sulpiride has been researched along with haloperidol in 569 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 268 (47.10) | 18.7374 |
1990's | 166 (29.17) | 18.2507 |
2000's | 84 (14.76) | 29.6817 |
2010's | 49 (8.61) | 24.3611 |
2020's | 2 (0.35) | 2.80 |
Authors | Studies |
---|---|
Campbell, BG; Kimes, AS; London, ED; Scheffel, U; Wilson, AA | 1 |
Clanton, JA; de Paulis, T; Janowsky, A; Kessler, RM; Smith, HE | 1 |
Angeby-Möller, K; de Paulis, T; Florvall, L; Hall, H; Johansson, L; Kumar, Y; Ogren, SO; Rämsby, S | 1 |
Hasegawa, O; Hirata, Y; Iwanami, S; Takashima, M; Usuda, S | 1 |
Florvall, L; Ogren, SO | 1 |
Ahern, DG; Filer, CN; Grigoriadis, D; Guan, JH; Lilly, L; Neumeyer, JL; Seeman, P; Watanabe, M | 1 |
Audiau, F; Carpy, A; Guérémy, C; Le Fur, G; Léger, JM; Uzan, A | 1 |
Topliss, JG; Yoshida, F | 1 |
Fang, X; Hu, Z; Levant, B; Min, J; Varady, J; Wang, S; Wu, X | 1 |
Boeckler, F; Gmeiner, P; Lanig, H | 1 |
Caron, G; Ermondi, G | 1 |
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J | 1 |
Bleich, S; Gulbins, E; Kornhuber, J; Reichel, M; Terfloth, L; Tripal, P; Wiltfang, J | 1 |
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV | 1 |
Chen, L; He, Z; Li, H; Liu, J; Liu, X; Sui, X; Sun, J; Wang, Y; Zhang, W | 1 |
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A | 1 |
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV | 1 |
Boriss, H; Braggio, S; Corbioli, S; Fontana, S; Helmdach, L; Longhi, R; Schiller, J; Vinco, F | 1 |
Annand, R; Gozalbes, R; Jacewicz, M; Pineda-Lucena, A; Tsaioun, K | 1 |
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ | 1 |
Chen, L; Fei, J; Mei, Y; Ren, S; Yan, SF; Zeng, J; Zhang, JZ | 1 |
Bartholini, G | 1 |
Ackenheil, M; von Stralendorff, B; Zimmermann, J | 1 |
Bonollo, L; Cassano, GB; Castrogiovanni, P; Conti, L | 2 |
Costa, E | 1 |
Di Chiara, G; Loddo, P; Spano, PF; Tonon, GC; Trabucchi, M | 1 |
Cianchetti, C; Corsini, GU; Del Zompo, M; Gessa, GL; Manconi, S; Mangoni, A | 1 |
Dedek, J; Korf, J; Scatton, B | 2 |
Costall, B; Naylor, RJ; Nohria, V; Owen, RT | 1 |
Munday, KA; Poat, JA; Sumners, C; Woodruff, GN | 1 |
Horowski, R | 1 |
Bronzetti, B; Ciriaco, E; Germanà, G; Nisticó, G; Rotiroti, D; Scapagnini, U | 1 |
Hashimoto, M; Honda, F; Mori, J; Mukumoto, S | 1 |
Bellodi, L; Fabio, G; Rugarli, C; Sacchetti, E; Scorza-Smeraldi, R; Smeraldi, E | 1 |
Beckett, PR; Nahorski, SR; Roberts, DJ; Salazar, W | 1 |
Liebman, J; Moen, NJ; Neale, R | 1 |
Cianchetti, C; Corsini, GU; Gessa, G; Mangoni, A; Masala, C; Onali, P | 1 |
Fresia, P; Longoni, R; Spano, PF; Trabucchi, M | 1 |
Honda, F; Mori, J; Satoh, H; Satoh, Y | 1 |
Arimura, A; Dupont, A; Linthicum, GL; Redding, TW; Schally, AV | 1 |
Bentolila, A; Coll-García, E; Lechin, F; Peña, F; Rivas, C; van der Dijs, B | 1 |
Lechin, F; Van Der Dijs, B | 4 |
Honda, F; Kato, R; Noguchi, H; Satoh, H; Satoh, Y; Shimomura, K; Uchida, S | 1 |
Angeby, T; Haglund, L; Köhler, C; Ogren, SO | 2 |
Scatton, B | 1 |
Garau, L; Govoni, S; Spano, PF; Stefanini, E; Trabucchi, M | 1 |
Cassano, GB; Castrogiovanni, P; Conti, L | 1 |
Bonollo, L; Cassano, GB; Castrogiovanni, P; Conti, L; Maggini, C; Sarteschi, P | 1 |
Costall, B; Naylor, RJ | 3 |
Caroli, F; Deniker, P; Ginestet, D; Littre-Poirier, MF | 1 |
Loizzo, A; Longo, VG; Mora, S | 1 |
Baudry, M; Martres, MP; Schwartz, JC | 1 |
Boissier, JR; Puech, AJ; Simon, P | 1 |
Korf, J; Westerink, BH | 1 |
Roufogalis, BD; Thornton, M; Wade, DN | 1 |
Maître, L; Waldmeier, PC | 1 |
Brion, S; Chevalier, JF; Ginestet, D; Guerin, R | 1 |
Gräf, HJ; Horowski, R | 1 |
Abe, K; de Francisco, CP | 1 |
Fukushima, H; Honma, T | 1 |
Cianchetti, C; Corsini, GU; Mangoni, A; Zompo, MD | 1 |
Arhem, P; Elinder, F; Ericsson, G; Sandell, L; Westlind-Danielsson, A | 1 |
Ciancone, MT; Haracz, JL; Rebec, GV; White, IM | 1 |
Damsma, G; De Boer, P; Schram, Q; Stoof, JC; Westerink, BH; Zaagsma, J | 1 |
Fujiwara, H | 1 |
Buckland, PR; McGuffin, P; O'Donovan, MC | 2 |
Bambrick, M; Wilson, D | 1 |
Britton, DR; Buckley, M; Curzon, P; Nadzan, A; Tufano, M; Yahiro, L | 1 |
Amenta, F; Cerulli, L; Mancino, R; Ricci, A | 1 |
Gerbrandy-Colijn, A; Ottervanger, JP; Stricker, BH | 1 |
Niu, X; Wang, X | 1 |
Verhoeff, NP | 1 |
Chipkin, RE; Crosby, G; Iorio, LC; Tedford, CE | 1 |
Levant, B; Nemeroff, CB | 1 |
Bissette, G; Levant, B; Nemeroff, CB; Widerlöv, E | 1 |
Miura, O; Suzuki, A; Takase, H; Tatsumi, Y; Yumioka, E | 1 |
Lawrence, MS; Redmond, DE | 1 |
Edinger, H; Siegel, A; Sweidan, S | 1 |
Diana, M; Groves, PM; Young, SJ | 1 |
Watts, D | 1 |
Bogdanov, MB; Guinetdinov, RR; Kudrin, VS; Pogorelov, VM; Rayevsky, KS | 1 |
Abraini, JH; Rostain, JC; Tomei, C | 1 |
Stárková, L; Wiedermann, J | 1 |
Borzecki, Z; Kaliszuk, S; Swies, Z | 1 |
Oblin, A; Zivkovic, B | 1 |
Bourguignon, JJ; Gobaille, S; Hechler, V; Maitre, M; Schmidt, C; Schmitt, M | 1 |
Gonon, F; Ponec, J; Suaud-Chagny, MF | 1 |
Dai, JL; Xu, SF | 1 |
Narkevich, VB; Prikhozhan, AV; Raevskiĭ, KS | 1 |
Li, BH; Li, Q | 1 |
Tepper, JM; Trent, F | 1 |
Enero, MA; Nowicki, S | 1 |
Amano, H; Koizumi, Y; Naruse, T | 1 |
Cabib, S; Castellano, C; Cestari, V; Filibeck, U; Puglisi-Allegra, S | 1 |
Axelrod, J; Briley, EM; Felder, CC; Kanterman, RY; Mahan, LC; Monsma, FJ; Sibley, DR | 1 |
Glowinski, J; Godbout, R; Mantz, J; Pirot, S; Thierry, AM | 1 |
Libertun, C; Lux-Lantos, V; Rey, E; Somoza, G | 1 |
Fink, H; Morgenstern, R; Ott, T; Schremmer, C | 1 |
Dall'Olio, R; Gandolfi, O; Montanaro, N; Roncada, P; Vaccheri, A | 1 |
Bunney, BS; Moghaddam, B | 2 |
Boyer, P; Lecrubier, Y; Puech, AJ | 1 |
Bruno, JP; Hadjiconstantinou, M; Weihmuller, FB | 2 |
Delcker, A; Gaertner, HJ; Oczkowski, B; Schoon, ML | 1 |
Altar, CA; Boyar, WC; Kim, HS | 1 |
Karcz, M; Ossowska, K; Wardas, J; Wolfarth, S | 1 |
Enquist, M; Ljungberg, T | 1 |
Kobayashi, T; Shimizu, H; Toru, M | 1 |
Evans, AM; Green, KL | 2 |
Hama, H; Yamaguchi, K | 1 |
Schneider, T; Zrenner, E | 1 |
Feldon, J; Weiner, I | 1 |
Randall, PK; Yurek, DM | 2 |
Damsma, G; de Boer, P; de Vries, JB; Fibiger, HC; Timmerman, W; Westerink, BH | 1 |
McDougall, SA; Zolman, JF | 1 |
Baamonde, A; Daugé, V; Féger, J; Maldonado, R | 1 |
Hasegawa, Y; Kurachi, M; Otomo, S | 1 |
Daugé, V; Feger, J; Maldonado, R; Roques, BP | 1 |
Butkerait, P; Friedman, E; Wang, HY | 1 |
Argiolas, A; Gessa, GL; Melis, MR; Stancampiano, R | 1 |
Pranzatelli, MR | 1 |
Cooper, SM; McClelland, GR; Pilgrim, AJ | 1 |
Berger, W; Dietz, V; Feuerstein, TJ | 1 |
Bruhwyler, J; Chleide, E; Delarge, J; Liégeois, JF; Mercier, M | 1 |
Kubota, K; Matsumura, M; Sawaguchi, T | 1 |
Arai, I; Higuchi, T; Kazawa, T; Mikuni, M; Takahashi, K; Yamauchi, T | 1 |
Brodin, E; Lindefors, N; Ungerstedt, U | 1 |
Jenner, P; Marsden, CD; Rose, S; Weller, ME | 1 |
Bigornia, L; Napp, D; Ryan, KA; Schneider, AS; Suozzo, M | 1 |
Iwamoto, ET | 1 |
Csernansky, JG; Prosser, ES; Pruthi, R | 1 |
Bush, LG; Gibb, JW; Hanson, GR; Merchant, KM | 1 |
Higashi, H; Inanaga, K; Nishi, S; Uchimura, N | 1 |
Ebadi, M; Govitrapong, P; Hama, Y; Pfeiffer, R | 1 |
Ljungberg, T | 2 |
Bijak, M; Smiałowski, A | 3 |
McKenzie, GM; Warenycia, MW | 1 |
Chivers, JK; Jenner, P; Marsden, CD; Reavill, C | 2 |
Haikala, H | 1 |
Pfaus, JG; Phillips, AG | 1 |
Davis, KL; Guerin, JJ; Halperin, R | 1 |
Barta, L; Masserano, JM | 1 |
Badia, A; Cuffí, ML; Vila, E | 1 |
Argiolas, A; Gessa, GL; Melis, MR | 2 |
Cardinali, DP; Chuluyan, HE; Rosenstein, RE | 1 |
Imazu, Y; Kobayashi, K; Shohmori, T | 1 |
Faltus, F; Jirák, R; Pavlovský, P | 1 |
Buda, M; Gonon, FG; Suaud-Chagny, MF | 1 |
Hietala, J | 1 |
Collu, M; Diena, A; Fanni, B; Glasser, A; Mereu, G | 1 |
Di Chiara, G; Imperato, A | 3 |
Borsini, F; Nowakowska, E; Pulvirenti, L; Samanin, R | 1 |
Compton, DR; Johnson, KM | 1 |
Klassen, NE; Zharkovskiĭ, AM; Zharkovskiĭ, TA | 1 |
Ferrari, F | 1 |
Fleminger, S; Hall, MD; Jenner, P; Kelly, E; Kilpatrick, G; Marsden, CD; Rupniak, NM | 1 |
el Mestikawy, S; Glowinski, J; Hamon, M | 1 |
Andree, TH; Koenig, JI; Meltzer, HY; Mikuni, M; Tong, CY | 1 |
Carruba, MO; Memo, M; Missale, C; Picotti, GB; Pizzi, M; Spano, PF | 1 |
Jauregui, J; Kelley, AE; Nadaud, D; Stinus, L | 1 |
Lazareno, S; Marriott, DB; Nahorski, SR | 1 |
Bowers, MB; Hoffman, FJ | 1 |
Pich, EM; Samanin, R | 1 |
Blanchard, JC; Boireau, A; Carruette, AM; Chambry, J; Dubedat, P; Farges, G; Zundel, JL | 1 |
Ståhle, L; Ungerstedt, U | 1 |
Fujita, M; Horikomi, K | 1 |
Bagetta, G; Corasaniti, MT; Nisticò, G; Sakurada, S; Strongoli, MC | 1 |
Lindefors, N; Tossman, U; Ungerstedt, U | 1 |
Fukuda, T; Matsubara, S; Mikuni, M; Odagaki, Y; Setoguchi, M; Yamashita, I | 1 |
Wambebe, C | 1 |
Bourin, M; Larousse, C; Poisson, L | 1 |
Farde, L; Halldin, C; Sedvall, G; Wiesel, FA | 1 |
Collu, M; Fratta, W; Gessa, GL; Martellotta, MC; Muntoni, F; Pichiri, M | 1 |
Dinan, TG | 1 |
Horn, AS; Radhakishun, FS; Van Ree, JM | 1 |
Amore, M; Campanile, A; Campanile, S; Cerisoli, M | 1 |
Fitten, J; Gordon, LI; Kodama, CK; Menon, MK | 1 |
Kastin, AJ; Pulvirenti, L | 1 |
Aghajanian, GK; Rasmussen, K | 1 |
Biggio, G; Ongini, E; Porceddu, ML | 1 |
Gibbs, J; Schneider, LH; Smith, GP | 1 |
Barrett, RJ; Proakis, AG; Taylor, DR; Wright, KF | 1 |
Caporali, MG; Ongini, E | 1 |
Chiba, S; Furuta, S; Horiuchi, A; Iwatsuki, K; Oguchi, H | 1 |
Fowler, CJ; Magnusson, O; Mohringe, B | 1 |
Caporali, MG; Longo, VG; Ongini, E | 1 |
Cervo, L; Samanin, R | 1 |
Kurumiya, S; Nakajima, S | 1 |
Arbilla, S; Baud, P; Langer, SZ | 1 |
Gaginella, TS; Wahawisan, R; Wallace, LJ | 1 |
Alberch, J; Marsal, J; Solsona, C | 1 |
Glowinski, J; Le Douarin, C; Penit, J; Thierry, AM | 1 |
Fujiwara, M; Nishikawa, H; Yokotani, K | 1 |
Contreras, ML; Contreras, PC; Gehlert, DR; O'Donohue, TL; Quirion, R | 1 |
Benedí, J; Cantón, R; Grande, C; Manzanares, J; Zaragozá, F | 1 |
Ichihara, K; Kameyama, T; Nabeshima, T | 3 |
Burchill, SA; Thody, AJ | 1 |
Bowman, RE; Levin, ED; Vuchetich, J; Wegert, S | 1 |
Jenner, P; Marsden, CD; Rupniak, NM | 1 |
Chen, CC; Chen, IJ; Ko, WK; Yang, MJ | 1 |
Imazu, Y; Kobayashi, K; Shomori, T | 1 |
Anderson, D; Gordon, J; Herbster, G; Koller, W; Wack, R | 1 |
Chase, TN; Tamminga, CA; Tanimoto, K | 1 |
McKenzie, GM; Nakajima, S | 1 |
Biggio, G; Giorgi, O; Mele, S; Ongini, E; Porceddu, ML | 1 |
Carruba, MO; Liberini, P; Memo, M; Missale, C; Spano, P | 1 |
Biziere, K; Gueudet, C; Worms, P | 1 |
Barasi, S; Ben-Sreti, MM; Clatworthy, AL; Duggal, KN; Gonzalez, JP; Robertson, J; Rooney, KF; Sewell, RD | 1 |
Clopton, JK; Curtin, JC; Gordon, JH; Koller, WC | 1 |
Apud, JA; Masotto, C; Monopoli, A; Ongini, E; Racagni, G; Rovescalli, AC | 1 |
Radhakishun, FS; Van Ree, JM | 1 |
Kohjimoto, Y; Kuwaki, T; Nomura, Y; Ono, T; Satoh, H; Shibayama, F; Shirakawa, K | 1 |
Salama, AI; Saller, CF | 1 |
Daw, NW; Jensen, RJ | 2 |
Briggs, RS; Jenner, P; Mann, S; Marsden, CD; Petersen, MM; Reavill, C; Rupniak, NM | 1 |
Boismare, F; Chretien, P; Daoust, M; Moore, N; Saligaut, C | 1 |
D'Angio, M; Scatton, B; Serrano, A | 1 |
Govoni, S; Lucchi, L; Memo, M; Missale, C; Spano, PF; Trabucchi, M | 1 |
Arima, T; Nomura, Y; Samura, N; Segawa, T | 1 |
Jenner, P; Marsden, CD; Simpson, MD | 1 |
Lindefors, N; Sharp, T; Ungerstedt, U | 1 |
Ben Natan, L; Costentin, J; Gonzales-Rios, F; Protais, P; Vlaiculescu, A | 1 |
Hietala, J; MacDonald, E; Scheinin, M | 1 |
Horton, RW; Jenner, P; Marsden, CD; Prestwich, SA; Rupniak, NM | 1 |
Jenks, BG; Tonon, MC; Vaudry, H; Verburg-Van Kemenade, BM | 1 |
Anraku, S; Inanaga, K; Kojima, H; Nishi, S; Takamuki, K; Tsutsumi, T; Yamada, S; Yokoo, H | 1 |
Decker, H; Dimpfel, W | 1 |
Broekkamp, CL; Gower, AJ | 1 |
Powers, CA | 1 |
Biggio, G; Collu, M; Gessa, GL; Mereu, G; Ongini, E | 1 |
Behnke, K; Gerlach, J; Heltberg, J; Munk-Anderson, E; Nielsen, H | 1 |
Bonetti, AC; Canonico, PL; MacLeod, RM | 1 |
Costall, B; Eniojukan, JF; Naylor, RJ | 1 |
Gilbert, JC; Sawas, AH | 1 |
Ortmann, R | 1 |
Collu, M; Gessa, GL; Serra, G | 1 |
Borsini, F; Pulvirenti, L; Samanin, R | 1 |
Aleksić, J; Geber, J; Gjuris, V; Ivanović, D; Marović, A; Reić, P; Sikirić, P; Suchanek, E | 1 |
Buda, M; Gonon, F; le Moal, M; Louilot, A; Pujol, JF; Simon, H | 1 |
Drago, F; Scapagnini, U | 1 |
Horikawa, H; Konagaya, M; Mano, Y; Takayanagi, T | 1 |
Clemens, JA; Sawyer, BD; Smalstig, EB | 1 |
Sharp, T; Ungerstedt, U; Zetterström, T | 1 |
Guidotti, A | 1 |
Bronzetti, B; Ciriaco, E; Germanà, G; Nisticò, G | 1 |
Gômez, F; Lechin, E; Lechin, F; van der Dijs, B | 1 |
Maeno, H; Nishikori, K; Noshiro, O; Usuda, S | 1 |
Dyer, R; Hall, MD; Jenner, P; Leigh, N; Marsden, CD; Rupniak, NM | 1 |
Tissari, AH | 1 |
Dall'Olio, R; Gandolfi, O; Montanaro, N; Vaccheri, A | 3 |
Castelli, M; Genedani, S | 1 |
Duval, N; Langer, SZ; Massingham, R; Shepperson, NB | 1 |
Bracha, HS; Davis, KL; Kendler, KS | 1 |
Barrett, RJ; Ginos, JZ; Lokhandwala, MF | 1 |
Azuma, H; Iwai, K; Kikuta, M; Liu, HJ; Oshino, N; Sato, K | 1 |
De Gori, N; De Sarro, A; Nistico', G; Pujia, A; Urna, G | 1 |
Casu, M; Gessa, GL; Mereu, G | 1 |
Etienne, P; Lal, S; Nair, NP; Wood, PL | 1 |
Fleminger, S; Hall, MD; Jenner, P; Kerwin, R; Marsden, CD; Murugaiah, K; Rupniak, NM | 1 |
Fleminger, S; Hall, MD; Jenner, P; Marsden, CD; Rupniak, NM | 1 |
Pi, EH; Simpson, GM | 1 |
Borsini, F; Nowakowska, E; Samanin, R | 1 |
Jenner, P; Kerwin, RW; Marsden, CD; Rupniak, NM | 1 |
Guldvog, I; Linnestad, P; Schrumpf, E | 1 |
Planche, R | 1 |
Pinnock, RD | 1 |
Steranka, LR | 1 |
Costall, B; Domeney, AM; Naylor, RJ | 2 |
Dall'Olio, R; Gaggi, R; Gandolfi, O; Montanaro, N; Vaccheri, A | 1 |
Appel, JB; Callahan, PM; Cunningham, KA | 1 |
Angeby, K; Florvall, L; Hall, H; Köhler, C; Lindbom, LO; Magnusson, O; Ogren, SO | 1 |
Zharkovskaia, TA; Zharkovskiĭ, AM | 1 |
Davis, KL; Kendler, KS | 1 |
Agid, Y; Bokobza, B; Javoy-Agid, F; Montfort, JC; Ruberg, M | 1 |
Király, I; Van Ree, JM | 1 |
Albizzati, MG; Alemani, A; Bassi, S; Ferrarese, C; Frattola, L; Trabucchi, M | 1 |
Lee, T; Tang, SW | 1 |
Berzétei, IP; Csaba, G; Dobozy, O; Kurgyis, J; Rónai, AZ | 1 |
Cole, AE; Shinnick-Gallagher, P | 1 |
Arbilla, S; Kamal, LA; Langer, SZ | 1 |
Cubeddu, LX; Hoffmann, IS | 2 |
Anguera, P; Bulteau, J; Soubrier, JP | 1 |
Fujisawa, K | 1 |
Covelli, V; Lucchi, L; Petkov, VV; Spano, PF; Trabucchi, M | 1 |
Barger, AC; Dzau, VJ; Mizoguchi, H; Siwek, LG | 1 |
Behnke, K; Gerlach, J; Heltberg, J; Munk-Andersen, E; Nielsen, H | 1 |
Baggio, G; Ferrari, F | 2 |
Fleminger, S; Hall, MD; Jenner, P; Kilpatrick, G; Mann, S; Marsden, CD; Rupniak, NM | 1 |
Hall, MD; Jenner, P; Kilpatrick, G; Marsden, CD; Rupniak, NM | 1 |
Gold, R; Lemme, P; Mende, T; Morgenstern, R; Oelssner, W | 1 |
Bousquet, E; De Simone, D; Grasso, AA; Millia, CC; Rampello, L; Rapisarda, E; Reggio, A | 1 |
Condorelli, DF; Costa, G; Grasso, AA; Millia, C; Nicoletti, F; Patti, F; Rampello, L; Rapisarda, E; Scapagnini, U | 1 |
Fink, H; Morgenstern, R; Oelssner, W | 1 |
Durkin, TP; Ebel, A; Hashem-Zadeh, H; Kempf, J; Mandel, P | 1 |
Hanbauer, I; Memo, M | 1 |
Angeby, K; Ogren, SO; Rodebjer, A | 1 |
Angrist, BM | 1 |
Cianchetti, C; Gessa, GL; Mangoni, A; Masala, C | 1 |
Bailey, J; Bishop, M; Coppen, A; Rao, VA | 1 |
Argiolas, A; Fadda, F; Gessa, GL; Melis, MR; Serra, G | 1 |
Canonico, PL; Clementi, G; Di Giorgio, RM; Nicoletti, F; Patti, F; Prato, A; Rampello, L; Scapagnini, U | 1 |
Atzori, L; Galdieri, MT; Tissari, AH | 1 |
Akaike, A; Sasa, M; Takaori, S | 1 |
Arbilla, S; Galzin, AM; Langer, SZ; Nowak, JZ | 1 |
Agnati, LF; Andersson, K; Fuxe, K; Hall, H; Köhler, C; Ogren, SO; Schwarcz, R | 1 |
Canonico, PL; Condorelli, DF; Nicoletti, F; Patti, F; Scapagnini, U | 1 |
Azuma, H; Ishikawa, T; Miyazawa, T; Oshino, N | 1 |
Hall, MD; Jenner, P; Marsden, CD; Murugaiah, K; Rupniak, N; Theodorou, A | 1 |
Barbaccia, ML; Bosio, A; Lucchi, L; Spano, PF; Trabucchi, M | 1 |
Canonico, PL; Clementi, G; Condorelli, DF; di Giorgio, RM; Drago, F; Nicoletti, F; Patti, F; Prato, A | 1 |
Airaghi, ML; Lucchi, L; Memo, M; Spano, PF; Trabucchi, M | 1 |
Anraku, S; Inanaga, K; Kojima, H; Suetake, K; Yokoo, H; Yoshida, M | 1 |
Battistin, L; Gabana, MA; Saladini, M; Varotto, M; Zanchin, G | 1 |
Fink, H; Morgenstern, R | 1 |
Bannet, J; Belmaker, RH; Ebstein, RP; Gillis, S | 1 |
Aubineau, P; Boulu, RG; Oudart, N; Sercombe, R; Seylaz, J | 1 |
Condorelli, DF; Di Giorgio, RM; Giammona, G; Nicoletti, F; Patti, F; Rampello, L; Reggio, A | 1 |
Battaini, F; Memo, M; Spano, PF; Trabucchi, M | 1 |
Canonico, PL; Condorelli, DF; Di Giorgio, RM; Giammona, G; Nicoletti, F; Patti, F; Rampello, L; Scapagnini, U | 1 |
Condorelli, DF; Di Giorgio, RM; Giammona, G; Matera, M; Nicoletti, F; Patti, F; Rampello, L; Reggio, A | 1 |
Battaini, F; Memo, M; Reggiani, A; Spano, PF; Trabucchi, M | 1 |
Agnati, LF; Andersson, K; Benfenati, F; Cortelli, P; D'Alessandro, R; Fuxe, K; Ogren, SO | 1 |
Fujita, N; Hirata, A; Iwatsubo, K; Noguchi, Y; Saito, K; Yoshida, H | 1 |
Barbieri, C; Caldara, R; Ferrari, C; Romussi, M | 1 |
Lucchi, L; Memo, M; Spano, PF; Trabucchi, M | 1 |
Deutch, AY; Duman, RS; Ongür, D | 1 |
Deinum, ME; Schuiling, GA; Timmerman, W; Westerink, BH | 1 |
Bloch, B; Fournier, MC; Jaber, M; Tison, F | 1 |
Perrault, G; Sanger, DJ | 1 |
Middlemiss, DN; Reavill, C; Storey, VJ | 1 |
Kishioka, S; Masuda, Y; Miyamoto, Y; Ozaki, M; Yamamoto, H | 1 |
Kassir, S; Parsons, B; Przedborski, S; Togasaki, DM | 1 |
Takaki, T; Tanaka, M; Yamada, S; Yokoo, H | 1 |
Smiałowska, M | 1 |
Chien, CC; Pasternak, GW | 2 |
Andersson, I; Gustafsson, K; Westlind-Danielsson, A | 1 |
Elands, J; Gobaille, S; Grauffel, C; Knödgen, B; Moran, P; Sarhan, S; Seiler, N; van den Buuse, M | 1 |
de Koning, P; de Vries, MH | 1 |
Grafton, TF; Hansen, DK; Holson, RR; Webb, PJ | 1 |
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Kulkarni, SK; Sharma, A | 2 |
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Ahlenius, S; Ericson, E; Wijkström, A | 1 |
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Strange, PG | 1 |
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Hanaoka, Y; Matsukura, S; Ohi, T | 1 |
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Wang, HH; Xu, SF | 1 |
Juhnn, YS; Kim, YS; Park, JB; Shin, CJ | 1 |
Batrak, GN; Degtiar, VY; Hawryluk, BR; Luik, AI; Mogilevich, SE; Naydyenova, IY; Prokopenko, RA | 1 |
Barbosa-Coutinho, LM; Barros, HM; Moraes, JT; Oliveira, MC | 1 |
Cabib, S; Caccia, S; Castellano, C; Felici, A; Mele, A; Oliverio, A | 1 |
Bargas, J; Galarraga, E; Hernández-López, S; Pacheco-Cano, MT; Tapia, D | 1 |
Drago, F; Le Pira, F; Malaguarnera, M; Nicoletti, G; Raffaele, R; Rampello, L | 1 |
Alzheimer, C; Chesi, AJ; Feasey-Truger, KJ; ten Bruggencate, G | 1 |
Ito, C; Onodera, K; Sakurai, E; Sato, M; Watanabe, T | 1 |
Gerlach, J; Peacock, L | 1 |
Amenta, F; Barili, P; Zaccheo, D | 1 |
Obuchowicz, E | 2 |
Barik, S; de Beaurepaire, R | 2 |
Fukamauchi, F; Kito, S; Mataga, N; Miyoshi, R; Sakai, M; Semba, J | 1 |
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Asaba, H; Inayama, Y; Matsumura, H; Sakai, J; Sakai, T; Takahata, R; Toyoda, H; Yoneda, H | 1 |
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Katsumoto, E; Ozaki, T; Yamagami, S; Yokotani, N | 1 |
Freeman, HL | 1 |
Danion, JM; Grangé, D; Kauffmann-Muller, F; Patat, A; Peretti, CS; Rosenzweig, P | 1 |
Fang, H; Helmeste, DM; Li, M; Tang, SW | 1 |
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Adams, MR; Brandon, EP; Chartoff, EH; Dorsa, DM; Idzerda, RL; McKnight, GS | 1 |
Drucker-Colín, R; Lara-Lemus, A; Méndez-Franco, J; Palomero-Rivero, M; Pérez de la Mora, M | 1 |
Buckland, PR; D'Souza, U; Maher, NA; McGuffin, P | 1 |
George, B; Kulkarni, SK | 1 |
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Furutsuka, D; Katsumoto, E; Mui, K; Ozaki, T; Yamagami, S | 1 |
Gobaille, S; Hodé, Y; Kemmel, V; Maitre, M; Ratomponirina, C | 1 |
Belowski, D; Herman, ZS; Kowalski, J; Madej, A | 1 |
Fleurot, O; Puech, A; Rein, W | 1 |
Kulkarni, SK; Ninan, I | 1 |
Gioanni, Y; Glowinski, J; Tassin, JP; Thierry, AM | 1 |
Obuchowicz, E; Turchan, J | 2 |
Hayashi, T; Kagaya, A; Nishida, A; Shimizu, M; Su, TP; Yamawaki, S | 1 |
Chowdhury, SA; Huda, K; Kawashima, T; Matsunami, K; Salunga, TL | 1 |
de Groat, WC; Namiki, M; Yokoyama, O; Yoshiyama, M | 1 |
Mui, K; Ozaki, T; Yamagami, S | 1 |
Aguilar, MA; Manzanedo, C; Miñarro, J | 1 |
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de Bie, A; Louwerens, JW; Milius, H; Muntjewerff, ND; O'Hanlon, JF; Patat, A; Ramaekers, JG; Rosenzweig, P | 1 |
Kachalova, LM; Popova, NS | 1 |
Liu, ZH; Zhang, KG | 1 |
Horikomi, K; Iizuka, K; Mita, N; Miwa, T; Nagase, H; Sakai, K; Sonehara, K; Takagi, K; Takahashi, S | 1 |
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Cryan, JF; Harkin, A; Kelly, JP; Leonard, BE; Naughton, M | 1 |
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Aguilar, MA; Arenas, MC; Miñarro, J; Parra, A; Simón, VM; Vinader-Caerols, C | 1 |
Möller, HJ | 2 |
Coulouvrat, C; Dondey-Nouvel, L; Rein, W | 1 |
Colonna, L; Dondey-Nouvel, L; Rein, W; Saleem, P | 1 |
Fushiki, T; Imaizumi, M; Takeda, M | 1 |
Liu, W; Wu, CF; Zhang, HL | 1 |
Bergougnan, L; Canal, M; L'Heritier, C; Legangneux, E; McEwen, J; Miget, N; Pinquier, JL; Rosenzweig, P; Wesnes, KA | 1 |
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Hillefors, M; von Euler, G | 1 |
Goto, K; Nakamura, T; Nambu, T; Sakurai, T; Uramura, K; Yada, T; Yanagisawa, M | 1 |
Ozaki, T | 1 |
Kusayama, T; Watanabe, S | 1 |
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De Boer, P; De Vries, JB; Geels, C; Kawahara, Y; Kruse, CG; Long, SK; Van Kalkeren, A; Van Vliet, B; Westerink, BH; Wikström, HV | 1 |
Gálfi, M; Janáky, T; Juhász, A; László, FA; Prohászka, G; Tóth, R; Varga, C | 1 |
Hilger, E; Kasper, S | 1 |
Azorin, JM | 1 |
Fukamauchi, F; Ikawa, K; Kaneno, S; Komatsu, H; Koyama, K | 1 |
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Fu, D; Javitch, JA; Lin, H; Strange, PG; Wilson, J | 1 |
Basso, AM; Cancela, LM; Capriles, NR; Martijena, ID; Molina, VA | 1 |
Reuss, B; Unsicker, K | 1 |
Bridges, S; Miller, C; Thompson, TL | 1 |
Hatzimanolis, J; Lykouras, L; Markianos, M | 1 |
Alexandre, L; Allard, J; Benoit, G; Bernabé, J; Droupy, S; Giuliano, F; Rampin, O | 1 |
Dai, J; Fowler, WL; Ichikawa, J; Meltzer, HY; O'Laughlin, IA | 1 |
Bartholini, F; Casu, MA; Gessa, GL; Marchese, G; Pani, L; Ruiu, S; Saba, P | 1 |
Haasen, C; Krausz, M; Naber, D; Nika, E; Yagdiran, O | 1 |
Araujo, AP; Maia Filho, HS; Padua, PA | 1 |
Möller, HJ; Peuskens, J; Puech, A | 1 |
Conn, PJ; Marino, MJ; Wittmann, M | 1 |
Horikomi, K; Karasawa, J; Takagi, K; Takahashi, S | 1 |
Ohye, C; Shibazaki, T | 1 |
Chen, CC; Chen, KP; Chuang, CL; Shen, WW; Su, KP | 1 |
Basta-Kaim, A; Budziszewska, B; Jaworska-Feil, L; Kubera, M; Lasoń, W; Leśkiewicz, M; Tetich, M | 1 |
Benkert, O; Eich, FX; Müller, MJ; Puech, A; Rein, W; Wetzel, H | 1 |
Goudie, AJ; Smith, JA | 1 |
Biala, G; Duarte, C; Hamon, M; Le Bihan, C; Thiébot, MH | 1 |
Sugiyama, A | 1 |
Correll, CU; Kane, JM; Leucht, S | 1 |
Grigor'eva, EA; Ritskov, AS | 1 |
Ago, Y; Baba, A; Matsuda, T; Nakamura, S | 1 |
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Amann, B; Hegerl, U; Juckel, G; Möller, HJ; Mulert, C; Pogarell, O | 1 |
Lawrie, S; McIntosh, A; Nadeem, Z | 2 |
Gratton, A; Laplante, F; Quirion, R; Srivastava, LK; Stevenson, CW | 1 |
Barna, I; Gazdag, G; Iványi, Z; Tolna, J | 1 |
Axelrod, JD; Barghshoon, S; Chen, CK; Cheyette, BN; Ebert, J; Kovoor, A; Lester, HA; Schwarz, J; Schwarz, S; Seyffarth, P; Simon, MI | 1 |
Lawrie, S; McIntosh, A | 1 |
Taylor, GT; Yuede, CM | 1 |
Knecht, G; Naber, D; Veismann, S; Wolf, K | 1 |
Cummins, R; Gnoffo, Z; Kew, JN; Roberts, C | 1 |
Deshpande, C; Dhir, A; Kulkarni, SK | 1 |
Bastianetto, S; Danik, M; Mennicken, F; Quirion, R; Williams, S | 1 |
Cipriani, A; Geddes, JR; Rendell, JM | 1 |
Ohmori, T; Yamauchi, K | 1 |
Bäuml, J; Davis, JM; Engel, RR; Leucht, S | 1 |
Afsar, N; Dib, H; Günal, DI; Köseoglu, M; Midi, I | 1 |
Limosin, F | 1 |
Bezzina, G; Body, S; Bradshaw, CM; Cheung, TH; Fone, KC; Hampson, CL; Szabadi, E | 1 |
Boter, H; Davidson, M; Dollfus, S; Fleischhacker, WW; Gaebel, W; Galderisi, S; Gheorghe, MD; Grobbee, DE; Hranov, LG; Hummer, M; Kahn, RS; Keet, IP; Libiger, J; Lindefors, N; López-Ibor, JJ; Peuskens, J; Riecher-Rössler, A; Rybakowski, JK; Vergouwe, Y | 1 |
de Moura Linck, V; Elisabetsky, E; Goerck, GC; Herrmann, AP; Iwu, MM; Leal, MB; Okunji, CO | 1 |
Agai-Csongor, E; Bugovics, G; Domány, G; Fazekas, K; Gyertyán, I; Horváth, A; Kiss, B; Laszlovszky, I; Némethy, Z; Schmidt, E; Szombathelyi, Z | 1 |
Barlow, KB; Kapur, S; Natesan, S; Nobrega, JN; Reckless, GE | 1 |
Costa, E; Dong, E; Grayson, DR; Guidotti, A; Nelson, M | 1 |
Endo, S; Hamamura, T; Ishihara, T; Kuroda, S; Miyata, S; Taoka, H; Toma, K | 1 |
Dhir, A; Kulkarni, SK | 1 |
Bogo, MR; Bonan, CD; Dias, RD; Oliveira, Rda L; Rico, EP; Seibt, KJ | 1 |
Dietrich-Muszalska, A; Olas, B | 1 |
Ayesa, R; Crespo-Facorro, B; Martínez-Garcia, O; Mata, I; Pérez-Iglesias, R; Ramirez-Bonilla, M; Rodríguez-Sánchez, JM; Vázquez-Barquero, JL | 1 |
Goldberg, TE; Gomar, JJ | 1 |
Burns, T; Derks, EM; Fleischhacker, WW; Gaebel, W; Kahn, RS; Riesbeck, M; Rössler, W; von Wilmsdorff, M | 1 |
Kastania, A; Katsafouros, K; Laskos, E; Lykouras, L; Michalopoulou, PG; Papadopoulou, A; Rizos, EN; Vasilopoulos, D | 1 |
Cicale, M; de Bartolomeis, A; Fiore, G; Iasevoli, F; Muscettola, G | 1 |
Arakawa, R; Ito, H; Maeda, J; Okubo, Y; Okumura, M; Suhara, T; Takahashi, H; Takano, A; Takano, H | 1 |
Binfaré, RW; Budni, J; Mantovani, M; Rodrigues, AL; Santos, AR | 1 |
Araki, H; Hidaka, N; Suemaru, K | 1 |
Dietrich-Muszalska, A; Kontek, B; Olas, B; Rabe-Jabłońska, J | 1 |
Cho, HY; Kim, YH; Lee, BJ; Lee, JG; Park, SW; Seo, MK; Seol, W | 1 |
Bitter, I; Czobor, P; Derks, EM; Fleischhacker, WW; Kahn, RS; Libiger, J; Volavka, J | 1 |
Body, S; Bradshaw, CM; de Bruin, N; den Boon, FS; Hampson, CL; Szabadi, E | 1 |
Bonan, CD; Piato, AL; Savio, LE; Vuaden, FC; Wyse, AT | 1 |
Bonan, CD; da Luz Oliveira, R; Rosemberg, DB; Savio, LE; Scherer, EB; Schmitz, F; Seibt, KJ; Wyse, AT | 1 |
Dudova, I; Hrdlicka, M; Urbanek, T; Zedkova, I | 1 |
Czernikiewicz, A; Kucharska-Pietura, K; Mortimer, A; Tylec, A | 1 |
Chung, YC; Huang, GB; Lee, KH; Park, CH; Park, MS; Park, TW; Tong, Z; Yang, JC | 1 |
Chang, CH; Kao Yang, YH; Lai, EC; Lin, CY; Lin, SJ | 1 |
Bitter, I; Bucci, P; Fleischhacker, WW; Galderisi, S; Kahn, RS; Libiger, J; Mucci, A | 1 |
Kirchhoff, BA; Smith, SE; Taylor, GT | 1 |
Feng, Z; Hou, T; Li, Y | 1 |
Chung, YC; Han, EH; Huang, GB; Kang, NI; Li, CR; Sui, ZY; Zhao, T | 1 |
Chung, YC; Huang, GB; Kim, MG; Oh, KY; Park, TW; Yang, JC; Zhao, T | 1 |
Buonaguro, EF; de Bartolomeis, A; Iasevoli, F; Marmo, F; Rossi, R; Tomasetti, C | 1 |
Cheung, C; Chua, SE; Collier, DA; Deng, W; Gong, Q; Huang, C; Jiang, L; Li, M; Li, T; Ma, X; McAlonan, GM; Sham, PC; Wang, Q; Wang, Y | 1 |
Arvanitakis, P; Dimopoulou, K; Kalkavoura, CS; Lykouras, L; Michopoulos, I; Theodoropoulou, P; Tzebelikos, E | 1 |
Bogo, MR; Bonan, CD; Kist, LW; Pereira, TC; Rosemberg, DB; Savio, LE; Vuaden, FC; Wyse, AT | 1 |
Deslauriers, J; Desmarais, C; Grignon, S; Sarret, P | 1 |
Citrome, L; Czobor, P; Van Dorn, RA; Volavka, J | 1 |
Blanchet, PJ; Lévesque, D; Mahmoudi, S | 1 |
Bestmann, S; Galea, JM; Rothwell, J; Ruge, D | 1 |
Domínguez, R; Handal, A; Juárez, CE; Morán, C; Morán, JL; Padilla, JF; Rosas-Murrieta, NH; Venegas-Meneses, B | 1 |
Bogo, MR; Bonan, CD; Oliveira, Rda L; Seibt, KJ; Senger, MR | 1 |
Gao, N; Huang, JZ; Li, KQ; Liang, Y; Si, TM; Su, YA; Tang, MQ; Yang, FD; Yu, X; Zhao, ZG | 1 |
Bestmann, S; Galea, JM; Penny, W; Ruge, D; Tomassini, A | 1 |
Ananthan, S; Głowacka, U; Kosmowska, B; Ossowska, K; Wardas, J | 1 |
Antczak, A; Górski, P; Karbownik, MS; Kowalczyk, E; Pietras, T; Szemraj, J; Wieteska, Ł | 1 |
Buonaguro, EF; de Bartolomeis, A; Iasevoli, F; Latte, G; Marmo, F; Tomasetti, C | 1 |
Chan, HY; Chen, CH; Chen, JJ; Pan, YJ | 1 |
Barber, S; Cipriani, A; Corsi, M; Olotu, U | 1 |
Espinosa-Juárez, JV; Jaramillo-Morales, OA; López-Muñoz, FJ | 1 |
Jasińska-Stroschein, M; Jóźwiak-Bębenista, M; Kowalczyk, E | 1 |
Aguirre, C; Erezuma, I; Garcia, M; Hernandez, R; Lertxundi, U; Medrano, J | 1 |
Abbasi-Maleki, S; Mesbahzadeh, B; Moradi-Kor, N | 1 |
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Guo, Y; Li, T; Peng, X; Sun, X; Zhang, B | 1 |
21 review(s) available for sulpiride and haloperidol
Article | Year |
---|---|
Atypical neuroleptics: clozapine and the benzamides in the prevention and treatment of tardive dyskinesia.
Topics: Antipsychotic Agents; Benzamides; Clinical Trials as Topic; Clozapine; Dibenzazepines; Dose-Response Relationship, Drug; Dyskinesia, Drug-Induced; Haloperidol; Humans; Metoclopramide; Prospective Studies; Schizophrenia; Sulpiride; Tiapamil Hydrochloride | 1983 |
Intestinal pharmacomanometry and glucose tolerance: two kinds of dopaminergic mechanisms in the human.
Topics: Animals; Brain Chemistry; Colon; Dextroamphetamine; Dogs; Dopamine Antagonists; Drug Interactions; Gastrointestinal Motility; Glucose Tolerance Test; Haloperidol; Humans; Insulin; Receptors, Dopamine; Serotonin; Sulpiride | 1981 |
Dopamine receptors in the basal ganglia: relevance to Parkinson's disease.
Topics: Basal Ganglia; Basal Ganglia Diseases; Brain; Clozapine; Dopamine Agents; Dopamine D2 Receptor Antagonists; Female; Haloperidol; Humans; Levodopa; Male; Neostriatum; Neural Pathways; Parkinson Disease; Receptors, Dopamine D1; Receptors, Dopamine D2; Sulpiride | 1993 |
[Ballism, hemiballism].
Topics: Cerebrovascular Disorders; Chlorpromazine; Electromyography; Haloperidol; Humans; Movement Disorders; Sulpiride | 1993 |
New antipsychotics: the present status.
Topics: Antipsychotic Agents; Binding, Competitive; Clozapine; Dopamine Antagonists; Haloperidol; Humans; Psychotic Disorders; Sulpiride | 1995 |
Amisulpride compared with standard neuroleptics in acute exacerbations of schizophrenia: three efficacy studies.
Topics: Adult; Amisulpride; Antipsychotic Agents; Chronic Disease; Dose-Response Relationship, Drug; Double-Blind Method; Dyskinesia, Drug-Induced; Female; Flupenthixol; Haloperidol; Humans; Male; Middle Aged; Multicenter Studies as Topic; Neurologic Examination; Psychiatric Status Rating Scales; Randomized Controlled Trials as Topic; Sulpiride; Treatment Outcome | 1997 |
Amisulpride: a review of its efficacy in schizophrenia.
Topics: Acute Disease; Amisulpride; Antipsychotic Agents; Brief Psychiatric Rating Scale; Chronic Disease; Clinical Trials as Topic; Flupenthixol; Haloperidol; Humans; Risperidone; Schizophrenia; Sulpiride; Treatment Outcome | 2000 |
Safety profile of amisulpride in short- and long-term use.
Topics: Amisulpride; Antipsychotic Agents; Chronic Disease; Clinical Trials as Topic; Drug Administration Schedule; Female; Haloperidol; Humans; Male; Risperidone; Schizophrenia; Sulpiride; Treatment Outcome | 2000 |
Atypical antipsychotics: new directions and new challenges in the treatment of schizophrenia.
Topics: Amisulpride; Antipsychotic Agents; Benzodiazepines; Clozapine; Dibenzothiazepines; Dibenzothiepins; Dopamine Antagonists; Drug Monitoring; Haloperidol; Humans; Imidazoles; Indoles; Olanzapine; Piperazines; Pirenzepine; Quetiapine Fumarate; Receptors, Dopamine D2; Receptors, Dopamine D4; Risperidone; Schizophrenia; Schizophrenic Psychology; Serotonin Antagonists; Sulpiride; Thiazoles; Treatment Outcome | 2001 |
[Atypical neuroleptics: new approaches to drug therapy of schizophrenic disorders].
Topics: Aged; Amisulpride; Antipsychotic Agents; Benzodiazepines; Clozapine; Controlled Clinical Trials as Topic; Dibenzothiazepines; Dibenzothiepins; Haloperidol; Humans; Imidazoles; Indoles; Multicenter Studies as Topic; Olanzapine; Piperazines; Pirenzepine; Placebos; Quetiapine Fumarate; Risperidone; Schizophrenia; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Sulpiride; Thiazoles | 2000 |
[Effects of clinically available drugs on the repolarization process of the heart assessed by the in vivo canine models].
Topics: Action Potentials; Animals; Anti-Arrhythmia Agents; Antipsychotic Agents; Antitubercular Agents; Cation Transport Proteins; Cisapride; Disease Models, Animal; Dogs; Ether-A-Go-Go Potassium Channels; Fluoroquinolones; Gastrointestinal Agents; Haloperidol; Histamine H1 Antagonists; Long QT Syndrome; Potassium Channels; Potassium Channels, Voltage-Gated; Sulpiride; Terfenadine; Torsades de Pointes | 2003 |
Lower risk for tardive dyskinesia associated with second-generation antipsychotics: a systematic review of 1-year studies.
Topics: Adolescent; Adult; Aged; Amisulpride; Antipsychotic Agents; Benzodiazepines; Child; Dibenzothiazepines; Double-Blind Method; Dyskinesia, Drug-Induced; Haloperidol; Humans; Middle Aged; Neurologic Examination; Olanzapine; Piperazines; Quetiapine Fumarate; Randomized Controlled Trials as Topic; Risk; Sulpiride; Thiazoles | 2004 |
[The features of atypical neuroleptic amisulpride action].
Topics: Adolescent; Adult; Age Factors; Aged; Aged, 80 and over; Amisulpride; Antipsychotic Agents; Clinical Trials as Topic; Drug Interactions; Drug Therapy, Combination; Electrocardiography; Female; Haloperidol; Humans; Male; Middle Aged; Multicenter Studies as Topic; Risperidone; Schizophrenia; Sulpiride | 2004 |
[Psychotropics and weight gain].
Topics: Adolescent; Adult; Amisulpride; Antidepressive Agents; Antimanic Agents; Antipsychotic Agents; Aripiprazole; Benzodiazepines; Body Mass Index; Child; Clozapine; Dibenzothiazepines; Double-Blind Method; Female; Fructose; Haloperidol; Humans; Imidazoles; Indoles; Male; Obesity; Olanzapine; Piperazines; Placebos; Psychotropic Drugs; Quetiapine Fumarate; Quinolones; Randomized Controlled Trials as Topic; Risperidone; Socioeconomic Factors; Sulpiride; Thiazoles; Time Factors; Topiramate; Valproic Acid; Weight Gain | 2004 |
Schizophrenia.
Topics: Amisulpride; Antipsychotic Agents; Benzodiazepines; Chlorpromazine; Clozapine; Cognitive Behavioral Therapy; Dibenzothiepins; Haloperidol; Humans; Olanzapine; Patient Compliance; Perazine; Pimozide; Risperidone; Schizophrenia; Sulpiride | 2003 |
Schizophrenia.
Topics: Amisulpride; Antipsychotic Agents; Benzodiazepines; Chlorpromazine; Clozapine; Haloperidol; Humans; Olanzapine; Patient Compliance; Perazine; Pimozide; Risperidone; Schizophrenia; Sulpiride | 2004 |
Schizophrenia.
Topics: Amisulpride; Antipsychotic Agents; Chlorpromazine; Clozapine; Cognitive Behavioral Therapy; Dibenzothiepins; Family Therapy; Haloperidol; Humans; Patient Compliance; Risperidone; Schizophrenia; Secondary Prevention; Sulpiride; Thioridazine | 2005 |
Haloperidol alone or in combination for acute mania.
Topics: Amisulpride; Antipsychotic Agents; Aripiprazole; Benzodiazepines; Bipolar Disorder; Carbamazepine; Dibenzothiazepines; Drug Therapy, Combination; Haloperidol; Humans; Olanzapine; Piperazines; Quetiapine Fumarate; Quinolones; Randomized Controlled Trials as Topic; Risperidone; Sulpiride; Valproic Acid | 2006 |
[Two cases of tardive Tourette syndrome].
Topics: Adult; Akathisia, Drug-Induced; Alcoholism; Amantadine; Antipsychotic Agents; Cholinergic Antagonists; Dopamine Agents; Dopamine Antagonists; Haloperidol; Humans; Male; Middle Aged; Schizophrenia; Sulpiride; Tourette Syndrome | 2006 |
[The use of atypical antipsychotics in the long-term care of schizophrenia].
Topics: Amisulpride; Antipsychotic Agents; Aripiprazole; Basal Ganglia Diseases; Benzodiazepines; Clozapine; Cognition Disorders; Drug Tolerance; Dyskinesia, Drug-Induced; Haloperidol; Humans; Olanzapine; Piperazines; Quinolones; Risperidone; Schizophrenia; Sulpiride; Time Factors | 2006 |
Clozapine combined with different antipsychotic drugs for treatment-resistant schizophrenia.
Topics: Adult; Amisulpride; Antipsychotic Agents; Aripiprazole; Clozapine; Dibenzothiazepines; Drug Resistance; Drug Therapy, Combination; Female; Haloperidol; Humans; Male; Piperazines; Quetiapine Fumarate; Randomized Controlled Trials as Topic; Risperidone; Schizophrenia; Sulpiride; Thiazoles; Weight Gain | 2017 |
40 trial(s) available for sulpiride and haloperidol
Article | Year |
---|---|
Sulpiride--an antipsychotic agent: comparative trial vs. haloperidol.
Topics: Adult; Antipsychotic Agents; Clinical Trials as Topic; Double-Blind Method; Drug Evaluation; Female; Haloperidol; Humans; Male; Psychiatric Status Rating Scales; Schizophrenia; Sulpiride | 1977 |
Apomorphine hydrochloride-induced improvement in Huntington's chorea: stimulation of dopamine receptor.
Topics: Adult; Apomorphine; Clinical Trials as Topic; Dose-Response Relationship, Drug; Double-Blind Method; Female; Haloperidol; Humans; Huntington Disease; Male; Middle Aged; Premedication; Receptors, Dopamine; Sulpiride | 1978 |
Sulpiride versus haloperidol in schizophrenia: a double-blind comparative trial.
Topics: Adult; Aged; Analysis of Variance; Brief Psychiatric Rating Scale; Clinical Trials as Topic; Computers; Female; Haloperidol; Humans; Male; Middle Aged; Placebos; Psychiatric Status Rating Scales; Schizophrenia, Disorganized; Schizophrenia, Paranoid; Sulpiride | 1975 |
An automated diagnostic process (PDA) in clinical psychopharmacology. An exemplification of its use in a sulpiride versus haloperidol comparative trial.
Topics: Adult; Aged; Clinical Trials as Topic; Diagnosis, Computer-Assisted; Female; Haloperidol; Humans; Male; Mental Disorders; Middle Aged; Psychiatric Status Rating Scales; Sulpiride | 1976 |
[Trial of interruption of antiparkinson drugs in long term treatments with neuroleptics].
Topics: Adult; Antiparkinson Agents; Basal Ganglia Diseases; Chlorpromazine; Clinical Trials as Topic; Fluphenazine; Haloperidol; Humans; Long-Term Care; Male; Placebos; Psychotic Disorders; Recurrence; Substance Withdrawal Syndrome; Sulpiride; Tranquilizing Agents | 1975 |
Treatment of positive and negative symptoms: pharmacologic approaches.
Topics: Adult; Amisulpride; Antipsychotic Agents; Clinical Trials as Topic; Dose-Response Relationship, Drug; Double-Blind Method; Dyskinesia, Drug-Induced; Female; Fluphenazine; Haloperidol; Humans; Male; Middle Aged; Psychiatric Status Rating Scales; Schizophrenia; Schizophrenic Psychology; Sulpiride | 1990 |
Amisulpride versus haloperidol in treatment of schizophrenic patients--results of a double-blind study.
Topics: Adult; Amisulpride; Antipsychotic Agents; Basal Ganglia Diseases; Double-Blind Method; Female; Haloperidol; Hemodynamics; Humans; Male; Psychiatric Status Rating Scales; Randomized Controlled Trials as Topic; Schizophrenia; Schizophrenic Psychology; Sulpiride | 1990 |
A comparison of the central nervous system effects of haloperidol, chlorpromazine and sulpiride in normal volunteers.
Topics: Adult; Chlorpromazine; Double-Blind Method; Electroencephalography; Haloperidol; Humans; Male; Middle Aged; Pain Measurement; Psychomotor Performance; Reaction Time; Sulpiride | 1990 |
Sulpiride and haloperidol in schizophrenia: a double-blind cross-over study of therapeutic effect, side effects and plasma concentrations.
Topics: Adolescent; Adult; Aged; Clinical Trials as Topic; Double-Blind Method; Female; Haloperidol; Humans; Male; Middle Aged; Psychiatric Status Rating Scales; Schizophrenia; Schizophrenic Psychology; Sulpiride | 1985 |
Atypical neuroleptics: clozapine and the benzamides in the prevention and treatment of tardive dyskinesia.
Topics: Antipsychotic Agents; Benzamides; Clinical Trials as Topic; Clozapine; Dibenzazepines; Dose-Response Relationship, Drug; Dyskinesia, Drug-Induced; Haloperidol; Humans; Metoclopramide; Prospective Studies; Schizophrenia; Sulpiride; Tiapamil Hydrochloride | 1983 |
Acute treatment of Huntington's chorea with lisuride.
Topics: Clinical Trials as Topic; Ergolines; Female; Haloperidol; Humans; Huntington Disease; Lisuride; Male; Placebos; Sulpiride | 1983 |
[Comparative study of the effects of sultopride and haloperidol in agitation states. 94 cases at the psychiatric infirmary of the Paris police headquarters].
Topics: Amisulpride; Haloperidol; Humans; Psychomotor Agitation; Sulpiride | 1983 |
Sulpiride versus haloperidol, a clinical trial in schizophrenia. A preliminary report.
Topics: Adult; Autonomic Nervous System; Clinical Trials as Topic; Double-Blind Method; Female; Haloperidol; Humans; Male; Middle Aged; Parkinson Disease, Secondary; Schizophrenia; Sulpiride | 1984 |
Suppression of REM and delta sleep by apomorphine in man: a dopamine mimetic effect.
Topics: Adult; Apomorphine; Dopamine; Electroencephalography; Female; Haloperidol; Humans; Male; Sleep; Sleep, REM; Sulpiride; Time Factors | 1980 |
A clinical and pharmacodynamic evaluation of sulpiride.
Topics: Chronic Disease; Clinical Trials as Topic; Double-Blind Method; Female; Haloperidol; Humans; Middle Aged; Prolactin; Psychiatric Status Rating Scales; Schizophrenia; Sulpiride | 1981 |
A comparison of the neuro-endocrinological and temperature effects of DU 29894, flesinoxan, sulpiride and haloperidol in normal volunteers.
Topics: Administration, Oral; Adrenocorticotropic Hormone; Adult; Body Temperature; Chromatography, High Pressure Liquid; Cross-Over Studies; Dopamine Antagonists; Double-Blind Method; Enzyme-Linked Immunosorbent Assay; Growth Hormone; Haloperidol; Humans; Hydrocortisone; Male; Piperazines; Prolactin; Radioimmunoassay; Serotonin Receptor Agonists; Sulpiride | 1995 |
Are there dissociable roles of the mesostriatal and mesolimbocortical dopamine systems on temporal information processing in humans?
Topics: Adult; Arousal; Attention; Basal Ganglia; Cerebral Cortex; Corpus Striatum; Dopamine; Dopamine Antagonists; Dose-Response Relationship, Drug; Double-Blind Method; Flicker Fusion; Haloperidol; Humans; Limbic System; Male; Mesencephalon; Neural Pathways; Psychomotor Performance; Reaction Time; Receptors, Dopamine D2; Remoxipride; Sensory Thresholds; Sulpiride; Time Perception | 1997 |
Effects of haloperidol and amisulpride on motor and cognitive skill learning in healthy volunteers.
Topics: Adult; Amisulpride; Analysis of Variance; Antipsychotic Agents; Cognition; Female; Haloperidol; Humans; Learning; Male; Memory; Psychomotor Performance; Sulpiride | 1997 |
Improvement of acute exacerbations of schizophrenia with amisulpride: a comparison with haloperidol. PROD-ASLP Study Group.
Topics: Adult; Akathisia, Drug-Induced; Amisulpride; Antipsychotic Agents; Brief Psychiatric Rating Scale; Double-Blind Method; Female; Haloperidol; Humans; Male; Movement Disorders; Schizophrenia; Sulpiride | 1997 |
Changes in human motor cortex excitability induced by dopaminergic and anti-dopaminergic drugs.
Topics: Administration, Oral; Adult; Analysis of Variance; Bromocriptine; Dopamine Agonists; Dopamine Antagonists; Electromyography; Evoked Potentials, Motor; Female; Haloperidol; Humans; Levodopa; Magnetics; Male; Motor Cortex; Physical Stimulation; Reference Values; Selegiline; Sulpiride | 1997 |
Amisulpride, and atypical antipsychotic, in the treatment of acute episodes of schizophrenia: a dose-ranging study vs. haloperidol. The Amisulpride Study Group.
Topics: Acute Disease; Adult; Amisulpride; Antipsychotic Agents; Dose-Response Relationship, Drug; Double-Blind Method; Drug Administration Schedule; Female; Haloperidol; Humans; Male; Middle Aged; Neurologic Examination; Psychiatric Status Rating Scales; Schizophrenia; Sulpiride; Treatment Outcome | 1998 |
Psychomotor, Cognitive, extrapyramidal, and affective functions of healthy volunteers during treatment with an atypical (amisulpride) and a classic (haloperidol) antipsychotic.
Topics: Adult; Affective Disorders, Psychotic; Amisulpride; Antipsychotic Agents; Basal Ganglia Diseases; Cognition; Cross-Over Studies; Double-Blind Method; Female; Haloperidol; Humans; Male; Psychomotor Performance; Sulpiride | 1999 |
Quantitative EEG in schizophrenic patients before and during pharmacotherapy.
Topics: Adult; Antipsychotic Agents; Beta Rhythm; Delta Rhythm; Electroencephalography; Female; Fluphenazine; Fourier Analysis; Haloperidol; Humans; Male; Schizophrenia; Sulpiride | 2000 |
Long-term safety and efficacy of amisulpride in subchronic or chronic schizophrenia. Amisulpride Study Group.
Topics: Adolescent; Adult; Aged; Amisulpride; Antipsychotic Agents; Chronic Disease; Dyskinesia, Drug-Induced; Female; Haloperidol; Humans; Male; Middle Aged; Psychiatric Status Rating Scales; Schizophrenia; Sulpiride | 2000 |
The acute effects of amisulpride (50 mg and 200 mg) and haloperidol (2 mg) on cognitive function in healthy elderly volunteers.
Topics: Aged; Aged, 80 and over; Amisulpride; Antipsychotic Agents; Arousal; Cognition; Cross-Over Studies; Double-Blind Method; Female; Flicker Fusion; Haloperidol; Humans; Male; Mental Recall; Reaction Time; Sulpiride | 2000 |
Amisulpride has a superior benefit/risk profile to haloperidol in schizophrenia: results of a multicentre, double-blind study (the Amisulpride Study Group).
Topics: Adolescent; Adult; Amisulpride; Antipsychotic Agents; Brief Psychiatric Rating Scale; Double-Blind Method; Female; Haloperidol; Health Status; Humans; Male; Middle Aged; Quality of Life; Schizophrenia; Sulpiride; Surveys and Questionnaires; Treatment Outcome | 2000 |
Neuroendocrine responsivities of the pituitary dopamine system in male schizophrenic patients during treatment with clozapine, olanzapine, risperidone, sulpiride, or haloperidol.
Topics: Adult; Antipsychotic Agents; Benzodiazepines; Clozapine; Dopamine Antagonists; Dose-Response Relationship, Drug; Haloperidol; Humans; Male; Middle Aged; Olanzapine; Pirenzepine; Pituitary Gland; Prolactin; Receptors, Dopamine D2; Risperidone; Schizophrenia; Sulpiride | 2001 |
Amisulpride: efficacy in the management of chronic patients with predominant negative symptoms of schizophrenia.
Topics: Adolescent; Adult; Aged; Amisulpride; Antipsychotic Agents; Basal Ganglia Diseases; Chronic Disease; Double-Blind Method; Female; Haloperidol; Humans; Male; Middle Aged; Pilot Projects; Psychiatric Status Rating Scales; Schizophrenia; Schizophrenic Psychology; Sulpiride | 2001 |
A pilot cross-over design study on QTc interval prolongation associated with sulpiride and haloperidol.
Topics: Adolescent; Adult; Antipsychotic Agents; Cross-Over Studies; Female; Haloperidol; Heart Conduction System; Humans; Long QT Syndrome; Male; Middle Aged; Pilot Projects; Schizophrenia; Sulpiride | 2003 |
Dose-related effects of amisulpride on five dimensions of psychopathology in patients with acute exacerbation of schizophrenia.
Topics: Adolescent; Adult; Amisulpride; Antipsychotic Agents; Dose-Response Relationship, Drug; Female; Haloperidol; Humans; Male; Middle Aged; Psychiatric Status Rating Scales; Schizophrenia; Schizophrenic Psychology; Sulpiride; Treatment Outcome | 2002 |
Effectiveness of antipsychotic drugs in first-episode schizophrenia and schizophreniform disorder: an open randomised clinical trial.
Topics: Adolescent; Adult; Amisulpride; Antipsychotic Agents; Benzodiazepines; Dibenzothiazepines; Female; Haloperidol; Humans; Linear Models; Male; Olanzapine; Patient Compliance; Piperazines; Proportional Hazards Models; Quetiapine Fumarate; Schizophrenia; Sulpiride; Thiazoles; Treatment Outcome | 2008 |
Neurocognitive effectiveness of haloperidol, risperidone, and olanzapine in first-episode psychosis: a randomized, controlled 1-year follow-up comparison.
Topics: Adult; Amisulpride; Antipsychotic Agents; Benzodiazepines; Brain; Clozapine; Cognition Disorders; Female; Follow-Up Studies; Haloperidol; Humans; Male; Neuropsychological Tests; Olanzapine; Perphenazine; Piperazines; Prospective Studies; Psychotic Disorders; Risperidone; Severity of Illness Index; Sulpiride; Thiazoles | 2009 |
Drug attitude as predictor for effectiveness in first-episode schizophrenia: Results of an open randomized trial (EUFEST).
Topics: Adult; Amisulpride; Antipsychotic Agents; Benzodiazepines; Dibenzothiazepines; Female; Haloperidol; Humans; Male; Medication Adherence; Olanzapine; Piperazines; Psychiatric Status Rating Scales; Quetiapine Fumarate; ROC Curve; Schizophrenia; Schizophrenic Psychology; Sulpiride; Surveys and Questionnaires; Thiazoles; Treatment Outcome | 2010 |
Efficacy of antipsychotic drugs against hostility in the European First-Episode Schizophrenia Trial (EUFEST).
Topics: Adult; Aggression; Amisulpride; Antipsychotic Agents; Benzodiazepines; Dibenzothiazepines; Haloperidol; Hostility; Humans; Olanzapine; Piperazines; Psychiatric Status Rating Scales; Psychotic Disorders; Quetiapine Fumarate; Schizophrenia; Schizophrenic Psychology; Sulpiride; Thiazoles; Treatment Outcome | 2011 |
No negative symptoms in healthy volunteers after single doses of amisulpride, aripiprazole, and haloperidol: a double-blind placebo-controlled trial.
Topics: Adult; Amisulpride; Antipsychotic Agents; Aripiprazole; Cognitive Dysfunction; Dizziness; Double-Blind Method; Female; Haloperidol; Humans; Hypnotics and Sedatives; Male; Neurotoxicity Syndromes; Piperazines; Psychiatric Status Rating Scales; Quinolones; Risperidone; Severity of Illness Index; Sulpiride; Time Factors; Young Adult | 2012 |
Persistent negative symptoms in first episode patients with schizophrenia: results from the European First Episode Schizophrenia Trial.
Topics: Adolescent; Adult; Amisulpride; Antipsychotic Agents; Benzodiazepines; Cognition Disorders; Dibenzothiazepines; Female; Haloperidol; Humans; Male; Neuropsychological Tests; Olanzapine; Piperazines; Psychomotor Disorders; Psychotic Disorders; Quetiapine Fumarate; Schizophrenia; Schizophrenic Psychology; Sulpiride; Thiazoles; Treatment Outcome; Young Adult | 2013 |
Cognitive effects of a single dose of atypical antipsychotics in healthy volunteers compared with placebo or haloperidol.
Topics: Adult; Amisulpride; Antipsychotic Agents; Aripiprazole; Cognition; Double-Blind Method; Female; Haloperidol; Humans; Hypnotics and Sedatives; Male; Piperazines; Psychomotor Performance; Quinolones; Risperidone; Sulpiride; Treatment Outcome; Young Adult | 2012 |
Effectiveness of antipsychotic drugs against hostility in patients with schizophrenia in the Clinical Antipsychotic Trials of Intervention Effectiveness (CATIE) study.
Topics: Adult; Aggression; Amisulpride; Antipsychotic Agents; Benzodiazepines; Female; Haloperidol; Hostility; Humans; Male; Middle Aged; Olanzapine; Perphenazine; Piperazines; Quetiapine Fumarate; Risperidone; Schizophrenia; Schizophrenic Psychology; Sulpiride; Thiazoles | 2014 |
Acute Effects of Haloperidol, Amisulpride, and Quetiapine on Bone Turnover Markers in Patients With Schizophrenia.
Topics: Adult; Amisulpride; Antipsychotic Agents; Biomarkers; Bone Remodeling; Bone Resorption; Female; Haloperidol; Humans; Male; Osteogenesis; Prospective Studies; Quetiapine Fumarate; Schizophrenia; Sulpiride; Young Adult | 2015 |
The Role of Dopamine in Temporal Uncertainty.
Topics: Adult; Cross-Over Studies; Dopamine; Dopamine Antagonists; Double-Blind Method; Feedback; Female; Haloperidol; Humans; Intention; Male; Models, Psychological; Movement; Photic Stimulation; Reaction Time; Sulpiride; Time Factors; Time Perception; Uncertainty; Young Adult | 2016 |
509 other study(ies) available for sulpiride and haloperidol
Article | Year |
---|---|
Radiosynthesis, cerebral distribution, and binding of [125I]-1-(p-iodophenyl)-3-(1-adamantyl)guanidine, a ligand for sigma binding sites.
Topics: Animals; Autoradiography; Binding Sites; Binding, Competitive; Brain; Guanidines; Guinea Pigs; Iodobenzenes; Male; Mice; Receptors, sigma; Tissue Distribution | 1992 |
(S)-N-[(1-ethyl-2-pyrrolidinyl)methyl]-5-[125I]iodo- 2-methoxybenzamide hydrochloride, a new selective radioligand for dopamine D-2 receptors.
Topics: Animals; Benzamides; Chromatography, High Pressure Liquid; Isomerism; Kinetics; Male; Pyrrolidines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine | 1988 |
Potential neuroleptic agents. 3. Chemistry and antidopaminergic properties of substituted 6-methoxysalicylamides.
Topics: Animals; Apomorphine; Benzamides; Chemical Phenomena; Chemistry; Corpus Striatum; Dopamine Antagonists; Humans; Hyperkinesis; Magnetic Resonance Spectroscopy; Male; Rats; Rats, Inbred Strains; Salicylamides; Spiperone; Stereotyped Behavior; Structure-Activity Relationship | 1985 |
Synthesis and neuroleptic activity of benzamides. Cis-N-(1-benzyl-2-methylpyrrolidin-3-yl)-5-chloro-2-methoxy-4-(methylamino)benzamide and related compounds.
Topics: Animals; Antipsychotic Agents; Avoidance Learning; Benzamides; Catalepsy; Humans; Rats; Stereotyped Behavior; Structure-Activity Relationship | 1981 |
Potential neuroleptic agents. 2,6-Dialkoxybenzamide derivatives with potent dopamine receptor blocking activities.
Topics: Animals; Antipsychotic Agents; Apomorphine; Behavior, Animal; Benzamides; Catalepsy; Chemical Phenomena; Chemistry; Humans; Lethal Dose 50; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine | 1982 |
Aporphines. 58. N-(2-chloroethyl) [8,9-2H]norapomorphine, an irreversible ligand for dopamine receptors: synthesis and application.
Topics: Animals; Aporphines; Binding, Competitive; Corpus Striatum; Dogs; Pituitary Gland, Anterior; Receptors, Dopamine; Spiperone; Swine | 1984 |
2-Amino-6-chloro-4-(N-methylpiperazino)pyrimidines, inhibitors of spiroperidol binding.
Topics: Animals; Binding, Competitive; Butyrophenones; Chemical Phenomena; Chemistry; Clozapine; Corpus Striatum; Crystallography; Haloperidol; In Vitro Techniques; Molecular Conformation; Piperazines; Pyrimidines; Rats; Receptors, Dopamine; Spiperone; X-Ray Diffraction | 1982 |
QSAR model for drug human oral bioavailability.
Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship | 2000 |
Molecular modeling of the three-dimensional structure of dopamine 3 (D3) subtype receptor: discovery of novel and potent D3 ligands through a hybrid pharmacophore- and structure-based database searching approach.
Topics: Algorithms; Binding Sites; Computational Biology; Crystallography, X-Ray; Databases, Protein; Humans; Kinetics; Ligands; Lipid Bilayers; Models, Molecular; Molecular Conformation; Mutation; Receptors, Dopamine D2; Receptors, Dopamine D3; Reproducibility of Results; Solvents; Structure-Activity Relationship; Tetrahydronaphthalenes; Water | 2003 |
Modeling the similarity and divergence of dopamine D2-like receptors and identification of validated ligand-receptor complexes.
Topics: Amino Acid Sequence; Animals; Cattle; Conserved Sequence; Dopamine Antagonists; Humans; Ligands; Models, Molecular; Molecular Sequence Data; Mutation; Protein Conformation; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Dopamine D4; Rhodopsin; Sequence Alignment; Spiperone | 2005 |
Calculating virtual log P in the alkane/water system (log P(N)(alk)) and its derived parameters deltalog P(N)(oct-alk) and log D(pH)(alk).
Topics: 1-Octanol; Alkanes; Hydrogen-Ion Concentration; Least-Squares Analysis; Mathematics; Models, Chemical; Models, Molecular; Solvents; Water | 2005 |
Chemical genetics reveals a complex functional ground state of neural stem cells.
Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells | 2007 |
Identification of new functional inhibitors of acid sphingomyelinase using a structure-property-activity relation model.
Topics: Algorithms; Animals; Cell Line; Cell Line, Tumor; Chemical Phenomena; Chemistry, Physical; Enzyme Inhibitors; Humans; Hydrogen-Ion Concentration; Molecular Conformation; Quantitative Structure-Activity Relationship; Rats; Sphingomyelin Phosphodiesterase | 2008 |
Physicochemical determinants of human renal clearance.
Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight | 2009 |
Prediction of volume of distribution values in human using immobilized artificial membrane partitioning coefficients, the fraction of compound ionized and plasma protein binding data.
Topics: Blood Proteins; Chemistry, Physical; Computer Simulation; Humans; Membranes, Artificial; Models, Biological; Pharmaceutical Preparations; Protein Binding; Tissue Distribution | 2009 |
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship | 2010 |
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations | 2010 |
Brain tissue binding of drugs: evaluation and validation of solid supported porcine brain membrane vesicles (TRANSIL) as a novel high-throughput method.
Topics: Absorption; Albumins; Animals; Brain; Brain Chemistry; Cell Membrane; Chromatography, High Pressure Liquid; Drug Evaluation, Preclinical; In Vitro Techniques; Lipids; Male; Microdialysis; Pharmaceutical Preparations; Protein Binding; Rats; Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization; Swine; Tissue Distribution | 2011 |
QSAR-based permeability model for drug-like compounds.
Topics: Caco-2 Cells; Cell Membrane Permeability; Drug Discovery; Humans; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship | 2011 |
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship | 2012 |
Discovery and characterization of novel, potent, and selective cytochrome P450 2J2 inhibitors.
Topics: Chromatography, High Pressure Liquid; Cytochrome P-450 CYP2J2; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Drug Discovery; Enzyme Inhibitors; Humans; Inhibitory Concentration 50; Kinetics; Microsomes, Liver; Models, Molecular; Molecular Dynamics Simulation; Substrate Specificity | 2013 |
Differential effect of neuroleptic drugs on dopamine turnover in the extrapyramidal and limbic system.
Topics: Animals; Caudate Nucleus; Chlorpromazine; Clozapine; Dopamine; Extrapyramidal Tracts; Haloperidol; Homovanillic Acid; Limbic System; Male; Olfactory Bulb; Rats; Sulpiride; Thioridazine; Tranquilizing Agents | 1976 |
[Acute and chronic effects of carpipramine, clozapine, haloperidol and sulpiride on the metabolism of biogenic amines in the rat brain (author's transl)].
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Biogenic Amines; Brain; Brain Chemistry; Cerebral Cortex; Clozapine; Corpus Striatum; Dibenzazepines; Haloperidol; Homovanillic Acid; Hydroxyindoleacetic Acid; Limbic System; Male; Methoxyhydroxyphenylglycol; Rats; Sulpiride | 1976 |
Nonstriatal dopaminergic neurons: Section X. Morphine, amphetamine, and noncataleptogenic neuroleptics: Introduction: morphine, amphetamine, and noncataleptogenic neuroleptics.
Topics: Acetylcholine; Animals; Antipsychotic Agents; Brain; Clozapine; Corpus Striatum; Dextroamphetamine; Dopamine; gamma-Aminobutyric Acid; Glutamates; Haloperidol; Morphine; Neurotransmitter Agents; Rats; Receptors, Dopamine; Receptors, Opioid; Sulpiride | 1977 |
Dopamine-stimulated adenylate cyclase in rat substantia nigra: localization and effects of neuroleptics.
Topics: Adenylyl Cyclases; Animals; Antipsychotic Agents; Apomorphine; Chlorpromazine; Dopamine; Fluphenazine; Haloperidol; In Vitro Techniques; Isoproterenol; Male; Norepinephrine; Rats; Substantia Nigra; Sulpiride | 1977 |
Sedative, hypnotic, and antipsychotic effects of low doses of apomorphine in man.
Topics: Adolescent; Adult; Antipsychotic Agents; Apomorphine; Bipolar Disorder; Drug Interactions; Female; Haloperidol; Humans; Hypnotics and Sedatives; Male; Schizophrenia; Sulpiride | 1977 |
Dopamine metabolism in the rat retina and brain after acute and repeated treatment with neuroleptics.
Topics: Animals; Antipsychotic Agents; Brain; Dopamine; Dose-Response Relationship, Drug; Drug Tolerance; Haloperidol; Male; Rats; Retina; Sulpiride; Time Factors | 1978 |
Changes in dopamine-dependent motor behaviour caused by propranolol and its isomers.
Topics: Animals; Apomorphine; Dopamine; Dyskinesia, Drug-Induced; Guinea Pigs; Haloperidol; Mice; Motor Activity; Propranolol; Stereoisomerism; Sulpiride; Time Factors | 1978 |
The effect of neuroleptic drugs on drinking induced by central administration of angiotensin or carbachol.
Topics: Angiotensin II; Animals; Antipsychotic Agents; Carbachol; Chlorpromazine; Clozapine; Dopamine; Drinking Behavior; Flupenthixol; Fluphenazine; Haloperidol; Injections, Intraperitoneal; Injections, Intraventricular; Male; Pimozide; Rats; Sulpiride | 1979 |
Hypothermic action of lisuride in rats and differences to bromocriptine in the antagonistic effect of neuroleptics.
Topics: Animals; Antipsychotic Agents; Body Temperature; Bromocriptine; Cold Temperature; Depression, Chemical; Ergolines; Female; Haloperidol; Lisuride; Rats; Sulpiride; Time Factors | 1979 |
Crop-sac response after systemic and intraventricular administration of neuroleptic drugs.
Topics: Animals; Antipsychotic Agents; Clozapine; Columbidae; Crop, Avian; Female; Haloperidol; Injections, Intraventricular; Reserpine; Sulpiride | 1979 |
Amines and the rat exocrine pancreas: (2) Effects of receptor blockers on turnover of L-5HTP.
Topics: 5-Hydroxytryptophan; Adrenergic alpha-Antagonists; Animals; Cyproheptadine; Haloperidol; Histocytochemistry; Male; Methysergide; Microscopy, Fluorescence; Monoamine Oxidase Inhibitors; Pancreas; Pancreatic Juice; Rats; Receptors, Adrenergic; Receptors, Serotonin; Sulpiride | 1979 |
Interference between anti-HLA antibodies and adrenergic receptor-binding drugs.
Topics: Adrenergic beta-Antagonists; Antibodies; Apomorphine; Binding Sites, Antibody; Chlorpromazine; Cross Reactions; Dopamine; Epitopes; Female; Haloperidol; Histocompatibility Antigens; HLA Antigens; Humans; Immune Sera; Lymphocytes; Propranolol; Sulpiride | 1977 |
[Clebopride, a new orthopramide with potent and selective central antidopaminergic properties].
Topics: Alprenolol; Animals; Benzamides; Dihydroergotoxine; Haloperidol; Metoclopramide; Piperidines; Rats; Receptors, Dopamine; Sulpiride | 1978 |
Differential behavioral effects of sulpiride in the rat and squirrel monkey.
Topics: Animals; Avoidance Learning; Behavior, Animal; Benztropine; Haloperidol; Haplorhini; Male; Saimiri; Sulpiride; Time Factors | 1978 |
Sulpiride: a study of the effects on dopamine receptors in rat neostriatum and limbic forebrain.
Topics: Adenylyl Cyclases; Animals; Apomorphine; Corpus Striatum; Cyclic AMP; Dopamine; Haloperidol; Imipramine; Male; Olfactory Bulb; Rats; Receptors, Drug; Sulpiride | 1975 |
Amines and the rat exocrine pancreas: (3) Effects of amines on pancreatic secretion.
Topics: 5-Hydroxytryptophan; Amines; Animals; Bicarbonates; Haloperidol; Levodopa; Male; Monoamine Oxidase Inhibitors; Pancreatic Juice; Phenoxybenzamine; Phenylephrine; Proteins; Rats; Secretin; Secretory Rate; Sulpiride | 1979 |
Isolation of gamma-amino butyric acid from pig hypothalami and demonstration of its prolactin release-inhibiting (PIF) activity in vivo and in vitro.
Topics: Animals; Chlorpromazine; Culture Techniques; gamma-Aminobutyric Acid; Haloperidol; Hypothalamus; Monoiodotyrosine; Perphenazine; Pituitary Gland; Prolactin; Sulpiride; Swine | 1977 |
The effects of dopaminergic blocking agents on the glucose tolerance test in 6 humans and 6 dogs.
Topics: Animals; Blood Glucose; Dogs; Glucose Tolerance Test; Haloperidol; Humans; Species Specificity; Sulpiride | 1979 |
Effects of dopaminergic blocking agents on distal colon motility.
Topics: Adolescent; Adult; Biperiden; Colon; Dihydroergotamine; Dopamine Antagonists; Female; Gastrointestinal Motility; Haloperidol; Humans; Male; Middle Aged; Muscle Tonus; Pimozide; Sulpiride; Thioridazine | 1979 |
Effects of diphenylhydantoin (DPH) on distal colon motility.
Topics: Adult; Colon; Colon, Sigmoid; Female; Gastrointestinal Motility; Haloperidol; Humans; Male; Manometry; Phenytoin; Rectum; Sulpiride | 1979 |
Dopamine receptor blocking activity of sulpiride in the central nervous system.
Topics: Administration, Oral; Animals; Apomorphine; Behavior, Animal; Brain; Catalepsy; Cerebral Ventricles; Chlorpromazine; Compulsive Behavior; Haloperidol; Humans; Injections, Intravenous; Male; Methamphetamine; Rats; Receptors, Dopamine; Sulpiride | 1977 |
Regional displacement by sulpiride of [3H]spiperone binding in vivo. Biochemical and behavioural evidence for a preferential action of limbic and nigral dopamine receptors.
Topics: Animals; Apomorphine; Binding, Competitive; Brain; Butyrophenones; Catalepsy; Haloperidol; Humans; Male; Rats; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Sulpiride | 1979 |
Differential regional development of tolerance to increase in dopamine turnover upon repeated neuroleptic administration.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Brain; Dopamine; Drug Tolerance; Haloperidol; Homovanillic Acid; Male; Rats; Sulpiride; Time Factors | 1977 |
Dopamine receptors: pharmacological and anatomical evidences indicate that two distinct dopamine receptor populations are present in rat striatum.
Topics: Adenylyl Cyclases; Animals; Corpus Striatum; Haloperidol; Male; Rats; Receptors, Dopamine; Spiperone; Sulpiride; Time Factors | 1978 |
The computer diagnosis in a multicenter study of psychoactive agents.
Topics: Adult; Aged; Diagnosis, Computer-Assisted; Haloperidol; Humans; Middle Aged; Schizophrenia; Sulpiride | 1976 |
A comparison of the abilities of typical neuroleptic agents and of thioridazine, clozapine, sulpiride and metoclopramide to antagonise the hyperactivity induced by dopamine applied intracerebrally to areas of the extrapyramidal and mesolimbic systems.
Topics: Animals; Brain; Clozapine; Corpus Striatum; Dopamine Antagonists; Dose-Response Relationship, Drug; Extrapyramidal Tracts; Fluphenazine; Haloperidol; Limbic System; Male; Metoclopramide; Pimozide; Rats; Stereotaxic Techniques; Sulpiride; Thioridazine; Tranquilizing Agents | 1976 |
Central effects of thyrotropin-releasing factor (TRF); interaction with some antipsychotic drugs.
Topics: Animals; Behavior, Animal; Chlorpromazine; Drug Interactions; Haloperidol; Injections, Intraventricular; Levodopa; Mice; Reserpine; Sulpiride; Thyrotropin-Releasing Hormone; Time Factors | 1976 |
In vivo binding of 3H-pimozide in mouse striatum: effects of dopamine agonists and antagonists.
Topics: Animals; Apomorphine; Cerebellum; Cerebral Cortex; Corpus Striatum; Dextroamphetamine; Haloperidol; Homovanillic Acid; Levodopa; Male; Mice; Pimozide; Receptors, Dopamine; Sulpiride | 1977 |
Effect of single and repeated administration of haloperidol and sulpiride on striatal and retinal dopamine turnover in the rat.
Topics: Animals; Corpus Striatum; Dopamine; Drug Tolerance; Haloperidol; Male; Rats; Retina; Sulpiride | 1977 |
Antagonism by sulpiride of three apomorphine-induced effects in rodents.
Topics: Animals; Apomorphine; Behavior, Animal; Body Temperature; Depression, Chemical; Haloperidol; Humans; Male; Mice; Pimozide; Rats; Stereotyped Behavior; Sulpiride | 1976 |
Acidic dopamine metabolites in cortical areas of the rat brain: localization and effects of drug.
Topics: 3,4-Dihydroxyphenylacetic Acid; Amphetamine; Animals; Apomorphine; Cerebral Cortex; Clozapine; Corpus Striatum; Haloperidol; Homovanillic Acid; Male; Morphine; Olfactory Bulb; Oxotremorine; Phenylacetates; Probenecid; Rats; Sulpiride; Thioridazine | 1976 |
Specificity of the dopamine sensitive adenylate cyclase for antipsychotic antagonists.
Topics: Adenylyl Cyclases; Animals; Apomorphine; Chlorpromazine; Clozapine; Corpus Striatum; Dopamine; Dopamine Antagonists; Enzyme Activation; Haloperidol; Male; Metoclopramide; Rats; Sulpiride | 1976 |
On the relevance of preferential increases of mesolimbic versus striatal dopamine turnover for the prediction of antipsychotic activity of psychotropic drugs.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Anthracenes; Clozapine; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Haloperidol; Homovanillic Acid; Humans; Limbic System; Male; Methyltyrosines; Psychotic Disorders; Psychotropic Drugs; Rats; Sulpiride; Thioridazine | 1976 |
[Chemotherapy of melancholia by sequential neuroleptic-viloxazine association].
Topics: Adjustment Disorders; Adult; Bipolar Disorder; Chlorpromazine; Depression; Depressive Disorder, Major; Drug Therapy, Combination; Female; Haloperidol; Humans; Male; Methotrimeprazine; Middle Aged; Morpholines; Sulpiride; Tranquilizing Agents; Viloxazine | 1976 |
Influence of dopaminergic agonists and antagonists on serum prolactin concentrations in the rat.
Topics: Animals; Apomorphine; Benserazide; Clonidine; Dextroamphetamine; Dopamine; Female; Haloperidol; Hypophysectomy; Levodopa; Male; Methyltyrosines; Piribedil; Pituitary Gland; Prolactin; Rats; Reserpine; Sulpiride; Transplantation, Homologous | 1976 |
Therapeutic spectrum of sulpiride, haloperidol and lithium: a graphic representation by clinical observation.
Topics: Haloperidol; Humans; Lithium; Models, Theoretical; Psychotic Disorders; Sulpiride | 1976 |
Correlation between catalepsy and dopamine decrease in the rat striatum induced by neuroleptics.
Topics: Animals; Butyrophenones; Catalepsy; Chlorpromazine; Clozapine; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Haloperidol; Humans; Male; Rats; Sulpiride; Thioridazine; Time Factors; Tranquilizing Agents; Trifluperidol | 1976 |
Detection of the nueroleptic properties of clozapine, sulpiride and thioridazine.
Topics: Animals; Apomorphine; Behavior, Animal; Catalepsy; Clozapine; Dextroamphetamine; Dibenzazepines; Dose-Response Relationship, Drug; Drug Synergism; Fluphenazine; Haloperidol; Humans; Isoquinolines; Male; Methyltyrosines; Pimozide; Rats; Spiro Compounds; Stereotyped Behavior; Succinimides; Sulpiride; Thioridazine; Tranquilizing Agents | 1975 |
Therapeutical efficacy of a combination of apomorphine with sulpiride or metoclopramide in Parkinsonism.
Topics: Adult; Apomorphine; Drug Therapy, Combination; Haloperidol; Humans; Male; Metoclopramide; Parkinson Disease; Sleep; Sulpiride; Vomiting | 1976 |
High concentrations of the neuroleptic remoxipride block voltage-activated Na+ channels in central and peripheral nerve membranes.
Topics: Animals; Brain; Cerebral Cortex; Corpus Striatum; Dose-Response Relationship, Drug; Electrophysiology; Haloperidol; In Vitro Techniques; Male; Nerve Fibers, Myelinated; Potassium; Rats; Rats, Sprague-Dawley; Remoxipride; Sodium; Sodium Channels; Sulpiride; Xenopus laevis | 1992 |
A lever-release version of the conditioned avoidance response paradigm: effects of haloperidol, clozapine, sulpiride, and BMY-14802.
Topics: Animals; Antipsychotic Agents; Avoidance Learning; Clozapine; Dextroamphetamine; Dose-Response Relationship, Drug; Haloperidol; Male; Psychotropic Drugs; Pyrimidines; Rats; Rats, Inbred Strains; Stereotyped Behavior; Sulpiride | 1992 |
The effect of intrastriatal application of directly and indirectly acting dopamine agonists and antagonists on the in vivo release of acetylcholine measured by brain microdialysis. The importance of the post-surgery interval.
Topics: Acetylcholine; Amphetamine; Animals; Benzazepines; Corpus Striatum; Dopamine; Dopamine Agents; Dopamine Antagonists; Ergolines; Haloperidol; Indoles; Male; Oxidopamine; Phenanthridines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Sulpiride | 1992 |
Comparative studies of sulpiride and classical neuroleptics on induction of catalepsy, locomotor activity, and brain dopamine metabolism in mice.
Topics: Animals; Antipsychotic Agents; Brain Chemistry; Catalepsy; Dopamine; Haloperidol; Male; Mice; Mice, Inbred Strains; Motor Activity; Pimozide; Sulpiride | 1992 |
Changes in dopamine D1, D2 and D3 receptor mRNA levels in rat brain following antipsychotic treatment.
Topics: Animals; Antipsychotic Agents; Blotting, Northern; Brain Chemistry; Haloperidol; Loxapine; Male; Oligonucleotides; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; RNA, Messenger; Sulpiride | 1992 |
Recurrent neuroleptic malignant syndrome in a man with mild mental handicap.
Topics: Adult; Antipsychotic Agents; Carbamazepine; Dose-Response Relationship, Drug; Drug Therapy, Combination; Haloperidol; Humans; Intellectual Disability; Male; Neuroleptic Malignant Syndrome; Neurologic Examination; Orphenadrine; Recurrence; Sulpiride | 1992 |
Evaluation of a stable CCK agonist (A68552) in conditioned avoidance responding in mice, rats, and primates: comparison with typical and atypical antipsychotics.
Topics: Animals; Antipsychotic Agents; Avoidance Learning; Cholecystokinin; Clozapine; Dose-Response Relationship, Drug; Haloperidol; Macaca fascicularis; Male; Mice; Peptide Fragments; Rats; Sulpiride | 1992 |
Direct demonstration of dopamine D1-like receptor sites in the ciliary body of the rabbit eye by light microscope autoradiography.
Topics: Animals; Autoradiography; Benzazepines; Binding Sites; Binding, Competitive; Ciliary Body; Dopamine Agents; Drug Interactions; Haloperidol; Rabbits; Receptors, Dopamine D1; Sulpiride | 1992 |
Lack of effect of chronic antipsychotic treatment on dopamine D5 receptor mRNA level.
Topics: Animals; Antipsychotic Agents; Base Sequence; Brain Chemistry; Down-Regulation; Haloperidol; Loxapine; Male; Molecular Sequence Data; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D5; RNA, Messenger; Sulpiride | 1992 |
[Fever caused by neuroleptics].
Topics: Adult; Delayed-Action Preparations; Female; Fever; Haloperidol; Humans; Male; Middle Aged; Neuroleptic Malignant Syndrome; Solvents; Sulpiride | 1992 |
[The effects of dopamine D-1 and D-2 receptor antagonists on 3,4-dihydroxyphenylacetic acid (DOPAC) in rat striatum with differential normal pulse voltammetry].
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Benzazepines; Chlorpromazine; Corpus Striatum; Dopamine D2 Receptor Antagonists; Haloperidol; Male; Rats; Rats, Wistar; Receptors, Dopamine D1; Sulpiride | 1992 |
[The suppressed pill with far-reaching consequences].
Topics: Dystonia; Haloperidol; Humans; Receptors, Dopamine; Receptors, Dopamine D2; Sulpiride; Tomography, Emission-Computed, Single-Photon | 1992 |
Effect of SCH 39166, a novel dopamine D1 receptor antagonist, on [3H]acetylcholine release in rat striatal slices.
Topics: Acetylcholine; Animals; Apomorphine; Benzazepines; Choline; Corpus Striatum; Dopamine Antagonists; Electric Stimulation; Haloperidol; In Vitro Techniques; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Sulpiride | 1992 |
Further studies on the modulation of regional brain neurotensin concentrations by antipsychotic drugs: focus on haloperidol and BMY 14802.
Topics: Animals; Benzazepines; Brain; Drug Interactions; Haloperidol; Injections, Intraperitoneal; Male; Neurotensin; Psychotropic Drugs; Pyrimidines; Rats; Rats, Inbred Strains; Sulpiride | 1992 |
Alterations in regional brain neurotensin concentrations produced by atypical antipsychotic drugs.
Topics: Animals; Antipsychotic Agents; Benzamides; Carbazoles; Caudate Nucleus; Haloperidol; Male; Neurotensin; Nucleus Accumbens; Radioimmunoassay; Rats; Rats, Inbred Strains; Remoxipride; Sulpiride | 1991 |
[The mechanism of the inhibitory effects of oren-gedoku-to (OGT) on gastric acid secretion in rats].
Topics: Adrenergic alpha-Antagonists; Animals; Atropine; Baclofen; Depression, Chemical; Drugs, Chinese Herbal; Gastric Acid; Haloperidol; Male; Phentolamine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Dopamine; Sulpiride; Thyrotropin-Releasing Hormone; Yohimbine | 1991 |
MPTP lesions and dopaminergic drugs alter eye blink rate in African green monkeys.
Topics: Animals; Apomorphine; Blinking; Chlorocebus aethiops; Dopamine Agents; Haloperidol; Male; MPTP Poisoning; Oxazines; Parkinson Disease; Receptors, Dopamine; Substantia Nigra; Sulpiride | 1991 |
D2 dopamine receptor-mediated mechanisms in the medial preoptic-anterior hypothalamus regulate effective defense behavior in the cat.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Affect; Aggression; Analysis of Variance; Animals; Apomorphine; Benzazepines; Cats; Dopamine Agents; Dose-Response Relationship, Drug; Electric Stimulation; Ergolines; Female; Haloperidol; Hypothalamus, Anterior; Male; Organ Specificity; Preoptic Area; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D2; Sulpiride | 1991 |
Modulation of dopaminergic terminal excitability by D1 selective agents: further characterization.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; alpha-Methyltyrosine; Animals; Benzazepines; Corpus Striatum; Dopamine; Dopamine Agents; Electric Stimulation; Haloperidol; Kainic Acid; Male; Methyltyrosines; Nerve Endings; Pharmaceutical Vehicles; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Sulpiride; Tyrosine 3-Monooxygenase | 1991 |
Neuroleptic malignant syndrome in a case of acute post-traumatic psychosis.
Topics: Antipsychotic Agents; Carbamazepine; Diagnosis, Differential; Haloperidol; Humans; Middle Aged; Neurocognitive Disorders; Neuroleptic Malignant Syndrome; Neurologic Examination; Stress Disorders, Post-Traumatic; Sulpiride | 1991 |
Stereoisomers of the atypical neuroleptic carbidine modulate striatal dopamine release in awake rats.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Antipsychotic Agents; Carbolines; Corpus Striatum; Dialysis; Dopamine; Haloperidol; Homovanillic Acid; Male; Rats; Rats, Inbred Strains; Stereoisomerism; Sulpiride | 1991 |
Role of dopamine receptors in the occurrence of the behavioral motor disturbances in rats exposed to high pressure.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Atmospheric Pressure; Behavior, Animal; Dopamine Agents; Epilepsies, Myoclonic; Ergolines; Haloperidol; High Pressure Neurological Syndrome; Injections, Intraventricular; Male; Motor Activity; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sulpiride; Tremor | 1991 |
Our experience with incisive neuroleptic drugs in child psychiatry.
Topics: Antipsychotic Agents; Autistic Disorder; Child; Haloperidol; Humans; Mental Disorders; Obsessive-Compulsive Disorder; Penfluridol; Pimozide; Psychotic Disorders; Sulpiride; Tic Disorders | 1991 |
The influence of agonists and antagonists of dopaminergic system on the formation of audiogenic seizures in rats during the ethanol abstinence period.
Topics: Amantadine; Animals; Bromocriptine; Dopamine Agents; Dopamine Antagonists; Ethanol; Haloperidol; Male; Metoclopramide; Rats; Rats, Wistar; Substance Withdrawal Syndrome; Sulpiride | 1990 |
Tachykinins in the rat substantia nigra: effects of selective dopamine receptor antagonists.
Topics: Amino Acid Sequence; Animals; Benzazepines; Chromatography, High Pressure Liquid; Dopamine Antagonists; Haloperidol; Male; Molecular Sequence Data; Neurokinin B; Radioimmunoassay; Rats; Rats, Inbred Strains; Substance P; Substantia Nigra; Sulpiride; Tachykinins | 1991 |
Anti-sedative and anti-cataleptic properties of NCS-382, a gamma-hydroxybutyrate receptor antagonist.
Topics: Animals; Anticonvulsants; Benzocycloheptenes; Catalepsy; Dose-Response Relationship, Drug; Haloperidol; Hypnotics and Sedatives; Male; Psychomotor Performance; Rats; Rats, Inbred Strains; Sodium Oxybate; Sulpiride; Swimming | 1991 |
Presynaptic autoinhibition of the electrically evoked dopamine release studied in the rat olfactory tubercle by in vivo electrochemistry.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Dopamine; Electric Stimulation; Ergolines; Evoked Potentials; Haloperidol; Male; Microelectrodes; Olfactory Bulb; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Secretory Rate; Sulpiride | 1991 |
Effects of phencyclidine on contractile forces of isolated rabbit papillary muscles.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Benzazepines; Dextrorphan; Female; Haloperidol; Male; Myocardial Contraction; Papillary Muscles; Phencyclidine; Rabbits; Stimulation, Chemical; Sulpiride | 1991 |
[An experimental study of the antidepressive properties of captopril].
Topics: Amitriptyline; Animals; Antidepressive Agents; Apomorphine; Captopril; Haloperidol; Male; Mice; Motor Activity; Physical Exertion; Stereotyped Behavior; Sulpiride; Swimming | 1991 |
[Comparison of central stimulating effects between ephedrine and apomorphine].
Topics: Animals; Apomorphine; Blepharoptosis; Catalepsy; Ephedrine; Haloperidol; Male; Mice; Motor Activity; Prazosin; Rats; Rats, Inbred Strains; Stereotyped Behavior; Sulpiride; Vomiting | 1991 |
Dorsal raphé stimulation modifies striatal-evoked antidromic invasion of nigral dopaminergic neurons in vivo.
Topics: Animals; Corpus Striatum; Dopamine; Electric Stimulation; Electrodes; Fenclonine; Haloperidol; Male; Metergoline; Neurons; Raphe Nuclei; Rats; Rats, Inbred Strains; Serotonin; Substantia Nigra; Sulpiride | 1991 |
Role of dopamine1-receptors in mediating renal responses to furosemide in the rat.
Topics: Animals; Benzazepines; Blood Pressure; Dopamine; Female; Furosemide; Haloperidol; Kidney; Potassium; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Sodium; Sulpiride | 1991 |
Possible involvement of dopamine D-1 and D-2 receptors in diazepam-induced hyperphagia in rats.
Topics: alpha-Methyltyrosine; Animals; Benzamides; Benzazepines; Diazepam; Domperidone; Dose-Response Relationship, Drug; Feeding Behavior; Haloperidol; Hyperphagia; Injections, Subcutaneous; Male; Methyltyrosines; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Sulpiride | 1991 |
D1 and D2 receptor antagonists differently affect cocaine-induced locomotor hyperactivity in the mouse.
Topics: Animals; Benzazepines; Cocaine; Dopamine Antagonists; Dose-Response Relationship, Drug; Haloperidol; Male; Metoclopramide; Mice; Mice, Inbred C57BL; Motor Activity; Receptors, Dopamine D1; Receptors, Dopamine D2; Stimulation, Chemical; Sulpiride | 1991 |
Transfected D2 dopamine receptors mediate the potentiation of arachidonic acid release in Chinese hamster ovary cells.
Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Apomorphine; Arachidonic Acid; Arachidonic Acids; Calcimycin; Cricetinae; Cricetulus; Cyclic AMP; Dopamine; Drug Synergism; Ergolines; Haloperidol; In Vitro Techniques; Melitten; Pertussis Toxin; Protein Kinase C; Quinpirole; Receptors, Dopamine; Sulpiride; Tetradecanoylphorbol Acetate; Transfection; Virulence Factors, Bordetella | 1991 |
Inhibitory influence of the mesocortical dopaminergic neurons on their target cells: electrophysiological and pharmacological characterization.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Dopamine; Electric Stimulation; Ergolines; Frontal Lobe; Haloperidol; Iontophoresis; Isoproterenol; Male; Norepinephrine; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Dopamine; Sulpiride | 1991 |
Further evidence for the inhibitory action of baclofen on a prolactin-releasing factor.
Topics: alpha-Methyltyrosine; Animals; Baclofen; Dose-Response Relationship, Drug; Female; Haloperidol; Male; Methyltyrosines; Prolactin; Rats; Rats, Inbred Strains; Serotonin; Sulpiride; Thyrotropin-Releasing Hormone | 1991 |
Atypical neuroleptics suppress dopaminergic behavioral supersensitivity.
Topics: Animals; Antipsychotic Agents; Apomorphine; Behavior, Animal; Clozapine; Cyproheptadine; Haloperidol; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Ritanserin; Serotonin Antagonists; Sulpiride; Thioridazine | 1990 |
Repeated treatment with (-)-sulpiride plus a low dose of SCH 23390 displays wider neuroleptic activity without inducing dopaminergic supersensitivity.
Topics: Animals; Antipsychotic Agents; Apomorphine; Benzazepines; Corpus Striatum; Dopamine Agents; Haloperidol; Male; Rats; Rats, Inbred Strains; Stereotyped Behavior; Sulpiride; Synaptic Transmission | 1990 |
Acute effects of typical and atypical antipsychotic drugs on the release of dopamine from prefrontal cortex, nucleus accumbens, and striatum of the rat: an in vivo microdialysis study.
Topics: Animals; Antipsychotic Agents; Clozapine; Corpus Striatum; Dialysis; Dopamine; Frontal Lobe; Haloperidol; Male; Nucleus Accumbens; Rats; Rats, Inbred Strains; Septal Nuclei; Sulpiride | 1990 |
Dopamine receptors and sensorimotor behavior in MPTP-treated mice.
Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Arousal; Benzazepines; Discrimination Learning; Dopamine Agents; Dopamine Antagonists; Dose-Response Relationship, Drug; Ergolines; Haloperidol; Male; Mice; Mice, Inbred Strains; Motor Activity; Orientation; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Sulpiride | 1990 |
Discriminatory roles for D1 and D2 dopamine receptor subtypes in the in vivo control of neostriatal cyclic GMP.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Corpus Striatum; Cyclic GMP; Dopamine Agents; Dose-Response Relationship, Drug; Drug Interactions; Ergolines; Haloperidol; Male; Mice; Quinpirole; Receptors, Dopamine; Sulpiride | 1990 |
Striatal and nucleus accumbens D1/D2 dopamine receptors in neuroleptic catalepsy.
Topics: Animals; Antipsychotic Agents; Benzazepines; Catalepsy; Corpus Striatum; Dose-Response Relationship, Drug; Haloperidol; Male; Nucleus Accumbens; Rats; Rats, Inbred Strains; Receptors, Dopamine; Septal Nuclei; Sulpiride | 1990 |
Effects of dopamine D-1 and D-2 antagonists on decision making by rats: no reversal of neuroleptic-induced attenuation by scopolamine.
Topics: Animals; Antipsychotic Agents; Benzazepines; Conditioning, Operant; Decision Making; Dopamine; Drinking Behavior; Extinction, Psychological; Haloperidol; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Dopamine; Scopolamine; Sulpiride | 1990 |
[The inhibition of dopamine D1 and D2 receptors in human putamen by antipsychotic drugs].
Topics: Aged; Aged, 80 and over; Antipsychotic Agents; Benzamides; Benzazepines; Chlorpromazine; Depression, Chemical; Female; Haloperidol; Humans; In Vitro Techniques; Putamen; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Sulpiride | 1990 |
The action of dopamine receptor antagonists on the secretory response of the cockroach salivary gland in vitro.
Topics: Animals; Benzazepines; Binding, Competitive; Chlorpromazine; Cockroaches; Domperidone; Dopamine; Dopamine Antagonists; Haloperidol; Metoclopramide; Salivary Glands; Sulpiride | 1990 |
Participation of periventricular dopamine receptors in vasopressin secretion elicited by hypertonicity of systemic blood in rats.
Topics: Animals; Benzazepines; Chlorides; Dopamine; Dose-Response Relationship, Drug; Haloperidol; Hypothalamus; Injections, Intraventricular; Male; Osmolar Concentration; Rats; Rats, Inbred Strains; Receptors, Dopamine; Saline Solution, Hypertonic; Sodium; Sulpiride; Vasopressins | 1991 |
Effects of D-1 and D-2 dopamine antagonists on ERG and optic nerve response of the cat.
Topics: Animals; Cats; Electrophysiology; Electroretinography; Fluphenazine; Haloperidol; Optic Nerve; Receptors, Dopamine; Retina; Sulpiride | 1991 |
The latent inhibition model of schizophrenic attention disorder. Haloperidol and sulpiride enhance rats' ability to ignore irrelevant stimuli.
Topics: Animals; Appetitive Behavior; Arousal; Association Learning; Attention; Brain; Conditioning, Classical; Disease Models, Animal; Dose-Response Relationship, Drug; Haloperidol; Humans; Inhibition, Psychological; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Schizophrenic Psychology; Sulpiride | 1991 |
Striatal depth EEG reveals postsynaptic activity of striatal neurons following dopamine receptor stimulation and blockade.
Topics: Animals; Apomorphine; Corpus Striatum; Dopamine Antagonists; Electrodes, Implanted; Electroencephalography; Electrophysiology; Fourier Analysis; Haloperidol; Male; Mice; Mice, Inbred C57BL; Neurons; Receptors, Dopamine; Stereotyped Behavior; Sulpiride; Synapses | 1991 |
Dopaminergic-cholinergic interactions in the striatum: the critical significance of calcium concentrations in brain microdialysis.
Topics: Acetylcholine; Animals; Apomorphine; Atropine; Calcium; Corpus Striatum; Dextroamphetamine; Dialysis Solutions; Dopamine; Haloperidol; Interneurons; Male; Neostigmine; Nomifensine; Perfusion; Rats; Rats, Inbred Strains; Sodium Chloride; Sulpiride; Tetrahydronaphthalenes; Thiophenes | 1990 |
Utilization of microdialysis for assessing the release of mesotelencephalic dopamine following clozapine and other antipsychotic drugs.
Topics: Animals; Cerebral Cortex; Clozapine; Corpus Striatum; Dialysis; Dopamine; Haloperidol; Mesencephalon; Microchemistry; Nucleus Accumbens; Organ Specificity; Rats; Sulpiride; Telencephalon | 1990 |
Dopamine antagonists produce an age-dependent increase in the responding of the young chick.
Topics: Age Factors; Animals; Appetitive Behavior; Arousal; Avoidance Learning; Brain; Chickens; Conditioning, Classical; Dose-Response Relationship, Drug; Haloperidol; Mental Recall; Receptors, Dopamine; Receptors, Dopamine D2; Sulpiride | 1990 |
Effects induced by chronic treatment with selective D1 or D2 antagonists on open-field behavior and colonic temperature.
Topics: Animals; Behavior, Animal; Benzazepines; Body Temperature; Colon; Dopamine Antagonists; Drug Administration Schedule; Haloperidol; Locomotion; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Dopamine D1; Receptors, Dopamine D2; Sulpiride | 1990 |
Dopamine D2 receptors and spinal cord excitation in mice.
Topics: Animals; Apomorphine; Benzazepines; Dopamine Antagonists; Haloperidol; Injections, Spinal; Injections, Subcutaneous; Male; Mice; Mice, Inbred ICR; Morphine; Receptors, Dopamine; Receptors, Dopamine D2; Reflex; Spinal Cord; Sulpiride | 1990 |
Chronic blockade of D2 but not D1 dopamine receptors facilitates behavioural responses to endogenous enkephalins, protected by kelatorphan, administered in the accumbens in rats.
Topics: Animals; Behavior, Animal; Benzazepines; Dipeptides; Dose-Response Relationship, Drug; Enkephalin, Leucine; Enkephalins; Haloperidol; Injections; Male; Motor Activity; Narcotic Antagonists; Nucleus Accumbens; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Opioid; Receptors, Opioid, delta; Sulpiride | 1990 |
Decreased striatal release of acetylcholine following withdrawal from long-term treatment with haloperidol: modulation by cholinergic, dopamine-D1 and -D2 mechanisms.
Topics: Acetylcholine; Animals; Benzazepines; Corpus Striatum; Haloperidol; In Vitro Techniques; Male; Parasympathetic Nervous System; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Muscarinic; Substance Withdrawal Syndrome; Sulpiride | 1990 |
Effect of apomorphine on oxytocin concentrations in different brain areas and plasma of male rats.
Topics: Animals; Apomorphine; Benzazepines; Brain Chemistry; Haloperidol; Hippocampus; Hypothalamus; Male; Oxytocin; Radioimmunoassay; Rats; Rats, Inbred Strains; Sulpiride | 1990 |
Evidence for involvement of 5-HT2 and 5-HT1C receptors in the behavioral effects of the 5-HT agonist 1-(2,5-dimethoxy-4-iodophenyl aminopropane)-2 (DOI).
Topics: Amphetamines; Animals; Body Temperature; Dioxanes; Haloperidol; Male; Methysergide; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Spiro Compounds; Stereotyped Behavior; Sulpiride | 1990 |
Characterization of the dopamine receptor mediating the hyperpolarization of cockroach salivary gland acinar cells in vitro.
Topics: Animals; Benzazepines; Chlorpromazine; Cockroaches; Domperidone; Electric Stimulation; Haloperidol; In Vitro Techniques; Kinetics; Metoclopramide; Receptors, Dopamine; Salivary Glands; Sulpiride | 1990 |
Significance of dopamine receptor antagonists in human postural control.
Topics: Adult; Diazepam; Domperidone; Flupenthixol; Haloperidol; Humans; Muscles; Posture; Proprioception; Receptors, Dopamine; Reflex; Sulpiride | 1990 |
Anxiolytic potential of sulpiride, clozapine and derivatives in the open-field test.
Topics: Animals; Chlordiazepoxide; Clozapine; Defecation; Dibenzazepines; Exploratory Behavior; Haloperidol; Rats; Rats, Inbred Strains; Structure-Activity Relationship; Sulpiride | 1990 |
Effects of dopamine antagonists on neuronal activity related to a delayed response task in monkey prefrontal cortex.
Topics: Animals; Behavior, Animal; Dopamine; Dopamine Antagonists; Fluphenazine; Frontal Lobe; Haloperidol; Male; Neurons; Sulpiride | 1990 |
Characterization of sulpiride-displaceable 3H-YM-09151-2 binding sites in rat frontal cortex and the effects of subchronic treatment with haloperidol on cortical D-2 dopamine receptors.
Topics: Animals; Benzamides; Binding Sites; Corpus Striatum; Dopamine Antagonists; Frontal Lobe; Haloperidol; In Vitro Techniques; Ketanserin; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sulpiride | 1990 |
Neuroleptic treatment induces region-specific changes in levels of neurokinin A and substance P in rat brain.
Topics: Animals; Brain; Cerebral Cortex; Chromatography, High Pressure Liquid; Corpus Striatum; Haloperidol; Male; Nerve Tissue Proteins; Neurokinin A; Nucleus Accumbens; Organ Specificity; Radioimmunoassay; Rats; Rats, Inbred Strains; Substance P; Substantia Nigra; Sulpiride | 1986 |
In vitro characterisation of dopamine receptors in the superior colliculus of the rat.
Topics: Animals; Apomorphine; Binding, Competitive; Butaclamol; Catecholamines; Corpus Striatum; Haloperidol; In Vitro Techniques; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Serotonin; Spiperone; Sulpiride; Superior Colliculi; Synaptosomes | 1987 |
Dopamine receptors on adrenal chromaffin cells modulate calcium uptake and catecholamine release.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenal Glands; Animals; Apomorphine; Butaclamol; Calcium; Calcium Radioisotopes; Catecholamines; Cattle; Cells, Cultured; Chromaffin System; Electric Conductivity; Haloperidol; Ion Channels; Nicotine; Potassium; Receptors, Dopamine; Spiperone; Sulpiride | 1988 |
Evidence for a model of activation of central sigma systems.
Topics: Animals; Benzazepines; Benzomorphans; Butaclamol; Carbazoles; Dopamine Antagonists; Haloperidol; Kinetics; Male; Models, Biological; Motor Activity; Naltrexone; Narcotic Antagonists; Phenazocine; Pyrimidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Sulpiride | 1989 |
Differences in the time course of dopaminergic supersensitivity following chronic administration of haloperidol, molindone, or sulpiride.
Topics: Animals; Corpus Striatum; Haloperidol; In Vitro Techniques; Indoles; Limbic System; Male; Molindone; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereotyped Behavior; Sulpiride | 1989 |
Dopamine D2 receptors exert tonic regulation over discrete neurotensin systems of the rat brain.
Topics: Animals; Corpus Striatum; Haloperidol; Hydroxydopamines; Male; Neurotensin; Nucleus Accumbens; Oxidopamine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Reserpine; Septal Nuclei; Sulpiride | 1989 |
Enhancement of dopamine actions on rat nucleus accumbens neurones in vitro after methamphetamine pre-treatment.
Topics: Action Potentials; Animals; Bucladesine; Calcium; Colforsin; Dopamine; Dose-Response Relationship, Drug; Haloperidol; In Vitro Techniques; Male; Membrane Potentials; Methamphetamine; Nucleus Accumbens; Rats; Rats, Inbred Strains; Receptors, Dopamine; Septal Nuclei; Sulpiride | 1989 |
Status of dopamine in bovine pineal glands and the stimulation of N-acetyltransferase activity by D2-dopaminergic receptor agonists in the rat pineal glands in culture.
Topics: Acetyltransferases; Animals; Cattle; Dopamine; Dopamine Agents; Haloperidol; Melatonin; Norepinephrine; Organ Culture Techniques; Pineal Gland; Rats; Rats, Inbred Strains; Serotonin; Sulpiride | 1989 |
Dopamine D-2 antagonists reverse apomorphine-induced decreased water intake in the rat: prediction of antipsychotic drugs with few extrapyramidal side-effects?
Topics: Animals; Antipsychotic Agents; Apomorphine; Domperidone; Dose-Response Relationship, Drug; Drinking Behavior; Haloperidol; Male; Metoclopramide; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Sulpiride | 1989 |
Functional supersensitivity of the hippocampal dopaminergic system after prolonged treatment with haloperidol.
Topics: Animals; Apomorphine; Dopamine; Dopamine Agents; Ergolines; Haloperidol; Hippocampus; In Vitro Techniques; Male; Neurons; Quinpirole; Rats; Rats, Inbred Strains; Sulpiride; Time Factors | 1989 |
Pharmacological activity profiles of dopamine D-1 and D-2 reception agonists and antagonists on striatal neuronal activity and the response to dexamphetamine in freely moving rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Benzazepines; Corpus Striatum; Dextroamphetamine; Dopamine Agents; Dopamine Antagonists; Ergolines; Haloperidol; Male; Neurons; Quinpirole; Rats; Sulpiride | 1989 |
Definition of the in-vivo binding of [3H]spiperone in rat brain using substituted benzamide drugs.
Topics: Amisulpride; Animals; Apomorphine; Benzamides; Binding, Competitive; Brain Chemistry; Female; Haloperidol; Rats; Rats, Inbred Strains; Spiperone; Stereotyped Behavior; Sulpiride | 1989 |
Dual effects of nicotine on neuroleptic-induced changes of striatal dopamine metabolism in mice.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Antipsychotic Agents; Apomorphine; Body Temperature; Corpus Striatum; Dopamine; Haloperidol; Homovanillic Acid; Male; Mice; Nicotine; Sodium Oxybate; Sulpiride | 1989 |
Differential effects of dopamine receptor antagonists on the sexual behavior of male rats.
Topics: Animals; Antipsychotic Agents; Clozapine; Ejaculation; Female; Haloperidol; Male; Metoclopramide; Pimozide; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sexual Behavior, Animal; Sulpiride | 1989 |
Regional differences in the induction of behavioral supersensitivity by prolonged treatment with atypical neuroleptics.
Topics: Animals; Antipsychotic Agents; Behavior, Animal; Body Weight; Clozapine; Corpus Striatum; Dopamine; Haloperidol; Humans; Injections; Metoclopramide; Motor Activity; Nucleus Accumbens; Rats; Rats, Inbred Strains; Stereotyped Behavior; Sulpiride | 1989 |
Effects of dopaminergic and GABAergic antagonists on methamphetamine-induced locomotor activity in mice selectively bred for their differences in locomotor activity.
Topics: Animals; Bicuculline; Dopamine Agents; GABA Antagonists; Haloperidol; Methamphetamine; Mice; Motor Activity; Sulpiride | 1989 |
Effects of some antipsychotic drugs on cardiovascular catecholamine receptors in the rat.
Topics: Animals; Antipsychotic Agents; Blood Pressure; Chlorpromazine; Haloperidol; Heart Rate; Male; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Dopamine; Sulpiride; Thioridazine; Xylazine | 1989 |
Apomorphine increases plasma oxytocin concentration in male rats.
Topics: Animals; Apomorphine; Benzazepines; Dopamine; Haloperidol; Male; Oxytocin; Pituitary Gland, Posterior; Radioimmunoassay; Rats; Rats, Inbred Strains; Sulpiride | 1989 |
Serotonin release mechanisms in bovine pineal gland: stimulation by norepinephrine and dopamine.
Topics: Animals; Benzazepines; Calcium; Cattle; Clonidine; Dopamine; Dopamine Antagonists; Haloperidol; Isoproterenol; Kinetics; Norepinephrine; Phentolamine; Phenylephrine; Pineal Gland; Prazosin; Propranolol; Serotonin; Sulpiride | 1989 |
Dissociation between biochemical and behavioral recovery in MPTP-treated mice.
Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; 3,4-Dihydroxyphenylacetic Acid; Animals; Benzazepines; Corpus Striatum; Dopamine; Dopamine Antagonists; Drug Interactions; Haloperidol; Male; Mice; Phenylacetates; Psychomotor Performance; Sulpiride; Time Factors | 1989 |
Comparative study of sulpiride and haloperidol on dopamine turnover in the rat brain.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Apomorphine; Brain; Dopamine; Haloperidol; Levodopa; Male; Rats; Rats, Inbred Strains; Sulpiride | 1989 |
[Sulpiride in psychiatric practice].
Topics: Anorexia Nervosa; Bulimia; Haloperidol; Humans; Schizophrenia; Sulpiride | 1989 |
Pharmacology of electrically evoked dopamine release studied in the rat olfactory tubercle by in vivo electrochemistry.
Topics: 3,4-Dihydroxyphenylacetic Acid; Amphetamine; Animals; Apomorphine; Dopamine; Electric Stimulation; Electrochemistry; Electrodes; Haloperidol; Male; Medial Forebrain Bundle; Methylphenidate; Nomifensine; Olfactory Bulb; Rats; Reserpine; Sulpiride | 1989 |
Central dopamine-oxytocin-adrenocorticotropin link in the expression of yawning and penile erection.
Topics: Adrenocorticotropic Hormone; Animals; Animals, Newborn; Apomorphine; Cosyntropin; Dopamine; Dopamine Antagonists; Haloperidol; Hypothalamus; Male; Oxytocin; Penile Erection; Rats; Rats, Inbred Strains; Sodium Glutamate; Sulpiride; Yawning | 1988 |
Effects of DA-1- and DA-2-dopamine antagonists on apomorphine-induced inhibition of peripheral sympathetic neurotransmission.
Topics: Animals; Apomorphine; Blood Pressure; Domperidone; Dopamine Antagonists; Electric Stimulation; Fluphenazine; Haloperidol; Male; Peripheral Nerves; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Sulpiride; Sympathetic Nervous System; Synaptic Transmission; Vasoconstriction | 1988 |
Zetidoline, a novel neuroleptic, activates nigral dopaminergic neurons in rats.
Topics: Animals; Antipsychotic Agents; Apomorphine; Dopamine; Electrophysiology; Haloperidol; Imidazoles; Male; Neurons; Rats; Rats, Inbred Strains; Substantia Nigra; Sulpiride | 1985 |
Dopamine release and metabolism in awake rats after systemic neuroleptics as studied by trans-striatal dialysis.
Topics: 4-Butyrolactone; Animals; Antipsychotic Agents; Basal Metabolism; Consciousness; Dialysis; Dopamine; Drug Interactions; Flupenthixol; Haloperidol; Injections, Subcutaneous; Male; Rats; Sulpiride | 1985 |
Repeated treatment with amitriptyline reduces immobility in the behavioural 'despair' test in rats by activating dopaminergic and beta-adrenergic mechanisms.
Topics: Amitriptyline; Animals; Behavior, Animal; Haloperidol; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Dopamine; Sulpiride | 1985 |
Striatal synaptosomal dopamine synthesis: evidence against direct regulation by an autoreceptor mechanism.
Topics: Animals; Chlorpromazine; Corpus Striatum; Dopamine; Dopamine Antagonists; Haloperidol; Hydroxylation; In Vitro Techniques; Male; Nomifensine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sulpiride; Synaptosomes; Tyrosine 3-Monooxygenase | 1985 |
[Effect of carbidine on the dopamine and serotonin receptors of the central nervous system].
Topics: Animals; Antipsychotic Agents; Brain; Carbolines; Central Nervous System; Haloperidol; Humans; Indoles; Male; Mice; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Serotonin; Spiperone; Stereotyped Behavior; Sulpiride | 1985 |
Sexual excitement and stretching and yawning induced by B-HT 920.
Topics: Adrenergic alpha-Agonists; Animals; Azepines; Behavior, Animal; Haloperidol; Humans; Male; Penis; Prazosin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sexual Behavior, Animal; Stereotyped Behavior; Sulpiride; Yohimbine | 1985 |
Mesolimbic dopamine function is not altered during continuous chronic treatment of rats with typical or atypical neuroleptic drugs.
Topics: Adenylyl Cyclases; Animals; Antipsychotic Agents; Clozapine; Dopamine; Haloperidol; Male; Motor Activity; Nucleus Accumbens; Rats; Rats, Inbred Strains; Receptors, Dopamine; Septal Nuclei; Sulpiride | 1985 |
Rapid tolerance to neuroleptic-induced stimulation of dopamine release in freely moving rats.
Topics: Animals; Antipsychotic Agents; Dopamine; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Tolerance; Flupenthixol; Haloperidol; Injections, Subcutaneous; Male; Rats; Rats, Inbred Strains; Sulpiride; Time Factors | 1985 |
Presynaptic dopamine autoreceptors control tyrosine hydroxylase activation in depolarized striatal dopaminergic terminals.
Topics: Amphetamine; Animals; Bucladesine; Cerebral Cortex; Clozapine; Corpus Striatum; Dopamine; Enzyme Activation; Haloperidol; Hippocampus; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Sulpiride; Synapses; Synaptosomes; Tyrosine 3-Monooxygenase; Veratridine | 1986 |
Differential effect of subchronic treatment with various neuroleptic agents on serotonin2 receptors in rat cerebral cortex.
Topics: 5,7-Dihydroxytryptamine; Animals; Antipsychotic Agents; Cerebral Cortex; Chlorpromazine; Clozapine; Female; Haloperidol; Imipramine; Ketanserin; Loxapine; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Spiperone; Sulpiride | 1986 |
Postsynaptic D1 and D2 dopamine receptors are present in rabbit renal and mesenteric arteries.
Topics: Adenylyl Cyclases; Animals; Benzazepines; Bromocriptine; Fenoldopam; Haloperidol; Hydroxydopamines; Mesenteric Arteries; Oxidopamine; Rabbits; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Renal Artery; Sulpiride | 1985 |
Chronic treatment with five different neuroleptics elicits behavioral supersensitivity to opiate infusion into the nucleus accumbens.
Topics: Animals; Antipsychotic Agents; Enkephalin, Methionine; Flupenthixol; Fluphenazine; Haloperidol; Male; Nucleus Accumbens; Perphenazine; Phenothiazines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Septal Nuclei; Sulpiride; Time Factors | 1986 |
Differential effects of selective and non-selective neuroleptics on intracellular and extracellular cyclic AMP accumulation in rat striatal slices.
Topics: Animals; Antipsychotic Agents; Corpus Striatum; Culture Media; Cyclic AMP; Domperidone; Dopamine; Flupenthixol; Haloperidol; In Vitro Techniques; Male; Rats; Rats, Inbred Strains; Structure-Activity Relationship; Sulpiride | 1985 |
Homovanillic acid in caudate and pre-frontal cortex following acute and chronic neuroleptic administration.
Topics: Animals; Antipsychotic Agents; Caudate Nucleus; Cerebral Cortex; Fluphenazine; Haloperidol; Homovanillic Acid; Male; Rats; Rats, Inbred Strains; Sulpiride; Time Factors | 1986 |
Disinhibitory effects of buspirone and low doses of sulpiride and haloperidol in two experimental anxiety models in rats: possible role of dopamine.
Topics: Animals; Anti-Anxiety Agents; Apomorphine; Behavior, Animal; Buspirone; Drug Interactions; Exploratory Behavior; Haloperidol; Male; Motor Activity; Pyrimidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sulpiride | 1986 |
Enhancing effect of dopamine blockers on evoked acetylcholine release in rat striatal slices: a classical D-2 antagonist response?
Topics: Acetylcholine; Animals; Benzazepines; Chlorpromazine; Corpus Striatum; Domperidone; Dopamine Antagonists; Haloperidol; In Vitro Techniques; Male; Phenothiazines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Sulpiride | 1986 |
Effects of neuroleptic drugs on the inhibition of exploratory behaviour induced by a low dose of apomorphine: implications for the identity of dopamine receptors.
Topics: Animals; Antipsychotic Agents; Apomorphine; Benzazepines; Drug Interactions; Exploratory Behavior; Flupenthixol; Haloperidol; Male; Metoclopramide; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sulpiride | 1986 |
[Comparative study of the pharmacological properties of sultopride sulpiride and other antipsychotic drugs: influence of sultopride, sulpiride and other antipsychotic drugs on spontaneous locomotor activity and changes in locomotor activity induced by apo
Topics: Amisulpride; Animals; Antipsychotic Agents; Apomorphine; Chlorpromazine; Clonidine; Drug Interactions; Haloperidol; Imipramine; Male; Mice; Motor Activity; Pimozide; Sulpiride; Yohimbine | 1986 |
Electrocortical spectrum power effects of different classes of neuroleptics in rats.
Topics: Animals; Antipsychotic Agents; Cerebral Ventricles; Chlorpromazine; Electroencephalography; Haloperidol; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sleep; Sulpiride | 1987 |
Subchronic haloperidol and sulpiride treatment induces region-specific changes in tissue levels of putative amino acid transmitters in rat brain.
Topics: Amino Acids; Animals; Aspartic Acid; Brain; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Glutamine; Haloperidol; Male; Neurotransmitter Agents; Rats; Rats, Inbred Strains; Sulpiride | 1987 |
Pharmacological and biochemical properties of iminodibenzyl antipsychotic drugs including Y-516 and clocapramine.
Topics: Animals; Antipsychotic Agents; Behavior, Animal; Benzazepines; Benzylamines; Dibenzazepines; Haloperidol; Male; Promazine; Rats; Rats, Inbred Strains; Sulpiride | 1986 |
Influence of (-)-sulpiride and YM-09151-2 on stereotyped behavior in chicks and catalepsy in rats.
Topics: Aging; Animals; Antipsychotic Agents; Benzamides; Catalepsy; Chickens; Dextroamphetamine; Fenclonine; Haloperidol; Male; Rats; Rats, Inbred Strains; Stereoisomerism; Stereotyped Behavior; Sulpiride | 1987 |
Piracetam interactions with neuroleptics in psychopharmacological tests.
Topics: Amphetamines; Animals; Antipsychotic Agents; Apomorphine; Behavior, Animal; Drug Interactions; Fluphenazine; Haloperidol; Hypothermia; Male; Mice; Piracetam; Pyrrolidinones; Sulpiride | 1986 |
Blockade by neuroleptics of water intake and operant responding for water in the rat: anhedonia, motor deficit, or both?
Topics: Animals; Antipsychotic Agents; Conditioning, Operant; Consummatory Behavior; Drinking; Haloperidol; Male; Metoclopramide; Motivation; Motor Activity; Rats; Rats, Inbred Strains; Sulpiride | 1987 |
Central D2-dopamine receptor occupancy in schizophrenic patients treated with antipsychotic drugs.
Topics: Adult; Antipsychotic Agents; Brain; Carbon Radioisotopes; Dopamine Antagonists; Female; Haloperidol; Humans; Male; Middle Aged; Nortriptyline; Putamen; Radiography; Receptors, Dopamine; Schizophrenia; Sulpiride; Tomography, Emission-Computed | 1988 |
Stress-induced insomnia: opioid-dopamine interactions.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Appetite Depressants; Benzazepines; gamma-Aminobutyric Acid; Haloperidol; Male; Naloxone; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Opioid; Sleep Deprivation; Sleep Initiation and Maintenance Disorders; Sleep, REM; Stress, Psychological; Sulpiride | 1987 |
Neuroleptic effects on platelet aggregation: a study in normal volunteers and schizophrenics.
Topics: Adolescent; Adult; Antipsychotic Agents; Chlorpromazine; Delayed-Action Preparations; Flupenthixol; Fluphenazine; Haloperidol; Humans; Male; Platelet Aggregation; Procyclidine; Schizophrenia; Sulpiride; Trifluoperazine | 1987 |
Desenkephalin-gamma-endorphin and neuroleptics counteract the DP-7-ATN-induced hypomotility after intra-accumbens treatment.
Topics: Animals; Antipsychotic Agents; beta-Endorphin; Haloperidol; Injections; Male; Motor Activity; Naphthalenes; Nucleus Accumbens; Rats; Rats, Inbred Strains; Sulpiride; Tetrahydronaphthalenes | 1988 |
Pisa syndrome. Report of a case.
Topics: Adult; Amisulpride; Antipsychotic Agents; Dyskinesia, Drug-Induced; Haloperidol; Humans; Male; Schizophrenia; Sulpiride; Syndrome | 1988 |
Influence of D-1 receptor system on the D-2 receptor-mediated hypothermic response in mice.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Anti-Anxiety Agents; Apomorphine; Benzamides; Benzazepines; Dopamine; Dopamine Antagonists; Ergolines; Haloperidol; Hypothermia; Male; Mice; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Sulpiride | 1988 |
Blockade of brain dopamine receptors antagonizes the anti-immobility effect of MIF-1 and Tyr-MIF-1 in rats.
Topics: Animals; Antidepressive Agents; Behavior, Animal; Depression; Haloperidol; Immobilization; Male; MSH Release-Inhibiting Hormone; Rats; Receptors, Dopamine; Sulpiride | 1988 |
Effects of locally applied D-1 and D-2 receptor agonists and antagonists studied with brain dialysis.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Azepines; Benzazepines; Brain; Dialysis; Dopamine; Dopamine Agents; Dopamine Antagonists; Ergolines; Haloperidol; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sulpiride | 1988 |
Definition of the in-vivo accumulation of [3H]spiperone in brain using haloperidol and sulpiride to determine functional dopamine receptor occupation.
Topics: Animals; Apomorphine; Brain Chemistry; Corpus Striatum; Female; Haloperidol; Homovanillic Acid; Limbic System; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Sulpiride | 1988 |
Potency of antipsychotics in reversing the effects of a hallucinogenic drug on locus coeruleus neurons correlates with 5-HT2 binding affinity.
Topics: Amphetamines; Animals; Antipsychotic Agents; Chlorpromazine; Clozapine; DOM 2,5-Dimethoxy-4-Methylamphetamine; Electric Stimulation; Evoked Potentials; Haloperidol; Locus Coeruleus; Male; Neurons; Rats; Rats, Inbred Strains; Receptors, Serotonin; Sciatic Nerve; Spiperone; Sulpiride | 1988 |
[3H]SCH 23390 binding sites increase after chronic blockade of D-1 dopamine receptors.
Topics: Adenylyl Cyclases; Animals; Benzazepines; Binding Sites; Haloperidol; In Vitro Techniques; Kinetics; Male; Membranes; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Sulpiride | 1985 |
D-2 selective receptor antagonists suppress sucrose sham feeding in the rat.
Topics: Amisulpride; Animals; Feeding Behavior; Food Deprivation; Haloperidol; Male; Pimozide; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Reward; Stereoisomerism; Sucrose; Sulpiride; Taste; Water Deprivation | 1986 |
Involvement of dopamine receptor subtypes in dopaminergic modulation of aldosterone secretion in rats.
Topics: Aldosterone; Animals; Blood; Domperidone; Dopamine; Haloperidol; Male; Metoclopramide; Osmolar Concentration; Potassium; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Sodium; Sulpiride | 1987 |
Differential effects of dopamine D-1 and D-2 receptor agonists on EEG activity and behaviour in the rabbit.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Behavior, Animal; Benzazepines; Electroencephalography; Ergolines; Haloperidol; Male; Quinpirole; Rabbits; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Stereotyped Behavior; Sulpiride | 1987 |
Effects of human atrial natriuretic polypeptide on pancreatic exocrine secretion in the dog.
Topics: Animals; Atrial Natriuretic Factor; Atropine; Bicarbonates; Cimetidine; Dogs; Ethacrynic Acid; Female; Haloperidol; Injections, Intra-Arterial; Male; Pancreatic Juice; Pancreatin; Perfusion; Phentolamine; Propranolol; Proteins; Secretin; Sodium; Sulpiride | 1987 |
Comparison of the effects of dopamine D1 and D2 receptor antagonists on rat striatal, limbic and nigral dopamine synthesis and utilisation.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Benzamides; Benzazepines; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Haloperidol; Homovanillic Acid; Male; Olfactory Bulb; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Remoxipride; Substantia Nigra; Sulpiride | 1987 |
Excitatory and inhibitory action of dopamine on hippocampal neurons in vitro. Involvement of D2 and D1 receptors.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Culture Techniques; Dopamine; Dopamine Antagonists; Haloperidol; Hippocampus; Male; Neurons; Pergolide; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Sulpiride | 1987 |
Blockade of D-1 dopamine receptors by SCH 23390 prevents EEG and behavioral activation induced by L-dopa.
Topics: Animals; Behavior, Animal; Benzazepines; Electroencephalography; Haloperidol; Levodopa; Male; Rabbits; Receptors, Dopamine; Receptors, Dopamine D1; Sulpiride | 1987 |
Potential antidepressant properties of 8-hydroxy-2-(di-n-propylamino)tetralin, a selective serotonin1A receptor agonist.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Drug Interactions; Haloperidol; Male; Methiothepin; Naphthalenes; Physical Exertion; Rats; Receptors, Serotonin; Serotonin; Sulpiride; Swimming; Tetrahydronaphthalenes | 1987 |
Dopamine D1 receptors in the nucleus accumbens: involvement in the reinforcing effect of tegmental stimulation.
Topics: Animals; Benzazepines; Conditioning, Operant; Dopamine Antagonists; Electric Stimulation; Haloperidol; Male; Nucleus Accumbens; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Reinforcement, Psychology; Septal Nuclei; Sulpiride | 1988 |
Inhibition of the electrically evoked release of [3H]acetylcholine in rat striatal slices: an experimental model for drugs that enhance dopaminergic neurotransmission.
Topics: Acetylcholine; Amphetamine; Animals; Chlorpromazine; Clozapine; Cocaine; Corpus Striatum; Dopamine; Electric Stimulation; Haloperidol; Male; Nomifensine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sulpiride; Synaptic Transmission | 1985 |
Jejunal-ileal differences in dopaminergic but not alpha-adrenergic antisecretory effects.
Topics: Animals; Apomorphine; Bucladesine; Clonidine; Haloperidol; Ileum; Intestinal Absorption; Jejunum; Male; Phentolamine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Dopamine; Sulpiride; Water-Electrolyte Balance | 1985 |
Modulation of the endogenous acetylcholine release from rat striatal slices.
Topics: Acetylcholine; Animals; Apomorphine; Corpus Striatum; Dopamine; Haloperidol; In Vitro Techniques; Male; Potassium; Rats; Rats, Inbred Strains; Sulpiride; Synaptic Transmission | 1985 |
Effects of ventro-medial mesencephalic tegmentum (VMT) stimulation on the spontaneous activity of nucleus accumbens neurones: influence of the dopamine system.
Topics: Animals; Dopamine; Electric Stimulation; Haloperidol; Hydroxydopamines; Male; Neural Inhibition; Neural Pathways; Nucleus Accumbens; Oxidopamine; Rats; Rats, Inbred Strains; Septal Nuclei; Sulpiride; Synaptic Transmission; Tegmentum Mesencephali | 1986 |
Catecholamine receptors involved in the inhibitory effects of dopamine on vagally stimulated gastric acid secretion and mucosal blood flow in rats.
Topics: Animals; Domperidone; Dopamine; Gastric Acid; Gastric Mucosa; Haloperidol; Male; Metoclopramide; Phentolamine; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Catecholamine; Regional Blood Flow; Sulpiride; Vagus Nerve | 1987 |
Autoradiographic distribution of non-dopaminergic binding sites labeled by [3H]haloperidol in rat brain.
Topics: Animals; Autoradiography; Benzazepines; Binding, Competitive; Brain; Haloperidol; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Opioid; Receptors, sigma; Spiperone; Sulpiride | 1987 |
Levels of insulin in the brains of rats modified by chronic administration of amphetamine, haloperidol and sulpiride.
Topics: Amphetamine; Animals; Brain; Female; Haloperidol; Insulin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sulpiride | 1988 |
Effects of haloperidol, sulpiride and SCH 23390 on passive avoidance learning in mice.
Topics: Animals; Avoidance Learning; Benzazepines; Electroshock; Haloperidol; Male; Memory; Mice; Motor Activity; Sulpiride | 1988 |
Dopaminergic inhibition of tyrosinase activity in hair follicular melanocytes of the mouse.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Aging; Animals; Benzazepines; Bromocriptine; Catechol Oxidase; Depression, Chemical; Dopamine; Ergolines; Female; Hair; Haloperidol; Male; Melanocytes; Mice; Mice, Inbred C3H; Monophenol Monooxygenase; Quinpirole; Skin; Spiperone; Sulpiride | 1986 |
Psychopharmacological investigations of a lead-induced long-term cognitive deficit in monkeys.
Topics: Acetylcholine; Amphetamine; Animals; Behavior, Animal; Cognition Disorders; Dopamine; Haloperidol; Lead Poisoning; Levodopa; Macaca mulatta; Physostigmine; Scopolamine; Sulpiride | 1987 |
Differential alteration of striatal D-1 and D-2 receptors induced by the long-term administration of haloperidol, sulpiride or clozapine to rats.
Topics: Animals; Apomorphine; Clozapine; Corpus Striatum; Dibenzazepines; Dose-Response Relationship, Drug; Haloperidol; Humans; Kinetics; Long-Term Care; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Stereotyped Behavior; Sulpiride; Thioxanthenes | 1985 |
Opposite effects induced by low and high doses of apomorphine on single-trial passive avoidance learning in mice.
Topics: Animals; Apomorphine; Avoidance Learning; Dose-Response Relationship, Drug; Haloperidol; Male; Mice; Mice, Inbred Strains; Retention, Psychology; Sulpiride; Vocalization, Animal | 1988 |
The effects of haloperidol and sulpiride on apomorphine-induced locomotor activity in rats.
Topics: Animals; Apomorphine; Haloperidol; Male; Motor Activity; Rats; Rats, Inbred Strains; Sulpiride | 1988 |
[Difference in mechanism of action of sulpiride and haloperidol on dopamine brain turnover].
Topics: Animals; Brain; Dopamine; Haloperidol; Levodopa; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sulpiride | 1988 |
The effect of acute and prolonged treatment with citalopram on the action of dopamine and SKF 38393 in rat hippocampal slices.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antidepressive Agents; Appetite Depressants; Benzazepines; Citalopram; Dopamine; Ergolines; Haloperidol; Hippocampus; In Vitro Techniques; Male; Motor Activity; Neurons; Propylamines; Quinpirole; Rats; Rats, Inbred Strains; Sulpiride | 1988 |
Quinpirole hydrochloride, a potential anti-parkinsonism drug.
Topics: Animals; Benzazepines; Corpus Striatum; Dogs; Dose-Response Relationship, Drug; Ergolines; Grooming; Haloperidol; Male; Motor Activity; Parkinson Disease; Quinpirole; Rats; Rats, Inbred Strains; Spiperone; Stereotyped Behavior; Sulpiride | 1987 |
Elevation of plasma prolactin concentrations by intravenous SCH 23390 and SKF 38393 in conscious rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Haloperidol; Injections, Intravenous; Male; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sulpiride | 1987 |
Reduction of the rewarding effect of brain stimulation by a blockade of dopamine D1 receptor with SCH 23390.
Topics: Animals; Benzazepines; Brain; Brain Mapping; Haloperidol; Hypothalamic Area, Lateral; Male; Raphe Nuclei; Rats; Receptors, Dopamine; Reward; Self Stimulation; Sulpiride; Tegmentum Mesencephali | 1986 |
3H-SCH 23390 binding sites in the rat substantia nigra: evidence for a presynaptic localization and innervation by dopamine.
Topics: Animals; Benzazepines; Dopamine; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Haloperidol; Kainic Acid; Male; Membranes; Rats; Receptors, Dopamine; Substantia Nigra; Sulpiride; Synapses | 1986 |
Characterization of dopamine receptors associated with aldosterone secretion in rat adrenal glomerulosa.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Adrenal Cortex; Aldosterone; Animals; Benzazepines; Bromocriptine; Dihydroergotoxine; Haloperidol; Lisuride; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism; Sulpiride | 1986 |
Induction of turning by direct intrastriatal injection of dopaminomimetic drugs in mice: pharmacological analysis of a simple screening model.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Bromocriptine; Dextroamphetamine; Dopamine; Female; Haloperidol; Mice; Nomifensine; Posture; Pyridazines; Stereotyped Behavior; Sulpiride; Time Factors | 1986 |
Dopamine receptor-mediated spinal antinociception in the normal and haloperidol pretreated rat: effects of sulpiride and SCH 23390.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Benzofurans; Dopamine Antagonists; Haloperidol; Male; Pain; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spinal Cord; Sulpiride | 1987 |
Chronic autoreceptor blockade and neuroleptic-induced dopamine receptor hypersensitivity.
Topics: Animals; Apomorphine; Dose-Response Relationship, Drug; Haloperidol; Male; Metoclopramide; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereotyped Behavior; Sulpiride; Synapses | 1987 |
Effects of repeated tiapride administration on anterior pituitary dopamine receptors and prolactin release in the rat.
Topics: Animals; Benzamides; Corpus Striatum; Dose-Response Relationship, Drug; Haloperidol; Male; Pituitary Gland, Anterior; Prolactin; Rats; Receptors, Dopamine; Secretory Rate; Sulpiride; Tiapamil Hydrochloride; Time Factors | 1987 |
The hypomotility elicited by small doses of apomorphine seems exclusively mediated by dopaminergic systems in the nucleus accumbens.
Topics: Analysis of Variance; Animals; Apomorphine; beta-Endorphin; Endorphins; Haloperidol; Male; Motor Activity; Nucleus Accumbens; Rats; Rats, Inbred Strains; Receptors, Dopamine; Septal Nuclei; Stereotyped Behavior; Sulpiride | 1987 |
Effect of long-term dosing with tiapride on brain dopamine receptors and metabolism in rats. Comparative study with sulpiride and haloperidol.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Antiparkinson Agents; Apomorphine; Benzamides; Brain Chemistry; Dopamine; Haloperidol; Homovanillic Acid; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Sulpiride; Tiapamil Hydrochloride | 1987 |
Apomorphine enantiomers' effects on dopamine metabolism: receptor and non-receptor related actions.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Apomorphine; Biopterins; Corpus Striatum; Dopamine; Haloperidol; Homovanillic Acid; Male; Pterins; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism; Sulpiride; Synaptosomes | 1986 |
Effects of dopamine and its agonists and antagonists on the receptive field properties of ganglion cells in the rabbit retina.
Topics: Action Potentials; Animals; Apomorphine; Dopamine; Dopamine Antagonists; Flupenthixol; Fluphenazine; Haloperidol; Photic Stimulation; Rabbits; Reaction Time; Receptors, Dopamine; Retina; Retinal Ganglion Cells; Sulpiride; Visual Fields | 1986 |
Differential alterations in striatal acetylcholine function in rats during 12 months' continuous administration of haloperidol, sulpiride, or clozapine.
Topics: Acetylcholine; Acetylcholinesterase; Animals; Choline O-Acetyltransferase; Clozapine; Corpus Striatum; Dibenzazepines; Dyskinesia, Drug-Induced; Haloperidol; Male; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Sulpiride | 1986 |
Survival time in hypoxic mice: differentiation between apomorphine-induced hypothermia and antihypoxic properties.
Topics: Animals; Apomorphine; Body Temperature; Domperidone; Drug Interactions; Female; Haloperidol; Hypoxia; Mice; Social Isolation; Sulpiride | 1986 |
In vivo voltammetric measurement of extracellular DOPAC levels in the anteromedial prefrontal cortex of the rat.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Benzylamines; Bis(4-Methyl-1-Homopiperazinylthiocarbonyl)disulfide; Electrochemistry; Frontal Lobe; Haloperidol; Male; Phenylacetates; Rats; Rats, Inbred Strains; Sulpiride | 1986 |
Effect of lead exposure on dopaminergic receptors in rat striatum and nucleus accumbens.
Topics: Adenylyl Cyclases; Animals; Binding, Competitive; Corpus Striatum; Female; Haloperidol; Lead Poisoning; Male; Nucleus Accumbens; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Rats, Inbred Strains; Receptors, Dopamine; Septal Nuclei; Spiperone; Sulpiride | 1986 |
Comparison of effects of tiapride and sulpiride on D-1, D-2, D-3 and D-4 subtypes of dopamine receptors in rat striatal and bovine caudate nucleus membranes.
Topics: Animals; Benzamides; Caudate Nucleus; Corpus Striatum; Dopamine; Haloperidol; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sulpiride; Tiapamil Hydrochloride | 1986 |
Hyperprolactinaemia does not alter specific striatal 3H-spiperone binding in the rat.
Topics: Animals; Corpus Striatum; Dopamine; Haloperidol; In Vitro Techniques; Male; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Sulpiride; Tritium | 1986 |
Effects of subchronic haloperidol and sulpiride on regional brain dopamine metabolism in the rat.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Brain; Dopamine; Haloperidol; Homovanillic Acid; Male; Rats; Rats, Inbred Strains; Sulpiride; Tissue Distribution | 1986 |
Dissociated effects of apomorphine on various nociceptive responses in mice.
Topics: Analgesics; Animals; Apomorphine; Body Temperature; Domperidone; Dopamine; Haloperidol; Male; Mice; Naloxone; Pain Measurement; Sulpiride | 1986 |
Presynaptic dopamine receptors in the pithed rat: characterization with apomorphine and comparison with central dopamine autoreceptors.
Topics: Animals; Apomorphine; Atropine; Decerebrate State; Electric Stimulation; Haloperidol; Hemodynamics; Male; Motor Activity; Phenylephrine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sulpiride; Yohimbine | 1986 |
Alterations in cerebral glutamic acid decarboxylase and 3H-flunitrazepam binding during continuous treatment of rats for up to 1 year with haloperidol, sulpiride or clozapine.
Topics: Animals; Body Weight; Brain; Clozapine; Flunitrazepam; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Haloperidol; Kinetics; Male; Psychotropic Drugs; Rats; Rats, Inbred Strains; Sulpiride; Time Factors | 1987 |
Characteristics of receptors for dopamine in the pars intermedia of the amphibian Xenopus laevis.
Topics: Animals; Apomorphine; Benzamides; Domperidone; Dopamine; Drug Interactions; Ergolines; Haloperidol; Melanocyte-Stimulating Hormones; Pituitary Gland, Anterior; Quinpirole; Receptors, Dopamine; Sulpiride; Xenopus laevis | 1986 |
Effects of neuroleptics on dopamine release from striatal slices.
Topics: Animals; Chlorpromazine; Corpus Striatum; Dopamine; Haloperidol; In Vitro Techniques; Male; Methamphetamine; Psychotropic Drugs; Rats; Rats, Inbred Strains; Sulpiride | 1985 |
Classification of sulpiride, clozapine and haloperidol by toposelective recording from different brain structures in the immobilized rat (stereo-EEG).
Topics: Animals; Brain; Clozapine; Corpus Striatum; Dibenzazepines; Electroencephalography; Haloperidol; Male; Motor Cortex; Rats; Reticular Formation; Somatosensory Cortex; Sulpiride | 1985 |
Dopaminergic agents including 3-PPP and its enantiomers on medial septal self-stimulation.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Appetite Depressants; Benzazepines; Dextroamphetamine; Drug Interactions; Haloperidol; Male; Nomifensine; Piperidines; Rats; Receptors, Dopamine; Self Stimulation; Stereoisomerism; Sulpiride; Tetrahydronaphthalenes | 1985 |
Dopamine receptor blockade increases glandular kallikrein-like activity in the neurointermediate lobe of the rat pituitary.
Topics: Animals; Haloperidol; Kallikreins; Male; Peptide Hydrolases; Perphenazine; Pituitary Gland; Promethazine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sulpiride | 1985 |
SCH 23390, a selective dopamine D1 antagonist, activates dopamine neurons but fails to prevent their inhibition by apomorphine.
Topics: Action Potentials; Animals; Apomorphine; Benzazepines; Haloperidol; Male; Neurons; Rats; Receptors, Dopamine; Substantia Nigra; Sulpiride | 1985 |
Brain cortex phosphatidylserine inhibits phosphatidylinositol turnover in rat anterior pituitary glands.
Topics: Animals; Cattle; Cerebral Cortex; Dopamine; Female; Haloperidol; In Vitro Techniques; Kinetics; Phosphatidylinositols; Phosphatidylserines; Phosphorus Radioisotopes; Pimozide; Pituitary Gland, Anterior; Rats; Rats, Inbred Strains; Sulpiride; Thyrotropin-Releasing Hormone | 1985 |
Dopamine agonist action in mesolimbic, cortical and extrapyramidal areas to modify spontaneous climbing behaviour of the mouse.
Topics: Animals; Apomorphine; Cerebral Cortex; Dopamine; Dose-Response Relationship, Drug; Extrapyramidal Tracts; Female; Haloperidol; Limbic System; Mice; Motor Activity; Prazosin; Sulpiride; Yohimbine | 1985 |
Lipid peroxidation as a possible mechanism for the neurotoxic and nephrotoxic effects of a combination of lithium carbonate and haloperidol.
Topics: Animals; Cerebral Cortex; Drug Interactions; Haloperidol; In Vitro Techniques; Kidney; Lipid Peroxides; Lithium; Lithium Carbonate; Male; Rats; Rats, Inbred Strains; Sulpiride; Synaptosomes; Time Factors | 1985 |
The conditioned place preference paradigm in rats: effect of bupropion.
Topics: Animals; Bupropion; Conditioning, Psychological; Haloperidol; Male; Motor Activity; Propiophenones; Rats; Sulpiride | 1985 |
Dopamine receptors mediating yawning: are they autoreceptors?
Topics: Animals; Domperidone; Drug Synergism; Haloperidol; Male; Methyltyrosines; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reflex; Reserpine; Stereoisomerism; Sulpiride | 1986 |
Evidence of dopamine involvement in the effect of repeated treatment with various antidepressants in the behavioural 'despair' test in rats.
Topics: Animals; Antidepressive Agents; Antidepressive Agents, Tricyclic; Behavior, Animal; Dibenzocycloheptenes; Haloperidol; Male; Motor Activity; Nomifensine; Rats; Receptors, Dopamine; Sulpiride | 1985 |
The role of dopamine in the formation of gastric ulcers in rats.
Topics: Animals; Apomorphine; Bromocriptine; Domperidone; Dopamine; Female; Haloperidol; Levodopa; Male; Rats; Rats, Inbred Strains; Stomach Ulcer; Sulpiride | 1985 |
Effect of haloperidol and sulpiride on dopamine metabolism in nucleus accumbens and olfactory tubercle: a study by in vivo voltammetry.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Catechols; Chloral Hydrate; Dopamine; Drug Interactions; Electrochemistry; Haloperidol; Male; Nucleus Accumbens; Olfactory Bulb; Rats; Rats, Inbred Strains; Septal Nuclei; Sulpiride | 1985 |
Side effects of drugs stimulating prolactin secretion on the behavior of male rats.
Topics: Animals; Domperidone; Haloperidol; Male; Motor Activity; Pituitary Gland; Prolactin; Rats; Rats, Inbred Strains; Sexual Behavior, Animal; Sulpiride | 1985 |
[Three cases of lingual ballistic movement followed by a rigid-dystonic state of the tongue].
Topics: Aged; Basal Ganglia Diseases; Dyskinesia, Drug-Induced; Female; Haloperidol; Humans; Male; Movement Disorders; Sulpiride; Tongue | 1985 |
Simultaneous catalepsy and apomorphine-induced stereotypic behavior in mice.
Topics: Animals; Apomorphine; Catalepsy; Chlorpromazine; Domperidone; Drug Interactions; Haloperidol; Injections, Intraventricular; Mice; Spiperone; Stereotyped Behavior; Sulpiride | 1985 |
Antipsychotic drugs stimulate prolactin release.
Topics: Animals; Chlorpromazine; Dopamine; Female; Fluphenazine; Haloperidol; Male; Phenothiazines; Pimozide; Prolactin; Promethazine; Rats; Receptors, Drug; Sex Factors; Stimulation, Chemical; Sulpiride; Thiethylperazine; Thioridazine; Tranquilizing Agents | 1974 |
Effect of neuroleptic drugs on striatal dopamine release and metabolism in the awake rat studied by intracerebral dialysis.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Antipsychotic Agents; Catalepsy; Corpus Striatum; Dialysis; Dopamine; Flupenthixol; Haloperidol; Homovanillic Acid; Humans; Hydroxyindoleacetic Acid; In Vitro Techniques; Male; Rats; Rats, Inbred Strains; Sulpiride | 1984 |
Regulation of tyrosine hydroxylase after chronic treatment with classic and atypical antischizophrenic drugs.
Topics: Animals; Antipsychotic Agents; Brain; Clozapine; Corpus Striatum; Haloperidol; Male; Nucleus Accumbens; Rats; Sulpiride; Time Factors; Tyrosine 3-Monooxygenase | 1980 |
Morphological changes of pigeon crop-sac mucosa and pituitary lactotrophs after systemic and intraventricular administration of neuroleptic drugs.
Topics: Animals; Antipsychotic Agents; Clozapine; Columbidae; Crop, Avian; Female; Haloperidol; Mucous Membrane; Pituitary Gland, Anterior; Prolactin; Reserpine; Sulpiride | 1980 |
Distal colon motility in schizophrenic patients.
Topics: Adolescent; Adrenergic alpha-Antagonists; Adult; Aged; Colon; Dopamine; Female; Gastrointestinal Motility; Haloperidol; Humans; Male; Middle Aged; Norepinephrine; Schizophrenia; Sulpiride; Sympathetic Nervous System | 1980 |
Neuroleptic properties of cis-N-(1-benzyl-2-methylpyrrolidin-3-yl)-5-chloro-2-methoxy-4-methylaminobenzamide (YM-09151-2) with selective antidopaminergic activity.
Topics: Animals; Antipsychotic Agents; Apomorphine; Benzamides; Chlorpropamide; Dogs; Drug Evaluation, Preclinical; Female; Haloperidol; Humans; Hypothermia; Male; Methamphetamine; Mice; Mice, Inbred ICR; Receptors, Dopamine; Stereotyped Behavior; Sulpiride; Vomiting | 1981 |
Hypophysectomy does not prevent development of striatal dopamine receptor supersensitivity induced by repeated neuroleptic treatment.
Topics: Animals; Antipsychotic Agents; Corpus Striatum; Drug Resistance; Haloperidol; Humans; Hypophysectomy; Luteinizing Hormone; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Sulpiride | 1981 |
Increase of dopamine synthesis in synaptosomes from rats treated with neuroleptics or reserpine.
Topics: 4-Butyrolactone; Animals; Antipsychotic Agents; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Haloperidol; Kinetics; Male; Rats; Rats, Inbred Strains; Reserpine; Sulpiride; Synaptosomes; Temperature; Tyrosine 3-Monooxygenase | 1982 |
Neuroleptic versus antidepressant activity of sulpiride isomers in the rat.
Topics: Animals; Antidepressive Agents; Antipsychotic Agents; Apomorphine; Behavior, Animal; Depression; Exploratory Behavior; Haloperidol; Humans; Male; Motor Activity; Rats; Rats, Inbred Strains; Stereoisomerism; Sulpiride | 1982 |
Phentolamine inhibition of rat seminal vesicle response to dopamine-mimetic drugs: alpha-adrenoceptor implication or lack of specificity?
Topics: Animals; Apomorphine; Carbachol; Catecholamines; Dopamine; Haloperidol; Imidazolines; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Phentolamine; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Seminal Vesicles; Sulpiride | 1982 |
Differential blocking effects of several dopamine receptor antagonists for peripheral pre- and postsynaptic dopamine receptors in the anesthetized dog.
Topics: Anesthesia; Animals; Aporphines; Dinoprostone; Dogs; Epinephrine; Haloperidol; Heart Rate; In Vitro Techniques; Nictitating Membrane; Prostaglandins E; Receptors, Dopamine; Sulpiride; Synapses; Yohimbine | 1982 |
Dopamine autoreceptor and postsynaptic receptor blocking potency of neuroleptics.
Topics: Animals; Antipsychotic Agents; Apomorphine; Fluphenazine; Haloperidol; Male; Metoclopramide; Mice; Molindone; Motor Activity; Receptors, Dopamine; Sulpiride; Synapses | 1982 |
Evaluation of peripheral dopamine receptor and alpha-adrenoceptor blocking activity of sulpiride.
Topics: Adrenergic alpha-Antagonists; Animals; Aporphines; Dogs; Electric Stimulation; Female; Haloperidol; Heart Rate; Male; Pimozide; Receptors, Dopamine; Sulpiride; Sympathetic Nervous System; Synaptic Transmission | 1982 |
[Suppressive effects of lisuride on the synthesis, release and metabolism of dopamine in rat brain].
Topics: Animals; Apomorphine; Brain; Depression, Chemical; Dihydroergotoxine; Dopamine; Ergolines; Female; Haloperidol; Histocytochemistry; Homovanillic Acid; Lisuride; Metoclopramide; Nucleus Accumbens; Olfactory Bulb; Rats; Sulpiride; Tyrosine 3-Monooxygenase | 1982 |
Optic tectum adenylate cyclase activity from goldfish (Carassius auratus) as a model to assess dopamine receptor agonists and antagonists.
Topics: Adenylyl Cyclases; Animals; Chlorpromazine; Cyclic AMP; Cyprinidae; Dose-Response Relationship, Drug; Goldfish; Haloperidol; Models, Biological; Neurotransmitter Agents; Phentolamine; Propranolol; Receptors, Dopamine; Sulpiride; Superior Colliculi | 1983 |
(-)-Sulpiride activates the firing rate and tyrosine hydroxylase activity of dopaminergic neurons in unanesthetized rats.
Topics: Animals; Apomorphine; Dopamine; Electric Stimulation; Evoked Potentials; Haloperidol; Isomerism; Male; Neurons; Rats; Rats, Inbred Strains; Substantia Nigra; Sulpiride; Tyrosine 3-Monooxygenase | 1983 |
Buspirone: a potential atypical neuroleptic.
Topics: Animals; Antipsychotic Agents; Buspirone; Clozapine; Dopamine; Dose-Response Relationship, Drug; Haloperidol; Male; Pyrimidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Substantia Nigra; Sulpiride; Time Factors | 1983 |
Long-term adaptive changes in striatal dopamine function in response to chronic neuroleptic intake in rats.
Topics: Acetylcholine; Animals; Antipsychotic Agents; Apomorphine; Corpus Striatum; Glutamates; Glutamic Acid; Haloperidol; Rats; Receptors, Dopamine; Spiperone; Sulpiride | 1983 |
Changes in apomorphine-induced stereotypy as a result of subacute neuroleptic treatment correlates with increased D-2 receptors, but not with increases in D-1 receptors.
Topics: Animals; Antipsychotic Agents; Apomorphine; Brain; Drug Synergism; Flupenthixol; Haloperidol; Humans; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Stereotyped Behavior; Sulpiride; Thioxanthenes | 1983 |
Effect of repeated treatment with desipramine in the behavioral "despair" test in rats: antagonism by "atypical" but not "classical" neuroleptics or antiadrenergic drugs.
Topics: Adrenergic alpha-Antagonists; Animals; Antipsychotic Agents; Butyrophenones; Chlorpromazine; Clonidine; Clozapine; Depressive Disorder; Desipramine; Dibenzazepines; Haloperidol; Humans; Male; Metoclopramide; Phentolamine; Prazosin; Propranolol; Rats; Sulpiride | 1984 |
A comparison of the effects of acute and one year's continuous neuroleptic treatment on the release of [3H]glutamate and [3H]acetylcholine from rat striatal slices.
Topics: Acetylcholine; Animals; Antipsychotic Agents; Calcium; Clozapine; Corpus Striatum; Dopamine; Glutamates; Glutamic Acid; Haloperidol; In Vitro Techniques; Male; Potassium; Rats; Rats, Inbred Strains; Sulpiride; Trifluoperazine | 1984 |
Effects of dopamine and dopamine antagonists on postprandial release of pancreatic polypeptide in dogs and in healthy volunteers.
Topics: Adrenergic beta-Antagonists; Adult; Animals; Dogs; Dopamine; Female; Food; Haloperidol; Humans; Male; Pancreatic Polypeptide; Phentolamine; Propranolol; Receptors, Dopamine; Sulpiride | 1983 |
[Long-term use of 200 mg Dogmatil. Apropos of 13 cases].
Topics: Adult; Amitriptyline; Antipsychotic Agents; Bipolar Disorder; Borderline Personality Disorder; Drug Evaluation; Drug Therapy, Combination; Female; Haloperidol; Humans; Male; Middle Aged; Neurotic Disorders; Paranoid Disorders; Schizophrenia; Sulpiride; Time Factors; Trifluperidol; Trimipramine | 1984 |
The actions of antipsychotic drugs on dopamine receptors in the rat substantia nigra.
Topics: Action Potentials; Animals; Antipsychotic Agents; Dopamine; Dopamine Antagonists; Flupenthixol; Haloperidol; In Vitro Techniques; Male; Neurons; Rats; Receptors, Dopamine; Stereoisomerism; Substantia Nigra; Sulpiride | 1984 |
Effects of antipsychotic drugs on the long-term effects of amphetamine on nigro-striatal dopamine neurons in iprindole-treated rats.
Topics: Analysis of Variance; Animals; Antipsychotic Agents; Behavior, Animal; Brain; Clozapine; Corpus Striatum; Dextroamphetamine; Dopamine; Haloperidol; Indoles; Iprindole; Male; Methyltyrosines; Neurons; Rats; Rats, Inbred Strains; Sulpiride | 1984 |
Long-term consequences of antagonism by neuroleptics of behavioural events occurring during mesolimbic dopamine infusion.
Topics: Animals; Antiparkinson Agents; Antipsychotic Agents; Apomorphine; Dopamine; Dopamine Antagonists; Female; Haloperidol; Injections; Methysergide; Motor Activity; Nucleus Accumbens; Rats; Rats, Inbred Strains; Septal Nuclei; Sulpiride; Time Factors | 1984 |
Antidepressant versus neuroleptic activities of sulpiride isomers on four animal models of depression.
Topics: Animals; Antidepressive Agents; Antipsychotic Agents; Apomorphine; Behavior, Animal; Body Temperature; Depressive Disorder; Desipramine; Haloperidol; Helplessness, Learned; Humans; Hypnotics and Sedatives; Male; Rats; Rats, Inbred Strains; Stereoisomerism; Sulpiride | 1984 |
Discriminative stimulus properties of lergotrile.
Topics: Animals; Apomorphine; Discrimination Learning; Dose-Response Relationship, Drug; Ergolines; Ergonovine; Haloperidol; Lisuride; Lysergic Acid Diethylamide; Male; Piperidines; Pizotyline; Quipazine; Rats; Rats, Inbred Strains; Sulpiride | 1984 |
Remoxipride, a new potential antipsychotic compound with selective antidopaminergic actions in the rat brain.
Topics: Adenylyl Cyclases; Animals; Antipsychotic Agents; Apomorphine; Behavior, Animal; Benzamides; Binding, Competitive; Brain Chemistry; Catalepsy; Chlorpromazine; Dogs; Female; Haloperidol; Histocytochemistry; Humans; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Remoxipride; Spiperone; Sulpiride; Thioridazine; Vomiting | 1984 |
[Changes in the number of benzodiazepine receptors in different parts of the brain of rats after neuroleptic withdrawal].
Topics: Animals; Antipsychotic Agents; Brain; Clozapine; Flunitrazepam; Haloperidol; Humans; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substance Withdrawal Syndrome; Sulpiride; Time Factors | 1984 |
Acute and chronic effects of neuroleptic drugs on plasma and brain homovanillic acid in the rat.
Topics: Animals; Antipsychotic Agents; Brain Chemistry; Chlorpromazine; Fluphenazine; Haloperidol; Homovanillic Acid; Loxapine; Male; Metoclopramide; Molindone; Phenylacetates; Rats; Rats, Inbred Strains; Sulpiride | 1984 |
[3H]spiperone binding in the nigrostriatal system in human brain.
Topics: Aged; Apomorphine; Binding, Competitive; Butaclamol; Butyrophenones; Caudate Nucleus; Cinanserin; Corpus Striatum; Domperidone; Female; Haloperidol; Humans; In Vitro Techniques; Kinetics; Male; Nerve Endings; Phentolamine; Postmortem Changes; Putamen; Spiperone; Substantia Nigra; Sulpiride; Time Factors | 1984 |
Non-opiate beta-endorphin fragments and dopamine--VI. Behavioural analysis of the interaction between gamma-type endorphins and dopaminergic systems in the nucleus accumbens of rats.
Topics: Amphetamine; Animals; Apomorphine; Behavior, Animal; beta-Endorphin; Bromocriptine; Dopamine; Endorphins; Ergolines; Fluphenazine; gamma-Endorphin; Haloperidol; Male; Motor Activity; Nucleus Accumbens; Rats; Rats, Inbred Strains; Septal Nuclei; Sulpiride | 1984 |
Loxapine and clozapine decrease serotonin (S2) but do not elevate dopamine (D2) receptor numbers in the rat brain.
Topics: Animals; Clozapine; Dibenzazepines; Dibenzoxazepines; Haloperidol; Loxapine; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Serotonin; Sulpiride; Time Factors | 1984 |
The effect of neonatal treatment of mice with opioid and dopaminergic agents on the late responsiveness of vasa deferentia to opioids in vitro.
Topics: Animals; Animals, Newborn; Dopamine; Endorphins; Enkephalin, Methionine; Haloperidol; Male; Mice; Morphine; Naloxone; Piribedil; Sulpiride; Time Factors; Vas Deferens | 1984 |
Alpha-adrenoceptor and dopamine receptor antagonists do not block the slow inhibitory postsynaptic potential in sympathetic ganglia.
Topics: Animals; Atropine; Dose-Response Relationship, Drug; Evoked Potentials; Ganglia, Sympathetic; Haloperidol; Male; Neural Inhibition; Phenoxybenzamine; Phentolamine; Propranolol; Rabbits; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Dopamine; Receptors, Muscarinic; Sulpiride; Synapses; Yohimbine | 1980 |
Presynaptic modulation of the release of dopamine from the rabbit caudate nucleus: differences between electrical stimulation, amphetamine and tyramine.
Topics: Amphetamine; Animals; Apomorphine; Calcium; Caudate Nucleus; Dopamine; Electric Stimulation; Haloperidol; In Vitro Techniques; Male; Rabbits; Receptors, Adrenergic, alpha; Receptors, Dopamine; Sulpiride; Tyramine | 1981 |
Operational characteristics of the inhibitory feedback mechanism for regulation of dopamine release via presynaptic receptors.
Topics: Animals; Apomorphine; Calcium; Caudate Nucleus; Corpus Striatum; Dopamine; Electric Stimulation; Feedback; Haloperidol; Putamen; Rabbits; Receptors, Neurotransmitter; Sulpiride | 1982 |
Effects of dopamine on neuromuscular transmission in the guinea-pig mesenteric artery.
Topics: Action Potentials; Animals; Dopamine; Guinea Pigs; Haloperidol; In Vitro Techniques; Mesenteric Arteries; Muscle, Smooth, Vascular; Neuromuscular Junction; Phentolamine; Receptors, Adrenergic, alpha; Receptors, Dopamine; Sulpiride; Synaptic Transmission | 1983 |
Effects of ethanol, given during pregnancy, on the offspring dopaminergic system.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Corpus Striatum; Dextroamphetamine; Dopamine; Ethanol; Female; Haloperidol; Kinetics; Motor Activity; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Rats, Inbred Strains; Spiperone; Sulpiride; Synaptic Transmission | 1983 |
Effect of intrarenal administration of dopamine on renin release in conscious dogs.
Topics: Animals; Dogs; Dopamine; Haloperidol; Infusions, Intra-Arterial; Natriuresis; Phentolamine; Propranolol; Renal Artery; Renal Circulation; Renin; Sulpiride; Vascular Resistance | 1983 |
The role of dopaminergic receptors in the behavioral effects induced by lisuride in male rats.
Topics: Aggression; Animals; Behavior, Animal; Dose-Response Relationship, Drug; Ergolines; Haloperidol; Humans; Lisuride; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sexual Behavior, Animal; Stereotyped Behavior; Sulpiride | 1983 |
Differential effects of continuous administration for 1 year of haloperidol or sulpiride on striatal dopamine function in the rat.
Topics: Acetylcholine; Animals; Apomorphine; Body Weight; Corpus Striatum; Haloperidol; Humans; Kinetics; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Sulpiride | 1984 |
Differential alterations in striatal dopamine receptor sensitivity induced by repeated administration of clinically equivalent doses of haloperidol, sulpiride or clozapine in rats.
Topics: Animals; Apomorphine; Clozapine; Corpus Striatum; Dibenzazepines; Haloperidol; Humans; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Sulpiride | 1984 |
Effects of dopamine antagonists on receptive fields of brisk cells and directionally selective cells in the rabbit retina.
Topics: Animals; Dopamine Antagonists; Flupenthixol; Fluphenazine; Haloperidol; Metoclopramide; Rabbits; Receptors, Dopamine; Retina; Retinal Ganglion Cells; Sulpiride | 1984 |
Drug-induced modulation of locomotor hyperactivity induced by picrotoxin in nucleus accumbens.
Topics: Animals; Apomorphine; Carbachol; Clozapine; Diazepam; Haloperidol; Lisuride; Lysergic Acid Diethylamide; Male; Motor Activity; Nucleus Accumbens; Picrotoxin; Rats; Rats, Inbred Strains; Reserpine; Septal Nuclei; Sulpiride | 1984 |
[Effects of dopaminergic drugs on the concentrations of PGE2 and PGF2alpha in various brain regions].
Topics: Animals; Apomorphine; Brain Chemistry; Dinoprost; Dinoprostone; Dopamine; Haloperidol; Male; Prostaglandins E; Prostaglandins F; Rats; Rats, Inbred Strains; Sulpiride | 1983 |
Effects of dopaminergic drugs on cerebellar prostaglandin concentrations.
Topics: Animals; Apomorphine; Brain; Dinoprost; Dinoprostone; Haloperidol; Male; Prostaglandins; Prostaglandins E; Prostaglandins F; Rats; Rats, Inbred Strains; Sulpiride | 1983 |
LSD-potentiated apomorphine hypermotility: a model for differentiating antipsychotic drugs.
Topics: Animals; Apomorphine; Chlorpromazine; Clozapine; Disease Models, Animal; Drug Antagonism; Haloperidol; Humans; Hyperkinesis; Lysergic Acid Diethylamide; Male; Motor Activity; Rats; Rats, Inbred Strains; Sulpiride | 1983 |
Genotypic variation in the dopaminergic inhibitory control of striatal and hippocampal cholinergic activity in mice.
Topics: Acetylcholine; Adenylyl Cyclases; Animals; Apomorphine; Choline; Corpus Striatum; Dopamine; Genetic Variation; Genotype; Haloperidol; Hippocampus; Humans; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Motor Activity; Stereotyped Behavior; Sulpiride | 1983 |
Phosphorylation of membrane proteins in response to persistent stimulation of adenylate cyclase-linked dopamine receptors in slices of striatum.
Topics: Adenylyl Cyclases; Animals; Corpus Striatum; Dopamine; Haloperidol; In Vitro Techniques; Male; Membrane Proteins; Phosphorylation; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sulpiride | 1984 |
The 'presynaptic' blocking potency of sulpiride and haloperidol in the rat is age-dependent.
Topics: Age Factors; Animals; Ergolines; Haloperidol; Male; Models, Neurological; Models, Psychological; Motor Activity; Pergolide; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sulpiride | 1984 |
The neurobiologically active benzamides and related compounds: some historical aspects.
Topics: Benzamides; Chlorpromazine; Haloperidol; History, 20th Century; Humans; Metoclopramide; Nervous System; Procainamide; Sulpiride | 1982 |
Effect of dopamine agonists and antagonists on DOPA formation in the substantia nigra.
Topics: Animals; Apomorphine; Caudate Nucleus; Dextroamphetamine; Dihydroxyphenylalanine; Dopamine; Haloperidol; Male; Monoamine Oxidase Inhibitors; Pargyline; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Substantia Nigra; Sulpiride | 1982 |
Influence of lisuride on morphine withdrawal signs in the rat: a dopamine-mimetic effect.
Topics: Aggression; Animals; Apomorphine; Dopamine; Ergolines; Haloperidol; Humans; Lisuride; Male; Morphine Dependence; Naloxone; Rats; Rats, Inbred Strains; Substance Withdrawal Syndrome; Sulpiride | 1982 |
Effects of hyper- and hypoprolactinemia on glutamate decarboxylase activity in medial basal hypothalamus of male rat.
Topics: Animals; Apomorphine; Carboxy-Lyases; Domperidone; Glutamate Decarboxylase; Haloperidol; Hypophysectomy; Hypothalamus; Male; Prolactin; Rats; Sulpiride | 1983 |
Inhibition of dopamine synthesis in striatal synaptosomes by lisuride: stereospecific reversal by (-)-sulpiride.
Topics: Animals; Corpus Striatum; Dopamine; Ergolines; Haloperidol; In Vitro Techniques; Lisuride; Male; Rats; Rats, Inbred Strains; Stereoisomerism; Sulpiride; Synaptosomes | 1983 |
Effects of haloperidol and sulpiride on dopamine-induced inhibition of nucleus accumbens neurons.
Topics: Animals; Dopamine; Drug Interactions; Haloperidol; Male; Neurons; Nucleus Accumbens; Rats; Rats, Inbred Strains; Septal Nuclei; Sulpiride | 1983 |
Frequency-dependent release of acetylcholine and dopamine from rabbit striatum: its modulation by dopaminergic receptors.
Topics: Acetylcholine; Animals; Apomorphine; Benztropine; Caudate Nucleus; Corpus Striatum; Dopamine; Electric Stimulation; Haloperidol; In Vitro Techniques; Putamen; Rabbits; Receptors, Dopamine; Sulpiride | 1983 |
Changes in sensitivity of release modulating dopamine autoreceptors after chronic treatment with haloperidol.
Topics: Animals; Apomorphine; Caudate Nucleus; Dopamine; Electric Stimulation; Haloperidol; Hypothalamus; Male; Norepinephrine; Rabbits; Receptors, Dopamine; Sulpiride | 1983 |
Stimulation of rat spontaneous locomotion by low doses of haloperidol and (-)-sulpiride: importance of animal selection and measurement technique.
Topics: Animals; Apomorphine; Dextroamphetamine; Female; Haloperidol; Motor Activity; Rats; Rats, Inbred Strains; Sulpiride | 1983 |
Differential enhancement of behavioral sensitivity to apomorphine following chronic treatment of rats with (-)-sulpiride and haloperidol.
Topics: Animals; Apomorphine; Behavior, Animal; Exploratory Behavior; Haloperidol; Humans; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereotyped Behavior; Substance Withdrawal Syndrome; Sulpiride | 1982 |
Effects of chronic treatment with l-sulpiride and haloperidol on central monoaminergic mechanisms.
Topics: 5-Hydroxytryptophan; Animals; Apomorphine; Behavior, Animal; Biogenic Amines; Brain; Haloperidol; Hydroxydopamines; Ibotenic Acid; Male; Nerve Degeneration; Rats; Sulpiride; Time Factors | 1980 |
Possible involvement of prolactin in sulpiride-induced changes in nigral and striatal GAD activity.
Topics: Animals; Carboxy-Lyases; Corpus Striatum; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Haloperidol; Male; Prolactin; Rats; Substantia Nigra; Sulpiride | 1982 |
[Effects of an ergot derivative, lisuride, on the central nervous system -- stimulatory effect on local cerebral glucose utilization in the rat].
Topics: 4-Butyrolactone; Animals; Brain; Dihydroergotoxine; Ergolines; Glucose; Haloperidol; Lisuride; Male; Rats; Rats, Inbred Strains; Stimulation, Chemical; Substantia Nigra; Sulpiride | 1982 |
Behavioral supersensitivity to methamphetamine following chronic treatment with (--)-sulpiride in the rat.
Topics: Animals; Behavior, Animal; Drug Interactions; Haloperidol; Humans; Male; Methamphetamine; Motor Activity; Rats; Substance Withdrawal Syndrome; Sulpiride | 1981 |
Regional blockade by neuroleptic drugs of in vivo 3H-spiperone binding in the rat brain. Relation to blockade of apomorphine induced hyperactivity and stereotypies.
Topics: Animals; Apomorphine; Binding, Competitive; Brain; Butyrophenones; Chlorpromazine; Clozapine; Haloperidol; Humans; Hyperkinesis; Kinetics; Organ Specificity; Rats; Receptors, Dopamine; Receptors, Drug; Spiperone; Stereotyped Behavior; Sulpiride; Thioridazine | 1981 |
Repeated administration of sulpiride for three weeks produces behavioural and biochemical evidence for cerebral dopamine receptor supersensitivity.
Topics: Adenylyl Cyclases; Animals; Apomorphine; Brain; Haloperidol; Humans; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereotyped Behavior; Sulpiride | 1982 |
Neuronal mechanisms regulating ethanol effects on the dopaminergic system.
Topics: 3,4-Dihydroxyphenylacetic Acid; Alcoholism; Animals; Dopamine; Ethanol; Haloperidol; Humans; Male; Morphine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Sulpiride | 1982 |
Possible role of prolactin in the modification of medial basal hypothalamic glutamic acid decarboxylase activity.
Topics: Animals; Apomorphine; Carboxy-Lyases; Glutamate Decarboxylase; Haloperidol; Hypothalamus; Male; Prolactin; Rats; Sulpiride | 1981 |
Chronic lead treatment induces in rat a specific and differential effect on dopamine receptors in different brain areas.
Topics: Adenylyl Cyclases; Animals; Brain; Dopamine; Haloperidol; Kinetics; Lead Poisoning; Motor Activity; Organ Specificity; Rats; Receptors, Dopamine; Spiperone; Sulpiride; Tritium | 1981 |
The acute effects of sulpiride on the central dopamine turnover in rats: a quantitative histochemical study.
Topics: Animals; Brain; Caudate Nucleus; Dopamine; Haloperidol; Male; Microscopy, Fluorescence; Organ Specificity; Putamen; Rats; Sulpiride | 1981 |
[Pharmacological influences on the brain level and transport of GABA. II) Effect of various psychoactive drugs on brain level and uptake of GABA].
Topics: Amitriptyline; Animals; Biological Transport; Brain; gamma-Aminobutyric Acid; Haloperidol; Methotrimeprazine; Mice; Sulpiride | 1981 |
Scopolamine-induced hypermotility in rats is mediated via a dopaminergic system.
Topics: Animals; Apomorphine; Haloperidol; Lysergic Acid Diethylamide; Male; Motor Activity; Rats; Receptors, Cholinergic; Receptors, Dopamine; Scopolamine; Sulpiride | 1980 |
Effect of chronic sulpiride on striatal spiperone binding.
Topics: Animals; Butyrophenones; Corpus Striatum; Haloperidol; Rats; Spiperone; Sulpiride; Tritium; Visual Cortex | 1980 |
Relaxation by dopaminergic agonists in cerebral and peripheral arteries (in vitro).
Topics: Animals; Cerebral Arteries; Dopamine; Dopamine Antagonists; Droperidol; Drug Interactions; Haloperidol; In Vitro Techniques; Propranolol; Rabbits; Sulpiride; Vasodilator Agents | 1981 |
Effects of chronic haloperidol and sulpiride treatment on rat nigral GABA content.
Topics: Animals; gamma-Aminobutyric Acid; Haloperidol; Male; Rats; Rats, Inbred Strains; Substantia Nigra; Sulpiride | 1981 |
Intestinal pharmacomanometry and glucose tolerance: evidence for two antagonistic dopaminergic mechanisms in the human.
Topics: Animals; Blood Glucose; Colon; Dopamine; Dopamine Antagonists; Gastrointestinal Motility; Haloperidol; Humans; Manometry; Receptors, Dopamine; Rectum; Serotonin; Sulpiride | 1981 |
Sulpiride and the role of dopaminergic receptor blockade in the antipsychotic activity of neuroleptics.
Topics: Adenylyl Cyclases; Animals; Corpus Striatum; Drug Interactions; Haloperidol; Male; Rats; Receptors, Dopamine; Spiperone; Sulpiride | 1981 |
Comparative effects of chronic haloperidol and sulpiride treatment on nigral and striatal GABA content.
Topics: Animals; Corpus Striatum; gamma-Aminobutyric Acid; Haloperidol; Male; Rats; Rats, Inbred Strains; Substantia Nigra; Sulpiride | 1981 |
Effects of different doses of apomorphine on GAD activity in rat substantia nigra.
Topics: Animals; Apomorphine; Carboxy-Lyases; Glutamate Decarboxylase; Haloperidol; Male; Rats; Rats, Inbred Strains; Substantia Nigra; Sulpiride | 1981 |
Effect of long-term treatment with haloperidol and sulpiride on different types of dopaminergic receptors.
Topics: Adenylyl Cyclases; Animals; Corpus Striatum; Haloperidol; Kinetics; Male; Membranes; Pituitary Gland; Rats; Receptors, Dopamine; Sulpiride | 1980 |
Effects of chronic treatment with 1-sulpiride and haloperidol on central dopamine turnover evaluated in dopamine cell body and nerve terminal-rich areas.
Topics: Animals; Brain; Catecholamines; Caudate Nucleus; Dopamine; Haloperidol; Male; Nerve Endings; Nucleus Accumbens; Rats; Sulpiride; Time Factors | 1980 |
Effects of dopaminergic agonists and antagonists on [3H]apomorphine binding to striatal membranes: sulpiride lack of interactions with positive cooperative [3H]apomorphine binding.
Topics: Adenylyl Cyclases; Animals; Apomorphine; Binding, Competitive; Cell Membrane; Corpus Striatum; Haloperidol; Kinetics; Male; Rats; Receptors, Dopamine; Sulpiride; Tritium | 1980 |
Effect of four dopamine receptor antagonists on gastrin secretion in healthy subjects.
Topics: Adult; Female; Gastrins; Haloperidol; Humans; Male; Metoclopramide; Middle Aged; Pimozide; Receptors, Dopamine; Secretory Rate; Sulpiride; Time Factors | 1980 |
Aging process affects a single class of dopamine receptors.
Topics: 3,4-Dihydroxyphenylacetic Acid; Adenylyl Cyclases; Aging; Animals; Corpus Striatum; Haloperidol; Humans; Male; Receptors, Dopamine; Spiperone; Sulpiride | 1980 |
Antipsychotic drugs induce Fos protein in the thalamic paraventricular nucleus: a novel locus of antipsychotic drug action.
Topics: Animals; Antipsychotic Agents; Blotting, Western; Clozapine; Haloperidol; Immunohistochemistry; Male; Muscarinic Antagonists; Prazosin; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Ritanserin; Scopolamine; Serotonin Antagonists; Sulpiride; Thalamic Nuclei | 1995 |
Lack of evidence for dopamine autoreceptors in the mediobasal hypothalamus: a microdialysis study in awake rats.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Benzazepines; Consciousness; Dopamine Antagonists; Haloperidol; Hypothalamus, Middle; Male; Microdialysis; Nomifensine; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine; Salicylamides; Sulpiride | 1995 |
Differential influence of haloperidol and sulpiride on dopamine receptors and peptide mRNA levels in the rat striatum and pituitary.
Topics: Animals; Blotting, Northern; Corpus Striatum; Enkephalins; Gene Expression Regulation; Growth Hormone; Haloperidol; In Situ Hybridization; Interleukin-6; Male; Neuropeptides; Pituitary Gland; Pituitary Hormones, Anterior; Pro-Opiomelanocortin; Prolactin; Protein Precursors; Rats; Receptors, Dopamine; Substance P; Sulpiride; Up-Regulation | 1994 |
Effects of typical and atypical antipsychotic drugs on response decrement patterns in rats.
Topics: Animals; Antipsychotic Agents; Clozapine; Conditioning, Operant; Dose-Response Relationship, Drug; Haloperidol; Isoxazoles; Male; Piperidines; Rats; Rats, Wistar; Remoxipride; Risperidone; Serotonin Antagonists; Sulpiride | 1995 |
Effect of haloperidol and (-)-sulpiride on dopamine agonist-induced hypoactivity.
Topics: Animals; Apomorphine; Benzopyrans; Dopamine Agonists; Dose-Response Relationship, Drug; Ergolines; Haloperidol; Male; Motor Activity; Oxazines; Quinolines; Quinpirole; Rats; Rats, Sprague-Dawley; Sulpiride; Tetrahydronaphthalenes | 1995 |
The dopaminergic system modulates the endogenous opioid system in guinea-pig isolated ileal longitudinal muscle.
Topics: Amisulpride; Animals; Antipsychotic Agents; Dopamine; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; Haloperidol; Ileum; Male; Models, Neurological; Muscle Contraction; Opioid Peptides; Sulpiride | 1995 |
Neuroleptics up-regulate adenosine A2a receptors in rat striatum: implications for the mechanism and the treatment of tardive dyskinesia.
Topics: Animals; Antipsychotic Agents; Binding Sites; Binding, Competitive; Corpus Striatum; Dyskinesia, Drug-Induced; Fluphenazine; Haloperidol; Male; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; Sulpiride; Up-Regulation | 1995 |
Differential effects of dopamine antagonists on evoked dopamine release from slices of striatum and nucleus accumbens in rats.
Topics: Animals; Binding, Competitive; Clozapine; Corpus Striatum; Dopamine; Dopamine Antagonists; Electric Stimulation; Haloperidol; Male; Nucleus Accumbens; Rats; Rats, Wistar; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Sulpiride | 1995 |
An inhibitory dopaminergic regulation of the neuropeptide Y immunoreactivity expression in the rat cerebral cortex neurons.
Topics: Animals; Benzazepines; Cerebral Cortex; Dopamine; Dopamine D2 Receptor Antagonists; Gene Expression Regulation; Haloperidol; Immunohistochemistry; Kinetics; Male; Neurons; Neuropeptide Y; Phenoxybenzamine; Propranolol; Rats; Rats, Wistar; Receptors, Dopamine D1; Reserpine; Sulpiride; Time Factors | 1995 |
Sigma antagonists potentiate opioid analgesia in rats.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Drug Synergism; Haloperidol; Morphine; Naloxone; Narcotics; Pain Measurement; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, sigma; Sulpiride | 1995 |
Remoxipride shows low propensity to block functional striatal dopamine D2 receptors in vitro.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Action Potentials; Animals; Calcium; Colforsin; Corpus Striatum; Cyclic AMP; Dopamine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Haloperidol; In Vitro Techniques; Male; Pergolide; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Remoxipride; Salicylamides; Structure-Activity Relationship; Sulpiride | 1994 |
Suppression of haloperidol-induced oral dyskinesias in rats by vigabatrin.
Topics: 4-Aminobutyrate Transaminase; Animals; Anticonvulsants; Body Weight; Brain; Dyskinesia, Drug-Induced; Eating; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Haloperidol; Male; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Stereotyped Behavior; Sulpiride; Vigabatrin | 1995 |
Prenatal neuroleptic exposure and growth stunting in the rat: an in vivo and in vitro examination of sensitive periods and possible mechanisms.
Topics: Analysis of Variance; Animals; Antipsychotic Agents; Benzazepines; Body Weight; Brain; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Embryonic and Fetal Development; Feeding Behavior; Female; Gestational Age; Growth; Haloperidol; Male; Organ Size; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Rats, Inbred Strains; Receptors, Dopamine D1; Reproducibility of Results; Reserpine; Sex Characteristics; Sulpiride; Teratogens | 1994 |
Lack of effect of antipsychotic and antidepressant drugs on glutamate receptor mRNA levels in rat brains.
Topics: Animals; Antidepressive Agents; Antipsychotic Agents; Base Sequence; Brain Chemistry; Citalopram; Clozapine; Gene Expression Regulation; Haloperidol; Male; Mianserin; Molecular Sequence Data; Nerve Tissue Proteins; Rats; Rats, Wistar; Receptors, Glutamate; Receptors, N-Methyl-D-Aspartate; RNA, Messenger; Schizophrenia; Sulpiride | 1994 |
Neuroleptics cause stimulation of dopamine D1 receptors and their desensitization after chronic treatment.
Topics: Acetylcholine; Animals; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine Antagonists; Drug Tolerance; Haloperidol; Male; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Sulpiride | 1994 |
Atypical antipsychotics, clozapine and sulpiride do not antagonise amphetamine-induced stereotyped locomotion.
Topics: Amphetamine; Animals; Antipsychotic Agents; Clozapine; Haloperidol; Male; Motor Activity; Rats; Rats, Wistar; Stereotyped Behavior; Sulpiride | 1994 |
The role of D1-dopamine receptor in working memory: local injections of dopamine antagonists into the prefrontal cortex of rhesus monkeys performing an oculomotor delayed-response task.
Topics: Animals; Antipsychotic Agents; Appetitive Behavior; Attention; Benzazepines; Dominance, Cerebral; Dopamine; Dopamine Antagonists; Eye Movements; Fixation, Ocular; Haloperidol; Injections; Ketanserin; Macaca mulatta; Male; Mental Recall; Orientation; Prefrontal Cortex; Raclopride; Reaction Time; Receptors, Dopamine D1; Saccades; Salicylamides; Sulpiride | 1994 |
Endogenous dopamine inhibits the release of enkephalin-like immunoreactivity from amacrine cells of the chicken retina in the light.
Topics: Animals; Benzazepines; Chickens; Chlorpromazine; Darkness; Dopamine; Dopamine Agents; Dopamine Antagonists; Enkephalins; Haloperidol; Light; Radioimmunoassay; Retina; Sulpiride; Tetrahydronaphthalenes | 1994 |
Dopaminergic stimulation of subthalamic nucleus elicits oral dyskinesia in rats.
Topics: Animals; Apomorphine; Benzazepines; Dopamine Agents; Dyskinesia, Drug-Induced; Haloperidol; Kainic Acid; Male; Mouth Diseases; Rats; Rats, Sprague-Dawley; Sulpiride; Thalamic Nuclei | 1994 |
Opposing roles for dopamine D2 and D3 receptors on neurotensin mRNA expression in nucleus accumbens.
Topics: Animals; Benzazepines; Haloperidol; Male; Neurotensin; Nucleus Accumbens; Rats; Rats, Wistar; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; RNA, Messenger; Sulpiride; Transcription, Genetic | 1994 |
Evidence that systemically administered dopamine antagonists activate dopamine neuron firing primarily by blockade of somatodendritic autoreceptors.
Topics: Animals; Autoreceptors; Corpus Striatum; Dopamine Antagonists; Dose-Response Relationship, Drug; Haloperidol; Male; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Substantia Nigra; Sulpiride | 1994 |
Differential regulation of glutamate decarboxylase and preproenkephalin mRNA levels in the rat striatum.
Topics: Aging; Animals; Animals, Newborn; Autoradiography; Dopamine; Enkephalins; Female; Glutamate Decarboxylase; Haloperidol; In Situ Hybridization; Neostriatum; Neurons; Oxidopamine; Pertussis Toxin; Pregnancy; Protein Precursors; Rats; Rats, Sprague-Dawley; RNA, Messenger; Sulpiride; Virulence Factors, Bordetella | 1994 |
Dopamine receptor mediated antidepressant action of B-HT 920 in mice.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antidepressive Agents; Azepines; Desipramine; Drug Interactions; Escape Reaction; Female; Haloperidol; Male; Mice; Motor Activity; Receptors, Dopamine; Reserpine; Sulpiride; Swimming; Yohimbine | 1994 |
On the characterization of dopamine-induced contractile response of rat anococcygeus muscle preparation.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Azepines; Benzazepines; Desipramine; Dioxanes; Dopamine; Female; Haloperidol; Idazoxan; Male; Muscle Contraction; Prazosin; Rats; Receptors, Adrenergic; Receptors, Dopamine; Reserpine; Sulpiride; Yohimbine | 1994 |
Convergent regulation by ciliary neurotrophic factor and dopamine of tyrosine hydroxylase expression in cultures of rat substantia nigra.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Cells, Cultured; Ciliary Neurotrophic Factor; Dopamine; Dose-Response Relationship, Drug; Embryo, Mammalian; Ergolines; Glial Fibrillary Acidic Protein; Haloperidol; Kinetics; Nerve Growth Factors; Nerve Tissue Proteins; Neurons; Neurotransmitter Agents; Phosphopyruvate Hydratase; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Recombinant Proteins; Spiperone; Substantia Nigra; Sulpiride; Time Factors; Tyrosine 3-Monooxygenase | 1993 |
Discriminative stimulus properties of cocaine in the rat using a two-choice discrete-trial avoidance paradigm.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Avoidance Learning; Benzazepines; Cocaine; Discrimination Learning; Discrimination, Psychological; Dopamine Agents; Dose-Response Relationship, Drug; Electroshock; Ergolines; Haloperidol; Male; Methamphetamine; Neurotransmitter Uptake Inhibitors; Piperazines; Quinpirole; Rats; Sulpiride | 1993 |
Dopamine D3 receptor mRNA and binding sites in human brain.
Topics: Aminoquinolines; Binding Sites; Binding, Competitive; Brain Chemistry; Corpus Striatum; DNA; Domperidone; Dopamine; Dopamine Agents; Ergolines; Gene Expression Regulation; Haloperidol; Humans; Nerve Tissue Proteins; Organ Specificity; Protein Binding; Quinpirole; Receptors, Dopamine; RNA, Messenger; Sulpiride | 1993 |
Lack of interaction between alpha 2-adrenoceptors and dopamine D2-receptors in mediating their inhibitory effects on [3H]dopamine release from rat nucleus accumbens slices.
Topics: Adrenergic alpha-Agonists; Animals; Apomorphine; Binding, Competitive; Brimonidine Tartrate; Dopamine; Electric Stimulation; Ergolines; GTP-Binding Proteins; Haloperidol; In Vitro Techniques; Male; Nucleus Accumbens; Pergolide; Quinoxalines; Quinpirole; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Receptors, Dopamine D2; Signal Transduction; Sulpiride | 1993 |
Mediation of dopamine D1 and D2 receptors in the effects of GBR 12909 on latent learning and locomotor activity in mice.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Dopamine Agents; Drinking Behavior; Ergolines; Exploratory Behavior; Haloperidol; Learning; Male; Mice; Mice, Inbred Strains; Motor Activity; Neurotransmitter Uptake Inhibitors; Piperazines; Quinpirole; Receptors, Dopamine D1; Receptors, Dopamine D2; Sulpiride | 1993 |
Stimulation of brain dopamine autoreceptors by remoxipride administration in reserpine-treated male rats.
Topics: 5-Hydroxytryptophan; Animals; Aromatic Amino Acid Decarboxylase Inhibitors; Brain Chemistry; Chromatography, High Pressure Liquid; Dihydroxyphenylalanine; Dopamine; Electrochemistry; Haloperidol; Hydrazines; Male; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Remoxipride; Reserpine; Stimulation, Chemical; Sulpiride | 1993 |
Characterisation of a chimeric hD3/D2 dopamine receptor expressed in CHO cells.
Topics: Adenylyl Cyclases; Amino Acid Sequence; Animals; Arachidonic Acid; Base Sequence; Calcimycin; Cell Membrane; CHO Cells; Colforsin; Cricetinae; Dopamine; Dopamine Agents; Dopamine Antagonists; Haloperidol; Humans; Kinetics; Ligands; Molecular Sequence Data; Oligodeoxyribonucleotides; Polymerase Chain Reaction; Protein Structure, Secondary; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Recombinant Fusion Proteins; Sulpiride; Transfection | 1993 |
Functional antagonism of morphine analgesia by (+)-pentazocine: evidence for an anti-opioid sigma 1 system.
Topics: Analgesia; Animals; Dopamine D2 Receptor Antagonists; Drug Interactions; Haloperidol; Male; Mice; Morphine; Pentazocine; Receptors, sigma; Stereoisomerism; Sulpiride | 1993 |
Dopamine D1 receptors are involved in the ACTH-induced reversal of hemorrhagic shock.
Topics: Analysis of Variance; Animals; Benzazepines; Cosyntropin; Dose-Response Relationship, Drug; Female; Haloperidol; Injections, Intravenous; Injections, Subcutaneous; Male; Peptide Fragments; Rats; Rats, Wistar; Receptors, Dopamine D1; Shock, Hemorrhagic; Sulpiride | 1994 |
Central dopaminergic origin of bromocriptine induced tachycardia in normotensive rats.
Topics: Adrenalectomy; Animals; Blood Pressure; Bromocriptine; Domperidone; Dopamine D2 Receptor Antagonists; Haloperidol; Heart Rate; Male; Metoclopramide; Rats; Rats, Wistar; Sulpiride; Tachycardia | 1993 |
Chronic treatment with haloperidol modifies the sensitivity of autoreceptors that modulate dopamine release in rat striatum.
Topics: Animals; Apomorphine; Corpus Striatum; Dopamine; Electric Stimulation; Haloperidol; In Vitro Techniques; Male; Rats; Rats, Wistar; Receptors, Dopamine; Sulpiride; Time Factors | 1993 |
Aromatic L-amino acid decarboxylase activity of mouse striatum is modulated via dopamine receptors.
Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Aromatic-L-Amino-Acid Decarboxylases; Benzazepines; Bromocriptine; Corpus Striatum; Cycloheximide; Dopamine Antagonists; Haloperidol; Kinetics; Levodopa; Male; Mice; Pyridoxal Phosphate; Receptors, Dopamine; Reserpine; Sulpiride; Time Factors | 1993 |
[Effect of D1 and D2 dopamine receptor antagonists on acupuncture analgesia].
Topics: Acupuncture Analgesia; Animals; Benzazepines; Clozapine; Domperidone; Dopamine D2 Receptor Antagonists; Electroacupuncture; Female; Haloperidol; Male; Pain Threshold; Rabbits; Receptors, Dopamine D1; Sulpiride | 1993 |
Changes in G protein levels in the hippocampus and the striatum of rat brain after chronic treatment with haloperidol and sulpiride.
Topics: Animals; Corpus Striatum; GTP-Binding Proteins; Haloperidol; Hippocampus; Male; Rats; Rats, Sprague-Dawley; Sulpiride | 1995 |
Behavioural interactions between 5-hydroxytryptophan, neuroleptic agents and 5-HT receptor antagonists in modifying rodent responding to aversive situations.
Topics: Animals; Antipsychotic Agents; Avoidance Learning; Benperidol; Clozapine; Drug Interactions; Haloperidol; Male; Mice; Mice, Inbred Strains; Rats; Rats, Inbred Strains; Ritanserin; Serotonin; Serotonin Antagonists; Social Behavior; Sulpiride; Thioridazine | 1995 |
Effects of haloperidol and chlorpromazine on smooth muscle contractility, platelet aggregation and neuronal calcium current.
Topics: Animals; Antipsychotic Agents; Butyrophenones; Calcium Channel Blockers; Calcium Channels; Calmodulin; Chlorpromazine; Droperidol; Electric Stimulation; Guinea Pigs; Haloperidol; In Vitro Techniques; Isometric Contraction; Male; Muscle, Smooth; Neurons; Phenothiazines; Platelet Aggregation; Platelet Aggregation Inhibitors; Prazosin; Rats; Rats, Wistar; Snails; Sulpiride; Thrombin; Ureter; Verapamil | 1995 |
Effect of estrogen and neuroleptics on prolactin secretion and immunoreactive prolactin cells.
Topics: Animals; Antipsychotic Agents; Estrogens; Fluphenazine; Haloperidol; Male; Metoclopramide; Pituitary Gland; Prolactin; Rats; Rats, Wistar; Sulpiride | 1996 |
Dopamine-N-methyl-D-aspartate interactions in the modulation of locomotor activity and memory consolidation in mice.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Avoidance Learning; Benzazepines; Dizocilpine Maleate; Dopamine Agonists; Dopamine Antagonists; Excitatory Amino Acid Antagonists; Haloperidol; Male; Memory; Mice; Mice, Inbred Strains; Motor Activity; Piperazines; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, N-Methyl-D-Aspartate; Sulpiride | 1996 |
Inhibitory action of dopamine involves a subthreshold Cs(+)-sensitive conductance in neostriatal neurons.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Action Potentials; Animals; Benzazepines; Cesium; Cyclic AMP; Dopamine; Dopamine Agonists; Electric Stimulation; Electrophysiology; Evoked Potentials; Haloperidol; In Vitro Techniques; Ion Channels; Membrane Potentials; Neostriatum; Neurons; Patch-Clamp Techniques; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Sulpiride; Tetrodotoxin | 1996 |
Hysterical neurosis of the conversion type: therapeutic activity of neuroleptics with different hyperprolactinemic potency.
Topics: Adult; Antipsychotic Agents; Female; Haloperidol; Humans; Hysteria; Male; Middle Aged; Prolactin; Sulpiride | 1996 |
Dopamine autoreceptor sensitivity is unchanged in rat nucleus accumbens after chronic haloperidol treatment: an in vivo and in vitro voltammetric study.
Topics: Animals; Autoreceptors; Dopamine; Dopamine Agonists; Dose-Response Relationship, Drug; Ergolines; Haloperidol; Male; Nucleus Accumbens; Quinpirole; Rats; Sulpiride; Time Factors | 1995 |
Effects of dopamine antagonists on neuronal histamine release in the striatum of rats subjected to acute and chronic treatments with methamphetamine.
Topics: Animals; Corpus Striatum; Dopamine Antagonists; Haloperidol; Histamine Release; Male; Methamphetamine; Rats; Rats, Wistar; Receptors, Dopamine D2; Stereotyped Behavior; Sulpiride | 1996 |
Pharmacological characterization and autoradiographic localization of dopamine receptors in the rat adrenal medulla.
Topics: Adrenal Medulla; Animals; Autoradiography; Benzazepines; Butaclamol; Corpus Striatum; Haloperidol; Male; Radioligand Assay; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Sulpiride | 1996 |
Long-term treatment with chlorpromazine and haloperidol but not with sulpiride and clozapine markedly elevates neuropeptide Y-like immunoreactivity in the rat hypothalamus.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Antipsychotic Agents; Benzazepines; Chlorpromazine; Clozapine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Gene Expression Regulation; Haloperidol; Hypothalamus; Male; Neuropeptide Y; Prazosin; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Sulpiride | 1996 |
Evidence for a functional role of the dopamine D3 receptors in the cerebellum.
Topics: Amisulpride; Animals; Antipsychotic Agents; Apomorphine; Behavior, Animal; Cerebellum; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Female; Haloperidol; Locomotion; Naphthalenes; Nucleus Accumbens; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Sulpiride | 1996 |
Differential expression of c-fos mRNA in rat prefrontal cortex, striatum, N. accumbens and lateral septum after typical and atypical antipsychotics: an in situ hybridization study.
Topics: Animals; Antipsychotic Agents; Aripiprazole; Brain; Clozapine; Corpus Striatum; Fluphenazine; Genes, fos; Haloperidol; In Situ Hybridization; Nucleus Accumbens; Piperazines; Prefrontal Cortex; Quinolones; Rats; RNA, Messenger; Septum Pellucidum; Sulpiride | 1996 |
Effect of chronic treatment with typical and atypical neuroleptics on the expression of dopamine D2 and D3 receptors in rat brain.
Topics: Animals; Antipsychotic Agents; Clozapine; Haloperidol; In Situ Hybridization; Limbic System; Male; Neostriatum; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; RNA, Messenger; Sulpiride | 1996 |
[Difference in prolaction response of schizophrenic patients to equivalent doses of haloperidol, remoxipride and sulpiride].
Topics: Adult; Age Factors; Aged; Antipsychotic Agents; Female; Haloperidol; Humans; Male; Middle Aged; Prolactin; Remoxipride; Schizophrenia; Sex Factors; Sulpiride | 1996 |
BMY-14802 reversed the sigma receptor agonist-induced neck dystonia in rats.
Topics: Animals; Antipsychotic Agents; Dibenzothiepins; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dystonia; Guanidines; Haloperidol; Male; Microinjections; Nerve Tissue Proteins; Perphenazine; Piperidines; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, sigma; Red Nucleus; Sulpiride; Torticollis | 1996 |
Antipsychotics with inverse agonist activity at the dopamine D3 receptor.
Topics: Animals; Antipsychotic Agents; Calcium; CHO Cells; Clozapine; Colforsin; Cricetinae; Cyclic AMP; DNA Replication; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Flupenthixol; Glioma; Haloperidol; Humans; Hybrid Cells; Naphthalenes; Neuroblastoma; Pertussis Toxin; Phenothiazines; Pimozide; Pyrrolidines; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3; Recombinant Proteins; Risperidone; Salicylamides; Second Messenger Systems; Sulpiride; Tetrahydronaphthalenes; Tumor Cells, Cultured; Virulence Factors, Bordetella | 1996 |
Effect of antipsychotic drugs on the gene expression of NMDA receptor subunits in rats.
Topics: Animals; Antipsychotic Agents; Brain; Gene Expression Regulation; Haloperidol; Male; Peptide Fragments; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Sulpiride | 1997 |
The behavioural effects of pramipexole, a novel dopamine receptor agonist.
Topics: Animals; Antiparkinson Agents; Benzazepines; Benzothiazoles; Body Temperature; Catalepsy; Clozapine; Dopamine Agents; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Dyskinesia, Drug-Induced; Haloperidol; Injections, Subcutaneous; Levodopa; Male; Mice; Motor Activity; Pramipexole; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Spiperone; Stereotyped Behavior; Sulpiride; Thiazoles | 1997 |
The comparative effects of haloperidol, (-)-sulpiride, and SCH23390 on c-fos and c-jun mRNA expressions, and AP-1 DNA binding activity.
Topics: Animals; Benzazepines; DNA; Dopamine Antagonists; Electrophoresis, Polyacrylamide Gel; Haloperidol; Image Processing, Computer-Assisted; Male; Mice; Mice, Inbred Strains; Nuclear Proteins; Proto-Oncogene Proteins c-fos; Proto-Oncogene Proteins c-jun; Ribonucleases; RNA Probes; RNA, Messenger; Sulpiride; Transcription Factor AP-1 | 1997 |
Multiple [3H]-nemonapride binding sites in calf brain.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Adrenergic alpha-Antagonists; Animals; Anticonvulsants; Benzamides; Binding, Competitive; Brain; Cattle; Cerebellum; Cerebral Cortex; Corpus Striatum; Dioxanes; Dopamine Agonists; Dopamine Antagonists; Guanidines; Haloperidol; In Vitro Techniques; Isotope Labeling; Narcotic Antagonists; Pentazocine; Piperidines; Propylamines; Pyrrolidines; Receptors, Dopamine D2; Receptors, sigma; Sulpiride; Tritium | 1997 |
Bidirectional effects of dopamine D2 receptor antagonists on responding for a conditioned reinforcer.
Topics: Amphetamine; Animals; Benzazepines; Conditioning, Operant; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Female; Haloperidol; Motivation; Pimozide; Raclopride; Rats; Reinforcement, Psychology; Reward; Salicylamides; Sulpiride | 1997 |
Involvement of activation of dopaminergic neuronal system in learning and memory deficits associated with experimental mild traumatic brain injury.
Topics: Animals; Apomorphine; Benzazepines; Brain Injuries; Dopamine; Dopamine Agonists; Dopamine Antagonists; Exploratory Behavior; Haloperidol; Learning Disabilities; Male; Memory Disorders; Mice; Mice, Inbred Strains; Neurons; Retention, Psychology; Sulpiride | 1997 |
Regulation of D2 and D3 receptors in transfected cells by agonists and antagonists.
Topics: Adenylyl Cyclase Inhibitors; Brain; Cell Line; Dopamine Agonists; Dopamine Antagonists; GTP-Binding Proteins; Haloperidol; Humans; Kinetics; Receptors, Dopamine D2; Receptors, Dopamine D3; Recombinant Proteins; Salicylamides; Sulpiride; Transfection; Up-Regulation; Virulence Factors, Bordetella | 1998 |
Loss of haloperidol induced gene expression and catalepsy in protein kinase A-deficient mice.
Topics: Animals; Antipsychotic Agents; Behavior, Animal; Catalepsy; Corpus Striatum; Cyclic AMP-Dependent Protein Kinase RIIbeta Subunit; Cyclic AMP-Dependent Protein Kinases; Gene Expression Regulation; Haloperidol; Mice; Mice, Mutant Strains; Neurotensin; Proto-Oncogene Proteins c-fos; Receptors, Dopamine D2; RNA, Messenger; Signal Transduction; Sulpiride; Transcription, Genetic; Transcriptional Activation | 1997 |
Effects of REM sleep deprivation on the d-amphetamine-induced self-mutilating behavior.
Topics: Animals; Benzazepines; Central Nervous System Stimulants; Dextroamphetamine; Dopamine; Dopamine Antagonists; Haloperidol; Male; Rats; Rats, Wistar; Receptors, Dopamine; Self-Injurious Behavior; Sleep Deprivation; Sleep, REM; Sulpiride | 1997 |
The effects of antipsychotic drugs on the mRNA levels of serotonin 5HT2A and 5HT2C receptors.
Topics: Animals; Antipsychotic Agents; Brain; Chlorpromazine; Clozapine; Down-Regulation; Haloperidol; Male; Organ Specificity; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; RNA, Messenger; Sulpiride; Time Factors; Transcription, Genetic; Up-Regulation | 1997 |
Dopaminergic modulation of lithium/pilocarpine-induced status epilepticus in rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Azepines; Benzazepines; Disease Models, Animal; Dopamine Agonists; Dopamine Antagonists; Haloperidol; Lipid Peroxidation; Lithium; Male; Muscarinic Agonists; Pilocarpine; Rats; Rats, Wistar; Status Epilepticus; Sulpiride | 1997 |
Distribution of Fos- and Jun-related proteins and activator protein-1 composite factors in mouse brain induced by neuroleptics.
Topics: Animals; Antipsychotic Agents; Benzazepines; Brain Chemistry; Electrophoresis, Polyacrylamide Gel; Haloperidol; Immunohistochemistry; Male; Mice; Nuclear Proteins; Proto-Oncogene Proteins c-fos; Proto-Oncogene Proteins c-jun; Sulpiride; Transcription Factor AP-1 | 1998 |
Sulpiride, but not haloperidol, up-regulates gamma-hydroxybutyrate receptors in vivo and in cultured cells.
Topics: Animals; Brain Chemistry; Cell Line; Cells, Cultured; Dopamine Antagonists; Haloperidol; Injections, Intraventricular; Kinetics; Male; Rats; Rats, Wistar; Receptors, Cell Surface; Sodium Oxybate; Sulpiride; Up-Regulation | 1998 |
Influence of neuroleptics on cytotoxic activity of macrophages in rats.
Topics: Animals; Antipsychotic Agents; Chlorpromazine; Cytotoxicity, Immunologic; Haloperidol; In Vitro Techniques; Macrophages; Male; Rats; Rats, Wistar; Sulpiride | 1998 |
Preferential blockade by clozapine of hyperlocomotion induced by non-competitive NMDA antagonist MK-801.
Topics: Analysis of Variance; Animals; Antipsychotic Agents; Benzazepines; Clozapine; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Interactions; Haloperidol; Hyperkinesis; Mice; Mice, Inbred BALB C; N-Methylaspartate; Neuroprotective Agents; Rats; Rats, Wistar; Stereotyped Behavior; Sulpiride | 1998 |
Alpha1-adrenergic, D1, and D2 receptors interactions in the prefrontal cortex: implications for the modality of action of different types of neuroleptics.
Topics: Animals; Antipsychotic Agents; Benzazepines; Cerebral Cortex; Clozapine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Electric Stimulation; Electrophysiology; Haloperidol; Injections, Intravenous; Iontophoresis; Neural Inhibition; Prazosin; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Receptors, Dopamine D1; Receptors, Dopamine D2; Sulpiride | 1998 |
Influence of typical and atypical antipsychotics on neuropeptide Y-like immunoreactivity and NPY mRNA expression in rat striatum.
Topics: Adrenergic Antagonists; Animals; Antipsychotic Agents; Chlorpromazine; Clozapine; Corpus Striatum; Dopamine Antagonists; Haloperidol; In Situ Hybridization; Injections, Intraperitoneal; Male; Neuropeptide Y; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Dopamine; Receptors, Serotonin; RNA, Messenger; Serotonin Antagonists; Sulpiride | 1998 |
Neuroleptics with differential affinities at dopamine D2 receptors and sigma receptors affect differently the N-methyl-D-aspartate-induced increase in intracellular calcium concentration: involvement of protein kinase.
Topics: Animals; Antipsychotic Agents; Calcium; Cells, Cultured; Chlorpromazine; Clozapine; Dopamine Antagonists; Frontal Lobe; Guanidines; Haloperidol; N-Methylaspartate; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, sigma; Sulpiride | 1999 |
Effects of acute or long-term treatment with chlorpromazine, haloperidol or sulpiride on neuropeptide Y-like immunoreactivity concentrations in the nucleus accumbens of rat.
Topics: Animals; Antipsychotic Agents; Chlorpromazine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Haloperidol; Immunohistochemistry; In Situ Hybridization; Male; Neuropeptide Y; Nucleus Accumbens; Rats; Rats, Wistar; Receptors, Dopamine D1; RNA, Messenger; Substance Withdrawal Syndrome; Sulpiride; Time Factors | 1999 |
Dopaminergic modulation of transcallosal activity of cat motor cortical neurons.
Topics: Action Potentials; Animals; Benzazepines; Cats; Corpus Callosum; Dopamine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Electric Stimulation; Haloperidol; Motor Cortex; Neurons; Pyramidal Tracts; Reaction Time; Receptors, Dopamine D1; Sulpiride | 1999 |
Glutamatergic and dopaminergic contributions to rat bladder hyperactivity after cerebral artery occlusion.
Topics: Animals; Arterial Occlusive Diseases; Benzazepines; Cerebral Infarction; Cerebrovascular Disorders; Dizocilpine Maleate; Dopamine; Dopamine Antagonists; Drug Interactions; Excitatory Amino Acid Antagonists; Female; Glutamic Acid; Haloperidol; Rats; Rats, Sprague-Dawley; Sulpiride; Urinary Bladder; Urinary Bladder, Neurogenic | 1999 |
Comparison of the effects of dopamine D1 and D2 receptor antagonists on nerve growth factor mRNA expression.
Topics: Animals; Benzazepines; Cerebral Cortex; Corpus Striatum; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Gene Expression; Gene Expression Regulation; Haloperidol; Hippocampus; In Situ Hybridization; Male; Mice; Nerve Growth Factors; Nucleus Accumbens; Receptors, Dopamine D1; RNA, Messenger; Sulpiride; Time Factors | 1999 |
The effects of dopamine D2 and D3 antagonists on spontaneous motor activity and morphine-induced hyperactivity in male mice.
Topics: Animals; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Haloperidol; Indans; Male; Mice; Morphine; Motor Activity; Narcotics; Receptors, Dopamine D3; Sulpiride | 1999 |
A mixed D1 and D2 antagonist does not replay pattern electroretinogram alterations observed with a selective D2 antagonist in normal humans: relationship with Parkinson's disease pattern electroretinogram alterations.
Topics: Adult; Brain; Electroencephalography; Electroretinography; Haloperidol; Humans; Parkinson Disease; Reference Values; Sulpiride | 1999 |
[Intercentral interactions during typical and atypical neuroleptics administration].
Topics: Animals; Antipsychotic Agents; Avoidance Learning; Brain; Dogs; Electric Stimulation; Electroencephalography; Evoked Potentials; Haloperidol; Photic Stimulation; Reaction Time; Sulpiride; Time | 1999 |
Dihydroetorphine-induced place preference was mediated by dopamine D1 receptors in rats.
Topics: Animals; Behavior, Animal; Benzazepines; Dopamine Agonists; Etorphine; Haloperidol; Male; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Sulpiride | 1999 |
Pharmacological profile of MS-377, a novel antipsychotic agent with selective affinity for sigma receptors.
Topics: Amisulpride; Animals; Antipsychotic Agents; Apomorphine; Catalepsy; Dopamine Agonists; Free Radical Scavengers; Guinea Pigs; Haloperidol; Head Movements; Male; Mice; Phenazocine; Phencyclidine; Piperazines; Pyrrolidines; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Serotonin; Receptors, sigma; Risperidone; Serotonin; Serotonin Antagonists; Stereotyped Behavior; Sulpiride; Tartrates | 1999 |
Pentadecapeptide BPC 157 attenuates disturbances induced by neuroleptics: the effect on catalepsy and gastric ulcers in mice and rats.
Topics: Animals; Anti-Ulcer Agents; Antipsychotic Agents; Catalepsy; Clozapine; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Fluphenazine; Haloperidol; Male; Mice; Orientation; Peptic Ulcer; Peptide Fragments; Proteins; Rats; Rats, Wistar; Sulpiride; Time Factors | 1999 |
Long-term treatment with antidepressants increases glucocorticoid receptor binding and gene expression in cultured rat hippocampal neurones.
Topics: Amitriptyline; Animals; Antidepressive Agents, Tricyclic; Cells, Cultured; Desipramine; Dexamethasone; Gene Expression Regulation; Haloperidol; Hippocampus; Ketanserin; Mianserin; Neurons; Paroxetine; Phentolamine; Propranolol; Radioligand Assay; Rats; Receptors, Glucocorticoid; Receptors, Mineralocorticoid; RNA, Messenger; Sulpiride; Transcription, Genetic; Tritium | 1999 |
Dopamine receptor antagonists modulate glucose uptake in rat pheochromocytoma (PC12) cells.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Benzazepines; Biological Transport; Chlorpromazine; Clozapine; Dizocilpine Maleate; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Excitatory Amino Acid Antagonists; Fluphenazine; Glucose; Haloperidol; PC12 Cells; Pimozide; Rats; Receptors, Dopamine D2; Spiperone; Sulpiride; Tritium | 1999 |
Chronic effect of antidopaminergic drugs or estrogen on male wistar rat lactotrophs and somatotrophs.
Topics: Animals; Dopamine Antagonists; Estrogens; Fluphenazine; Growth Hormone; Haloperidol; Hyperprolactinemia; Male; Pituitary Gland; Prolactin; Rats; Rats, Wistar; Sulpiride | 1999 |
Cortically driven Fos induction in the striatum is amplified by local dopamine D2-class receptor blockade.
Topics: Animals; Cerebral Cortex; Corpus Striatum; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Gene Expression Regulation; Haloperidol; Injections, Epidural; Oncogene Proteins v-fos; Picrotoxin; Rats; Rats, Sprague-Dawley; Sulpiride | 1999 |
Differential behavioural effect of quinpirole in neuroleptic-pretreated rats - role of alpha(1)-adrenoceptor.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Antipsychotic Agents; Behavior, Animal; Chlorpromazine; Dopamine Agonists; Drug Synergism; Haloperidol; Injections, Intraperitoneal; Male; Motor Activity; Prazosin; Quinpirole; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Sodium Chloride; Sulpiride | 1999 |
Characterization of D-fenfluramine-induced hypothermia: evidence for multiple sites of action.
Topics: Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Benzofurans; Body Temperature; Cerebral Cortex; Dopamine Antagonists; Dose-Response Relationship, Drug; Fenclonine; Fenfluramine; Haloperidol; Hydroxyindoleacetic Acid; Hypothalamus; Hypothermia; Ketanserin; Male; Piperazines; Pyridines; Rats; Rats, Sprague-Dawley; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Sertraline; Sulpiride; Yohimbine | 2000 |
Predicting how equipotent doses of chlorpromazine, haloperidol, sulpiride, raclopride and clozapine reduce locomotor activity in mice.
Topics: Animals; Antipsychotic Agents; Chlorpromazine; Clozapine; Female; Haloperidol; Male; Mice; Motor Activity; Raclopride; Sulpiride | 2000 |
Effects of oil intake in the conditioned place preference test in mice.
Topics: Animals; Behavior, Animal; Benzazepines; Brain Chemistry; Conditioning, Psychological; Corn Oil; Dopamine Antagonists; Eating; Haloperidol; Indoles; Male; Mice; Piperidines; Receptors, Dopamine D1; Reward; Space Perception; Sulpiride | 2000 |
Potentiation of ethanol-induced loss of the righting reflex by ascorbic acid in mice: interaction with dopamine antagonists.
Topics: Animals; Ascorbic Acid; Benzazepines; Clozapine; Dopamine Antagonists; Drug Synergism; Ethanol; Female; Haloperidol; Mice; Receptors, Dopamine D2; Reflex; Sleep; Sulpiride | 2000 |
Modulation of long-term depression by dopamine in the mesolimbic system.
Topics: Animals; Benzazepines; Conditioning, Psychological; Dopamine; Dopamine Agonists; Dopamine Antagonists; Haloperidol; Limbic System; Long-Term Potentiation; Mesencephalon; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Neural Inhibition; Neuronal Plasticity; Neurons; Nucleus Accumbens; Patch-Clamp Techniques; Quinpirole; Salicylamides; Substance-Related Disorders; Sulpiride; Ventral Tegmental Area | 2000 |
Pharmacology of [3H]R(+)-7-OH-DPAT binding in the rat caudate-putamen.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Benzopyrans; Binding, Competitive; Caudate Nucleus; Clozapine; Dopamine; Dopamine Agonists; Dopamine Antagonists; Guanidines; Guanosine Triphosphate; Haloperidol; Heterotrimeric GTP-Binding Proteins; Indans; Kinetics; Magnesium; Male; Oxazines; Protein Binding; Putamen; Quinpirole; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Remoxipride; Sodium; Specific Pathogen-Free Organisms; Sulfones; Sulpiride; Tetrahydronaphthalenes | 2001 |
Orexin-induced hyperlocomotion and stereotypy are mediated by the dopaminergic system.
Topics: Animals; Axons; Behavior, Animal; Benzazepines; Carrier Proteins; Dopamine; Dopamine Antagonists; Haloperidol; Intracellular Signaling Peptides and Proteins; Male; Motor Activity; Nerve Endings; Neurons; Neuropeptides; Orexins; Rats; Rats, Wistar; Stereotyped Behavior; Sulpiride; Tegmentum Mesencephali; Tyrosine 3-Monooxygenase | 2000 |
Comparative effects of dopamine D(1) and D(2) receptor antagonists on nerve growth factor protein induction.
Topics: Animals; Antipsychotic Agents; Benzazepines; Blotting, Western; Brain Chemistry; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Gene Expression Regulation; Genes, fos; Genes, jun; Haloperidol; Immunohistochemistry; Male; Mice; Nerve Growth Factor; Receptors, Dopamine D1; RNA, Messenger; Sulpiride | 2000 |
Reinforcing effects of methamphetamine in planarians.
Topics: Amphetamine-Related Disorders; Animals; Behavior, Animal; Benzazepines; Brain; Conditioning, Psychological; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Haloperidol; Methamphetamine; Planarians; Receptors, Dopamine D1; Receptors, Dopamine D2; Reinforcement, Psychology; Sulpiride | 2000 |
Antipsychotic drugs classified by their effects on the release of dopamine and noradrenaline in the prefrontal cortex and striatum.
Topics: Animals; Antipsychotic Agents; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Haloperidol; Male; Norepinephrine; Prefrontal Cortex; Raclopride; Rats; Rats, Wistar; Receptors, Serotonin; Sulpiride | 2001 |
Effects of dopamine and dopamine-active compounds on oxytocin and vasopressin production in rat neurohypophyseal tissue cultures.
Topics: Animals; Apomorphine; Butaclamol; Chlorpromazine; Culture Techniques; Dopamine; Dopamine Agonists; Dopamine Antagonists; Drug Synergism; Haloperidol; Male; Neuroglia; Oxytocin; Pituitary Gland; Rats; Rats, Wistar; Sulpiride; Vasopressins | 2001 |
Acute phase of schizophrenia: impact of atypical antipsychotics.
Topics: Acute Disease; Amisulpride; Antipsychotic Agents; Haloperidol; Humans; Prognosis; Recurrence; Risperidone; Schizophrenia; Severity of Illness Index; Sulpiride | 2000 |
Reversal effect of sulpiride on rotational behaviour of rats with unilateral frontal cortex ablation: an alternative explanation for the pharmacological mechanism of its antidepressant effect.
Topics: Animals; Antidepressive Agents, Second-Generation; Brain Chemistry; Central Nervous System Stimulants; Dopamine Antagonists; Functional Laterality; Glutathione; Haloperidol; Male; Methamphetamine; Prefrontal Cortex; Rats; Rats, Wistar; Rotation; Stereotyped Behavior; Sulpiride | 2001 |
The changes of biological markers and treatment efficacy in schizophrenia.
Topics: Acute Disease; Adult; Amisulpride; Antipsychotic Agents; Biomarkers; Brain; Cognition; Dexamethasone; Follow-Up Studies; Haloperidol; Humans; Hydrocortisone; Inpatients; Memory; Perphenazine; Psychological Tests; Psychomotor Performance; Reaction Time; Schizophrenia; Schizophrenic Psychology; Sulpiride; Time Factors; Tomography, X-Ray Computed | 2001 |
Mechanisms of inverse agonism of antipsychotic drugs at the D(2) dopamine receptor: use of a mutant D(2) dopamine receptor that adopts the activated conformation.
Topics: 1-Methyl-3-isobutylxanthine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antipsychotic Agents; Apomorphine; Binding, Competitive; Bromocriptine; Butaclamol; Chlorpromazine; CHO Cells; Clozapine; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; GTP-Binding Proteins; Haloperidol; Humans; Macromolecular Substances; Mutagenesis, Site-Directed; Phenethylamines; Piperidines; Protein Binding; Protein Conformation; Radioligand Assay; Receptors, Dopamine D2; Recombinant Fusion Proteins; Sodium; Spiperone; Structure-Activity Relationship; Sulpiride; Transfection; Tyramine | 2001 |
A dopaminergic mechanism is involved in the 'anxiogenic-like' response induced by chronic amphetamine treatment: a behavioral and neurochemical study.
Topics: Amphetamine; Amphetamine-Related Disorders; Animals; Anxiety; Behavior, Animal; Benzazepines; Brain; Brain Chemistry; Chloride Channels; Chlorides; Dopamine; Dopamine Antagonists; Drug Administration Schedule; Drug Interactions; gamma-Aminobutyric Acid; Haloperidol; Male; Maze Learning; Neurons; Rats; Rats, Wistar; Receptors, Dopamine; Sulpiride | 2001 |
Atypical neuroleptic drugs downregulate dopamine sensitivity in rat cortical and striatal astrocytes.
Topics: Adrenergic beta-Antagonists; Animals; Animals, Newborn; Antipsychotic Agents; Astrocytes; Benzodiazepines; Calcium; Calcium Signaling; Cells, Cultured; Cerebral Cortex; Clozapine; Dopamine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Down-Regulation; Haloperidol; Intracellular Fluid; Neostriatum; Olanzapine; Pirenzepine; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D4; Risperidone; Serotonin Antagonists; Sulpiride | 2001 |
Modulation of dopamine uptake in rat nucleus accumbens: effect of specific dopamine receptor antagonists and sigma ligands.
Topics: Animals; Antipsychotic Agents; Carbazoles; Dopamine; Dopamine Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Female; Haloperidol; Ligands; Neurons; Nomifensine; Nucleus Accumbens; Phenazocine; Progesterone; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, sigma; Spiperone; Sulpiride; Synaptosomes; Tritium | 2001 |
Pro-erectile effect of systemic apomorphine: existence of a spinal site of action.
Topics: Animals; Apomorphine; Benzazepines; Binding Sites; Blood Pressure; Domperidone; Haloperidol; Hexamethonium; Injections, Intravenous; Male; Penile Erection; Penis; Rats; Rats, Sprague-Dawley; Spinal Cord; Spinal Cord Injuries; Sulpiride | 2002 |
Atypical, but not typical, antipsychotic drugs increase cortical acetylcholine release without an effect in the nucleus accumbens or striatum.
Topics: Acetylcholine; Acetylcholinesterase; Animals; Antipsychotic Agents; Benzodiazepines; Cerebral Cortex; Cholinesterase Inhibitors; Clozapine; Corpus Striatum; Haloperidol; Male; Nucleus Accumbens; Olanzapine; Oxotremorine; Piperazines; Pirenzepine; Rats; Rats, Sprague-Dawley; Risperidone; Scopolamine; Sulpiride; Thiazoles; Thioridazine | 2002 |
Sub-chronic treatment with classical but not atypical antipsychotics produces morphological changes in rat nigro-striatal dopaminergic neurons directly related to "early onset" vacuous chewing.
Topics: Amisulpride; Animals; Antipsychotic Agents; Clozapine; Dopamine; Dose-Response Relationship, Drug; Drug Administration Schedule; Dyskinesia, Drug-Induced; Haloperidol; Male; Mastication; Neostriatum; Nerve Degeneration; Neural Pathways; Neurons; Rats; Rats, Sprague-Dawley; Risperidone; Substance Withdrawal Syndrome; Substantia Nigra; Sulpiride | 2002 |
Switching to amisulpride due to hepatic complications.
Topics: Adult; Amisulpride; Antipsychotic Agents; Chemical and Drug Induced Liver Injury; Flupenthixol; Haloperidol; Humans; Male; Perazine; Schizophrenia; Sulpiride | 2002 |
Management of rheumatic chorea: an observational study.
Topics: Anti-Dyskinesia Agents; Child; Chorea; Cross-Sectional Studies; Diazepam; Female; Haloperidol; Humans; Male; Sulpiride; Valproic Acid | 2002 |
Amisulpride improves depressive symptoms in acute exacerbations of schizophrenia: comparison with haloperidol and risperidone.
Topics: Adult; Amisulpride; Antipsychotic Agents; Brief Psychiatric Rating Scale; Depression; Double-Blind Method; Female; Haloperidol; Humans; Male; Middle Aged; Multicenter Studies as Topic; Randomized Controlled Trials as Topic; Risperidone; Schizophrenia; Sulpiride; Treatment Outcome | 2002 |
Dopamine modulates the function of group II and group III metabotropic glutamate receptors in the substantia nigra pars reticulata.
Topics: Animals; Benzazepines; Bridged Bicyclo Compounds; Dopamine; Dopamine Agonists; Excitatory Amino Acid Agonists; Haloperidol; Neurons; Rats; Receptors, Metabotropic Glutamate; Substantia Nigra; Sulpiride; Synaptic Transmission | 2002 |
Effects of sigma(1) receptor ligand MS-377 on D(2) antagonists-induced behaviors.
Topics: Amisulpride; Animals; Antipsychotic Agents; Apomorphine; Behavior, Animal; Catalepsy; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Drug Interactions; Female; Haloperidol; Male; Mice; Nootropic Agents; Phenazocine; Piperazines; Pyridines; Pyrrolidines; Rats; Receptors, sigma; Serotonin Antagonists; Sigma-1 Receptor; Sulpiride; Tartrates | 2002 |
Lesioning the thalamus for dyskinesia.
Topics: Antiparkinson Agents; Antipsychotic Agents; Dyskinesia, Drug-Induced; Dyskinesias; Electrocoagulation; Haloperidol; Humans; Levodopa; Male; Middle Aged; Parkinson Disease; Parkinsonian Disorders; Reoperation; Retrospective Studies; Schizophrenia; Stereotaxic Techniques; Sulpiride; Torticollis; Treatment Outcome; Tremor; Ventral Thalamic Nuclei | 2001 |
Chlorpromazine inhibits the glucocorticoid receptor-mediated gene transcription in a calcium-dependent manner.
Topics: Animals; Antipsychotic Agents; Calcimycin; Calcium; Calcium Channel Blockers; Cell Line; Cell Line, Transformed; Chloramphenicol O-Acetyltransferase; Chlorpromazine; Clozapine; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Inhibitors; Estrenes; Fibroblasts; Gene Expression Regulation; Genes, Reporter; Haloperidol; Histamine; Histamine H1 Antagonists; Ionophores; Mammary Tumor Virus, Mouse; Mice; Nifedipine; Phorbol Esters; Phosphodiesterase Inhibitors; Protein Kinase C; Protein Kinase C-alpha; Pyrilamine; Pyrrolidinones; Raclopride; Receptors, Glucocorticoid; Remoxipride; Sulfonamides; Sulpiride; Tetradecanoylphorbol Acetate; Thionucleotides; Transcription, Genetic; Type C Phospholipases | 2002 |
Discriminative stimulus properties in rats of the novel antipsychotic quetiapine.
Topics: Amisulpride; Analysis of Variance; Animals; Antipsychotic Agents; Chlorpromazine; Clozapine; Dibenzothiazepines; Discrimination Learning; Discrimination, Psychological; Dose-Response Relationship, Drug; Female; Generalization, Psychological; Haloperidol; Loxapine; Quetiapine Fumarate; Quinoxalines; Rats; Rats, Wistar; Risperidone; Sulpiride | 2002 |
Respective roles of dopamine D2 and D3 receptors in food-seeking behaviour in rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Amisulpride; Analysis of Variance; Animals; Apomorphine; Benzazepines; Benzopyrans; Conditioning, Operant; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Synergism; Feeding Behavior; Haloperidol; Male; Naphthalenes; Pyrroles; Pyrrolidines; Quinolines; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Reinforcement, Psychology; Sulpiride; Tetrahydronaphthalenes | 2003 |
Sulpiride in combination with fluvoxamine increases in vivo dopamine release selectively in rat prefrontal cortex.
Topics: Animals; Antidepressive Agents, Second-Generation; Dopamine; Dopamine Agonists; Dopamine Antagonists; Fluvoxamine; Haloperidol; Male; Microdialysis; Neostriatum; Piperazines; Prefrontal Cortex; Pyridines; Rats; Rats, Wistar; Serotonin; Serotonin Antagonists; Sulpiride | 2005 |
EEG abnormalities under treatment with atypical antipsychotics: effects of olanzapine and amisulpride as compared to haloperidol.
Topics: Adult; Amisulpride; Antipsychotic Agents; Benzodiazepines; Chi-Square Distribution; Dose-Response Relationship, Drug; Electroencephalography; Female; Follow-Up Studies; Haloperidol; Humans; Male; Middle Aged; Olanzapine; Schizophrenia; Sulpiride | 2004 |
Effects of neonatal ventral hippocampal lesion in rats on stress-induced acetylcholine release in the prefrontal cortex.
Topics: Acetylcholine; Animals; Animals, Newborn; Benzazepines; Brain Diseases; Dopamine; Dopamine Antagonists; Haloperidol; Hippocampus; Microdialysis; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Stress, Physiological; Sulpiride | 2004 |
The impact of neuroleptic medication on seizure threshold and duration in electroconvulsive therapy.
Topics: Adult; Aged; Antipsychotic Agents; Benzodiazepines; Brain; Clopenthixol; Clozapine; Dibenzothiazepines; Electric Impedance; Electroconvulsive Therapy; Electroencephalography; Electromyography; Female; Fluphenazine; Haloperidol; Humans; Male; Middle Aged; Olanzapine; Quetiapine Fumarate; Risperidone; Seizures; Sulpiride | 2004 |
D2 dopamine receptors colocalize regulator of G-protein signaling 9-2 (RGS9-2) via the RGS9 DEP domain, and RGS9 knock-out mice develop dyskinesias associated with dopamine pathways.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antiparkinson Agents; Antipsychotic Agents; Apomorphine; Corpus Striatum; Dopamine; Dopamine Agents; Dopamine Antagonists; Dyskinesia, Drug-Induced; Female; Haloperidol; Humans; Mice; Mice, Knockout; Movement Disorders; Parkinson Disease; Patch-Clamp Techniques; Protein Interaction Mapping; Protein Structure, Tertiary; Quinpirole; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, G-Protein-Coupled; Recombinant Fusion Proteins; Reserpine; RGS Proteins; Subcellular Fractions; Sulpiride; Transfection | 2005 |
Behaviorally timid rats respond differentially to conventional and atypical neuroleptics.
Topics: Analysis of Variance; Animals; Antipsychotic Agents; Behavior, Animal; Clozapine; Female; Haloperidol; Ovariectomy; Random Allocation; Rats; Rats, Long-Evans; Social Behavior; Sulpiride; Time Factors | 2005 |
Dopamine D3 modulation of locomotor activity and sleep in the nucleus accumbens and in lobules 9 and 10 of the cerebellum in the rat.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Amisulpride; Amphetamine; Animals; Cerebellum; Dopamine Agonists; Dopamine Antagonists; Dopamine Uptake Inhibitors; Female; Haloperidol; Microinjections; Motor Activity; Naphthalenes; Nucleus Accumbens; Pyrrolidines; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Sleep; Sulpiride; Tetrahydronaphthalenes | 2005 |
[Treatment resistant schizophrenia, residual subtype: symptom improvement after additional treatment with amisulpride].
Topics: Adult; Amisulpride; Antipsychotic Agents; Benzodiazepines; Clozapine; Commitment of Mentally Ill; Drug Resistance; Drug Therapy, Combination; Follow-Up Studies; Haloperidol; Homicide; Humans; Insanity Defense; Male; Olanzapine; Prisoners; Schizophrenia, Paranoid; Sulpiride; Treatment Outcome | 2006 |
Dopamine D3 receptor modulation of dopamine efflux in the rat nucleus accumbens.
Topics: Animals; Antipsychotic Agents; Clozapine; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Electric Stimulation; Haloperidol; Male; Nitriles; Nucleus Accumbens; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Sulpiride; Tetrahydroisoquinolines; Tetrahydronaphthalenes | 2006 |
Antagonistic activity of ascorbic acid (vitamin C) on dopaminergic modulation: apomorphine-induced stereotypic behavior in mice.
Topics: Animals; Antioxidants; Antipsychotic Agents; Apomorphine; Ascorbic Acid; Azepines; Benzazepines; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Combinations; Haloperidol; Male; Mice; Reserpine; Stereotyped Behavior; Sulpiride | 2006 |
Prototypical antipsychotic drugs protect hippocampal neuronal cultures against cell death induced by growth medium deprivation.
Topics: Animals; Anisoles; Antipsychotic Agents; Benzazepines; Butaclamol; Caspase Inhibitors; Cell Death; Cells, Cultured; Chlorpromazine; Clozapine; Domperidone; Dopamine Antagonists; Excitatory Amino Acid Antagonists; Ginkgo biloba; Haloperidol; Hippocampus; Indans; Isoxazoles; Neurons; Neuroprotective Agents; Peptides; Piperidines; Plant Extracts; Propylamines; Raclopride; Rats; Rats, Sprague-Dawley; Reactive Oxygen Species; Receptors, N-Methyl-D-Aspartate; Remoxipride; Risperidone; Sulpiride | 2006 |
Is the superior efficacy of new generation antipsychotics an artifact of LOCF?
Topics: Amisulpride; Artifacts; Benzodiazepines; Bias; Flupenthixol; Haloperidol; Humans; Olanzapine; Patient Dropouts; Psychiatric Status Rating Scales; Psychotropic Drugs; Randomized Controlled Trials as Topic; Schizophrenia; Schizophrenic Psychology; Sulpiride; Treatment Outcome | 2007 |
Hemichorea associated with polycythaemia vera.
Topics: Acute Disease; Aged; Anti-Dyskinesia Agents; Chorea; Dopamine Antagonists; Female; Haloperidol; Humans; Phlebotomy; Polycythemia Vera; Sulpiride | 2006 |
Effect of quinpirole on timing behaviour in the free-operant psychophysical procedure: evidence for the involvement of D2 dopamine receptors.
Topics: Animals; Behavior, Animal; Conditioning, Operant; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Drug Interactions; Female; Haloperidol; Quinpirole; Rats; Rats, Wistar; Reaction Time; Salicylamides; Sulpiride | 2007 |
The putative antipsychotic alstonine reverses social interaction withdrawal in mice.
Topics: Animals; Anti-Anxiety Agents; Antipsychotic Agents; Clozapine; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Haloperidol; Interpersonal Relations; Male; Mice; Motor Activity; Secologanin Tryptamine Alkaloids; Social Behavior Disorders; Sulpiride | 2008 |
Subnanomolar dopamine D3 receptor antagonism coupled to moderate D2 affinity results in favourable antipsychotic-like activity in rodent models: I. neurochemical characterisation of RG-15.
Topics: Amisulpride; Animals; CHO Cells; Cricetinae; Cricetulus; Dopamine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Haloperidol; Humans; Inhibitory Concentration 50; Male; Mice; Nitriles; Prolactin; Pyridines; Rats; Rats, Wistar; Receptors, Dopamine D3; Sulfonamides; Sulpiride; Tetrahydroisoquinolines | 2008 |
Amisulpride the 'atypical' atypical antipsychotic--comparison to haloperidol, risperidone and clozapine.
Topics: Amisulpride; Amphetamine; Animals; Antipsychotic Agents; Basal Ganglia; Behavior, Animal; Blood-Brain Barrier; Brain; Clozapine; Conditioning, Psychological; Haloperidol; Male; Models, Animal; Motor Activity; Phencyclidine; Prefrontal Cortex; Prolactin; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Serotonin; Risperidone; Sulpiride | 2008 |
Clozapine and sulpiride but not haloperidol or olanzapine activate brain DNA demethylation.
Topics: Acetylation; Animals; Benzodiazepines; Brain; Cell Adhesion Molecules, Neuronal; Clozapine; DNA Methylation; Extracellular Matrix Proteins; Glutamate Decarboxylase; Haloperidol; Histones; Lysine; Male; Mice; Nerve Tissue Proteins; Olanzapine; Promoter Regions, Genetic; Reelin Protein; Serine Endopeptidases; Sulpiride; Valproic Acid | 2008 |
Antipsychotics possessing antidepressive efficacy increase Golf protein in rat striatum.
Topics: Amisulpride; Animals; Antipsychotic Agents; Benzodiazepines; Blotting, Western; Clozapine; Corpus Striatum; Depressive Disorder; Dose-Response Relationship, Drug; GTP-Binding Protein alpha Subunits; Haloperidol; Injections, Intraperitoneal; Male; Olanzapine; Rats; Rats, Wistar; Risperidone; Sulpiride; Time Factors | 2008 |
Antidepressant-like effect of 17beta-estradiol: involvement of dopaminergic, serotonergic, and (or) sigma-1 receptor systems.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anti-Inflammatory Agents; Antidepressive Agents; Benzazepines; Cyclohexanols; Dopamine Antagonists; Dose-Response Relationship, Drug; Estradiol; Haloperidol; Hindlimb Suspension; Male; Mice; Motor Activity; Progesterone; Receptors, Dopamine; Receptors, Serotonin; Receptors, sigma; Selective Serotonin Reuptake Inhibitors; Serotonin Receptor Agonists; Sigma-1 Receptor; Sulpiride; Swimming; Venlafaxine Hydrochloride | 2008 |
Antipsychotic drugs inhibit nucleotide hydrolysis in zebrafish (Danio rerio) brain membranes.
Topics: 5'-Nucleotidase; Animals; Antipsychotic Agents; Benzodiazepines; Brain; Dose-Response Relationship, Drug; Enzyme Inhibitors; Female; Haloperidol; Hydrolysis; Intracellular Membranes; Male; Nucleoside-Triphosphatase; Olanzapine; Sulpiride; Zebrafish | 2009 |
Inhibitory effects of polyphenol compounds on lipid peroxidation caused by antipsychotics (haloperidol and amisulpride) in human plasma in vitro.
Topics: Adult; Amisulpride; Antioxidants; Antipsychotic Agents; Female; Haloperidol; Humans; In Vitro Techniques; Lipid Peroxidation; Male; Quercetin; Resveratrol; Stilbenes; Sulpiride; Thiobarbituric Acid Reactive Substances | 2010 |
Targeting cognition in schizophrenia research: from etiology to treatment.
Topics: Amisulpride; Antipsychotic Agents; Benzodiazepines; Cognition; Cognition Disorders; Dibenzothiazepines; Drug Administration Schedule; Haloperidol; Humans; Olanzapine; Piperazines; Quetiapine Fumarate; Reaction Time; Schizophrenia; Sulpiride; Thiazoles | 2009 |
Reduced serum BDNF levels in patients with chronic schizophrenic disorder in relapse, who were treated with typical or atypical antipsychotics.
Topics: Adult; Amisulpride; Antipsychotic Agents; Benzodiazepines; Brain-Derived Neurotrophic Factor; Case-Control Studies; Female; Haloperidol; Humans; Male; Middle Aged; Olanzapine; Risperidone; Schizophrenia; Sulpiride; Treatment Failure | 2010 |
Haloperidol induces higher Homer1a expression than risperidone, olanzapine and sulpiride in striatal sub-regions.
Topics: Animals; Antipsychotic Agents; Benzodiazepines; Brain Mapping; Carrier Proteins; Corpus Striatum; Gene Expression Regulation; Haloperidol; Homer Scaffolding Proteins; Male; Olanzapine; Random Allocation; Rats; Rats, Sprague-Dawley; Risperidone; RNA, Messenger; Sulpiride | 2010 |
Positron emission tomography measurement of dopamine D₂ receptor occupancy in the pituitary and cerebral cortex: relation to antipsychotic-induced hyperprolactinemia.
Topics: Adult; Antipsychotic Agents; Benzodiazepines; Carbon Radioisotopes; Cerebellar Cortex; Cerebral Cortex; Computer Graphics; Dopamine Antagonists; Dose-Response Relationship, Drug; Haloperidol; Humans; Hyperprolactinemia; Male; Mathematical Computing; Middle Aged; Olanzapine; Pituitary Gland; Positron-Emission Tomography; Prolactin; Pyrrolidines; Receptors, Dopamine D2; Risperidone; Salicylamides; Schizophrenia; Statistics as Topic; Sulpiride; Temporal Lobe; Young Adult | 2010 |
Involvement of dopamine receptors in the antidepressant-like effect of melatonin in the tail suspension test.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antidepressive Agents; Apomorphine; Benzazepines; Dopamine Agonists; Dopamine Antagonists; Drug Synergism; Fluoxetine; Haloperidol; Immobility Response, Tonic; Male; Melatonin; Mice; Motor Activity; Sulpiride | 2010 |
Serotonin-dopamine antagonism ameliorates impairments of spontaneous alternation and locomotor hyperactivity induced by repeated electroconvulsive seizures in rats.
Topics: Analysis of Variance; Animals; Behavior, Animal; Dopamine Antagonists; Electroshock; Haloperidol; Hyperkinesis; Ketanserin; Male; Motor Activity; Random Allocation; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Serotonin, 5-HT2; Risperidone; Seizures; Serotonin Antagonists; Sulpiride | 2010 |
Beta-glucan from Saccharomyces cerevisiae reduces plasma lipid peroxidation induced by haloperidol.
Topics: Adult; Amisulpride; Analysis of Variance; Antipsychotic Agents; beta-Glucans; Female; Haloperidol; Humans; Lipid Peroxidation; Male; Saccharomyces cerevisiae; Schizophrenia; Sulpiride; Thiobarbituric Acid Reactive Substances | 2011 |
Differential effects of amisulpride and haloperidol on dopamine D2 receptor-mediated signaling in SH-SY5Y cells.
Topics: Amisulpride; Arrestins; beta-Arrestin 2; beta-Arrestins; Cell Line, Tumor; Dopamine D2 Receptor Antagonists; Haloperidol; Humans; Neurites; Receptors, Dopamine D2; Signal Transduction; Sulpiride | 2011 |
Effects of amisulpride and aripiprazole on progressive-ratio schedule performance: comparison with clozapine and haloperidol.
Topics: Amisulpride; Animals; Antipsychotic Agents; Aripiprazole; Behavior, Animal; Clozapine; Conditioning, Operant; Dopamine Antagonists; Dose-Response Relationship, Drug; Female; Haloperidol; Kinetics; Models, Biological; Motor Activity; Motor Skills; Piperazines; Quinolones; Rats; Rats, Wistar; Reaction Time; Reinforcement Schedule; Serotonin Antagonists; Sulpiride | 2012 |
Behavioral changes induced by long-term proline exposure are reversed by antipsychotics in zebrafish.
Topics: 1-Pyrroline-5-Carboxylate Dehydrogenase; Amino Acid Metabolism, Inborn Errors; Animals; Antipsychotic Agents; Anxiety; Disease Models, Animal; Drug Interactions; Female; Haloperidol; Locomotion; Male; Proline; Proline Oxidase; Social Behavior; Sulpiride; Time Factors; Zebrafish | 2012 |
MK-801 alters Na+, K+-ATPase activity and oxidative status in zebrafish brain: reversal by antipsychotic drugs.
Topics: Animals; Antipsychotic Agents; Benzodiazepines; Brain Chemistry; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Female; Fluoresceins; Haloperidol; Lipid Peroxidation; Male; Membranes; Nerve Tissue Proteins; Olanzapine; Oxidative Stress; Reactive Nitrogen Species; Reactive Oxygen Species; Sodium-Potassium-Exchanging ATPase; Sulpiride; Thiobarbituric Acid Reactive Substances; Zebrafish | 2012 |
Onset of action of atypical and typical antipsychotics in the treatment of adolescent schizophrenic psychoses.
Topics: Adolescent; Antipsychotic Agents; Benzodiazepines; Clozapine; Dibenzothiazepines; Female; Haloperidol; Humans; Male; Medical Records; Olanzapine; Perphenazine; Piperazines; Psychotic Disorders; Quetiapine Fumarate; Risperidone; Schizophrenia; Sulpiride; Thiazoles; Time Factors; Treatment Outcome | 2011 |
Attentional and emotional functioning in schizophrenia patients treated with conventional and atypical antipsychotic drugs.
Topics: Adult; Amisulpride; Analysis of Variance; Antipsychotic Agents; Attention; Benzodiazepines; Dibenzothiazepines; Emotions; Fluphenazine; Haloperidol; Humans; Memory; Middle Aged; Olanzapine; Perazine; Perphenazine; Quetiapine Fumarate; Recognition, Psychology; Risperidone; Schizophrenia; Sulpiride | 2012 |
Effectiveness of sulpiride in adult patients with schizophrenia.
Topics: Adolescent; Adult; Aged; Antipsychotic Agents; Benzodiazepines; Cohort Studies; Female; Haloperidol; Humans; Male; Middle Aged; Olanzapine; Proportional Hazards Models; Retrospective Studies; Risperidone; Schizophrenia; Sulpiride; Treatment Outcome; Young Adult | 2013 |
Differential effects of antipsychotics on lateral bias and social attention in female rats.
Topics: Animals; Antipsychotic Agents; Attention; Behavior, Animal; Clozapine; Disease Models, Animal; Female; Functional Laterality; Haloperidol; Rats; Rats, Long-Evans; Social Behavior; Sulpiride | 2013 |
Structure-based drug design for dopamine D3 receptor.
Topics: Animals; Combinatorial Chemistry Techniques; Drug Design; Haloperidol; Humans; Indoles; Mice; Models, Molecular; Molecular Structure; Piperazines; Piperidines; Pyrazoles; Pyridines; Receptors, Dopamine D3; Spiperone; Structure-Activity Relationship; Sulpiride; Thiophenes | 2012 |
Choline acetyltransferase expression in rat prefrontal cortex and hippocampus after acute and chronic exposure to amisulpride, haloperidol, and risperidone.
Topics: Amisulpride; Animals; Antipsychotic Agents; Choline O-Acetyltransferase; Dose-Response Relationship, Drug; Haloperidol; Hippocampus; Male; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Risperidone; Sulpiride; Time Factors | 2012 |
Imaging brain gene expression profiles by antipsychotics: region-specific action of amisulpride on postsynaptic density transcripts compared to haloperidol.
Topics: Amisulpride; Animals; Antipsychotic Agents; Cerebral Cortex; Corpus Striatum; Dopamine Antagonists; Dose-Response Relationship, Drug; Functional Neuroimaging; Gene Expression Profiling; Genes, Immediate-Early; Haloperidol; Limbic System; Male; Organ Specificity; Post-Synaptic Density; Rats; Sulpiride | 2013 |
White-matter microstructure in previously drug-naive patients with schizophrenia after 6 weeks of treatment.
Topics: Adolescent; Adult; Anisotropy; Antipsychotic Agents; Aripiprazole; Benzodiazepines; Brain; Brain Mapping; Case-Control Studies; Dibenzothiazepines; Diffusion Tensor Imaging; Female; Frontal Lobe; Gyrus Cinguli; Haloperidol; Humans; Image Processing, Computer-Assisted; Male; Nerve Fibers, Myelinated; Olanzapine; Piperazines; Quetiapine Fumarate; Quinolones; Risperidone; Schizophrenia; Schizophrenic Psychology; Sulpiride; Treatment Outcome; Young Adult | 2013 |
Effects of cabergoline on hyperprolactinemia, psychopathology, and sexual functioning in schizophrenic patients.
Topics: Adult; Amisulpride; Antipsychotic Agents; Cabergoline; Diagnostic and Statistical Manual of Mental Disorders; Dopamine Agonists; Dose-Response Relationship, Drug; Ergolines; Female; Haloperidol; Humans; Hyperprolactinemia; Longitudinal Studies; Maintenance Chemotherapy; Male; Middle Aged; Prolactin; Prospective Studies; Risperidone; Schizophrenia; Schizophrenic Psychology; Severity of Illness Index; Sexual Dysfunction, Physiological; Sulpiride | 2013 |
Proline-induced changes in acetylcholinesterase activity and gene expression in zebrafish brain: reversal by antipsychotic drugs.
Topics: Acetylcholinesterase; Animals; Antipsychotic Agents; Brain; Brain Chemistry; Female; Gene Expression; Haloperidol; In Vitro Techniques; Male; Nerve Tissue Proteins; Parasympathetic Nervous System; Proline; Real-Time Polymerase Chain Reaction; Sulpiride; Zebrafish | 2013 |
Implication of the ERK/MAPK pathway in antipsychotics-induced dopamine D2 receptor upregulation and in the preventive effects of (±)-α-lipoic acid in SH-SY5Y neuroblastoma cells.
Topics: Amisulpride; Antipsychotic Agents; Cell Line, Tumor; Cell Survival; Haloperidol; Humans; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Neurons; Neuroprotective Agents; Receptors, Dopamine D2; RNA, Messenger; Sulpiride; Thioctic Acid; Up-Regulation | 2014 |
Upregulation of dopamine D3, not D2, receptors correlates with tardive dyskinesia in a primate model.
Topics: Animals; Antipsychotic Agents; Brain; Cebus; Clozapine; Disease Models, Animal; Dopamine Antagonists; Enkephalins; Female; Haloperidol; Iodine Radioisotopes; Movement Disorders; Neurons; Ovariectomy; Protein Binding; Receptors, Dopamine D2; Receptors, Dopamine D3; Sulpiride; Tetrahydronaphthalenes; Up-Regulation | 2014 |
The role of dopamine in motor flexibility.
Topics: Adult; Anticipation, Psychological; Dopamine; Dopamine Agents; Double-Blind Method; Female; Haloperidol; Humans; Levodopa; Male; Probability; Psychomotor Performance; Reaction Time; Receptors, Dopamine D1; Receptors, Dopamine D2; Sulpiride | 2015 |
Effects of ovarian dopaminergic receptors on ovulation.
Topics: Animals; Benzazepines; Dopamine and cAMP-Regulated Phosphoprotein 32; Estradiol; Estrous Cycle; Female; Gonadotropin-Releasing Hormone; Haloperidol; Ovarian Follicle; Ovulation; Progesterone; Random Allocation; Rats; Receptors, Dopamine; Sulpiride; Tyrosine 3-Monooxygenase | 2015 |
Investigation into effects of antipsychotics on ectonucleotidase and adenosine deaminase in zebrafish brain.
Topics: Adenosine Deaminase; Adenosine Triphosphatases; Animals; Antipsychotic Agents; Benzodiazepines; Brain; Female; Haloperidol; Hydrolysis; Male; Olanzapine; Sulpiride; Zebrafish; Zebrafish Proteins | 2015 |
Pramipexole at a Low Dose Induces Beneficial Effect in the Harmaline-induced Model of Essential Tremor in Rats.
Topics: Amisulpride; Animals; Anti-Dyskinesia Agents; Benzothiazoles; Disease Models, Animal; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Essential Tremor; Haloperidol; Harmaline; Imidazoles; Male; Movement; Nitriles; Pramipexole; Pyridines; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Sulpiride; Tetrahydroisoquinolines; Tetrahydronaphthalenes; Treatment Outcome | 2016 |
Antipsychotic Drugs Differentially Affect mRNA Expression of Genes Encoding the Neuregulin 1-Downstream ErbB4-PI3K Pathway.
Topics: Amisulpride; Antipsychotic Agents; Benzodiazepines; Cell Line, Tumor; Cell Survival; Clozapine; Gene Expression Regulation; Haloperidol; Humans; Neuregulin-1; Olanzapine; Phosphatidylinositol 3-Kinases; Quetiapine Fumarate; Receptor, ErbB-4; RNA, Messenger; Schizophrenia; Sulpiride | 2016 |
Switching antipsychotics: Imaging the differential effect on the topography of postsynaptic density transcripts in antipsychotic-naïve vs. antipsychotic-exposed rats.
Topics: Amisulpride; Animals; Antipsychotic Agents; Cerebral Cortex; Corpus Striatum; Cytoskeletal Proteins; Disks Large Homolog 4 Protein; Drug Resistance; Drug Substitution; Gene Expression; Haloperidol; Homer Scaffolding Proteins; Injections, Intraperitoneal; Intracellular Signaling Peptides and Proteins; Male; Membrane Proteins; Nerve Tissue Proteins; Post-Synaptic Density; Random Allocation; Rats, Sprague-Dawley; RNA, Messenger; Sulpiride | 2016 |
Time to Discontinuation of Second-Generation Antipsychotics Versus Haloperidol and Sulpiride in People With Schizophrenia: A Naturalistic, Comparative Study.
Topics: Adult; Antipsychotic Agents; Clozapine; Female; Haloperidol; Humans; Male; Medication Adherence; Retrospective Studies; Schizophrenia; Sulpiride; Taiwan; Time Factors; Young Adult | 2017 |
Haloperidol Decreases Hyperalgesia and Allodynia Induced by Chronic Constriction Injury.
Topics: Amines; Analgesics; Animals; Antipsychotic Agents; Chronic Disease; Constriction, Pathologic; Cyclohexanecarboxylic Acids; Dose-Response Relationship, Drug; Gabapentin; gamma-Aminobutyric Acid; Haloperidol; Hyperalgesia; Injections, Spinal; Male; Neuralgia; Pain Measurement; Piperazines; Rats; Rats, Wistar; Receptors, sigma; Sigma-1 Receptor; Sulpiride | 2017 |
Involvement of vascular endothelial growth factor (VEGF) and mitogen-activated protein kinases (MAPK) in the mechanism of neuroleptic drugs.
Topics: Amisulpride; Antipsychotic Agents; Benzodiazepines; Cell Line, Tumor; Haloperidol; Humans; Mitogen-Activated Protein Kinases; Neuroprotective Agents; Olanzapine; Pituitary Adenylate Cyclase-Activating Polypeptide; Signal Transduction; Sulpiride; Vascular Endothelial Growth Factor A | 2018 |
Antipsychotics and pituitary tumors: an analysis of the European pharmacovigilance database (EudraVigilance).
Topics: Adolescent; Adult; Aged; Amisulpride; Antipsychotic Agents; Child; Databases, Factual; Female; Haloperidol; Humans; Male; Middle Aged; Olanzapine; Paliperidone Palmitate; Pharmacovigilance; Pituitary Neoplasms; Pregnancy; Quetiapine Fumarate; Retrospective Studies; Risperidone; Sulpiride; Young Adult | 2019 |
Zinc enhances the expression of morphine-induced conditioned place preference through dopaminergic and serotonergic systems.
Topics: Animals; Benzazepines; Conditioning, Psychological; Dopamine Antagonists; Haloperidol; Ketanserin; Male; Morphine; Ondansetron; Piperazines; Rats; Rats, Wistar; Reward; Serotonin Antagonists; Sulpiride; Zinc | 2019 |
Letter to the Editor: Rethinking The Cost Of Antipsychotic Treatment: The Average Cost Of The Drugs Used In Turkey In 2020.
Topics: Adenosine Monophosphate; Adult; Amisulpride; Antipsychotic Agents; Aripiprazole; Benzodiazepines; Chlorpromazine; Clopenthixol; Clozapine; Flupenthixol; Fluphenazine; Haloperidol; Humans; Olanzapine; Paliperidone Palmitate; Pharmaceutical Preparations; Pimozide; Quetiapine Fumarate; Risperidone; Sulpiride; Trifluoperazine | 2022 |
Environmentally-relevant concentrations of the antipsychotic drugs sulpiride and clozapine induce abnormal dopamine and serotonin signaling in zebrafish brain.
Topics: Animals; Antipsychotic Agents; Brain; Clozapine; Dopamine; Haloperidol; Monoamine Oxidase; RNA, Messenger; Serotonin; Serotonin Plasma Membrane Transport Proteins; Sulpiride; Zebrafish | 2022 |