormone; Animals; Antidepressive Agents; Benzylamines; Corticosterone; Dexamethasone; Diazepam; Dose-Response Relationship, Drug; Male; Maprotiline; Metergoline; Naloxone; Piperidines; Pyrimidines; Radioimmunoassay; Rats; Rats, Inbred Strains; Serotonin Antagonists; Stereoisomerism; Sulpiride; Sympathomimetics

1991
[Study by the intracerebral microdialysis method of the effects of atypical neuroleptics and anxiolytics on striatal release and metabolism of dopamine in awake rats].
    Biulleten' eksperimental'noi biologii i meditsiny, 1991, Volume: 111, Issue:5

    Topics: Animals; Anti-Anxiety Agents; Antipsychotic Agents; Brain Chemistry; Buspirone; Corpus Striatum; Dialysis; Dopamine; In Vitro Techniques; Isoxazoles; Male; Methoxydimethyltryptamines; Piperidines; Rats; Rats, Inbred Strains; Risperidone; Ritanserin; Sulpiride; Wakefulness

1991
Atypical neuroleptics suppress dopaminergic behavioral supersensitivity.
    Psychopharmacology, 1990, Volume: 100, Issue:3

    Topics: Animals; Antipsychotic Agents; Apomorphine; Behavior, Animal; Clozapine; Cyproheptadine; Haloperidol; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Ritanserin; Serotonin Antagonists; Sulpiride; Thioridazine

1990
Inhibition of potassium currents by the sigma receptor ligand (+)-3-(3-hydroxyphenyl)-N-(1-propyl)piperidine in sympathetic neurons of the mouse isolated hypogastric ganglion.
    Neuroscience, 1990, Volume: 35, Issue:3

    Topics: Animals; Atropine; Carbazoles; Dopamine Agents; Evoked Potentials; Ganglia, Sympathetic; In Vitro Techniques; Male; Membrane Potentials; Mice; Mice, Inbred DBA; Neurons; Piperidines; Potassium Channels; Receptors, Opioid; Receptors, sigma; Sulpiride; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin

1990
Multiple sites of action of (+)-3-(3-hydroxyphenyl)-N-(1-propyl)piperidine ((+)-3PPP) in blood vessels.
    European journal of pharmacology, 1990, Nov-13, Volume: 190, Issue:3

    Topics: Animals; Arteries; Cocaine; Desoxycorticosterone; Ear; Male; Muscle Contraction; Muscle, Smooth, Vascular; Neuromuscular Junction; Norepinephrine; Piperidines; Rabbits; Rats; Rats, Inbred Strains; Stimulation, Chemical; Sulpiride; Tail

1990
D2-dopamine receptor specific brain uptake of carbon-11-labeled YM-09151-2.
    Journal of nuclear medicine : official publication, Society of Nuclear Medicine, 1989, Volume: 30, Issue:4

    Topics: Animals; Antipsychotic Agents; Benzamides; Brain; Carbon Radioisotopes; Cerebellum; Corpus Striatum; Dogs; Male; Piperidines; Radionuclide Imaging; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Ritanserin; Serotonin Antagonists; Spiperone; Sulpiride

1989
Brain dopamine and serotonin receptor sites revealed by digital subtraction autoradiography.
    Science (New York, N.Y.), 1985, May-03, Volume: 228, Issue:4699

    Topics: Animals; Autoradiography; Brain; Butaclamol; Computers; Ketanserin; Piperidines; Radiographic Image Enhancement; Radionuclide Imaging; Rats; Receptors, Dopamine; Receptors, Serotonin; Spiperone; Sulpiride

1985
Differential effect of subchronic treatment with various neuroleptic agents on serotonin2 receptors in rat cerebral cortex.
    Journal of neurochemistry, 1986, Volume: 46, Issue:1

    Topics: 5,7-Dihydroxytryptamine; Animals; Antipsychotic Agents; Cerebral Cortex; Chlorpromazine; Clozapine; Female; Haloperidol; Imipramine; Ketanserin; Loxapine; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Spiperone; Sulpiride

1986
Performance deficit induced by low doses of dopamine agonists in rats. Toward a model for approaching the neurobiology of negative schizophrenic symptomatology?
    Biological psychiatry, 1986, Volume: 21, Issue:1

    Topics: Amisulpride; Animals; Antipsychotic Agents; Apomorphine; Disease Models, Animal; Male; Phenothiazines; Pimozide; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reinforcement Schedule; Reinforcement, Psychology; Schizophrenia; Schizophrenic Psychology; Sulpiride

1986
Permissive role of D-1 receptor stimulation by endogenous dopamine for the expression of postsynaptic D-2-mediated behavioural responses. Yawning in rats.
    European journal of pharmacology, 1987, Feb-10, Volume: 134, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adrenergic alpha-Agonists; Animals; Azepines; Benzazepines; Brain Chemistry; Dopamine; Ergolines; Kainic Acid; Ketanserin; Male; Metergoline; Piperidines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Sulpiride; Yawning

1987
Comparisons between the in vitro binding of two substituted benzamides and two butyrophenones to dopamine-D2 receptors in the rat striatum.
    Acta pharmacologica et toxicologica, 1986, Volume: 58, Issue:5

    Topics: Animals; Benzamides; Butyrophenones; Corpus Striatum; Domperidone; In Vitro Techniques; Ketanserin; Kinetics; Male; Piperidines; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Salicylamides; Spiperone; Sulpiride

1986
Ventral tegmental area: site through which dopamine D2-receptor agonists evoke behavioural and electrocortical sleep in rats.
    British journal of pharmacology, 1988, Volume: 95, Issue:3

    Topics: Animals; Apomorphine; Cerebral Cortex; Electroencephalography; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Sleep; Sulpiride; Tegmentum Mesencephali

1988
Discriminative stimulus properties of lisuride revisited: involvement of dopamine D2 receptors.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:1

    Topics: Animals; Benzazepines; Discrimination Learning; Ergolines; Lisuride; Male; Neurons; Piperidines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sulpiride

1987
Neuroleptic malignant syndrome due to combination of penfluridol and sulpiride?
    Acta psychiatrica Scandinavica, 1987, Volume: 75, Issue:3

    Topics: Aged; Drug Interactions; Female; Humans; Middle Aged; Neuroleptic Malignant Syndrome; Penfluridol; Piperidines; Sulpiride

1987
Dopaminergic agents including 3-PPP and its enantiomers on medial septal self-stimulation.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 22, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Appetite Depressants; Benzazepines; Dextroamphetamine; Drug Interactions; Haloperidol; Male; Nomifensine; Piperidines; Rats; Receptors, Dopamine; Self Stimulation; Stereoisomerism; Sulpiride; Tetrahydronaphthalenes

1985
Dopamine receptors mediating yawning: are they autoreceptors?
    European journal of pharmacology, 1986, Jan-21, Volume: 120, Issue:2

    Topics: Animals; Domperidone; Drug Synergism; Haloperidol; Male; Methyltyrosines; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reflex; Reserpine; Stereoisomerism; Sulpiride

1986
Agonist and antagonist effects of 3-PPP enantiomers on functional dopamine autoreceptors and postsynaptic dopamine receptors in vitro.
    European journal of pharmacology, 1985, Jan-08, Volume: 107, Issue:3

    Topics: Acetylcholine; Animals; Cholera Toxin; Corpus Striatum; Dopamine; In Vitro Techniques; Male; Melanocyte-Stimulating Hormones; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism; Sulpiride

1985
Discriminative stimulus properties of lergotrile.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 230, Issue:1

    Topics: Animals; Apomorphine; Discrimination Learning; Dose-Response Relationship, Drug; Ergolines; Ergonovine; Haloperidol; Lisuride; Lysergic Acid Diethylamide; Male; Piperidines; Pizotyline; Quipazine; Rats; Rats, Inbred Strains; Sulpiride

1984
Assessment of dopamine autoreceptor agonist properties of apomorphine, (+)-3-PPP and (-)-3-PPP by recording of yawning behaviour in rats.
    European journal of pharmacology, 1984, Feb-17, Volume: 98, Issue:2

    Topics: Animals; Apomorphine; Behavior, Animal; Domperidone; Male; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism; Sulpiride

1984
Effects of typical and atypical antipsychotic drugs on response decrement patterns in rats.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 272, Issue:2

    Topics: Animals; Antipsychotic Agents; Clozapine; Conditioning, Operant; Dose-Response Relationship, Drug; Haloperidol; Isoxazoles; Male; Piperidines; Rats; Rats, Wistar; Remoxipride; Risperidone; Serotonin Antagonists; Sulpiride

1995
Further characterization of the effects of BMY 14802 on dopamine neuronal activity.
    Synapse (New York, N.Y.), 1993, Volume: 15, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Dopamine; Dopamine Agents; Ergolines; Injections, Intravenous; Iontophoresis; Male; Neurons; Piperidines; Pyrimidines; Quinpirole; Rats; Rats, Sprague-Dawley; Serotonin Antagonists; Stereoisomerism; Sulpiride

1993
Synthesis and in vitro evaluation of 5,6,7,8,9,10-hexahydro-7,10-iminocyclohept[b]indoles: high-affinity ligands for the N,N'-di-o-tolylguanidine-labeled sigma binding site.
    Journal of medicinal chemistry, 1993, Feb-05, Volume: 36, Issue:3

    Topics: Animals; Binding, Competitive; Brain; Carbolines; Guanidines; Guinea Pigs; In Vitro Techniques; Piperidines; Radioligand Assay; Rats; Receptors, Dopamine D2; Receptors, sigma; Stereoisomerism; Structure-Activity Relationship; Sulpiride; X-Ray Diffraction

1993
BMY-14802 reversed the sigma receptor agonist-induced neck dystonia in rats.
    Journal of neural transmission (Vienna, Austria : 1996), 1996, Volume: 103, Issue:10

    Topics: Animals; Antipsychotic Agents; Dibenzothiepins; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dystonia; Guanidines; Haloperidol; Male; Microinjections; Nerve Tissue Proteins; Perphenazine; Piperidines; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, sigma; Red Nucleus; Sulpiride; Torticollis

1996
Multiple [3H]-nemonapride binding sites in calf brain.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 356, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Adrenergic alpha-Antagonists; Animals; Anticonvulsants; Benzamides; Binding, Competitive; Brain; Cattle; Cerebellum; Cerebral Cortex; Corpus Striatum; Dioxanes; Dopamine Agonists; Dopamine Antagonists; Guanidines; Haloperidol; In Vitro Techniques; Isotope Labeling; Narcotic Antagonists; Pentazocine; Piperidines; Propylamines; Pyrrolidines; Receptors, Dopamine D2; Receptors, sigma; Sulpiride; Tritium

1997
Dopamine D(2) receptor antagonists prevent delta(9)-tetrahydrocannabinol-induced antinociception in rats.
    European journal of pharmacology, 1999, Nov-19, Volume: 384, Issue:2-3

    Topics: Analgesics, Non-Narcotic; Animals; Bromocriptine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dronabinol; Male; Nociceptors; Pain; Piperidines; Pyrazoles; Quinpirole; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Rimonabant; Sulpiride

1999
Control by GABA and tachykinins of the evoked release of acetylcholine in striatal compartments under different modalities of NMDA receptor stimulation.
    Brain research, 2000, Jan-17, Volume: 853, Issue:1

    Topics: Acetylcholine; Animals; Benzamides; Bicuculline; Cell Compartmentation; Cells, Cultured; Corpus Striatum; Dopamine Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; N-Methylaspartate; Piperidines; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Receptors, Neurokinin-2; Stimulation, Chemical; Sulpiride; Tachykinins

2000
Effects of oil intake in the conditioned place preference test in mice.
    Brain research, 2000, Jul-07, Volume: 870, Issue:1-2

    Topics: Animals; Behavior, Animal; Benzazepines; Brain Chemistry; Conditioning, Psychological; Corn Oil; Dopamine Antagonists; Eating; Haloperidol; Indoles; Male; Mice; Piperidines; Receptors, Dopamine D1; Reward; Space Perception; Sulpiride

2000
D(2) dopamine receptors enable delta(9)-tetrahydrocannabinol induced memory impairment and reduction of hippocampal extracellular acetylcholine concentration.
    British journal of pharmacology, 2000, Volume: 130, Issue:6

    Topics: Acetylcholine; Analgesics, Non-Narcotic; Animals; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Dronabinol; Extracellular Space; Hippocampus; Memory; Piperidines; Pyrazoles; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Cannabinoid; Receptors, Dopamine D2; Receptors, Drug; Rimonabant; Sulpiride; Time Factors

2000
Mechanisms of inverse agonism of antipsychotic drugs at the D(2) dopamine receptor: use of a mutant D(2) dopamine receptor that adopts the activated conformation.
    Journal of neurochemistry, 2001, Volume: 77, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antipsychotic Agents; Apomorphine; Binding, Competitive; Bromocriptine; Butaclamol; Chlorpromazine; CHO Cells; Clozapine; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; GTP-Binding Proteins; Haloperidol; Humans; Macromolecular Substances; Mutagenesis, Site-Directed; Phenethylamines; Piperidines; Protein Binding; Protein Conformation; Radioligand Assay; Receptors, Dopamine D2; Recombinant Fusion Proteins; Sodium; Spiperone; Structure-Activity Relationship; Sulpiride; Transfection; Tyramine

2001
Histamine H(3) receptor-mediated inhibition of depolarization-induced, dopamine D(1) receptor-dependent release of [(3)H]-gamma-aminobutryic acid from rat striatal slices.
    British journal of pharmacology, 2001, Volume: 133, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Calcium; Dopamine; Dopamine D2 Receptor Antagonists; gamma-Aminobutyric Acid; Histamine; Histamine Agonists; Histamine Antagonists; Imidazoles; In Vitro Techniques; Male; Membrane Potentials; Neostriatum; Piperidines; Potassium; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Histamine H3; Reserpine; Sulpiride; Thiourea

2001
D2 autoreceptor inhibition reveals oxygen-glucose deprivation-induced release of dopamine in guinea-pig cochlea.
    Neuroscience, 2005, Volume: 132, Issue:3

    Topics: Animals; Cochlea; Dopamine; Dopamine Antagonists; Dopamine Uptake Inhibitors; Drug Interactions; Electric Stimulation; Glucose; Guinea Pigs; Hypoxia; In Vitro Techniques; Indoles; Male; Neurons; Nomifensine; Piperidines; Receptors, Dopamine D2; Sulpiride; Tetrodotoxin; Time Factors; Tritium

2005
The role of 5-HT(2A) receptor antagonism in amphetamine-induced inhibition of A10 dopamine neurons in vitro.
    European journal of pharmacology, 2005, Sep-27, Volume: 520, Issue:1-3

    Topics: Action Potentials; Amphetamine; Animals; Antipsychotic Agents; Benzodiazepines; Clozapine; Dopamine; Dopamine D2 Receptor Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Fluorobenzenes; In Vitro Techniques; Male; Mesencephalon; Neural Inhibition; Neurons; Olanzapine; Piperidines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Dopamine D2; Serotonin 5-HT2 Receptor Antagonists; Sulpiride

2005
Dopamine modulation of state-dependent endocannabinoid release and long-term depression in the striatum.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, Nov-09, Volume: 25, Issue:45

    Topics: Animals; Aspartic Acid; Benzoxazines; Calcium Channel Blockers; Cannabinoid Receptor Modulators; Cerebellum; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Radiation; Electric Stimulation; Endocannabinoids; Epistasis, Genetic; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; In Vitro Techniques; Long-Term Synaptic Depression; Membrane Potentials; Methoxyhydroxyphenylglycol; Morpholines; Naphthalenes; Neurons; Nitrendipine; Patch-Clamp Techniques; Piperidines; Pyrazoles; Quinpirole; Rats; Rats, Sprague-Dawley; Sulpiride; Time Factors

2005
Prototypical antipsychotic drugs protect hippocampal neuronal cultures against cell death induced by growth medium deprivation.
    BMC neuroscience, 2006, Mar-30, Volume: 7

    Topics: Animals; Anisoles; Antipsychotic Agents; Benzazepines; Butaclamol; Caspase Inhibitors; Cell Death; Cells, Cultured; Chlorpromazine; Clozapine; Domperidone; Dopamine Antagonists; Excitatory Amino Acid Antagonists; Ginkgo biloba; Haloperidol; Hippocampus; Indans; Isoxazoles; Neurons; Neuroprotective Agents; Peptides; Piperidines; Plant Extracts; Propylamines; Raclopride; Rats; Rats, Sprague-Dawley; Reactive Oxygen Species; Receptors, N-Methyl-D-Aspartate; Remoxipride; Risperidone; Sulpiride

2006
Ethanol reverses the direction of long-term synaptic plasticity in the dorsomedial striatum.
    The European journal of neuroscience, 2007, Volume: 25, Issue:11

    Topics: Animals; Animals, Newborn; Central Nervous System Depressants; Corpus Striatum; Dopamine Antagonists; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Electric Stimulation; Ethanol; Evoked Potentials; In Vitro Techniques; Neuronal Plasticity; Neurons; Patch-Clamp Techniques; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Sulpiride; Synaptic Transmission; Time Factors

2007
Effects of cannabinoids infused into the dorsal hippocampus upon memory formation in 3-days apomorphine-treated rats.
    Neurobiology of learning and memory, 2009, Volume: 92, Issue:3

    Topics: Animals; Apomorphine; Avoidance Learning; Benzazepines; Benzoxazines; Cannabinoids; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Hippocampus; Male; Memory; Mental Recall; Morpholines; Naphthalenes; Neuropsychological Tests; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Sulpiride; Time Factors

2009
Dual motor response to l-dopa and nociceptin/orphanin FQ receptor antagonists in 1-methyl-4-phenyl-1,2,5,6-tetrahydropyridine (MPTP) treated mice: Paradoxical inhibition is relieved by D(2)/D(3) receptor blockade.
    Experimental neurology, 2010, Volume: 223, Issue:2

    Topics: Amisulpride; Animals; Antiparkinson Agents; Benzimidazoles; Benzothiazoles; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Drug Interactions; Drug Synergism; Levodopa; Male; Mice; Mice, Inbred C57BL; Motor Activity; Neural Inhibition; Nociceptin; Opioid Peptides; Parkinsonian Disorders; Piperidines; Pramipexole; Pyridines; Reaction Time; Receptors, Dopamine D3; Sulpiride

2010
Modulation of endocannabinoid-mediated long-lasting disinhibition of striatal output by cholinergic interneurons.
    Neuropharmacology, 2011, Volume: 61, Issue:8

    Topics: Animals; Animals, Newborn; Benzazepines; Bicuculline; Biophysics; Cannabinoid Receptor Modulators; Cholinergic Agents; Chromones; Corpus Striatum; Dopamine Antagonists; Electric Stimulation; Endocannabinoids; Excitatory Amino Acid Antagonists; GABA-A Receptor Antagonists; In Vitro Techniques; Interneurons; Long-Term Potentiation; Models, Neurological; Neural Inhibition; Piperidines; Pyrazoles; Pyridines; Rats; Rats, Wistar; Signal Transduction; Sulpiride; Valine

2011
Structure-based drug design for dopamine D3 receptor.
    Combinatorial chemistry & high throughput screening, 2012, Volume: 15, Issue:10

    Topics: Animals; Combinatorial Chemistry Techniques; Drug Design; Haloperidol; Humans; Indoles; Mice; Models, Molecular; Molecular Structure; Piperazines; Piperidines; Pyrazoles; Pyridines; Receptors, Dopamine D3; Spiperone; Structure-Activity Relationship; Sulpiride; Thiophenes

2012
Dopamine D2/3 receptor antagonism reduces activity-based anorexia.
    Translational psychiatry, 2015, Aug-04, Volume: 5

    Topics: Amisulpride; Animals; Anorexia Nervosa; Benzodiazepines; Disease Models, Animal; Dopamine D2 Receptor Antagonists; Eating; Female; Indoles; Mice; Mice, Inbred BALB C; Motor Activity; Nitriles; Olanzapine; Piperidines; Receptors, Dopamine D3; Salicylamides; Sulpiride; Tetrahydroisoquinolines; Weight Loss

2015
Genetic or pharmacological depletion of cannabinoid CB1 receptor protects against dopaminergic neurotoxicity induced by methamphetamine in mice.
    Free radical biology & medicine, 2017, Volume: 108

    Topics: Animals; Apoptosis; Butadienes; Cells, Cultured; Corpus Striatum; Dopamine; Extracellular Signal-Regulated MAP Kinases; Methamphetamine; Mice; Mice, Inbred C57BL; Mice, Knockout; Neurotoxicity Syndromes; Nitriles; Oxidative Stress; Piperidines; Protein Kinase C-delta; Pyrazoles; Receptor, Cannabinoid, CB1; Receptors, Dopamine D2; Rimonabant; Sulpiride

2017
Dopamine and ghrelin receptor co-expression and interaction in the spinal defecation centers.
    Neurogastroenterology and motility, 2021, Volume: 33, Issue:5

    Topics: Animals; Defecation; Dopamine; Dopamine Agonists; Dopamine Antagonists; Gastrointestinal Motility; Ghrelin; Humans; Piperidines; Pramipexole; Quinazolinones; Quinpirole; Rats; Receptors, Dopamine D2; Receptors, Ghrelin; Spinal Cord; Spinal Cord Lateral Horn; Sulpiride

2021
Flexible versus Fixed Spatial Self-Ordered Response Sequencing: Effects of Inactivation and Neurochemical Modulation of Ventrolateral Prefrontal Cortex.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2021, 08-25, Volume: 41, Issue:34

    Topics: Animals; Antipsychotic Agents; Baclofen; Callithrix; Cognition Disorders; Dopamine; Dopamine D2 Receptor Antagonists; Fluorobenzenes; GABA Agonists; gamma-Aminobutyric Acid; Goals; Memory, Short-Term; Muscimol; Piperidines; Prefrontal Cortex; Psychomotor Performance; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Spatial Behavior; Sulpiride

2021