Page last updated: 2024-08-16

sulpiride and ketanserin

sulpiride has been researched along with ketanserin in 28 studies

Research

Studies (28)

TimeframeStudies, this research(%)All Research%
pre-19906 (21.43)18.7374
1990's11 (39.29)18.2507
2000's4 (14.29)29.6817
2010's7 (25.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Guo, YZ; Kasliwal, R; Kung, HF; Kung, MP; Mach, RH; Pan, SG1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Pan, JT; Tai, MH1
Frau, M; Gessa, GL; Stefanini, E1
Arai, I; Higuchi, T; Kazawa, T; Mikuni, M; Takahashi, K; Yamauchi, T1
Altar, CA; Marshall, JF; O'Neil, S; Walter, RJ1
Andree, TH; Koenig, JI; Meltzer, HY; Mikuni, M; Tong, CY1
Di Chiara, G; Longoni, R; Spina, L1
Hall, H; Wedel, I1
Ozaki, L; Stern, N; Tuck, ML1
Goldman-Rakic, PS; Sawaguchi, T1
Nowak, JZ; Zawilska, JB1
Wallis, DI; Wang, XC; Wu, J1
Jeffrey, JJ; Rydelek-Fitzgerald, L; Teitler, M; Wilcox, BD1
Takeshita, N; Yamaguchi, I1
Deschaux, P; Ferriere, F; Khan, NA; Meyniel, JP1
Fujiseki, Y; Inagaki, C; Kinoshita, T; Okugawa, G; Omori, K; Suzukawa, J1
Cryan, JF; Harkin, A; Kelly, JP; Leonard, BE; Naughton, M1
Appel, SB; Brodie, MS; Bunney, EB2
Bonfante, V; Dall'Olio, R; Gaggi, R; Gandolfi, O1
Araki, H; Hidaka, N; Suemaru, K1
Krishnamurthy, S; Saxena, B; Singh, S1
Barchini, J; Jabbur, SJ; Linderoth, B; Meyerson, BA; Saadé, NE; Shamaa, F; Song, Z; Tchachaghian, S1
Matsumoto, K; Oka, JI; Sasaki-Hamada, S; Suzuki, A; Ueda, Y1
Abbasi-Maleki, S; Mesbahzadeh, B; Moradi-Kor, N1

Other Studies

28 other study(ies) available for sulpiride and ketanserin

ArticleYear
Dopamine D-2 receptor imaging radiopharmaceuticals: synthesis, radiolabeling, and in vitro binding of (R)-(+)- and (S)-(-)-3-iodo-2-hydroxy-6-methoxy-N- [(1-ethyl-2-pyrrolidinyl)methyl]benzamide.
    Journal of medicinal chemistry, 1988, Volume: 31, Issue:5

    Topics: Animals; Benzamides; Chemical Phenomena; Chemistry; Corpus Striatum; In Vitro Techniques; Iodine Radioisotopes; Male; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Stereoisomerism; Structure-Activity Relationship

1988
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Effects of ketanserin on DOI-, MCPP- and TRH-induced prolactin secretion in estrogen-treated rats.
    Life sciences, 1992, Volume: 51, Issue:11

    Topics: Amphetamines; Animals; Dopamine Antagonists; Drug Synergism; Estrogens; Female; Ketanserin; Piperazines; Prolactin; Rats; Rats, Inbred Strains; Serotonin Antagonists; Sulpiride; Thyrotropin-Releasing Hormone; Time Factors

1992
Increase in D2 dopamine receptors in the substantia nigra after chronic (-)-sulpiride treatment.
    Brain research, 1991, Aug-02, Volume: 555, Issue:2

    Topics: Animals; Caudate Nucleus; Ketanserin; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Substantia Nigra; Sulpiride; Up-Regulation

1991
Characterization of sulpiride-displaceable 3H-YM-09151-2 binding sites in rat frontal cortex and the effects of subchronic treatment with haloperidol on cortical D-2 dopamine receptors.
    Life sciences, 1990, Volume: 47, Issue:6

    Topics: Animals; Benzamides; Binding Sites; Corpus Striatum; Dopamine Antagonists; Frontal Lobe; Haloperidol; In Vitro Techniques; Ketanserin; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sulpiride

1990
Brain dopamine and serotonin receptor sites revealed by digital subtraction autoradiography.
    Science (New York, N.Y.), 1985, May-03, Volume: 228, Issue:4699

    Topics: Animals; Autoradiography; Brain; Butaclamol; Computers; Ketanserin; Piperidines; Radiographic Image Enhancement; Radionuclide Imaging; Rats; Receptors, Dopamine; Receptors, Serotonin; Spiperone; Sulpiride

1985
Differential effect of subchronic treatment with various neuroleptic agents on serotonin2 receptors in rat cerebral cortex.
    Journal of neurochemistry, 1986, Volume: 46, Issue:1

    Topics: 5,7-Dihydroxytryptamine; Animals; Antipsychotic Agents; Cerebral Cortex; Chlorpromazine; Clozapine; Female; Haloperidol; Imipramine; Ketanserin; Loxapine; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Spiperone; Sulpiride

1986
Permissive role of D-1 receptor stimulation by endogenous dopamine for the expression of postsynaptic D-2-mediated behavioural responses. Yawning in rats.
    European journal of pharmacology, 1987, Feb-10, Volume: 134, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adrenergic alpha-Agonists; Animals; Azepines; Benzazepines; Brain Chemistry; Dopamine; Ergolines; Kainic Acid; Ketanserin; Male; Metergoline; Piperidines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Sulpiride; Yawning

1987
Comparisons between the in vitro binding of two substituted benzamides and two butyrophenones to dopamine-D2 receptors in the rat striatum.
    Acta pharmacologica et toxicologica, 1986, Volume: 58, Issue:5

    Topics: Animals; Benzamides; Butyrophenones; Corpus Striatum; Domperidone; In Vitro Techniques; Ketanserin; Kinetics; Male; Piperidines; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Salicylamides; Spiperone; Sulpiride

1986
Evidence for dopaminergic binding sites in the human adrenal cortex.
    Metabolism: clinical and experimental, 1986, Volume: 35, Issue:12

    Topics: Adrenal Cortex; Adult; Aged; Apomorphine; Binding, Competitive; Bromocriptine; Domperidone; Dopamine; Epinephrine; Female; Humans; Ketanserin; Male; Metoclopramide; Middle Aged; Receptors, Dopamine; Spiperone; Sulpiride; Time Factors

1986
The role of D1-dopamine receptor in working memory: local injections of dopamine antagonists into the prefrontal cortex of rhesus monkeys performing an oculomotor delayed-response task.
    Journal of neurophysiology, 1994, Volume: 71, Issue:2

    Topics: Animals; Antipsychotic Agents; Appetitive Behavior; Attention; Benzazepines; Dominance, Cerebral; Dopamine; Dopamine Antagonists; Eye Movements; Fixation, Ocular; Haloperidol; Injections; Ketanserin; Macaca mulatta; Male; Mental Recall; Orientation; Prefrontal Cortex; Raclopride; Reaction Time; Receptors, Dopamine D1; Saccades; Salicylamides; Sulpiride

1994
Dopamine receptor regulating serotonin N-acetyltransferase activity in chick retina represents a D4-like subtype: pharmacological characterization.
    Neurochemistry international, 1994, Volume: 24, Issue:3

    Topics: Animals; Arylamine N-Acetyltransferase; Benzamides; Benzazepines; Chickens; Circadian Rhythm; Clozapine; Dopamine; Dopamine Antagonists; Ergolines; Ketanserin; Male; Quinpirole; Receptors, Dopamine; Retina; Spiperone; Sulpiride

1994
Is 5-hydroxytryptamine mediating descending inhibition in the neonatal rat spinal cord through different receptor subtypes?
    European journal of pharmacology, 1993, Dec-21, Volume: 250, Issue:3

    Topics: Animals; Animals, Newborn; Citalopram; Dioxanes; Dopamine Antagonists; Electric Stimulation; Ketanserin; Lumbar Vertebrae; Methiothepin; Methysergide; Rats; Receptors, Serotonin; Reflex, Monosynaptic; Serotonin; Spinal Cord; Spinal Nerve Roots; Spiperone; Spiro Compounds; Sulpiride; Sumatriptan

1993
Serotonin-mediated 5-HT2 receptor gene regulation in rat myometrial smooth muscle cells.
    Molecular and cellular endocrinology, 1993, Volume: 92, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Biguanides; Cells, Cultured; Cycloheximide; Female; Gene Expression Regulation; Ketanserin; Medroxyprogesterone Acetate; Myometrium; Piperazines; Quipazine; Rats; Receptors, Serotonin; RNA, Messenger; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Sulpiride; Transcription, Genetic; Up-Regulation

1993
Insulin attenuates formalin-induced nociceptive response in mice through a mechanism that is deranged by diabetes mellitus.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 281, Issue:1

    Topics: Analgesics; Animals; Blood Glucose; Diabetes Mellitus, Experimental; Female; Formaldehyde; Indoles; Insulin; Ketanserin; Male; Mice; Mice, Inbred C57BL; Naloxone; Pindolol; Streptozocin; Sulpiride; Tropisetron

1997
5-Hydroxytryptamine-induced calcium-channel gating in rainbow trout (Oncorhynchus mykiss) peripheral blood lymphocytes.
    The Biochemical journal, 1997, Apr-01, Volume: 323 ( Pt 1)

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Calcium Channels; Dopamine Antagonists; Ion Channel Gating; Ionomycin; Ionophores; Ketanserin; Lymphocytes; Metoclopramide; Oncorhynchus mykiss; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulpiride

1997
Long-term treatment with antidepressants increases glucocorticoid receptor binding and gene expression in cultured rat hippocampal neurones.
    Journal of neuroendocrinology, 1999, Volume: 11, Issue:11

    Topics: Amitriptyline; Animals; Antidepressive Agents, Tricyclic; Cells, Cultured; Desipramine; Dexamethasone; Gene Expression Regulation; Haloperidol; Hippocampus; Ketanserin; Mianserin; Neurons; Paroxetine; Phentolamine; Propranolol; Radioligand Assay; Rats; Receptors, Glucocorticoid; Receptors, Mineralocorticoid; RNA, Messenger; Sulpiride; Transcription, Genetic; Tritium

1999
Characterization of D-fenfluramine-induced hypothermia: evidence for multiple sites of action.
    European journal of pharmacology, 2000, Mar-03, Volume: 390, Issue:3

    Topics: Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Benzofurans; Body Temperature; Cerebral Cortex; Dopamine Antagonists; Dose-Response Relationship, Drug; Fenclonine; Fenfluramine; Haloperidol; Hydroxyindoleacetic Acid; Hypothalamus; Hypothermia; Ketanserin; Male; Piperazines; Pyridines; Rats; Rats, Sprague-Dawley; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Sertraline; Sulpiride; Yohimbine

2000
Cocaine potentiates ethanol-induced excitation of dopaminergic reward neurons in the ventral tegmental area.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 293, Issue:2

    Topics: Animals; Central Nervous System Depressants; Cocaine; Dopamine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dopamine Uptake Inhibitors; Drug Synergism; Ethanol; Extracellular Space; Ketanserin; Neurons; Rats; Rats, Inbred F344; Reward; Serotonin Antagonists; Sulpiride; Ventral Tegmental Area

2000
The non-competitive NMDA receptor blocker dizocilpine potentiates serotonergic function.
    Behavioural pharmacology, 1999, Volume: 10, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Benzazepines; Dizocilpine Maleate; Dopamine Antagonists; Excitatory Amino Acid Antagonists; Ketanserin; Male; Motor Activity; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Dopamine D1; Receptors, N-Methyl-D-Aspartate; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Receptor Agonists; Sulpiride

1999
Electrophysiological effects of cocaethylene, cocaine, and ethanol on dopaminergic neurons of the ventral tegmental area.
    The Journal of pharmacology and experimental therapeutics, 2001, Volume: 297, Issue:2

    Topics: Animals; Central Nervous System Depressants; Cocaine; Dopamine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Electrophysiology; Ethanol; Extracellular Space; In Vitro Techniques; Ketanserin; Neurons; Rats; Rats, Inbred F344; Serotonin Antagonists; Sulpiride; Ventral Tegmental Area

2001
Serotonin-dopamine antagonism ameliorates impairments of spontaneous alternation and locomotor hyperactivity induced by repeated electroconvulsive seizures in rats.
    Epilepsy research, 2010, Volume: 90, Issue:3

    Topics: Analysis of Variance; Animals; Behavior, Animal; Dopamine Antagonists; Electroshock; Haloperidol; Hyperkinesis; Ketanserin; Male; Motor Activity; Random Allocation; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Serotonin, 5-HT2; Risperidone; Seizures; Serotonin Antagonists; Sulpiride

2010
Gastroprotective potential of risperidone, an atypical antipsychotic, against stress and pyloric ligation induced gastric lesions.
    Chemico-biological interactions, 2011, Apr-25, Volume: 190, Issue:2-3

    Topics: Animals; Antipsychotic Agents; Capillary Permeability; Dinoprostone; Disease Models, Animal; Dopamine D2 Receptor Antagonists; Glyburide; Hexosamines; Indomethacin; KATP Channels; Ketanserin; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Rats; Receptors, Dopamine D2; Receptors, Serotonin, 5-HT2; Risperidone; Stomach Ulcer; Stress, Physiological; Sulfhydryl Compounds; Sulpiride

2011
Spinal segmental and supraspinal mechanisms underlying the pain-relieving effects of spinal cord stimulation: an experimental study in a rat model of neuropathy.
    Neuroscience, 2012, Jul-26, Volume: 215

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Analysis of Variance; Animals; Baclofen; Bicuculline; Disease Models, Animal; Dopamine Antagonists; Electrodes; Female; GABA Antagonists; Hyperalgesia; Ketanserin; Methysergide; Neuralgia; Pain Measurement; Pain Threshold; Phentolamine; Propranolol; Rats; Rats, Sprague-Dawley; Serotonin Antagonists; Spinal Cord; Sulpiride; Time Factors; Transcutaneous Electric Nerve Stimulation

2012
Serotonergic and dopaminergic systems are implicated in antidepressant-like effects of chotosan, a Kampo formula, in mice.
    Journal of pharmacological sciences, 2017, Volume: 133, Issue:2

    Topics: Animals; Antidepressive Agents; Disease Models, Animal; Dopamine Agents; Drugs, Chinese Herbal; Fenclonine; Imipramine; Ketanserin; Locomotion; Male; Medicine, Kampo; Metergoline; Mice; Piperazines; Pyridines; Serotonin Agents; Sulpiride; Swimming; Yohimbine

2017
Zinc enhances the expression of morphine-induced conditioned place preference through dopaminergic and serotonergic systems.
    Biomolecular concepts, 2019, Apr-03, Volume: 10, Issue:1

    Topics: Animals; Benzazepines; Conditioning, Psychological; Dopamine Antagonists; Haloperidol; Ketanserin; Male; Morphine; Ondansetron; Piperazines; Rats; Rats, Wistar; Reward; Serotonin Antagonists; Sulpiride; Zinc

2019