Page last updated: 2024-08-16

sulpiride and clozapine

sulpiride has been researched along with clozapine in 234 studies

Research

Studies (234)

TimeframeStudies, this research(%)All Research%
pre-199047 (20.09)18.7374
1990's45 (19.23)18.2507
2000's88 (37.61)29.6817
2010's48 (20.51)24.3611
2020's6 (2.56)2.80

Authors

AuthorsStudies
Audiau, F; Carpy, A; Guérémy, C; Le Fur, G; Léger, JM; Uzan, A1
Bechelli, S; Cagnotto, A; Campiani, G; Ciani, SM; de Boer, P; Fiorini, I; Garofalo, A; Liao, Y; Mennini, T; Nacci, V; Tepper, PG; Wikström, H1
Topliss, JG; Yoshida, F1
Faller, B; Wohnsland, F1
Fang, X; Hu, Z; Levant, B; Min, J; Varady, J; Wang, S; Wu, X1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Bleich, S; Gulbins, E; Kornhuber, J; Reichel, M; Terfloth, L; Tripal, P; Wiltfang, J1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chen, L; He, Z; Li, H; Liu, J; Liu, X; Sui, X; Sun, J; Wang, Y; Zhang, W1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Alelyunas, YW; Bui, K; Empfield, JR; McCarthy, D; Pelosi-Kilby, L; Shen, C; Spreen, RC1
Boriss, H; Braggio, S; Corbioli, S; Fontana, S; Helmdach, L; Longhi, R; Schiller, J; Vinco, F1
Barber, J; Dawson, S; Kenna, JG; Paul, N; Stahl, S1
Ambroso, JL; Ayrton, AD; Baines, IA; Bloomer, JC; Chen, L; Clarke, SE; Ellens, HM; Harrell, AW; Lovatt, CA; Reese, MJ; Sakatis, MZ; Taylor, MA; Yang, EY1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Chen, L; Fei, J; Mei, Y; Ren, S; Yan, SF; Zeng, J; Zhang, JZ1
Bartholini, G1
Ackenheil, M; von Stralendorff, B; Zimmermann, J1
Costa, E1
Munday, KA; Poat, JA; Sumners, C; Woodruff, GN1
Bronzetti, B; Ciriaco, E; Germanà, G; Nisticó, G; Rotiroti, D; Scapagnini, U1
Krause, R; Lotz, W1
Costall, B; Naylor, RJ4
Korf, J; Westerink, BH1
Roufogalis, BD; Thornton, M; Wade, DN1
Maître, L; Waldmeier, PC1
Fukushima, H; Honma, T1
Asenbaum, S; Brücke, T; Podreka, I; Roth, J; Strobl, R; Wenger, S1
Ciancone, MT; Haracz, JL; Rebec, GV; White, IM1
Budygin, EA; Gaĭnetdinov, RR; Kovalev, GI; Kudrin, VS; Raevskiĭ, KS1
Britton, DR; Buckley, M; Curzon, P; Nadzan, A; Tufano, M; Yahiro, L1
Bakhtiar, R; Bull, DR; Sheehan, MJ1
Fink, H; Morgenstern, R; Ott, T; Schremmer, C1
Bunney, BS; Moghaddam, B2
Bruhwyler, J; Chleide, E; Delarge, J; Liégeois, JF; Mercier, M1
Pfaus, JG; Phillips, AG1
Davis, KL; Guerin, JJ; Halperin, R1
Brugger, AJ; Martínez, JA; Milanés, MV; Pérez, D; Vargas, ML1
Fleminger, S; Hall, MD; Jenner, P; Kelly, E; Kilpatrick, G; Marsden, CD; Rupniak, NM1
el Mestikawy, S; Glowinski, J; Hamon, M1
Andree, TH; Koenig, JI; Meltzer, HY; Mikuni, M; Tong, CY1
Chang, KJ; Ferris, RM; Russell, A; Tang, FL1
Meltzer, HY1
Cools, AR1
Aghajanian, GK; Rasmussen, K1
Arbilla, S; Baud, P; Langer, SZ1
Yang, WJ1
Jenner, P; Marsden, CD; Rupniak, NM1
Halliday, CA; Leonard, MN; Marriott, AS; Strange, PG1
Briggs, RS; Jenner, P; Mann, S; Marsden, CD; Petersen, MM; Reavill, C; Rupniak, NM1
Horton, RW; Jenner, P; Marsden, CD; Prestwich, SA; Rupniak, NM1
Decker, H; Dimpfel, W1
Guidotti, A1
Bronzetti, B; Ciriaco, E; Germanà, G; Nisticò, G1
Kuribara, H; Tadokoro, S1
Aghajanian, GK; Marwaha, J1
Colboc, O; Costentin, J; Dubuc, I; Protais, P1
Etienne, P; Lal, S; Nair, NP; Wood, PL1
Pi, EH; Simpson, GM1
Borsini, F; Nowakowska, E; Samanin, R1
Jenner, P; Kerwin, RW; Marsden, CD; Rupniak, NM1
Steranka, LR1
Zharkovskaia, TA; Zharkovskiĭ, AM1
Lee, T; Tang, SW1
Hall, MD; Jenner, P; Kilpatrick, G; Marsden, CD; Rupniak, NM1
Gold, R; Lemme, P; Mende, T; Morgenstern, R; Oelssner, W1
Fink, H; Morgenstern, R; Oelssner, W1
Angeby, T; Haglund, L; Köhler, C; Ogren, SO1
Deutch, AY; Duman, RS; Ongür, D1
Baldessarini, RJ; Gardner, DM; Garver, DL1
Perrault, G; Sanger, DJ1
Takaki, T; Tanaka, M; Yamada, S; Yokoo, H1
de Angelis, L1
Buckland, PR; McGuffin, P; Oretti, RG; Spurlock, G1
Kenyon, P; Moore, S1
Buckland, PR; McGuffin, P; O'Donovan, MC1
Celander, M; Svartengren, J1
Nowak, JZ; Zawilska, JB1
Strange, PG1
Wang, HH; Xu, SF1
Imagawa, Y; Okuyama, S; Tomisawa, K1
Gerlach, J; Peacock, L1
Obuchowicz, E1
Fukamauchi, F; Kito, S; Mataga, N; Miyoshi, R; Sakai, M; Semba, J1
Hurley, MJ; Jenner, P; Marsden, CD; Stubbs, CM1
Griffon, N; Pilon, C; Sautel, F; Schwartz, JC; Sokoloff, P1
Derbiszewska, T; Nowak, JZ; Zawilska, JB1
Kołodziejczyk, K; Maj, J; Rogóz, Z; Skuza, G1
Buckland, PR; D'Souza, U; Maher, NA; McGuffin, P1
Aizenberg, D; Dorfman-Etrog, P; Khaikin, M; Modai, I; Radwan, M; Schwartz, B; Shiloh, R; Weizman, A; Zemishlany, Z1
Attar-Levy, D; Martinot, JL; Monnet, F; Paillère-Martinot, ML; Recassens, C; Trichard, C1
Hoes, MJ1
Kulkarni, SK; Ninan, I1
Procopio, M1
Gioanni, Y; Glowinski, J; Tassin, JP; Thierry, AM1
Obuchowicz, E; Turchan, J1
Hayashi, T; Kagaya, A; Nishida, A; Shimizu, M; Su, TP; Yamawaki, S1
Müssigbrodt, HE; Wetterling, T1
Buljat, G; Dodig, G; Jelovac, N; Marovic, A; Miklic, P; Mise, S; Perovic, D; Petek, M; Prkacin, I; Rucman, R; Seiwerth, S; Sikiric, P; Turkovic, B1
Bradley, RJ; Dwyer, DS; Liu, Y1
Bayle, FJ; Ghaoui, S; Olie, JP1
Gobbi, G; Janiri, L1
Aguilar, MA; Arenas, MC; Miñarro, J; Parra, A; Simón, VM; Vinader-Caerols, C1
Naber, D1
Möller, HJ1
McAskill, R; Taylor, DM1
Liu, W; Wu, CF; Zhang, HL1
Hillefors, M; von Euler, G1
Haw, CM; Mountjoy, CQ; Staley, CJ; Stubbs, JH1
Bebbington, P; Freemantle, N; Geddes, J; Harrison, P1
Braus, DF; Jatzko, A; Ries, S; Schreiner, A1
Kapur, S; Remington, G2
Agelink, MW; Klieser, E; Linka, T; Lukas, K; Majewski, T; Ullrich, H; Wurthmann, C1
Hilger, E; Kasper, S1
Fu, D; Javitch, JA; Lin, H; Strange, PG; Wilson, J1
Kruse, CG; Long, SK; Nievelstein, H; Wadman, WJ; Werkman, TR1
Reuss, B; Unsicker, K1
Pittman, QJ; Price, CJ1
Hatzimanolis, J; Lykouras, L; Markianos, M1
Dai, J; Fowler, WL; Ichikawa, J; Meltzer, HY; O'Laughlin, IA1
Bartholini, F; Casu, MA; Gessa, GL; Marchese, G; Pani, L; Ruiu, S; Saba, P1
Miledi, R; Nguyen, QT; Yang, J1
Bayle, FJ; Chereau, I; Lancon, C; Llorca, PM1
Bottlender, R; Dobmeier, P; Hofschuster, E; Jäger, M; Möller, HJ1
Jørgensen, JI; Sindø, I1
Basta-Kaim, A; Budziszewska, B; Jaworska-Feil, L; Kubera, M; Lasoń, W; Leśkiewicz, M; Tetich, M1
Goudie, AJ; Smith, JA1
Castle, DJ; Lambert, TJ1
Abou El Ela, A; Galla, HJ; Härtter, S; Hiemke, C; Hüwel, S; Langguth, P; Lohmann, T1
Henn, FA; Knopf, U; Thome, J; Zink, M1
Bitter, I1
Agelink, MW; Ak, I; Kavuk, I1
Freudenreich, O; Goff, D; Stahl, S1
Beer, MD; Cobb, AM; Kerwin, R; Launer, M; Matthiasson, P; Munro, J; Osborne, S; Purcell, S; Travis, M1
Bryois, Ch; Sahli, Ch1
Lawrie, S; McIntosh, A; Nadeem, Z2
Barna, I; Gazdag, G; Iványi, Z; Tolna, J1
Cowan, C; George, S1
Croissant, B; Hermann, D; Olbrich, R1
Agelink, MW; Kämpf, P; Naber, D1
Cook, B; Hoogenboom, G1
Lawrie, S; McIntosh, A1
Taylor, GT; Yuede, CM1
Berk, M; Bourin, M; Dodd, S; Ivanovski, B; Lagopoulos, J; Malhi, GS; Mitchell, PB1
Epshtein, S; Kreinin, A; Sheinkman, A; Tell, E1
Kruse, CG; McCreary, AC; Olijslagers, JE; Perlstein, B; Siarey, R; Wadman, WJ; Werkman, TR1
Bergemann, N; Frick, A; Kopitz, J; Kress, KR1
Brown, D; Fraser, K; Martin, M; Taylor, M; Turner, M; Watt, L1
Frecska, E1
Knecht, G; Naber, D; Veismann, S; Wolf, K1
Kreinin, A; Novitski, D; Weizman, A1
Cummins, R; Gnoffo, Z; Kew, JN; Roberts, C1
Bastianetto, S; Danik, M; Mennicken, F; Quirion, R; Williams, S1
Guo, WB; Guo, XF; Liu, ZN; Tang, JS; Wu, RR; Zhai, JG; Zhao, JP1
Baumgartner, S; Ebenbichler, C; Edlinger, M; Fleischhacker, WW; Hofer, A; Hummer, M; Kemmler, G; Lechleitner, M; Rettenbacher, MA1
Baumgartner, S; Ebenbichler, C; Edlinger, M; Hofer, A; Hummer, M; Kemmler, G; Lechleitner, M; Rettenbacher, MA; Wolfgang Fleischhacker, W1
Heidari, P; Riazi, G; Sahebgharani, M; Zarrindast, MR1
Alonso, J; Haro, JM; Lépine, JP; Novick, D; Ratcliffe, M; Suarez, D1
Heidari, P; Malekmohamadi, N; Sahebgharani, M; Zarrindast, MR1
Limosin, F1
Benitez, J; Daskalakis, ZJ; Egan, GF; Fitzgerald, PB; Jackson, G; Kulkarni, J; Sritharan, A1
Danovich, L; Gavish, M; Lahav, M; Leschiner, S; Shuster, V; Veenman, L; Weizman, A1
Bret, MC; Bret, P; Fourier-Réglat, A; Pariente, A1
Cazali, J; Dervaux, A1
Cai, ZJ; He, JL; Li, WB; Ungvari, GS; Xiang, YT1
Assion, HJ; Basilowski, M; Juckel, G; Lemanski, S; Reinbold, H1
Lang, UE; Malte Tugtekin, S; Matschke, K; Schmeisser, A; von Golitschek, R; Willbring, M1
Lawrie, SM; Shajahan, P; Taylor, M1
de Moura Linck, V; Elisabetsky, E; Goerck, GC; Herrmann, AP; Iwu, MM; Leal, MB; Okunji, CO1
Agai Csongor, E; Domány, G; Elekes, O; Gémesi, LI; Gyertyán, I; Kapás, M; Kedves, R; Kiss, B; Laszy, J; Pásztor, G; Sághy, K; Szombathelyi, Z; Zájer-Balázs, M1
Barlow, KB; Kapur, S; Natesan, S; Nobrega, JN; Reckless, GE1
Costa, E; Dong, E; Grayson, DR; Guidotti, A; Nelson, M1
Endo, S; Hamamura, T; Ishihara, T; Kuroda, S; Miyata, S; Taoka, H; Toma, K1
Akyildiz, U; Balci, V; Sevincok, L1
Kumar, R; Sachdev, PS1
Ayesa, R; Crespo-Facorro, B; Martínez-Garcia, O; Mata, I; Pérez-Iglesias, R; Ramirez-Bonilla, M; Rodríguez-Sánchez, JM; Vázquez-Barquero, JL1
Praharaj, SK; Sarkar, S; Sinha, VK1
Barbui, C; Boso, M; Cipriani, A1
Bhoopathi, PS; Hunger, H; Kissling, W; Komossa, K; Leucht, S; Rummel-Kluge, C; Schwarz, S1
Fenton, M; Omori, IM; Soares, B; Wang, J2
Gandotra, S; Praharaj, SK; Ray, P1
Duggan, L; Hunger, H; Kissling, W; Komossa, K; Leucht, S; Rummel-Kluge, C; Schmid, F; Schwarz, S1
Chen, CC; Chen, YY; Hung, GC1
Aggarwal, A; Sharma, DD1
Davis, JM; Hunger, H; Kissling, W; Komossa, K; Leucht, S; Lobos, CA; Rummel-Kluge, C; Schmid, F; Schwarz, S1
Bergman, J; Kreinin, A; Lerner, V; Libov, I; Miodownik, C; Shestakova, D; Sokolik, S1
Eberle, MC; Fallgatter, AJ; Plewnia, C; Wasserka, B; Wildgruber, D1
Claes, S; De Hert, M; Martens, GJ; Moons, T; Peuskens, J; Van Loo, KM; Van Schijndel, JE; van Winkel, R1
Hunger, H; Kissling, W; Komossa, K; Leucht, S; Rummel-Kluge, C; Schmid, F; Schwarz, S1
Begemann, MJ; Leucht, S; Sommer, IE; Temmerman, A1
Englisch, S; Esslinger, C; Meyer-Lindenberg, A; Rausch, F; Schirmbeck, F; Zink, M1
Ekström, J; Godoy, T; Riva, A2
Chiu, HW; Huang, HT; Ku, YC; Li, TC1
Body, S; Bradshaw, CM; de Bruin, N; den Boon, FS; Hampson, CL; Szabadi, E1
Dudova, I; Hrdlicka, M; Urbanek, T; Zedkova, I1
Alm, B; Englisch, S; Meyer-Lindenberg, A; Zink, M1
Chang, YT; Chen, CC; Chen, WJ; Kuo, CJ; Lee, WC; Liao, YT; Shau, WY; Tsai, SY; Yang, SY1
Kirchhoff, BA; Smith, SE; Taylor, GT1
Bowskill, SV; Flanagan, RJ; Handley, SA; Patel, MX1
Blagojević, D; Lečić-Toševski, D; Miljević, Č; Niketić, V; Nikolić, M; Nikolić-Kokić, A; Spasić, MB1
Couchman, L; Fisher, DS; Flanagan, RJ; Handley, SA; Morgan, PE; Partridge, SJ1
Fisher, DS; Flanagan, RJ; Handley, SA; Partridge, SJ1
Tufan, AE; Yalug, I1
Cantisani, A; Ferrari, G; Grassi, G; Pallanti, S; Poli, L; Righi, L1
Basu, A; Brooman-White, RS; Das, M; Gupta, N; Hotham, JE; Humphreys, SA; Larkin, F; Ross, CC; Simpson, PJ1
Cao, B; Hou, R; Jian, J; Mi, G; Qiu, H; Tang, M; Wang, M1
Blanchet, PJ; Lévesque, D; Mahmoudi, S1
Eifler, S; Englisch, S; Esslinger, C; Kirsch, P; Meyer-Lindenberg, A; Mier, D; Rausch, F; Schirmbeck, F; Zink, M1
Bianchini, O; Porcelli, S; Serretti, A1
Joyce, DW; Mateos Fernandez, MJ; Sarkar, SN; Shergill, SS; Tracy, DK1
Hema, T; Maran, S; Subhashini, G1
Antczak, A; Górski, P; Karbownik, MS; Kowalczyk, E; Pietras, T; Szemraj, J; Wieteska, Ł1
Chen, WH; Hsieh, MH; Huang, WL1
Bas, A; Bas, TO; Duran, A; Emul, M; Gultekin, G; Incir, S1
Chan, HY; Chen, CH; Chen, JJ; Pan, YJ1
Beyer, C; Fisher, DS; Flanagan, RJ; Seedat, S; van Schalkwyk, G1
Barber, S; Cipriani, A; Corsi, M; Olotu, U1
Amos, T; Bagalkote, H; Barnes, TR; Davies, L; Fitzgerald, Z; Fridrich, P; Haddad, PM; Husni, M; Iqbal, K; Keown, P; Kumar, R; Leeson, VC; Marston, L; Osborn, D; Paton, C; Singh, V; Whittaker, W; Zafar, R1
Abdel-Daim, MM; Ali, HA; El-Serehy, HA; Elmowalid, GA; Khalil, SR; Mahmoud, FA; Mohammed, AT1
Claro, A; Corte-Real, F; Franco, J; Monteiro, C; Mustra, C; Proença, P1
Bećirović, E; Brigić, A; Hasanović, M; Pajević, I; Prljača, E1
Osman, E; Yıldız, M1
Hu, QY; Huang, Y; Jin, Y; Li, ZZ; Liu, MJ; Liu, ZJ; Lv, QY; Shi, DH; Tan, HY; Wu, FC; Yang, JY; Yi, ZH; Zhao, L; Zhu, MH; Zhu, N1
Guo, Y; Li, T; Peng, X; Sun, X; Zhang, B1

Reviews

34 review(s) available for sulpiride and clozapine

ArticleYear
Atypical neuroleptics: clozapine and the benzamides in the prevention and treatment of tardive dyskinesia.
    Modern problems of pharmacopsychiatry, 1983, Volume: 21

    Topics: Antipsychotic Agents; Benzamides; Clinical Trials as Topic; Clozapine; Dibenzazepines; Dose-Response Relationship, Drug; Dyskinesia, Drug-Induced; Haloperidol; Humans; Metoclopramide; Prospective Studies; Schizophrenia; Sulpiride; Tiapamil Hydrochloride

1983
Dopamine receptors in the basal ganglia: relevance to Parkinson's disease.
    Movement disorders : official journal of the Movement Disorder Society, 1993, Volume: 8, Issue:3

    Topics: Basal Ganglia; Basal Ganglia Diseases; Brain; Clozapine; Dopamine Agents; Dopamine D2 Receptor Antagonists; Female; Haloperidol; Humans; Levodopa; Male; Neostriatum; Neural Pathways; Parkinson Disease; Receptors, Dopamine D1; Receptors, Dopamine D2; Sulpiride

1993
New antipsychotics: the present status.
    International clinical psychopharmacology, 1995, Volume: 10 Suppl 3

    Topics: Antipsychotic Agents; Binding, Competitive; Clozapine; Dopamine Antagonists; Haloperidol; Humans; Psychotic Disorders; Sulpiride

1995
Recent developments in the management of psychosis.
    Pharmacy world & science : PWS, 1998, Volume: 20, Issue:3

    Topics: Antipsychotic Agents; Clozapine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Humans; Psychotic Disorders; Risperidone; Serotonin Antagonists; Sulpiride

1998
[New antipsychotic agents].
    L'Encephale, 1999, Volume: 25 Spec No 3

    Topics: Amisulpride; Antipsychotic Agents; Benzodiazepines; Clozapine; Dibenzothiazepines; Humans; Imidazoles; Indoles; Olanzapine; Piperazines; Pirenzepine; Psychotic Disorders; Quetiapine Fumarate; Risperidone; Sulpiride; Thiazoles

1999
[New i.e. atypical neuroleptic agents for negative symptoms of schizophrenia: results and methodological problems of evaluation].
    Der Nervenarzt, 2000, Volume: 71, Issue:5

    Topics: Amisulpride; Antipsychotic Agents; Benzodiazepines; Clozapine; Dibenzothiazepines; Dibenzothiepins; Double-Blind Method; Dyskinesia, Drug-Induced; Humans; Imidazoles; Indoles; Neurotransmitter Agents; Olanzapine; Piperazines; Pirenzepine; Quetiapine Fumarate; Randomized Controlled Trials as Topic; Risperidone; Schizophrenia; Schizophrenic Psychology; Sulpiride; Thiazoles

2000
Atypical antipsychotics and weight gain--a systematic review.
    Acta psychiatrica Scandinavica, 2000, Volume: 101, Issue:6

    Topics: Amisulpride; Antipsychotic Agents; Benzodiazepines; Clozapine; Dibenzothiazepines; Dibenzothiepins; Humans; Imidazoles; Indoles; Olanzapine; Piperazines; Pirenzepine; Quetiapine Fumarate; Risperidone; Sulpiride; Thiazoles; Weight Gain

2000
Augmentation with sulpiride for a schizophrenic patient partially responsive to clozapine.
    Acta psychiatrica Scandinavica, 2000, Volume: 102, Issue:5

    Topics: Antipsychotic Agents; Clozapine; Drug Therapy, Combination; Humans; Male; Middle Aged; Randomized Controlled Trials as Topic; Schizophrenia, Paranoid; Sulpiride; Treatment Outcome

2000
Atypical antipsychotics in the treatment of schizophrenia: systematic overview and meta-regression analysis.
    BMJ (Clinical research ed.), 2000, Dec-02, Volume: 321, Issue:7273

    Topics: Amisulpride; Antipsychotic Agents; Benzodiazepines; Clozapine; Dibenzothiazepines; Drug Costs; Humans; Imidazoles; Indoles; Olanzapine; Pirenzepine; Quetiapine Fumarate; Regression Analysis; Risperidone; Schizophrenia; Sulpiride

2000
Atypical antipsychotics: new directions and new challenges in the treatment of schizophrenia.
    Annual review of medicine, 2001, Volume: 52

    Topics: Amisulpride; Antipsychotic Agents; Benzodiazepines; Clozapine; Dibenzothiazepines; Dibenzothiepins; Dopamine Antagonists; Drug Monitoring; Haloperidol; Humans; Imidazoles; Indoles; Olanzapine; Piperazines; Pirenzepine; Quetiapine Fumarate; Receptors, Dopamine D2; Receptors, Dopamine D4; Risperidone; Schizophrenia; Schizophrenic Psychology; Serotonin Antagonists; Sulpiride; Thiazoles; Treatment Outcome

2001
[Atypical neuroleptics: new approaches to drug therapy of schizophrenic disorders].
    Wiener klinische Wochenschrift, 2000, Dec-22, Volume: 112, Issue:24

    Topics: Aged; Amisulpride; Antipsychotic Agents; Benzodiazepines; Clozapine; Controlled Clinical Trials as Topic; Dibenzothiazepines; Dibenzothiepins; Haloperidol; Humans; Imidazoles; Indoles; Multicenter Studies as Topic; Olanzapine; Piperazines; Pirenzepine; Placebos; Quetiapine Fumarate; Risperidone; Schizophrenia; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Sulpiride; Thiazoles

2000
Dopamine D(2) receptors and their role in atypical antipsychotic action: still necessary and may even be sufficient.
    Biological psychiatry, 2001, Dec-01, Volume: 50, Issue:11

    Topics: Amisulpride; Antipsychotic Agents; Benzodiazepines; Clozapine; Dibenzothiazepines; Humans; Models, Neurological; Olanzapine; Pirenzepine; Quetiapine Fumarate; Receptors, Dopamine D2; Risperidone; Schizophrenia; Sulpiride

2001
Tardive dyskinesias and antipsychotics: a review.
    European psychiatry : the journal of the Association of European Psychiatrists, 2002, Volume: 17, Issue:3

    Topics: Amisulpride; Antipsychotic Agents; Benzodiazepines; Clozapine; Dyskinesia, Drug-Induced; Humans; Olanzapine; Pirenzepine; Prevalence; Psychotic Disorders; Risperidone; Sulpiride

2002
[Treatment of tics in Tourette syndrome with atypical antipsychotic drugs].
    Ugeskrift for laeger, 2002, Aug-05, Volume: 164, Issue:32

    Topics: Antipsychotic Agents; Benzodiazepines; Clozapine; Dopamine Antagonists; Humans; Olanzapine; Pirenzepine; Risperidone; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Sulpiride; Tics; Tourette Syndrome

2002
Pharmacological approaches to the management of schizophrenia.
    The Medical journal of Australia, 2003, 05-05, Volume: 178, Issue:S9

    Topics: Amisulpride; Antipsychotic Agents; Basal Ganglia Diseases; Benzodiazepines; Clozapine; Dibenzothiazepines; Humans; Olanzapine; Pirenzepine; Quetiapine Fumarate; Risperidone; Schizophrenia; Sulpiride

2003
Combination of clozapine and amisulpride in treatment-resistant schizophrenia--case reports and review of the literature.
    Pharmacopsychiatry, 2004, Volume: 37, Issue:1

    Topics: Adult; Amisulpride; Antipsychotic Agents; Body Weight; Clozapine; Dose-Response Relationship, Drug; Drug Resistance; Drug Therapy, Combination; Female; Humans; Male; Middle Aged; Outcome Assessment, Health Care; Psychiatric Status Rating Scales; Retrospective Studies; Schizophrenia; Schizophrenic Psychology; Sulpiride

2004
[Current pharmacotherapy of schizophrenia].
    Orvosi hetilap, 2004, Jan-18, Volume: 145, Issue:3

    Topics: Amisulpride; Antipsychotic Agents; Benzodiazepines; Clozapine; Dibenzothiazepines; Humans; Olanzapine; Piperazines; Quetiapine Fumarate; Risperidone; Schizophrenia; Serotonin Antagonists; Sulpiride; Thiazoles

2004
[Psychotropics and weight gain].
    Praxis, 2004, Aug-25, Volume: 93, Issue:35

    Topics: Adolescent; Adult; Amisulpride; Antidepressive Agents; Antimanic Agents; Antipsychotic Agents; Aripiprazole; Benzodiazepines; Body Mass Index; Child; Clozapine; Dibenzothiazepines; Double-Blind Method; Female; Fructose; Haloperidol; Humans; Imidazoles; Indoles; Male; Obesity; Olanzapine; Piperazines; Placebos; Psychotropic Drugs; Quetiapine Fumarate; Quinolones; Randomized Controlled Trials as Topic; Risperidone; Socioeconomic Factors; Sulpiride; Thiazoles; Time Factors; Topiramate; Valproic Acid; Weight Gain

2004
Schizophrenia.
    Clinical evidence, 2003, Issue:10

    Topics: Amisulpride; Antipsychotic Agents; Benzodiazepines; Chlorpromazine; Clozapine; Cognitive Behavioral Therapy; Dibenzothiepins; Haloperidol; Humans; Olanzapine; Patient Compliance; Perazine; Pimozide; Risperidone; Schizophrenia; Sulpiride

2003
Schizophrenia.
    Clinical evidence, 2004, Issue:12

    Topics: Amisulpride; Antipsychotic Agents; Benzodiazepines; Chlorpromazine; Clozapine; Haloperidol; Humans; Olanzapine; Patient Compliance; Perazine; Pimozide; Risperidone; Schizophrenia; Sulpiride

2004
A typical mood stabilizers: a "typical role for atypical antipsychotics.
    Acta psychiatrica Scandinavica. Supplementum, 2005, Issue:426

    Topics: Affect; Amisulpride; Antipsychotic Agents; Aripiprazole; Benzodiazepines; Bipolar Disorder; Clozapine; Dibenzothiazepines; Olanzapine; Piperazines; Quetiapine Fumarate; Quinolones; Randomized Controlled Trials as Topic; Risperidone; Secondary Prevention; Sulpiride; Thiazoles

2005
[From cradle to grave? Expectations from atypical antipsychotics].
    Neuropsychopharmacologia Hungarica : a Magyar Pszichofarmakologiai Egyesulet lapja = official journal of the Hungarian Association of Psychopharmacology, 2005, Volume: 7, Issue:1

    Topics: Amisulpride; Antipsychotic Agents; Clozapine; Humans; Sulpiride

2005
Schizophrenia.
    Clinical evidence, 2005, Issue:14

    Topics: Amisulpride; Antipsychotic Agents; Chlorpromazine; Clozapine; Cognitive Behavioral Therapy; Dibenzothiepins; Family Therapy; Haloperidol; Humans; Patient Compliance; Risperidone; Schizophrenia; Secondary Prevention; Sulpiride; Thioridazine

2005
[The use of atypical antipsychotics in the long-term care of schizophrenia].
    L'Encephale, 2006, Volume: 32 Pt 3

    Topics: Amisulpride; Antipsychotic Agents; Aripiprazole; Basal Ganglia Diseases; Benzodiazepines; Clozapine; Cognition Disorders; Drug Tolerance; Dyskinesia, Drug-Induced; Haloperidol; Humans; Olanzapine; Piperazines; Quinolones; Risperidone; Schizophrenia; Sulpiride; Time Factors

2006
Akathisia and second-generation antipsychotic drugs.
    Current opinion in psychiatry, 2009, Volume: 22, Issue:3

    Topics: Amisulpride; Antipsychotic Agents; Aripiprazole; Benzodiazepines; Clozapine; Dibenzothiazepines; Humans; Isoxazoles; Olanzapine; Piperazines; Piperidines; Prevalence; Psychomotor Agitation; Psychotic Disorders; Quetiapine Fumarate; Quinolones; Risk Factors; Risperidone; Sulpiride; Thiazoles

2009
Clozapine combined with different antipsychotic drugs for treatment resistant schizophrenia.
    The Cochrane database of systematic reviews, 2009, 07-08, Issue:3

    Topics: Amisulpride; Antipsychotic Agents; Clozapine; Dibenzothiazepines; Drug Resistance; Drug Therapy, Combination; Female; Humans; Male; Piperazines; Quetiapine Fumarate; Randomized Controlled Trials as Topic; Risperidone; Schizophrenia; Sulpiride; Thiazoles

2009
Ziprasidone versus other atypical antipsychotics for schizophrenia.
    The Cochrane database of systematic reviews, 2009, Oct-07, Issue:4

    Topics: Amisulpride; Antipsychotic Agents; Benzodiazepines; Clozapine; Dibenzothiazepines; Humans; Olanzapine; Piperazines; Quetiapine Fumarate; Randomized Controlled Trials as Topic; Risperidone; Schizophrenia; Sulpiride; Thiazoles

2009
Sulpiride augmentation for schizophrenia.
    Schizophrenia bulletin, 2010, Volume: 36, Issue:2

    Topics: Antipsychotic Agents; Clozapine; Drug Therapy, Combination; Humans; Long-Term Care; Randomized Controlled Trials as Topic; Schizophrenia; Schizophrenic Psychology; Sulpiride

2010
Sulpiride augmentation for schizophrenia.
    The Cochrane database of systematic reviews, 2010, Jan-20, Issue:1

    Topics: Antipsychotic Agents; Clozapine; Drug Synergism; Drug Therapy, Combination; Humans; Randomized Controlled Trials as Topic; Schizophrenia; Sulpiride

2010
Olanzapine versus other atypical antipsychotics for schizophrenia.
    The Cochrane database of systematic reviews, 2010, Mar-17, Issue:3

    Topics: Amisulpride; Antipsychotic Agents; Aripiprazole; Benzodiazepines; Clozapine; Dibenzothiazepines; Humans; Olanzapine; Piperazines; Quetiapine Fumarate; Quinolones; Risperidone; Schizophrenia; Sulpiride; Thiazoles

2010
Head-to-head comparisons of metabolic side effects of second generation antipsychotics in the treatment of schizophrenia: a systematic review and meta-analysis.
    Schizophrenia research, 2010, Volume: 123, Issue:2-3

    Topics: Amisulpride; Antipsychotic Agents; Aripiprazole; Benzodiazepines; Blood Glucose; Cholesterol; Clinical Trials as Topic; Clozapine; Dibenzothiazepines; Humans; Imidazoles; Indoles; Olanzapine; Piperazines; Quetiapine Fumarate; Quinolones; Risperidone; Schizophrenia; Sulpiride; Thiazoles; Weight Gain

2010
Risperidone versus other atypical antipsychotics for schizophrenia.
    The Cochrane database of systematic reviews, 2011, Jan-19, Issue:1

    Topics: Amisulpride; Antipsychotic Agents; Aripiprazole; Benzodiazepines; Clozapine; Dibenzothiazepines; Humans; Imidazoles; Indoles; Olanzapine; Piperazines; Quetiapine Fumarate; Quinolones; Randomized Controlled Trials as Topic; Risperidone; Schizophrenia; Sulpiride; Thiazoles

2011
Pharmacological augmentation strategies for schizophrenia patients with insufficient response to clozapine: a quantitative literature review.
    Schizophrenia bulletin, 2012, Volume: 38, Issue:5

    Topics: Antipsychotic Agents; Brief Psychiatric Rating Scale; Citalopram; Clozapine; Dioxoles; Double-Blind Method; Drug Synergism; Drug Therapy, Combination; Fructose; Humans; Lamotrigine; Piperidines; Psychiatric Status Rating Scales; Psychotropic Drugs; Randomized Controlled Trials as Topic; Schizophrenia; Schizophrenic Psychology; Sulpiride; Topiramate; Treatment Outcome; Triazines

2012
Clozapine combined with different antipsychotic drugs for treatment-resistant schizophrenia.
    The Cochrane database of systematic reviews, 2017, 03-23, Volume: 3

    Topics: Adult; Amisulpride; Antipsychotic Agents; Aripiprazole; Clozapine; Dibenzothiazepines; Drug Resistance; Drug Therapy, Combination; Female; Haloperidol; Humans; Male; Piperazines; Quetiapine Fumarate; Randomized Controlled Trials as Topic; Risperidone; Schizophrenia; Sulpiride; Thiazoles; Weight Gain

2017

Trials

17 trial(s) available for sulpiride and clozapine

ArticleYear
[Three antipsychotic drugs in the treatment of schizophrenia--a controlled and double-blind study].
    Zhonghua shen jing jing shen ke za zhi = Chinese journal of neurology and psychiatry, 1988, Volume: 21, Issue:5

    Topics: Adolescent; Adult; Chlorpromazine; Clinical Trials as Topic; Clozapine; Dibenzazepines; Double-Blind Method; Female; Humans; Male; Middle Aged; Schizophrenia; Sulpiride

1988
Atypical neuroleptics: clozapine and the benzamides in the prevention and treatment of tardive dyskinesia.
    Modern problems of pharmacopsychiatry, 1983, Volume: 21

    Topics: Antipsychotic Agents; Benzamides; Clinical Trials as Topic; Clozapine; Dibenzazepines; Dose-Response Relationship, Drug; Dyskinesia, Drug-Induced; Haloperidol; Humans; Metoclopramide; Prospective Studies; Schizophrenia; Sulpiride; Tiapamil Hydrochloride

1983
Sulpiride augmentation in people with schizophrenia partially responsive to clozapine. A double-blind, placebo-controlled study.
    The British journal of psychiatry : the journal of mental science, 1997, Volume: 171

    Topics: Adult; Antipsychotic Agents; Clozapine; Dopamine Antagonists; Double-Blind Method; Drug Synergism; Drug Therapy, Combination; Female; Humans; Male; Middle Aged; Schizophrenia; Sulpiride; Treatment Outcome

1997
Effects of newer atypical antipsychotics on autonomic neurocardiac function: a comparison between amisulpride, olanzapine, sertindole, and clozapine.
    Journal of clinical psychopharmacology, 2001, Volume: 21, Issue:1

    Topics: Adult; Amisulpride; Antipsychotic Agents; Autonomic Nervous System; Benzodiazepines; Clozapine; Electrocardiography; Female; Heart; Heart Rate; Humans; Imidazoles; Indoles; Male; Middle Aged; Olanzapine; Pirenzepine; Prospective Studies; Sulpiride

2001
Neuroendocrine responsivities of the pituitary dopamine system in male schizophrenic patients during treatment with clozapine, olanzapine, risperidone, sulpiride, or haloperidol.
    European archives of psychiatry and clinical neuroscience, 2001, Volume: 251, Issue:3

    Topics: Adult; Antipsychotic Agents; Benzodiazepines; Clozapine; Dopamine Antagonists; Dose-Response Relationship, Drug; Haloperidol; Humans; Male; Middle Aged; Olanzapine; Pirenzepine; Pituitary Gland; Prolactin; Receptors, Dopamine D2; Risperidone; Schizophrenia; Sulpiride

2001
Clozapine with amisulpride for refractory schizophrenia.
    The American journal of psychiatry, 2004, Volume: 161, Issue:5

    Topics: Adult; Amisulpride; Antipsychotic Agents; Brief Psychiatric Rating Scale; Clozapine; Drug Therapy, Combination; Electrocardiography; Female; Heart Rate; Humans; Male; Middle Aged; Psychiatric Status Rating Scales; Psychotic Disorders; Schizophrenia; Schizophrenic Psychology; Sulpiride; Treatment Outcome

2004
Amisulpride augmentation of clozapine: an open non-randomized study in patients with schizophrenia partially responsive to clozapine.
    Acta psychiatrica Scandinavica, 2004, Volume: 110, Issue:4

    Topics: Amisulpride; Antipsychotic Agents; Brief Psychiatric Rating Scale; Clozapine; Diagnostic and Statistical Manual of Mental Disorders; Drug Synergism; Drug Therapy, Combination; Female; Humans; Male; Schizophrenia; Sulpiride

2004
Amisulpride has no effect on plasma clozapine concentrations.
    Journal of clinical psychopharmacology, 2005, Volume: 25, Issue:5

    Topics: Adult; Amisulpride; Antipsychotic Agents; Clozapine; Drug Combinations; Drug Interactions; Female; Half-Life; Humans; Male; Middle Aged; Psychotic Disorders; Spectrophotometry, Ultraviolet; Sulpiride

2005
Amisulpride treatment of clozapine-induced hypersalivation in schizophrenia patients: a randomized, double-blind, placebo-controlled cross-over study.
    International clinical psychopharmacology, 2006, Volume: 21, Issue:2

    Topics: Amisulpride; Antipsychotic Agents; Clozapine; Cross-Over Studies; Double-Blind Method; Female; Humans; Male; Placebos; Schizophrenia; Sialorrhea; Sulpiride

2006
Effects of typical and atypical antipsychotics on glucose-insulin homeostasis and lipid metabolism in first-episode schizophrenia.
    Psychopharmacology, 2006, Volume: 186, Issue:4

    Topics: Adult; Antipsychotic Agents; Benzodiazepines; Blood Glucose; Body Mass Index; C-Peptide; Cholesterol; Clozapine; Female; Homeostasis; Humans; Insulin; Insulin Resistance; Lipid Metabolism; Male; Metabolic Syndrome; Olanzapine; Prospective Studies; Risperidone; Schizophrenia; Sulpiride; Triglycerides; Waist-Hip Ratio

2006
Early changes of plasma lipids during treatment with atypical antipsychotics.
    International clinical psychopharmacology, 2006, Volume: 21, Issue:6

    Topics: Adolescent; Adult; Aged; Amisulpride; Analysis of Variance; Antipsychotic Agents; Benzodiazepines; Body Mass Index; Body Weight; Cholesterol; Clozapine; Humans; Lipids; Middle Aged; Olanzapine; Piperazines; Prospective Studies; Schizophrenia; Sulpiride; Thiazoles; Time Factors; Triglycerides

2006
A preliminary fMRI study of the effects on cortical activation of the treatment of refractory auditory hallucinations with rTMS.
    Psychiatry research, 2007, May-15, Volume: 155, Issue:1

    Topics: Adult; Amisulpride; Antipsychotic Agents; Clozapine; Combined Modality Therapy; Female; Functional Laterality; Hallucinations; Humans; Magnetic Resonance Imaging; Male; Middle Aged; Parietal Lobe; Reaction Time; Schizophrenia; Sulpiride; Temporal Lobe; Transcranial Magnetic Stimulation; Treatment Outcome

2007
Amisulpride augmentation in patients with schizophrenia partially responsive or unresponsive to clozapine. A randomized, double-blind, placebo-controlled trial.
    Pharmacopsychiatry, 2008, Volume: 41, Issue:1

    Topics: Adolescent; Adult; Aged; Amisulpride; Antipsychotic Agents; Brief Psychiatric Rating Scale; Clozapine; Dose-Response Relationship, Drug; Double-Blind Method; Drug Synergism; Evaluation Studies as Topic; Female; Humans; Male; Middle Aged; Pilot Projects; Schizophrenia; Sulpiride

2008
Neurocognitive effectiveness of haloperidol, risperidone, and olanzapine in first-episode psychosis: a randomized, controlled 1-year follow-up comparison.
    The Journal of clinical psychiatry, 2009, Apr-21, Volume: 70, Issue:5

    Topics: Adult; Amisulpride; Antipsychotic Agents; Benzodiazepines; Brain; Clozapine; Cognition Disorders; Female; Follow-Up Studies; Haloperidol; Humans; Male; Neuropsychological Tests; Olanzapine; Perphenazine; Piperazines; Prospective Studies; Psychotic Disorders; Risperidone; Severity of Illness Index; Sulpiride; Thiazoles

2009
Amisulpride versus moclobemide in treatment of clozapine-induced hypersalivation.
    The world journal of biological psychiatry : the official journal of the World Federation of Societies of Biological Psychiatry, 2011, Volume: 12, Issue:8

    Topics: Adult; Aged; Amisulpride; Antipsychotic Agents; Clozapine; Cross-Over Studies; Female; Humans; Male; Middle Aged; Moclobemide; Psychotic Disorders; Schizophrenia; Severity of Illness Index; Sialorrhea; Sulpiride

2011
Amisulpride augmentation in clozapine-unresponsive schizophrenia (AMICUS): a double-blind, placebo-controlled, randomised trial of clinical effectiveness and cost-effectiveness.
    Health technology assessment (Winchester, England), 2017, Volume: 21, Issue:49

    Topics: Adult; Amisulpride; Antipsychotic Agents; Clozapine; Cost-Benefit Analysis; Double-Blind Method; Drug Therapy, Combination; Female; Humans; Male; Psychiatric Status Rating Scales; Quality-Adjusted Life Years; Schizophrenia; Sulpiride; Technology Assessment, Biomedical; Treatment Outcome

2017
Amisulpride augmentation therapy improves cognitive performance and psychopathology in clozapine-resistant treatment-refractory schizophrenia: a 12-week randomized, double-blind, placebo-controlled trial.
    Military Medical Research, 2022, 10-18, Volume: 9, Issue:1

    Topics: Amisulpride; Antipsychotic Agents; Clozapine; Cognition; Humans; Schizophrenia; Schizophrenia, Treatment-Resistant; Sulpiride

2022

Other Studies

184 other study(ies) available for sulpiride and clozapine

ArticleYear
2-Amino-6-chloro-4-(N-methylpiperazino)pyrimidines, inhibitors of spiroperidol binding.
    Journal of medicinal chemistry, 1982, Volume: 25, Issue:12

    Topics: Animals; Binding, Competitive; Butyrophenones; Chemical Phenomena; Chemistry; Clozapine; Corpus Striatum; Crystallography; Haloperidol; In Vitro Techniques; Molecular Conformation; Piperazines; Pyrimidines; Rats; Receptors, Dopamine; Spiperone; X-Ray Diffraction

1982
New antipsychotic agents with serotonin and dopamine antagonist properties based on a pyrrolo[2,1-b][1,3]benzothiazepine structure.
    Journal of medicinal chemistry, 1998, Sep-24, Volume: 41, Issue:20

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Antipsychotic Agents; Brain; Catalepsy; Dopamine; Dopamine Antagonists; Dose-Response Relationship, Drug; Male; Motor Activity; Pyrroles; Rats; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Serotonin; Serotonin Antagonists; Stereoisomerism; Structure-Activity Relationship; Thiazepines

1998
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
High-throughput permeability pH profile and high-throughput alkane/water log P with artificial membranes.
    Journal of medicinal chemistry, 2001, Mar-15, Volume: 44, Issue:6

    Topics: Alkanes; Humans; Hydrogen-Ion Concentration; Intestinal Absorption; Membranes, Artificial; Octanols; Permeability; Pharmaceutical Preparations; Solubility; Water

2001
Molecular modeling of the three-dimensional structure of dopamine 3 (D3) subtype receptor: discovery of novel and potent D3 ligands through a hybrid pharmacophore- and structure-based database searching approach.
    Journal of medicinal chemistry, 2003, Oct-09, Volume: 46, Issue:21

    Topics: Algorithms; Binding Sites; Computational Biology; Crystallography, X-Ray; Databases, Protein; Humans; Kinetics; Ligands; Lipid Bilayers; Models, Molecular; Molecular Conformation; Mutation; Receptors, Dopamine D2; Receptors, Dopamine D3; Reproducibility of Results; Solvents; Structure-Activity Relationship; Tetrahydronaphthalenes; Water

2003
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Identification of new functional inhibitors of acid sphingomyelinase using a structure-property-activity relation model.
    Journal of medicinal chemistry, 2008, Jan-24, Volume: 51, Issue:2

    Topics: Algorithms; Animals; Cell Line; Cell Line, Tumor; Chemical Phenomena; Chemistry, Physical; Enzyme Inhibitors; Humans; Hydrogen-Ion Concentration; Molecular Conformation; Quantitative Structure-Activity Relationship; Rats; Sphingomyelin Phosphodiesterase

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Prediction of volume of distribution values in human using immobilized artificial membrane partitioning coefficients, the fraction of compound ionized and plasma protein binding data.
    European journal of medicinal chemistry, 2009, Volume: 44, Issue:11

    Topics: Blood Proteins; Chemistry, Physical; Computer Simulation; Humans; Membranes, Artificial; Models, Biological; Pharmaceutical Preparations; Protein Binding; Tissue Distribution

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Experimental solubility profiling of marketed CNS drugs, exploring solubility limit of CNS discovery candidate.
    Bioorganic & medicinal chemistry letters, 2010, Dec-15, Volume: 20, Issue:24

    Topics: Central Nervous System Agents; Drug Evaluation, Preclinical; Hydrogen-Ion Concentration; Pharmaceutical Preparations; Solubility

2010
Brain tissue binding of drugs: evaluation and validation of solid supported porcine brain membrane vesicles (TRANSIL) as a novel high-throughput method.
    Drug metabolism and disposition: the biological fate of chemicals, 2011, Volume: 39, Issue:2

    Topics: Absorption; Albumins; Animals; Brain; Brain Chemistry; Cell Membrane; Chromatography, High Pressure Liquid; Drug Evaluation, Preclinical; In Vitro Techniques; Lipids; Male; Microdialysis; Pharmaceutical Preparations; Protein Binding; Rats; Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization; Swine; Tissue Distribution

2011
In vitro inhibition of the bile salt export pump correlates with risk of cholestatic drug-induced liver injury in humans.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Cholestasis; Drug-Related Side Effects and Adverse Reactions; Humans; Insecta; Rats; Risk Factors

2012
Preclinical strategy to reduce clinical hepatotoxicity using in vitro bioactivation data for >200 compounds.
    Chemical research in toxicology, 2012, Oct-15, Volume: 25, Issue:10

    Topics: Chemical and Drug Induced Liver Injury; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Decision Trees; Drug Evaluation, Preclinical; Drug-Related Side Effects and Adverse Reactions; Glutathione; Humans; Liver; Pharmaceutical Preparations; Protein Binding

2012
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Discovery and characterization of novel, potent, and selective cytochrome P450 2J2 inhibitors.
    Drug metabolism and disposition: the biological fate of chemicals, 2013, Volume: 41, Issue:1

    Topics: Chromatography, High Pressure Liquid; Cytochrome P-450 CYP2J2; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Drug Discovery; Enzyme Inhibitors; Humans; Inhibitory Concentration 50; Kinetics; Microsomes, Liver; Models, Molecular; Molecular Dynamics Simulation; Substrate Specificity

2013
Differential effect of neuroleptic drugs on dopamine turnover in the extrapyramidal and limbic system.
    The Journal of pharmacy and pharmacology, 1976, Volume: 28, Issue:5

    Topics: Animals; Caudate Nucleus; Chlorpromazine; Clozapine; Dopamine; Extrapyramidal Tracts; Haloperidol; Homovanillic Acid; Limbic System; Male; Olfactory Bulb; Rats; Sulpiride; Thioridazine; Tranquilizing Agents

1976
[Acute and chronic effects of carpipramine, clozapine, haloperidol and sulpiride on the metabolism of biogenic amines in the rat brain (author's transl)].
    Arzneimittel-Forschung, 1976, Volume: 26, Issue:6

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Biogenic Amines; Brain; Brain Chemistry; Cerebral Cortex; Clozapine; Corpus Striatum; Dibenzazepines; Haloperidol; Homovanillic Acid; Hydroxyindoleacetic Acid; Limbic System; Male; Methoxyhydroxyphenylglycol; Rats; Sulpiride

1976
Nonstriatal dopaminergic neurons: Section X. Morphine, amphetamine, and noncataleptogenic neuroleptics: Introduction: morphine, amphetamine, and noncataleptogenic neuroleptics.
    Advances in biochemical psychopharmacology, 1977, Volume: 16

    Topics: Acetylcholine; Animals; Antipsychotic Agents; Brain; Clozapine; Corpus Striatum; Dextroamphetamine; Dopamine; gamma-Aminobutyric Acid; Glutamates; Haloperidol; Morphine; Neurotransmitter Agents; Rats; Receptors, Dopamine; Receptors, Opioid; Sulpiride

1977
The effect of neuroleptic drugs on drinking induced by central administration of angiotensin or carbachol.
    Psychopharmacology, 1979, Feb-28, Volume: 60, Issue:3

    Topics: Angiotensin II; Animals; Antipsychotic Agents; Carbachol; Chlorpromazine; Clozapine; Dopamine; Drinking Behavior; Flupenthixol; Fluphenazine; Haloperidol; Injections, Intraperitoneal; Injections, Intraventricular; Male; Pimozide; Rats; Sulpiride

1979
Crop-sac response after systemic and intraventricular administration of neuroleptic drugs.
    Neuroendocrinology, 1979, Volume: 29, Issue:6

    Topics: Animals; Antipsychotic Agents; Clozapine; Columbidae; Crop, Avian; Female; Haloperidol; Injections, Intraventricular; Reserpine; Sulpiride

1979
Correlation between the effects of neuroleptics on prolactin release, mammary stimulation and the vaginal cycle in rats.
    The Journal of endocrinology, 1978, Volume: 76, Issue:3

    Topics: Animals; Chlorpromazine; Clozapine; Estrus; Female; Luteinizing Hormone; Male; Mammary Glands, Animal; Ovulation; Pregnancy; Prolactin; Rats; Secretory Rate; Sulpiride; Tranquilizing Agents

1978
A comparison of the abilities of typical neuroleptic agents and of thioridazine, clozapine, sulpiride and metoclopramide to antagonise the hyperactivity induced by dopamine applied intracerebrally to areas of the extrapyramidal and mesolimbic systems.
    European journal of pharmacology, 1976, Volume: 40, Issue:1

    Topics: Animals; Brain; Clozapine; Corpus Striatum; Dopamine Antagonists; Dose-Response Relationship, Drug; Extrapyramidal Tracts; Fluphenazine; Haloperidol; Limbic System; Male; Metoclopramide; Pimozide; Rats; Stereotaxic Techniques; Sulpiride; Thioridazine; Tranquilizing Agents

1976
Acidic dopamine metabolites in cortical areas of the rat brain: localization and effects of drug.
    Brain research, 1976, Aug-27, Volume: 113, Issue:2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Amphetamine; Animals; Apomorphine; Cerebral Cortex; Clozapine; Corpus Striatum; Haloperidol; Homovanillic Acid; Male; Morphine; Olfactory Bulb; Oxotremorine; Phenylacetates; Probenecid; Rats; Sulpiride; Thioridazine

1976
Specificity of the dopamine sensitive adenylate cyclase for antipsychotic antagonists.
    Life sciences, 1976, Sep-15, Volume: 19, Issue:6

    Topics: Adenylyl Cyclases; Animals; Apomorphine; Chlorpromazine; Clozapine; Corpus Striatum; Dopamine; Dopamine Antagonists; Enzyme Activation; Haloperidol; Male; Metoclopramide; Rats; Sulpiride

1976
On the relevance of preferential increases of mesolimbic versus striatal dopamine turnover for the prediction of antipsychotic activity of psychotropic drugs.
    Journal of neurochemistry, 1976, Volume: 27, Issue:2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Anthracenes; Clozapine; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Haloperidol; Homovanillic Acid; Humans; Limbic System; Male; Methyltyrosines; Psychotic Disorders; Psychotropic Drugs; Rats; Sulpiride; Thioridazine

1976
Correlation between catalepsy and dopamine decrease in the rat striatum induced by neuroleptics.
    Neuropharmacology, 1976, Volume: 15, Issue:10

    Topics: Animals; Butyrophenones; Catalepsy; Chlorpromazine; Clozapine; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Haloperidol; Humans; Male; Rats; Sulpiride; Thioridazine; Time Factors; Tranquilizing Agents; Trifluperidol

1976
Detection of the nueroleptic properties of clozapine, sulpiride and thioridazine.
    Psychopharmacologia, 1975, Jul-23, Volume: 43, Issue:1

    Topics: Animals; Apomorphine; Behavior, Animal; Catalepsy; Clozapine; Dextroamphetamine; Dibenzazepines; Dose-Response Relationship, Drug; Drug Synergism; Fluphenazine; Haloperidol; Humans; Isoquinolines; Male; Methyltyrosines; Pimozide; Rats; Spiro Compounds; Stereotyped Behavior; Succinimides; Sulpiride; Thioridazine; Tranquilizing Agents

1975
Antagonism of the hyperactivity induced by dopamine applied intracerebrally to the nucleus accumbens septi by typical neuroleptics and by clozapine, sulpiride and thioridazine.
    European journal of pharmacology, 1976, Volume: 35, Issue:1

    Topics: Animals; Clozapine; Dibenzazepines; Dopamine; Dopamine Antagonists; Male; Motor Activity; Rats; Stimulation, Chemical; Sulpiride; Thioridazine; Time Factors; Tranquilizing Agents

1976
Striatal dopamine D2-receptor blockade by typical and atypical neuroleptics.
    Lancet (London, England), 1992, Feb-22, Volume: 339, Issue:8791

    Topics: Antipsychotic Agents; Clozapine; Corpus Striatum; Dopamine Antagonists; Humans; Receptors, Dopamine D2; Schizophrenia; Sulpiride

1992
A lever-release version of the conditioned avoidance response paradigm: effects of haloperidol, clozapine, sulpiride, and BMY-14802.
    Pharmacology, biochemistry, and behavior, 1992, Volume: 41, Issue:1

    Topics: Animals; Antipsychotic Agents; Avoidance Learning; Clozapine; Dextroamphetamine; Dose-Response Relationship, Drug; Haloperidol; Male; Psychotropic Drugs; Pyrimidines; Rats; Rats, Inbred Strains; Stereotyped Behavior; Sulpiride

1992
[Different effects of typical and atypical neuroleptics on K+-stimulated dopamine release from isolated rat striatum].
    Biulleten' eksperimental'noi biologii i meditsiny, 1992, Volume: 114, Issue:7

    Topics: Animals; Antipsychotic Agents; Carbolines; Clozapine; Corpus Striatum; Dopamine; Dopamine Antagonists; In Vitro Techniques; Male; Metoclopramide; Potassium; Raclopride; Rats; Rats, Wistar; Remoxipride; Salicylamides; Stimulation, Chemical; Sulpiride; Thioridazine; Tiapamil Hydrochloride; Trifluoperazine

1992
Evaluation of a stable CCK agonist (A68552) in conditioned avoidance responding in mice, rats, and primates: comparison with typical and atypical antipsychotics.
    Pharmacology, biochemistry, and behavior, 1992, Volume: 43, Issue:2

    Topics: Animals; Antipsychotic Agents; Avoidance Learning; Cholecystokinin; Clozapine; Dose-Response Relationship, Drug; Haloperidol; Macaca fascicularis; Male; Mice; Peptide Fragments; Rats; Sulpiride

1992
Characterization of dopamine autoreceptors in the amygdala: a fast cyclic voltammetric study in vitro.
    Neuroscience letters, 1991, Dec-16, Volume: 134, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 2H-Benzo(a)quinolizin-2-ol, 2-Ethyl-1,3,4,6,7,11b-hexahydro-3-isobutyl-9,10-dimethoxy-; Amygdala; Animals; Antipsychotic Agents; Benzazepines; Clozapine; Dopamine; Electric Stimulation; Ergolines; Male; Metoclopramide; Neurotransmitter Uptake Inhibitors; Nialamide; Piperazines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Secretory Rate; Sulpiride

1991
Atypical neuroleptics suppress dopaminergic behavioral supersensitivity.
    Psychopharmacology, 1990, Volume: 100, Issue:3

    Topics: Animals; Antipsychotic Agents; Apomorphine; Behavior, Animal; Clozapine; Cyproheptadine; Haloperidol; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Ritanserin; Serotonin Antagonists; Sulpiride; Thioridazine

1990
Acute effects of typical and atypical antipsychotic drugs on the release of dopamine from prefrontal cortex, nucleus accumbens, and striatum of the rat: an in vivo microdialysis study.
    Journal of neurochemistry, 1990, Volume: 54, Issue:5

    Topics: Animals; Antipsychotic Agents; Clozapine; Corpus Striatum; Dialysis; Dopamine; Frontal Lobe; Haloperidol; Male; Nucleus Accumbens; Rats; Rats, Inbred Strains; Septal Nuclei; Sulpiride

1990
Utilization of microdialysis for assessing the release of mesotelencephalic dopamine following clozapine and other antipsychotic drugs.
    Progress in neuro-psychopharmacology & biological psychiatry, 1990, Volume: 14 Suppl

    Topics: Animals; Cerebral Cortex; Clozapine; Corpus Striatum; Dialysis; Dopamine; Haloperidol; Mesencephalon; Microchemistry; Nucleus Accumbens; Organ Specificity; Rats; Sulpiride; Telencephalon

1990
Anxiolytic potential of sulpiride, clozapine and derivatives in the open-field test.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 36, Issue:1

    Topics: Animals; Chlordiazepoxide; Clozapine; Defecation; Dibenzazepines; Exploratory Behavior; Haloperidol; Rats; Rats, Inbred Strains; Structure-Activity Relationship; Sulpiride

1990
Differential effects of dopamine receptor antagonists on the sexual behavior of male rats.
    Psychopharmacology, 1989, Volume: 98, Issue:3

    Topics: Animals; Antipsychotic Agents; Clozapine; Ejaculation; Female; Haloperidol; Male; Metoclopramide; Pimozide; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sexual Behavior, Animal; Sulpiride

1989
Regional differences in the induction of behavioral supersensitivity by prolonged treatment with atypical neuroleptics.
    Psychopharmacology, 1989, Volume: 98, Issue:3

    Topics: Animals; Antipsychotic Agents; Behavior, Animal; Body Weight; Clozapine; Corpus Striatum; Dopamine; Haloperidol; Humans; Injections; Metoclopramide; Motor Activity; Nucleus Accumbens; Rats; Rats, Inbred Strains; Stereotyped Behavior; Sulpiride

1989
Effects of chronic treatment with atypical neuroleptics on the biosynthesis and release of opioid peptides in guinea-pig ileum.
    Regulatory peptides, 1985, Volume: 10, Issue:4

    Topics: Animals; Antipsychotic Agents; Clozapine; Cycloheximide; Dose-Response Relationship, Drug; Electric Stimulation; Endorphins; Enkephalin, Methionine; Female; Guinea Pigs; Ileum; In Vitro Techniques; Male; Myenteric Plexus; Naloxone; Neuromuscular Junction; Sulpiride

1985
Mesolimbic dopamine function is not altered during continuous chronic treatment of rats with typical or atypical neuroleptic drugs.
    Journal of neural transmission, 1985, Volume: 62, Issue:3-4

    Topics: Adenylyl Cyclases; Animals; Antipsychotic Agents; Clozapine; Dopamine; Haloperidol; Male; Motor Activity; Nucleus Accumbens; Rats; Rats, Inbred Strains; Receptors, Dopamine; Septal Nuclei; Sulpiride

1985
Presynaptic dopamine autoreceptors control tyrosine hydroxylase activation in depolarized striatal dopaminergic terminals.
    Journal of neurochemistry, 1986, Volume: 46, Issue:1

    Topics: Amphetamine; Animals; Bucladesine; Cerebral Cortex; Clozapine; Corpus Striatum; Dopamine; Enzyme Activation; Haloperidol; Hippocampus; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Sulpiride; Synapses; Synaptosomes; Tyrosine 3-Monooxygenase; Veratridine

1986
Differential effect of subchronic treatment with various neuroleptic agents on serotonin2 receptors in rat cerebral cortex.
    Journal of neurochemistry, 1986, Volume: 46, Issue:1

    Topics: 5,7-Dihydroxytryptamine; Animals; Antipsychotic Agents; Cerebral Cortex; Chlorpromazine; Clozapine; Female; Haloperidol; Imipramine; Ketanserin; Loxapine; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Spiperone; Sulpiride

1986
Evidence that the potential antipsychotic agent rimcazole (BW 234U) is a specific, competitive antagonist of sigma sites in brain.
    Life sciences, 1986, Jun-23, Volume: 38, Issue:25

    Topics: Animals; Antipsychotic Agents; Apomorphine; Binding, Competitive; Brain; Carbazoles; Clozapine; Guinea Pigs; Kinetics; Male; Methylphenidate; Mice; Phenazocine; Phencyclidine; Phenoxybenzamine; Propranolol; Receptors, Opioid; Receptors, sigma; Sulpiride

1986
Effect of neuroleptics on the schizophrenic syndrome.
    Psychopharmacology series, 1987, Volume: 3

    Topics: Adult; Antipsychotic Agents; Chlorpromazine; Chronic Disease; Clozapine; Female; Humans; Male; Schizophrenia; Sulpiride; Syndrome

1987
The nucleus accumbens and antidepressants: modulation of ergometrine-induced hyperactivity by typical and atypical antidepressants and neuroleptics in rats.
    Psychopharmacology, 1987, Volume: 92, Issue:3

    Topics: Amitriptyline; Animals; Antidepressive Agents; Antipsychotic Agents; Clorgyline; Clozapine; Desipramine; Ergonovine; Male; Mianserin; Nucleus Accumbens; Rats; Rats, Inbred Strains; Septal Nuclei; Sulpiride; Zimeldine

1987
Potency of antipsychotics in reversing the effects of a hallucinogenic drug on locus coeruleus neurons correlates with 5-HT2 binding affinity.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 1988, Volume: 1, Issue:2

    Topics: Amphetamines; Animals; Antipsychotic Agents; Chlorpromazine; Clozapine; DOM 2,5-Dimethoxy-4-Methylamphetamine; Electric Stimulation; Evoked Potentials; Haloperidol; Locus Coeruleus; Male; Neurons; Rats; Rats, Inbred Strains; Receptors, Serotonin; Sciatic Nerve; Spiperone; Sulpiride

1988
Inhibition of the electrically evoked release of [3H]acetylcholine in rat striatal slices: an experimental model for drugs that enhance dopaminergic neurotransmission.
    Journal of neurochemistry, 1985, Volume: 44, Issue:2

    Topics: Acetylcholine; Amphetamine; Animals; Chlorpromazine; Clozapine; Cocaine; Corpus Striatum; Dopamine; Electric Stimulation; Haloperidol; Male; Nomifensine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sulpiride; Synaptic Transmission

1985
Differential alteration of striatal D-1 and D-2 receptors induced by the long-term administration of haloperidol, sulpiride or clozapine to rats.
    Psychopharmacology. Supplementum, 1985, Volume: 2

    Topics: Animals; Apomorphine; Clozapine; Corpus Striatum; Dibenzazepines; Dose-Response Relationship, Drug; Haloperidol; Humans; Kinetics; Long-Term Care; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Stereotyped Behavior; Sulpiride; Thioxanthenes

1985
D2 dopamine receptors in rat striatum are homogeneous as revealed by ligand-binding studies.
    Biochemical pharmacology, 1988, Nov-15, Volume: 37, Issue:22

    Topics: Animals; Binding, Competitive; Clozapine; Corpus Striatum; Domperidone; Loxapine; Male; Rats; Receptors, Dopamine; Sulpiride

1988
Differential alterations in striatal acetylcholine function in rats during 12 months' continuous administration of haloperidol, sulpiride, or clozapine.
    Clinical neuropharmacology, 1986, Volume: 9, Issue:3

    Topics: Acetylcholine; Acetylcholinesterase; Animals; Choline O-Acetyltransferase; Clozapine; Corpus Striatum; Dibenzazepines; Dyskinesia, Drug-Induced; Haloperidol; Male; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Sulpiride

1986
Alterations in cerebral glutamic acid decarboxylase and 3H-flunitrazepam binding during continuous treatment of rats for up to 1 year with haloperidol, sulpiride or clozapine.
    Journal of neural transmission, 1987, Volume: 68, Issue:1-2

    Topics: Animals; Body Weight; Brain; Clozapine; Flunitrazepam; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Haloperidol; Kinetics; Male; Psychotropic Drugs; Rats; Rats, Inbred Strains; Sulpiride; Time Factors

1987
Classification of sulpiride, clozapine and haloperidol by toposelective recording from different brain structures in the immobilized rat (stereo-EEG).
    Neuropsychobiology, 1985, Volume: 14, Issue:3

    Topics: Animals; Brain; Clozapine; Corpus Striatum; Dibenzazepines; Electroencephalography; Haloperidol; Male; Motor Cortex; Rats; Reticular Formation; Somatosensory Cortex; Sulpiride

1985
Regulation of tyrosine hydroxylase after chronic treatment with classic and atypical antischizophrenic drugs.
    Advances in biochemical psychopharmacology, 1980, Volume: 24

    Topics: Animals; Antipsychotic Agents; Brain; Clozapine; Corpus Striatum; Haloperidol; Male; Nucleus Accumbens; Rats; Sulpiride; Time Factors; Tyrosine 3-Monooxygenase

1980
Morphological changes of pigeon crop-sac mucosa and pituitary lactotrophs after systemic and intraventricular administration of neuroleptic drugs.
    General and comparative endocrinology, 1980, Volume: 41, Issue:2

    Topics: Animals; Antipsychotic Agents; Clozapine; Columbidae; Crop, Avian; Female; Haloperidol; Mucous Membrane; Pituitary Gland, Anterior; Prolactin; Reserpine; Sulpiride

1980
Correlation between antiavoidance activities of antipsychotic drugs in rats and daily clinical doses.
    Pharmacology, biochemistry, and behavior, 1981, Volume: 14, Issue:2

    Topics: Animals; Antipsychotic Agents; Avoidance Learning; Butyrophenones; Clozapine; Discrimination Learning; Dose-Response Relationship, Drug; Electroshock; Male; Phenothiazines; Rats; Sulpiride; Thioxanthenes

1981
Typical and atypical neuroleptics are potent antagonists at alpha 1-adrenoceptors of the dorsal lateral geniculate nucleus. An electrophysiological study.
    Naunyn-Schmiedeberg's archives of pharmacology, 1982, Volume: 321, Issue:1

    Topics: Action Potentials; Adrenergic alpha-Antagonists; Animals; Antipsychotic Agents; Carbachol; Clozapine; Electrophysiology; Geniculate Bodies; Male; Phenothiazines; Phenylephrine; Rats; Rats, Inbred Strains; Sulpiride

1982
Antagonism of the apomorphine-induced yawning by "atypical" neuroleptics.
    Neuropharmacology, 1982, Volume: 21, Issue:11

    Topics: Animals; Antipsychotic Agents; Apomorphine; Behavior, Animal; Clozapine; Dopamine; Dose-Response Relationship, Drug; Male; Physostigmine; Rats; Rats, Inbred Strains; Sulpiride

1982
Buspirone: a potential atypical neuroleptic.
    Life sciences, 1983, Jul-18, Volume: 33, Issue:3

    Topics: Animals; Antipsychotic Agents; Buspirone; Clozapine; Dopamine; Dose-Response Relationship, Drug; Haloperidol; Male; Pyrimidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Substantia Nigra; Sulpiride; Time Factors

1983
Effect of repeated treatment with desipramine in the behavioral "despair" test in rats: antagonism by "atypical" but not "classical" neuroleptics or antiadrenergic drugs.
    Life sciences, 1984, Mar-19, Volume: 34, Issue:12

    Topics: Adrenergic alpha-Antagonists; Animals; Antipsychotic Agents; Butyrophenones; Chlorpromazine; Clonidine; Clozapine; Depressive Disorder; Desipramine; Dibenzazepines; Haloperidol; Humans; Male; Metoclopramide; Phentolamine; Prazosin; Propranolol; Rats; Sulpiride

1984
A comparison of the effects of acute and one year's continuous neuroleptic treatment on the release of [3H]glutamate and [3H]acetylcholine from rat striatal slices.
    Neuroscience, 1984, Volume: 11, Issue:1

    Topics: Acetylcholine; Animals; Antipsychotic Agents; Calcium; Clozapine; Corpus Striatum; Dopamine; Glutamates; Glutamic Acid; Haloperidol; In Vitro Techniques; Male; Potassium; Rats; Rats, Inbred Strains; Sulpiride; Trifluoperazine

1984
Effects of antipsychotic drugs on the long-term effects of amphetamine on nigro-striatal dopamine neurons in iprindole-treated rats.
    Naunyn-Schmiedeberg's archives of pharmacology, 1984, Volume: 325, Issue:3

    Topics: Analysis of Variance; Animals; Antipsychotic Agents; Behavior, Animal; Brain; Clozapine; Corpus Striatum; Dextroamphetamine; Dopamine; Haloperidol; Indoles; Iprindole; Male; Methyltyrosines; Neurons; Rats; Rats, Inbred Strains; Sulpiride

1984
[Changes in the number of benzodiazepine receptors in different parts of the brain of rats after neuroleptic withdrawal].
    Biulleten' eksperimental'noi biologii i meditsiny, 1984, Volume: 98, Issue:10

    Topics: Animals; Antipsychotic Agents; Brain; Clozapine; Flunitrazepam; Haloperidol; Humans; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substance Withdrawal Syndrome; Sulpiride; Time Factors

1984
Loxapine and clozapine decrease serotonin (S2) but do not elevate dopamine (D2) receptor numbers in the rat brain.
    Psychiatry research, 1984, Volume: 12, Issue:4

    Topics: Animals; Clozapine; Dibenzazepines; Dibenzoxazepines; Haloperidol; Loxapine; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Serotonin; Sulpiride; Time Factors

1984
Differential alterations in striatal dopamine receptor sensitivity induced by repeated administration of clinically equivalent doses of haloperidol, sulpiride or clozapine in rats.
    Psychopharmacology, 1984, Volume: 84, Issue:4

    Topics: Animals; Apomorphine; Clozapine; Corpus Striatum; Dibenzazepines; Haloperidol; Humans; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Sulpiride

1984
Drug-induced modulation of locomotor hyperactivity induced by picrotoxin in nucleus accumbens.
    Pharmacology, biochemistry, and behavior, 1984, Volume: 21, Issue:4

    Topics: Animals; Apomorphine; Carbachol; Clozapine; Diazepam; Haloperidol; Lisuride; Lysergic Acid Diethylamide; Male; Motor Activity; Nucleus Accumbens; Picrotoxin; Rats; Rats, Inbred Strains; Reserpine; Septal Nuclei; Sulpiride

1984
LSD-potentiated apomorphine hypermotility: a model for differentiating antipsychotic drugs.
    Pharmacology, biochemistry, and behavior, 1983, Volume: 18, Issue:1

    Topics: Animals; Apomorphine; Chlorpromazine; Clozapine; Disease Models, Animal; Drug Antagonism; Haloperidol; Humans; Hyperkinesis; Lysergic Acid Diethylamide; Male; Motor Activity; Rats; Rats, Inbred Strains; Sulpiride

1983
Regional blockade by neuroleptic drugs of in vivo 3H-spiperone binding in the rat brain. Relation to blockade of apomorphine induced hyperactivity and stereotypies.
    Journal of neural transmission, 1981, Volume: 52, Issue:3

    Topics: Animals; Apomorphine; Binding, Competitive; Brain; Butyrophenones; Chlorpromazine; Clozapine; Haloperidol; Humans; Hyperkinesis; Kinetics; Organ Specificity; Rats; Receptors, Dopamine; Receptors, Drug; Spiperone; Stereotyped Behavior; Sulpiride; Thioridazine

1981
Antipsychotic drugs induce Fos protein in the thalamic paraventricular nucleus: a novel locus of antipsychotic drug action.
    Neuroscience, 1995, Volume: 66, Issue:2

    Topics: Animals; Antipsychotic Agents; Blotting, Western; Clozapine; Haloperidol; Immunohistochemistry; Male; Muscarinic Antagonists; Prazosin; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Ritanserin; Scopolamine; Serotonin Antagonists; Sulpiride; Thalamic Nuclei

1995
Conversions from clozapine to other antipsychotic drugs.
    Archives of general psychiatry, 1995, Volume: 52, Issue:12

    Topics: Antipsychotic Agents; Clozapine; Humans; Receptors, Dopamine; Risk Factors; Sulpiride; Thioridazine

1995
Effects of typical and atypical antipsychotic drugs on response decrement patterns in rats.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 272, Issue:2

    Topics: Animals; Antipsychotic Agents; Clozapine; Conditioning, Operant; Dose-Response Relationship, Drug; Haloperidol; Isoxazoles; Male; Piperidines; Rats; Rats, Wistar; Remoxipride; Risperidone; Serotonin Antagonists; Sulpiride

1995
Differential effects of dopamine antagonists on evoked dopamine release from slices of striatum and nucleus accumbens in rats.
    The Journal of pharmacy and pharmacology, 1995, Volume: 47, Issue:3

    Topics: Animals; Binding, Competitive; Clozapine; Corpus Striatum; Dopamine; Dopamine Antagonists; Electric Stimulation; Haloperidol; Male; Nucleus Accumbens; Rats; Rats, Wistar; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Sulpiride

1995
Ascorbic acid and atypical antipsychotic drugs: modulation of amineptine-induced behavior in mice.
    Brain research, 1995, Jan-30, Volume: 670, Issue:2

    Topics: Animals; Antipsychotic Agents; Ascorbic Acid; Clozapine; Dibenzocycloheptenes; Dopamine; Female; Mice; Motor Activity; Remoxipride; Sulpiride

1995
Lack of effect of antipsychotic and antidepressant drugs on glutamate receptor mRNA levels in rat brains.
    Neuroscience letters, 1994, Aug-15, Volume: 177, Issue:1-2

    Topics: Animals; Antidepressive Agents; Antipsychotic Agents; Base Sequence; Brain Chemistry; Citalopram; Clozapine; Gene Expression Regulation; Haloperidol; Male; Mianserin; Molecular Sequence Data; Nerve Tissue Proteins; Rats; Rats, Wistar; Receptors, Glutamate; Receptors, N-Methyl-D-Aspartate; RNA, Messenger; Schizophrenia; Sulpiride

1994
Atypical antipsychotics, clozapine and sulpiride do not antagonise amphetamine-induced stereotyped locomotion.
    Psychopharmacology, 1994, Volume: 114, Issue:1

    Topics: Amphetamine; Animals; Antipsychotic Agents; Clozapine; Haloperidol; Male; Motor Activity; Rats; Rats, Wistar; Stereotyped Behavior; Sulpiride

1994
Clozapine and sulpiride up-regulate dopamine D3 receptor mRNA levels.
    Neuropharmacology, 1993, Volume: 32, Issue:9

    Topics: Animals; Aromatic-L-Amino-Acid Decarboxylases; Autoradiography; Base Sequence; Clozapine; Electrophoresis, Polyacrylamide Gel; Male; Molecular Sequence Data; Oligonucleotide Probes; Rats; Rats, Wistar; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; RNA, Messenger; Sulpiride; Tyrosine 3-Monooxygenase; Up-Regulation

1993
The limbic functional selectivity of amperozide is not mediated by dopamine D2 receptors as assessed by in vitro and in vivo binding.
    European journal of pharmacology, 1994, Mar-11, Volume: 254, Issue:1-2

    Topics: Animals; Antipsychotic Agents; Binding, Competitive; Clozapine; Dopamine; In Vitro Techniques; Limbic System; Male; Neostriatum; Piperazines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Spiperone; Sulpiride

1994
Dopamine receptor regulating serotonin N-acetyltransferase activity in chick retina represents a D4-like subtype: pharmacological characterization.
    Neurochemistry international, 1994, Volume: 24, Issue:3

    Topics: Animals; Arylamine N-Acetyltransferase; Benzamides; Benzazepines; Chickens; Circadian Rhythm; Clozapine; Dopamine; Dopamine Antagonists; Ergolines; Ketanserin; Male; Quinpirole; Receptors, Dopamine; Retina; Spiperone; Sulpiride

1994
[Effect of D1 and D2 dopamine receptor antagonists on acupuncture analgesia].
    Sheng li xue bao : [Acta physiologica Sinica], 1993, Volume: 45, Issue:1

    Topics: Acupuncture Analgesia; Animals; Benzazepines; Clozapine; Domperidone; Dopamine D2 Receptor Antagonists; Electroacupuncture; Female; Haloperidol; Male; Pain Threshold; Rabbits; Receptors, Dopamine D1; Sulpiride

1993
Behavioural interactions between 5-hydroxytryptophan, neuroleptic agents and 5-HT receptor antagonists in modifying rodent responding to aversive situations.
    British journal of pharmacology, 1995, Volume: 116, Issue:7

    Topics: Animals; Antipsychotic Agents; Avoidance Learning; Benperidol; Clozapine; Drug Interactions; Haloperidol; Male; Mice; Mice, Inbred Strains; Rats; Rats, Inbred Strains; Ritanserin; Serotonin; Serotonin Antagonists; Social Behavior; Sulpiride; Thioridazine

1995
Behavioral evidence for modulation by sigma ligands of (+)MK-801-induced hyperlocomotion in monoamine-depleted mice.
    Neuropharmacology, 1996, Volume: 35, Issue:4

    Topics: alpha-Methyltyrosine; Animals; Anisoles; Biogenic Monoamines; Brain; Catecholamines; Clozapine; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Male; Methyltyrosines; Mice; Mice, Inbred ICR; Motor Activity; Propylamines; Receptors, N-Methyl-D-Aspartate; Receptors, sigma; Reserpine; Sulpiride

1996
Long-term treatment with chlorpromazine and haloperidol but not with sulpiride and clozapine markedly elevates neuropeptide Y-like immunoreactivity in the rat hypothalamus.
    Neuropeptides, 1996, Volume: 30, Issue:5

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Antipsychotic Agents; Benzazepines; Chlorpromazine; Clozapine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Gene Expression Regulation; Haloperidol; Hypothalamus; Male; Neuropeptide Y; Prazosin; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Sulpiride

1996
Differential expression of c-fos mRNA in rat prefrontal cortex, striatum, N. accumbens and lateral septum after typical and atypical antipsychotics: an in situ hybridization study.
    Neurochemistry international, 1996, Volume: 29, Issue:4

    Topics: Animals; Antipsychotic Agents; Aripiprazole; Brain; Clozapine; Corpus Striatum; Fluphenazine; Genes, fos; Haloperidol; In Situ Hybridization; Nucleus Accumbens; Piperazines; Prefrontal Cortex; Quinolones; Rats; RNA, Messenger; Septum Pellucidum; Sulpiride

1996
Effect of chronic treatment with typical and atypical neuroleptics on the expression of dopamine D2 and D3 receptors in rat brain.
    Psychopharmacology, 1996, Volume: 128, Issue:4

    Topics: Animals; Antipsychotic Agents; Clozapine; Haloperidol; In Situ Hybridization; Limbic System; Male; Neostriatum; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; RNA, Messenger; Sulpiride

1996
Antipsychotics with inverse agonist activity at the dopamine D3 receptor.
    Journal of neural transmission (Vienna, Austria : 1996), 1996, Volume: 103, Issue:10

    Topics: Animals; Antipsychotic Agents; Calcium; CHO Cells; Clozapine; Colforsin; Cricetinae; Cyclic AMP; DNA Replication; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Flupenthixol; Glioma; Haloperidol; Humans; Hybrid Cells; Naphthalenes; Neuroblastoma; Pertussis Toxin; Phenothiazines; Pimozide; Pyrrolidines; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3; Recombinant Proteins; Risperidone; Salicylamides; Second Messenger Systems; Sulpiride; Tetrahydronaphthalenes; Tumor Cells, Cultured; Virulence Factors, Bordetella

1996
Pharmacological modifications in dopaminergic neurotransmission affect the quinpirole-evoked suppression of serotonin N-acetyltransferase activity in chick retina: an impact on dopamine D4-like receptors.
    Journal of neural transmission (Vienna, Austria : 1996), 1996, Volume: 103, Issue:12

    Topics: Animals; Antipsychotic Agents; Arylamine N-Acetyltransferase; Chickens; Circadian Rhythm; Clozapine; Dopamine Agents; Enzyme Inhibitors; Levodopa; Male; Quinpirole; Raclopride; Receptors, Dopamine D2; Receptors, Dopamine D4; Retina; Salicylamides; Sulpiride; Synaptic Transmission

1996
The behavioural effects of pramipexole, a novel dopamine receptor agonist.
    European journal of pharmacology, 1997, Apr-11, Volume: 324, Issue:1

    Topics: Animals; Antiparkinson Agents; Benzazepines; Benzothiazoles; Body Temperature; Catalepsy; Clozapine; Dopamine Agents; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Dyskinesia, Drug-Induced; Haloperidol; Injections, Subcutaneous; Levodopa; Male; Mice; Motor Activity; Pramipexole; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Spiperone; Stereotyped Behavior; Sulpiride; Thiazoles

1997
The effects of antipsychotic drugs on the mRNA levels of serotonin 5HT2A and 5HT2C receptors.
    Brain research. Molecular brain research, 1997, Volume: 48, Issue:1

    Topics: Animals; Antipsychotic Agents; Brain; Chlorpromazine; Clozapine; Down-Regulation; Haloperidol; Male; Organ Specificity; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; RNA, Messenger; Sulpiride; Time Factors; Transcription, Genetic; Up-Regulation

1997
Binding of antipsychotic drugs to cortical 5-HT2A receptors: a PET study of chlorpromazine, clozapine, and amisulpride in schizophrenic patients.
    The American journal of psychiatry, 1998, Volume: 155, Issue:4

    Topics: Adolescent; Adult; Amisulpride; Animals; Antipsychotic Agents; Cerebral Cortex; Chlorpromazine; Clozapine; Dose-Response Relationship, Drug; Drug Administration Schedule; Female; Fluorine Radioisotopes; Humans; Male; Pyrimidinones; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Schizophrenia; Sulpiride; Tomography, Emission-Computed

1998
Preferential blockade by clozapine of hyperlocomotion induced by non-competitive NMDA antagonist MK-801.
    Indian journal of physiology and pharmacology, 1998, Volume: 42, Issue:3

    Topics: Analysis of Variance; Animals; Antipsychotic Agents; Benzazepines; Clozapine; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Interactions; Haloperidol; Hyperkinesis; Mice; Mice, Inbred BALB C; N-Methylaspartate; Neuroprotective Agents; Rats; Rats, Wistar; Stereotyped Behavior; Sulpiride

1998
Sulpiride augmentation on schizophrenia.
    The British journal of psychiatry : the journal of mental science, 1998, Volume: 172

    Topics: Antipsychotic Agents; Clozapine; Humans; Schizophrenia; Sulpiride; Treatment Failure

1998
Alpha1-adrenergic, D1, and D2 receptors interactions in the prefrontal cortex: implications for the modality of action of different types of neuroleptics.
    Synapse (New York, N.Y.), 1998, Volume: 30, Issue:4

    Topics: Animals; Antipsychotic Agents; Benzazepines; Cerebral Cortex; Clozapine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Electric Stimulation; Electrophysiology; Haloperidol; Injections, Intravenous; Iontophoresis; Neural Inhibition; Prazosin; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Receptors, Dopamine D1; Receptors, Dopamine D2; Sulpiride

1998
Influence of typical and atypical antipsychotics on neuropeptide Y-like immunoreactivity and NPY mRNA expression in rat striatum.
    Neuropeptides, 1998, Volume: 32, Issue:5

    Topics: Adrenergic Antagonists; Animals; Antipsychotic Agents; Chlorpromazine; Clozapine; Corpus Striatum; Dopamine Antagonists; Haloperidol; In Situ Hybridization; Injections, Intraperitoneal; Male; Neuropeptide Y; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Dopamine; Receptors, Serotonin; RNA, Messenger; Serotonin Antagonists; Sulpiride

1998
Neuroleptics with differential affinities at dopamine D2 receptors and sigma receptors affect differently the N-methyl-D-aspartate-induced increase in intracellular calcium concentration: involvement of protein kinase.
    Synapse (New York, N.Y.), 1999, Volume: 31, Issue:1

    Topics: Animals; Antipsychotic Agents; Calcium; Cells, Cultured; Chlorpromazine; Clozapine; Dopamine Antagonists; Frontal Lobe; Guanidines; Haloperidol; N-Methylaspartate; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, sigma; Sulpiride

1999
Weight gain: side effect of atypical neuroleptics?
    Journal of clinical psychopharmacology, 1999, Volume: 19, Issue:4

    Topics: Adolescent; Adult; Adverse Drug Reaction Reporting Systems; Antipsychotic Agents; Body Mass Index; Clozapine; Delusions; Dibenzothiepins; Female; Humans; Long-Term Care; Male; Middle Aged; Psychotic Disorders; Retrospective Studies; Risperidone; Schizophrenia; Sulpiride; Weight Gain

1999
Pentadecapeptide BPC 157 attenuates disturbances induced by neuroleptics: the effect on catalepsy and gastric ulcers in mice and rats.
    European journal of pharmacology, 1999, Aug-20, Volume: 379, Issue:1

    Topics: Animals; Anti-Ulcer Agents; Antipsychotic Agents; Catalepsy; Clozapine; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Fluphenazine; Haloperidol; Male; Mice; Orientation; Peptic Ulcer; Peptide Fragments; Proteins; Rats; Rats, Wistar; Sulpiride; Time Factors

1999
Dopamine receptor antagonists modulate glucose uptake in rat pheochromocytoma (PC12) cells.
    Neuroscience letters, 1999, Oct-29, Volume: 274, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Benzazepines; Biological Transport; Chlorpromazine; Clozapine; Dizocilpine Maleate; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Excitatory Amino Acid Antagonists; Fluphenazine; Glucose; Haloperidol; PC12 Cells; Pimozide; Rats; Receptors, Dopamine D2; Spiperone; Sulpiride; Tritium

1999
Clozapine blocks dopamine, 5-HT2 and 5-HT3 responses in the medial prefrontal cortex: an in vivo microiontophoretic study.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 1999, Volume: 10, Issue:1

    Topics: Action Potentials; Amphetamines; Animals; Biguanides; Clozapine; Dopamine; Dopamine Agonists; Dopamine Antagonists; Iontophoresis; Neurons; Prefrontal Cortex; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Serotonin Receptor Agonists; Sodium Chloride; Sulpiride

1999
Predicting how equipotent doses of chlorpromazine, haloperidol, sulpiride, raclopride and clozapine reduce locomotor activity in mice.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 2000, Volume: 10, Issue:3

    Topics: Animals; Antipsychotic Agents; Chlorpromazine; Clozapine; Female; Haloperidol; Male; Mice; Motor Activity; Raclopride; Sulpiride

2000
[Atypical antipsychotics].
    Der Nervenarzt, 2000, Volume: 71, Issue:5

    Topics: Acute Disease; Amisulpride; Antipsychotic Agents; Benzodiazepines; Clozapine; Cost-Benefit Analysis; Dibenzothiazepines; Dibenzothiepins; Dyskinesia, Drug-Induced; Germany; Humans; Neurotransmitter Agents; Olanzapine; Patient Compliance; Pirenzepine; Quetiapine Fumarate; Randomized Controlled Trials as Topic; Risperidone; Schizophrenia; Sulpiride

2000
Potentiation of ethanol-induced loss of the righting reflex by ascorbic acid in mice: interaction with dopamine antagonists.
    Pharmacology, biochemistry, and behavior, 2000, Volume: 66, Issue:2

    Topics: Animals; Ascorbic Acid; Benzazepines; Clozapine; Dopamine Antagonists; Drug Synergism; Ethanol; Female; Haloperidol; Mice; Receptors, Dopamine D2; Reflex; Sleep; Sulpiride

2000
Pharmacology of [3H]R(+)-7-OH-DPAT binding in the rat caudate-putamen.
    Neurochemistry international, 2001, Volume: 38, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Benzopyrans; Binding, Competitive; Caudate Nucleus; Clozapine; Dopamine; Dopamine Agonists; Dopamine Antagonists; Guanidines; Guanosine Triphosphate; Haloperidol; Heterotrimeric GTP-Binding Proteins; Indans; Kinetics; Magnesium; Male; Oxazines; Protein Binding; Putamen; Quinpirole; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Remoxipride; Sodium; Specific Pathogen-Free Organisms; Sulfones; Sulpiride; Tetrahydronaphthalenes

2001
[Acute tongue and pharyngeal spasms during changeover from clozapine to amisulpride. A case example].
    Der Nervenarzt, 2000, Volume: 71, Issue:11

    Topics: Acute Disease; Adult; Amisulpride; Antipsychotic Agents; Clozapine; Drug Administration Schedule; Drug Therapy, Combination; Female; Humans; Pharyngeal Diseases; Psychotic Disorders; Receptors, Dopamine; Spasm; Sulpiride; Tongue Diseases

2000
Mechanisms of inverse agonism of antipsychotic drugs at the D(2) dopamine receptor: use of a mutant D(2) dopamine receptor that adopts the activated conformation.
    Journal of neurochemistry, 2001, Volume: 77, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antipsychotic Agents; Apomorphine; Binding, Competitive; Bromocriptine; Butaclamol; Chlorpromazine; CHO Cells; Clozapine; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; GTP-Binding Proteins; Haloperidol; Humans; Macromolecular Substances; Mutagenesis, Site-Directed; Phenethylamines; Piperidines; Protein Binding; Protein Conformation; Radioligand Assay; Receptors, Dopamine D2; Recombinant Fusion Proteins; Sodium; Spiperone; Structure-Activity Relationship; Sulpiride; Transfection; Tyramine

2001
In vitro modulation of the firing rate of dopamine neurons in the rat substantia nigra pars compacta and the ventral tegmental area by antipsychotic drugs.
    Neuropharmacology, 2001, Volume: 40, Issue:7

    Topics: Action Potentials; Animals; Antipsychotic Agents; Clozapine; Dose-Response Relationship, Drug; Male; Neurons; Rats; Rats, Wistar; Receptors, Dopamine D2; Risperidone; Substantia Nigra; Sulpiride; Ventral Tegmental Area

2001
Atypical neuroleptic drugs downregulate dopamine sensitivity in rat cortical and striatal astrocytes.
    Molecular and cellular neurosciences, 2001, Volume: 18, Issue:2

    Topics: Adrenergic beta-Antagonists; Animals; Animals, Newborn; Antipsychotic Agents; Astrocytes; Benzodiazepines; Calcium; Calcium Signaling; Cells, Cultured; Cerebral Cortex; Clozapine; Dopamine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Down-Regulation; Haloperidol; Intracellular Fluid; Neostriatum; Olanzapine; Pirenzepine; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D4; Risperidone; Serotonin Antagonists; Sulpiride

2001
Dopamine D4 receptor activation inhibits presynaptically glutamatergic neurotransmission in the rat supraoptic nucleus.
    Journal of neurophysiology, 2001, Volume: 86, Issue:3

    Topics: Animals; Benzamides; Benzazepines; Clozapine; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; Glutamic Acid; Male; Patch-Clamp Techniques; Piperazines; Presynaptic Terminals; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D4; Sulpiride; Supraoptic Nucleus; Synaptic Transmission

2001
Atypical, but not typical, antipsychotic drugs increase cortical acetylcholine release without an effect in the nucleus accumbens or striatum.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2002, Volume: 26, Issue:3

    Topics: Acetylcholine; Acetylcholinesterase; Animals; Antipsychotic Agents; Benzodiazepines; Cerebral Cortex; Cholinesterase Inhibitors; Clozapine; Corpus Striatum; Haloperidol; Male; Nucleus Accumbens; Olanzapine; Oxotremorine; Piperazines; Pirenzepine; Rats; Rats, Sprague-Dawley; Risperidone; Scopolamine; Sulpiride; Thiazoles; Thioridazine

2002
Sub-chronic treatment with classical but not atypical antipsychotics produces morphological changes in rat nigro-striatal dopaminergic neurons directly related to "early onset" vacuous chewing.
    The European journal of neuroscience, 2002, Volume: 15, Issue:7

    Topics: Amisulpride; Animals; Antipsychotic Agents; Clozapine; Dopamine; Dose-Response Relationship, Drug; Drug Administration Schedule; Dyskinesia, Drug-Induced; Haloperidol; Male; Mastication; Neostriatum; Nerve Degeneration; Neural Pathways; Neurons; Rats; Rats, Sprague-Dawley; Risperidone; Substance Withdrawal Syndrome; Substantia Nigra; Sulpiride

2002
Effects of atypical antipsychotics on vertebrate neuromuscular transmission.
    Neuropharmacology, 2002, Volume: 42, Issue:5

    Topics: Animals; Antipsychotic Agents; Benzodiazepines; Clozapine; Fluphenazine; In Vitro Techniques; Membrane Potentials; Motor Endplate; Neuromuscular Junction; Olanzapine; Pirenzepine; Rana pipiens; Rana temporaria; Risperidone; Sulpiride; Synaptic Transmission

2002
Neuroleptic malignant syndrome due to atypical neuroleptics: three episodes in one patient.
    Pharmacopsychiatry, 2002, Volume: 35, Issue:3

    Topics: Amisulpride; Antipsychotic Agents; Clozapine; Female; Humans; Middle Aged; Neuroleptic Malignant Syndrome; Risperidone; Schizophrenia; Sulpiride

2002
Chlorpromazine inhibits the glucocorticoid receptor-mediated gene transcription in a calcium-dependent manner.
    Neuropharmacology, 2002, Volume: 43, Issue:6

    Topics: Animals; Antipsychotic Agents; Calcimycin; Calcium; Calcium Channel Blockers; Cell Line; Cell Line, Transformed; Chloramphenicol O-Acetyltransferase; Chlorpromazine; Clozapine; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Inhibitors; Estrenes; Fibroblasts; Gene Expression Regulation; Genes, Reporter; Haloperidol; Histamine; Histamine H1 Antagonists; Ionophores; Mammary Tumor Virus, Mouse; Mice; Nifedipine; Phorbol Esters; Phosphodiesterase Inhibitors; Protein Kinase C; Protein Kinase C-alpha; Pyrilamine; Pyrrolidinones; Raclopride; Receptors, Glucocorticoid; Remoxipride; Sulfonamides; Sulpiride; Tetradecanoylphorbol Acetate; Thionucleotides; Transcription, Genetic; Type C Phospholipases

2002
Discriminative stimulus properties in rats of the novel antipsychotic quetiapine.
    Experimental and clinical psychopharmacology, 2002, Volume: 10, Issue:4

    Topics: Amisulpride; Analysis of Variance; Animals; Antipsychotic Agents; Chlorpromazine; Clozapine; Dibenzothiazepines; Discrimination Learning; Discrimination, Psychological; Dose-Response Relationship, Drug; Female; Generalization, Psychological; Haloperidol; Loxapine; Quetiapine Fumarate; Quinoxalines; Rats; Rats, Wistar; Risperidone; Sulpiride

2002
How does the benzamide antipsychotic amisulpride get into the brain?--An in vitro approach comparing amisulpride with clozapine.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2003, Volume: 28, Issue:11

    Topics: Amisulpride; Animals; Antipsychotic Agents; Benzamides; Brain; Caco-2 Cells; Clozapine; Dose-Response Relationship, Drug; Humans; Sulpiride; Swine

2003
A successful antipsychotic combination trial. Quo Vadis?
    Acta psychiatrica Scandinavica, 2004, Volume: 110, Issue:4

    Topics: Amisulpride; Antipsychotic Agents; Clozapine; Drug Synergism; Drug Therapy, Combination; Humans; Psychotic Disorders; Sulpiride

2004
The impact of neuroleptic medication on seizure threshold and duration in electroconvulsive therapy.
    Ideggyogyaszati szemle, 2004, Nov-20, Volume: 57, Issue:11-12

    Topics: Adult; Aged; Antipsychotic Agents; Benzodiazepines; Brain; Clopenthixol; Clozapine; Dibenzothiazepines; Electric Impedance; Electroconvulsive Therapy; Electroencephalography; Electromyography; Female; Fluphenazine; Haloperidol; Humans; Male; Middle Aged; Olanzapine; Quetiapine Fumarate; Risperidone; Seizures; Sulpiride

2004
Effectiveness of amisulpride augmentation of clozapine in a non-responder to either drug alone: a case report.
    Acta psychiatrica Scandinavica, 2005, Volume: 111, Issue:2

    Topics: Adult; Amisulpride; Antipsychotic Agents; Clozapine; Drug Administration Schedule; Drug Synergism; Drug Therapy, Combination; Female; Humans; Schizophrenia; Sulpiride

2005
Reduction of side effects by combining clozapine with amisulpride: case report and short review of clozapine-induced hypersalivation-a case report.
    Pharmacopsychiatry, 2005, Volume: 38, Issue:1

    Topics: Adult; Amisulpride; Antipsychotic Agents; Clozapine; Drug Therapy, Combination; Humans; Male; Schizophrenia, Paranoid; Sialorrhea; Sulpiride

2005
Augmentation of clozapine with amisulpride: a promising therapeutic approach to refractory schizophrenic symptoms.
    Pharmacopsychiatry, 2005, Volume: 38, Issue:1

    Topics: Adult; Amisulpride; Antipsychotic Agents; Clozapine; Drug Synergism; Drug Therapy, Combination; Humans; Schizophrenia; Schizophrenic Psychology; Sulpiride

2005
Combined use of amisulpride and clozapine for patients with treatment-resistant schizophrenia.
    Australasian psychiatry : bulletin of Royal Australian and New Zealand College of Psychiatrists, 2004, Volume: 12, Issue:1

    Topics: Adult; Amisulpride; Antipsychotic Agents; Clozapine; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Resistance; Drug Therapy, Combination; Female; Humans; Male; Middle Aged; Patient Satisfaction; Schizophrenia; Schizophrenic Psychology; Sulpiride; Treatment Outcome

2004
Behaviorally timid rats respond differentially to conventional and atypical neuroleptics.
    Pharmacology, biochemistry, and behavior, 2005, Volume: 81, Issue:3

    Topics: Analysis of Variance; Animals; Antipsychotic Agents; Behavior, Animal; Clozapine; Female; Haloperidol; Ovariectomy; Random Allocation; Rats; Rats, Long-Evans; Social Behavior; Sulpiride; Time Factors

2005
Sulpiride addition for the treatment of clozapine-induced hypersalivation: preliminary study.
    The Israel journal of psychiatry and related sciences, 2005, Volume: 42, Issue:1

    Topics: Adult; Antidepressive Agents, Second-Generation; Antipsychotic Agents; Clozapine; Female; Follow-Up Studies; Humans; Male; Schizophrenia; Sialorrhea; Sulpiride

2005
The role of 5-HT(2A) receptor antagonism in amphetamine-induced inhibition of A10 dopamine neurons in vitro.
    European journal of pharmacology, 2005, Sep-27, Volume: 520, Issue:1-3

    Topics: Action Potentials; Amphetamine; Animals; Antipsychotic Agents; Benzodiazepines; Clozapine; Dopamine; Dopamine D2 Receptor Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Fluorobenzenes; In Vitro Techniques; Male; Mesencephalon; Neural Inhibition; Neurons; Olanzapine; Piperidines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Dopamine D2; Serotonin 5-HT2 Receptor Antagonists; Sulpiride

2005
Atypical anti-psychotics in the real world--a naturalistic comparative outcome study.
    Scottish medical journal, 2005, Volume: 50, Issue:3

    Topics: Adolescent; Adult; Aged; Amisulpride; Antipsychotic Agents; Benzodiazepines; Clozapine; Dibenzothiazepines; Dose-Response Relationship, Drug; Drug Administration Schedule; Female; Follow-Up Studies; Humans; Male; Middle Aged; Olanzapine; Patient Compliance; Probability; Prospective Studies; Psychiatric Status Rating Scales; Psychotic Disorders; Quality of Life; Quetiapine Fumarate; Risk Assessment; Risperidone; Severity of Illness Index; Statistics, Nonparametric; Sulpiride; Treatment Outcome

2005
[Treatment resistant schizophrenia, residual subtype: symptom improvement after additional treatment with amisulpride].
    Psychiatrische Praxis, 2006, Volume: 33, Issue:1

    Topics: Adult; Amisulpride; Antipsychotic Agents; Benzodiazepines; Clozapine; Commitment of Mentally Ill; Drug Resistance; Drug Therapy, Combination; Follow-Up Studies; Haloperidol; Homicide; Humans; Insanity Defense; Male; Olanzapine; Prisoners; Schizophrenia, Paranoid; Sulpiride; Treatment Outcome

2006
Dopamine D3 receptor modulation of dopamine efflux in the rat nucleus accumbens.
    European journal of pharmacology, 2006, Mar-18, Volume: 534, Issue:1-3

    Topics: Animals; Antipsychotic Agents; Clozapine; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Electric Stimulation; Haloperidol; Male; Nitriles; Nucleus Accumbens; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Sulpiride; Tetrahydroisoquinolines; Tetrahydronaphthalenes

2006
Prototypical antipsychotic drugs protect hippocampal neuronal cultures against cell death induced by growth medium deprivation.
    BMC neuroscience, 2006, Mar-30, Volume: 7

    Topics: Animals; Anisoles; Antipsychotic Agents; Benzazepines; Butaclamol; Caspase Inhibitors; Cell Death; Cells, Cultured; Chlorpromazine; Clozapine; Domperidone; Dopamine Antagonists; Excitatory Amino Acid Antagonists; Ginkgo biloba; Haloperidol; Hippocampus; Indans; Isoxazoles; Neurons; Neuroprotective Agents; Peptides; Piperidines; Plant Extracts; Propylamines; Raclopride; Rats; Rats, Sprague-Dawley; Reactive Oxygen Species; Receptors, N-Methyl-D-Aspartate; Remoxipride; Risperidone; Sulpiride

2006
Alterations of glucose metabolism during treatment with clozapine or amisulpride: results from a prospective 16-week study.
    Journal of psychopharmacology (Oxford, England), 2007, Volume: 21, Issue:4

    Topics: Adolescent; Adult; Aged; Amisulpride; Antipsychotic Agents; Body Mass Index; Clozapine; Female; Glucose; Glucose Metabolism Disorders; Homeostasis; Humans; Insulin; Insulin Resistance; Male; Middle Aged; Prospective Studies; Risk Factors; Schizophrenia; Sulpiride

2007
Influence of morphine and dopamine receptor sensitization on locomotor activity in mice.
    Pharmacology, 2006, Volume: 78, Issue:4

    Topics: Animals; Clozapine; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Tolerance; GABA Antagonists; Male; Mice; Morphine; Motor Activity; Receptors, Dopamine; Receptors, Opioid, mu; Reverse Transcriptase Polymerase Chain Reaction; Sulpiride

2006
Remission and relapse in the outpatient care of schizophrenia: three-year results from the Schizophrenia Outpatient Health Outcomes study.
    Journal of clinical psychopharmacology, 2006, Volume: 26, Issue:6

    Topics: Adult; Ambulatory Care; Amisulpride; Antipsychotic Agents; Benzodiazepines; Clozapine; Cohort Studies; Dibenzothiazepines; Europe; Female; Follow-Up Studies; Humans; Kaplan-Meier Estimate; Logistic Models; Male; Olanzapine; Prospective Studies; Quetiapine Fumarate; Recurrence; Risk Factors; Risperidone; Schizophrenia; Sulpiride; Time Factors; Treatment Outcome

2006
Effects of clozapine and sulpiride on morphine state-dependent memory in the step-down passive avoidance test.
    Pharmacology, 2007, Volume: 79, Issue:3

    Topics: Analgesics, Opioid; Animals; Antipsychotic Agents; Avoidance Learning; Behavior, Animal; Clozapine; Dose-Response Relationship, Drug; Injections, Intraperitoneal; Injections, Subcutaneous; Male; Mental Recall; Mice; Mice, Inbred Strains; Morphine; Receptors, Dopamine D4; Sulpiride; Time Factors

2007
The influence of clozapine treatment and other antipsychotics on the 18 kDa translocator protein, formerly named the peripheral-type benzodiazepine receptor, and steroid production.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 2008, Volume: 18, Issue:1

    Topics: Adrenal Glands; Animals; Antipsychotic Agents; Brain; Cell Line; Clozapine; Corticosterone; Humans; Isoquinolines; Male; Mice; Mitochondria; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Receptors, GABA; Risperidone; Steroids; Sulpiride; Testis; Testosterone; Thioridazine

2008
The use of atypical antipsychotics in French psychiatric hospitals.
    Pharmacy world & science : PWS, 2007, Volume: 29, Issue:5

    Topics: Adult; Age Factors; Amisulpride; Antimanic Agents; Antiparkinson Agents; Antipsychotic Agents; Benzodiazepines; Bipolar Disorder; Clozapine; Cross-Sectional Studies; Dose-Response Relationship, Drug; Drug Therapy, Combination; Female; France; Hospitals, Psychiatric; Humans; Male; Mental Disorders; Middle Aged; Olanzapine; Practice Patterns, Physicians'; Psychotic Disorders; Risperidone; Sex Factors; Sulpiride

2007
Clozapine and amisulpride in refractory schizophrenia and alcohol dependence.
    Journal of clinical psychopharmacology, 2007, Volume: 27, Issue:5

    Topics: Alcoholism; Amisulpride; Antipsychotic Agents; Behavior, Addictive; Blood Glucose; Clozapine; Comorbidity; Diabetes Mellitus; Diagnosis, Dual (Psychiatry); Drug Therapy, Combination; Humans; Male; Middle Aged; Schizophrenia; Sulpiride

2007
Hemoperfusion in the treatment of acute clozapine intoxication in China.
    Journal of clinical psychopharmacology, 2007, Volume: 27, Issue:6

    Topics: Acute Disease; Adult; Alprazolam; Antipsychotic Agents; China; Clonazepam; Clozapine; Depressive Disorder; Dose-Response Relationship, Drug; Drug Overdose; Emergency Service, Hospital; Hemoperfusion; Humans; Medical History Taking; Middle Aged; Pulmonary Edema; Retrospective Studies; Schizophrenia; Stress Disorders, Post-Traumatic; Suicide, Attempted; Sulpiride; Unconsciousness; Wine

2007
Clozapine-induced myocarditis after long-term treatment: case presentation and clinical perspectives.
    Journal of psychopharmacology (Oxford, England), 2008, Volume: 22, Issue:5

    Topics: Amisulpride; Antipsychotic Agents; Clozapine; Dibenzothiazepines; Humans; Male; Middle Aged; Myocarditis; Quetiapine Fumarate; Schizophrenia; Sulpiride

2008
Comparing the use and discontinuation of antipsychotics in clinical practice: an observational study.
    The Journal of clinical psychiatry, 2008, Volume: 69, Issue:2

    Topics: Adult; Aged; Amisulpride; Antipsychotic Agents; Benzodiazepines; Bipolar Disorder; Clozapine; Dibenzothiazepines; Drug Administration Schedule; Female; Humans; Male; Medical Records; Middle Aged; Olanzapine; Patient Admission; Polypharmacy; Practice Patterns, Physicians'; Quetiapine Fumarate; Research Design; Retrospective Studies; Risperidone; Schizophrenia; Scotland; Sulpiride

2008
The putative antipsychotic alstonine reverses social interaction withdrawal in mice.
    Progress in neuro-psychopharmacology & biological psychiatry, 2008, Aug-01, Volume: 32, Issue:6

    Topics: Animals; Anti-Anxiety Agents; Antipsychotic Agents; Clozapine; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Haloperidol; Interpersonal Relations; Male; Mice; Motor Activity; Secologanin Tryptamine Alkaloids; Social Behavior Disorders; Sulpiride

2008
Subnanomolar dopamine D3 receptor antagonism coupled to moderate D2 affinity results in favourable antipsychotic-like activity in rodent models: II. behavioural characterisation of RG-15.
    Naunyn-Schmiedeberg's archives of pharmacology, 2008, Volume: 378, Issue:5

    Topics: Amisulpride; Animals; Antipsychotic Agents; Avoidance Learning; Benzodiazepines; Biological Availability; Catalepsy; Clozapine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Male; Motor Activity; Olanzapine; Pyridines; Rats; Rats, Wistar; Receptors, Dopamine D3; Sulfonamides; Sulpiride; Tissue Distribution

2008
Amisulpride the 'atypical' atypical antipsychotic--comparison to haloperidol, risperidone and clozapine.
    Schizophrenia research, 2008, Volume: 105, Issue:1-3

    Topics: Amisulpride; Amphetamine; Animals; Antipsychotic Agents; Basal Ganglia; Behavior, Animal; Blood-Brain Barrier; Brain; Clozapine; Conditioning, Psychological; Haloperidol; Male; Models, Animal; Motor Activity; Phencyclidine; Prefrontal Cortex; Prolactin; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Serotonin; Risperidone; Sulpiride

2008
Clozapine and sulpiride but not haloperidol or olanzapine activate brain DNA demethylation.
    Proceedings of the National Academy of Sciences of the United States of America, 2008, Sep-09, Volume: 105, Issue:36

    Topics: Acetylation; Animals; Benzodiazepines; Brain; Cell Adhesion Molecules, Neuronal; Clozapine; DNA Methylation; Extracellular Matrix Proteins; Glutamate Decarboxylase; Haloperidol; Histones; Lysine; Male; Mice; Nerve Tissue Proteins; Olanzapine; Promoter Regions, Genetic; Reelin Protein; Serine Endopeptidases; Sulpiride; Valproic Acid

2008
Antipsychotics possessing antidepressive efficacy increase Golf protein in rat striatum.
    Psychopharmacology, 2008, Volume: 201, Issue:2

    Topics: Amisulpride; Animals; Antipsychotic Agents; Benzodiazepines; Blotting, Western; Clozapine; Corpus Striatum; Depressive Disorder; Dose-Response Relationship, Drug; GTP-Binding Protein alpha Subunits; Haloperidol; Injections, Intraperitoneal; Male; Olanzapine; Rats; Rats, Wistar; Risperidone; Sulpiride; Time Factors

2008
Tardive dystonia associated with low-dose of amisulpride: a case report.
    Journal of clinical psychopharmacology, 2008, Volume: 28, Issue:5

    Topics: Adult; Amisulpride; Antipsychotic Agents; Clozapine; Dyskinesia, Drug-Induced; Dystonia; Humans; Male; Schizophrenia, Paranoid; Sulpiride

2008
Amisulpride treatment for clozapine-induced sialorrhea.
    Journal of clinical psychopharmacology, 2009, Volume: 29, Issue:2

    Topics: Adult; Amisulpride; Antipsychotic Agents; Clozapine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Humans; Male; Receptors, Dopamine D3; Schizophrenia, Paranoid; Sialorrhea; Sulpiride

2009
Neuroleptics: necrotising enterocolitis.
    Prescrire international, 2009, Volume: 18, Issue:100

    Topics: Antipsychotic Agents; Atropine; Benzodiazepines; Clozapine; Drug Therapy, Combination; Enterocolitis, Necrotizing; France; Humans; Risperidone; Sulpiride

2009
Amisulpride improved debilitating clozapine-induced sialorrhea.
    American journal of therapeutics, 2011, Volume: 18, Issue:3

    Topics: Antipsychotic Agents; Clozapine; Dopamine Antagonists; Humans; Male; Middle Aged; Randomized Controlled Trials as Topic; Sialorrhea; Sulpiride

2011
Tardive dystonia induced by switch of atypical antipsychotics.
    Pharmacopsychiatry, 2010, Volume: 43, Issue:5

    Topics: Amisulpride; Antipsychotic Agents; Benzodiazepines; Clozapine; Dyskinesia, Drug-Induced; Female; Humans; Middle Aged; Olanzapine; Schizophrenia; Sulpiride

2010
Amisulpride for clozapine induced sialorrhea.
    Psychopharmacology bulletin, 2009, Volume: 42, Issue:4

    Topics: Adult; Amisulpride; Antipsychotic Agents; Clozapine; Female; Humans; Sialorrhea; Sulpiride

2009
Relief from chronic intractable auditory hallucinations after long-term bilateral theta burst stimulation.
    The American journal of psychiatry, 2010, Volume: 167, Issue:11

    Topics: Amisulpride; Antipsychotic Agents; Clozapine; Cognitive Behavioral Therapy; Combined Modality Therapy; Dominance, Cerebral; Follow-Up Studies; Hallucinations; Humans; Middle Aged; Parietal Lobe; Schizophrenia, Paranoid; Sulpiride; Temporal Lobe; Theta Rhythm; Transcranial Magnetic Stimulation; Treatment Outcome

2010
Clock genes and body composition in patients with schizophrenia under treatment with antipsychotic drugs.
    Schizophrenia research, 2011, Volume: 125, Issue:2-3

    Topics: Adult; Age Factors; Alleles; Amisulpride; Anthropometry; Antipsychotic Agents; Aripiprazole; Benzodiazepines; Body Composition; Body Mass Index; CLOCK Proteins; Clozapine; Dibenzothiazepines; Drug Therapy, Combination; Female; Genetic Association Studies; Genetic Carrier Screening; Genotype; Humans; Long-Term Care; Male; Middle Aged; Mutation, Missense; Olanzapine; Period Circadian Proteins; Piperazines; Polymorphism, Single Nucleotide; Psychotic Disorders; Quetiapine Fumarate; Quinolones; Receptor, Melanocortin, Type 3; Receptors, Glucocorticoid; Receptors, Leptin; Risperidone; Schizophrenia; Sex Factors; Sulpiride; Syndecan-3

2011
Antiserotonergic antipsychotics are associated with obsessive-compulsive symptoms in schizophrenia.
    Psychological medicine, 2011, Volume: 41, Issue:11

    Topics: Adult; Amisulpride; Antipsychotic Agents; Aripiprazole; Benzodiazepines; Clozapine; Comorbidity; Female; Germany; Humans; Male; Matched-Pair Analysis; Obsessive-Compulsive Disorder; Olanzapine; Piperazines; Prevalence; Quinolones; Schizophrenia; Serotonin Antagonists; Severity of Illness Index; Sulpiride

2011
Clozapine-induced salivation: interaction with N-desmethylclozapine and amisulpride in an experimental rat model.
    European journal of oral sciences, 2011, Volume: 119, Issue:4

    Topics: Abdomen; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Amisulpride; Animals; Antipsychotic Agents; Blood Pressure; Chorda Tympani Nerve; Clozapine; Female; Lingual Nerve; Liver Circulation; Methacholine Chloride; Models, Animal; Muscarinic Agonists; Parasympathectomy; Phentolamine; Propranolol; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M1; Receptor, Muscarinic M3; Saliva; Salivation; Submandibular Gland; Sulpiride; Time Factors

2011
Amisulpride augmentation of clozapine in refractory schizophrenia.
    The Journal of neuropsychiatry and clinical neurosciences, 2011,Summer, Volume: 23, Issue:3

    Topics: Amisulpride; Antipsychotic Agents; Clozapine; Drug Synergism; Humans; Male; Middle Aged; Schizophrenia; Sulpiride

2011
Effects of amisulpride and aripiprazole on progressive-ratio schedule performance: comparison with clozapine and haloperidol.
    Journal of psychopharmacology (Oxford, England), 2012, Volume: 26, Issue:9

    Topics: Amisulpride; Animals; Antipsychotic Agents; Aripiprazole; Behavior, Animal; Clozapine; Conditioning, Operant; Dopamine Antagonists; Dose-Response Relationship, Drug; Female; Haloperidol; Kinetics; Models, Biological; Motor Activity; Motor Skills; Piperazines; Quinolones; Rats; Rats, Wistar; Reaction Time; Reinforcement Schedule; Serotonin Antagonists; Sulpiride

2012
Onset of action of atypical and typical antipsychotics in the treatment of adolescent schizophrenic psychoses.
    Neuro endocrinology letters, 2011, Volume: 32, Issue:5

    Topics: Adolescent; Antipsychotic Agents; Benzodiazepines; Clozapine; Dibenzothiazepines; Female; Haloperidol; Humans; Male; Medical Records; Olanzapine; Perphenazine; Piperazines; Psychotic Disorders; Quetiapine Fumarate; Risperidone; Schizophrenia; Sulpiride; Thiazoles; Time Factors; Treatment Outcome

2011
Pregabalin-associated increase of clozapine serum levels.
    Journal of clinical psychopharmacology, 2012, Volume: 32, Issue:1

    Topics: Antimanic Agents; Antipsychotic Agents; Anxiety Disorders; Clozapine; Female; gamma-Aminobutyric Acid; Humans; Lithium Compounds; Male; Schizophrenia; Sulpiride

2012
Second-generation antipsychotic medications and risk of pneumonia in schizophrenia.
    Schizophrenia bulletin, 2013, Volume: 39, Issue:3

    Topics: Adult; Amisulpride; Antipsychotic Agents; Benzodiazepines; Case-Control Studies; Clozapine; Cohort Studies; Dibenzothiazepines; Dibenzothiepins; Drug Therapy, Combination; Female; Humans; Logistic Models; Male; Middle Aged; Olanzapine; Pneumonia; Quetiapine Fumarate; Risk Factors; Risperidone; Schizophrenia; Sulpiride; Taiwan

2013
Atypical antipsychotics--effects of amisulpride on salivary secretion and on clozapine-induced sialorrhea.
    Oral diseases, 2012, Volume: 18, Issue:7

    Topics: Amisulpride; Amylases; Animals; Antipsychotic Agents; Autonomic Agents; Bethanechol; Clozapine; Denervation; Female; Isoproterenol; Methacholine Chloride; Parasympathetic Nervous System; Parotid Gland; Raclopride; Rats; Rats, Sprague-Dawley; Saliva; Salivation; Sialorrhea; Submandibular Gland; Substance P; Sulpiride; Sympathetic Nervous System

2012
Differential effects of antipsychotics on lateral bias and social attention in female rats.
    Psychopharmacology, 2013, Volume: 225, Issue:2

    Topics: Animals; Antipsychotic Agents; Attention; Behavior, Animal; Clozapine; Disease Models, Animal; Female; Functional Laterality; Haloperidol; Rats; Rats, Long-Evans; Social Behavior; Sulpiride

2013
Plasma amisulpride in relation to prescribed dose, clozapine augmentation, and other factors: data from a therapeutic drug monitoring service, 2002-2010.
    Human psychopharmacology, 2012, Volume: 27, Issue:5

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Amisulpride; Antipsychotic Agents; Clozapine; Dose-Response Relationship, Drug; Drug Interactions; Drug Monitoring; Female; Humans; Linear Models; Male; Middle Aged; Smoking; Sulpiride; Young Adult

2012
Effect of atypical antipsychotics on antioxidant enzyme activities in human erythrocytes (in vitro study).
    Human psychopharmacology, 2013, Volume: 28, Issue:1

    Topics: Adult; Amisulpride; Antioxidants; Antipsychotic Agents; Aripiprazole; Benzodiazepines; Catalase; Clozapine; Dibenzothiazepines; Enzyme Activation; Erythrocytes; Glutathione Peroxidase; Glutathione Reductase; Humans; Imidazoles; Indoles; Male; Olanzapine; Piperazines; Quetiapine Fumarate; Quinolones; Sulpiride; Superoxide Dismutase; Superoxide Dismutase-1; Thiazoles; Treatment Outcome; Young Adult

2013
LC-MS/MS of some atypical antipsychotics in human plasma, serum, oral fluid and haemolysed whole blood.
    Forensic science international, 2013, Jun-10, Volume: 229, Issue:1-3

    Topics: Amisulpride; Antipsychotic Agents; Aripiprazole; Benzodiazepines; Chromatography, Liquid; Clozapine; Dibenzothiazepines; Female; Forensic Toxicology; Hemolysis; Humans; Isoxazoles; Male; Olanzapine; Paliperidone Palmitate; Piperazines; Pyrimidines; Quetiapine Fumarate; Quinolones; Reproducibility of Results; Risperidone; Saliva; Serum; Sulpiride; Tandem Mass Spectrometry

2013
Stability of some atypical antipsychotics in human plasma, haemolysed whole blood, oral fluid, human serum and calf serum.
    Forensic science international, 2013, Jun-10, Volume: 229, Issue:1-3

    Topics: Amisulpride; Animals; Antipsychotic Agents; Aripiprazole; Benzodiazepines; Cattle; Chromatography, Liquid; Clozapine; Dibenzothiazepines; Drug Stability; Female; Forensic Toxicology; Hemolysis; Humans; Isoxazoles; Male; Olanzapine; Paliperidone Palmitate; Piperazines; Pyrimidines; Quetiapine Fumarate; Quinolones; Reproducibility of Results; Risperidone; Saliva; Serum; Sulpiride; Tandem Mass Spectrometry

2013
Clozapine augmented with amisulpride in 3 cases of treatment-resistant early- and very early-onset schizophrenia.
    Journal of clinical psychopharmacology, 2013, Volume: 33, Issue:4

    Topics: Adolescent; Amisulpride; Antipsychotic Agents; Clozapine; Drug Resistance; Drug Therapy, Combination; Female; Humans; Male; Schizophrenia, Childhood; Schizophrenic Psychology; Sulpiride; Treatment Outcome

2013
Hypochondriasis and obsessive-compulsive disorder in schizophrenic patients treated with clozapine vs other atypical antipsychotics.
    CNS spectrums, 2014, Volume: 19, Issue:4

    Topics: Adult; Amisulpride; Antipsychotic Agents; Aripiprazole; Benzodiazepines; Clozapine; Comorbidity; Female; Humans; Hypochondriasis; Male; Middle Aged; Obsessive-Compulsive Disorder; Olanzapine; Paliperidone Palmitate; Prevalence; Quetiapine Fumarate; Risperidone; Schizophrenia; Schizophrenic Psychology; Sulpiride

2014
Augmentation of clozapine with amisulpride: an effective therapeutic strategy for violent treatment-resistant schizophrenia patients in a UK high-security hospital.
    CNS spectrums, 2014, Volume: 19, Issue:5

    Topics: Adult; Aggression; Amisulpride; Antipsychotic Agents; Blood Glucose; Body Mass Index; Cholesterol; Cholesterol, HDL; Clozapine; Cohort Studies; Drug Therapy, Combination; Hospitals, Psychiatric; Humans; Male; Retrospective Studies; Schizophrenia; Schizophrenic Psychology; Security Measures; Sulpiride; Treatment Outcome; United Kingdom; Violence; Young Adult

2014
Effects of antipsychotics on bone mineral density and prolactin levels in patients with schizophrenia: a 12-month prospective study.
    Human psychopharmacology, 2014, Volume: 29, Issue:2

    Topics: Adult; Alkaline Phosphatase; Antipsychotic Agents; Aripiprazole; Bone Density; Chlorpromazine; Clozapine; Dibenzothiazepines; Estrogens; Female; Humans; Male; Middle Aged; Osteoporosis; Perphenazine; Piperazines; Prolactin; Prospective Studies; Quetiapine Fumarate; Quinolones; Risk Factors; Schizophrenia; Sulpiride

2014
Upregulation of dopamine D3, not D2, receptors correlates with tardive dyskinesia in a primate model.
    Movement disorders : official journal of the Movement Disorder Society, 2014, Volume: 29, Issue:9

    Topics: Animals; Antipsychotic Agents; Brain; Cebus; Clozapine; Disease Models, Animal; Dopamine Antagonists; Enkephalins; Female; Haloperidol; Iodine Radioisotopes; Movement Disorders; Neurons; Ovariectomy; Protein Binding; Receptors, Dopamine D2; Receptors, Dopamine D3; Sulpiride; Tetrahydronaphthalenes; Up-Regulation

2014
Increased orbitofrontal cortex activation associated with "pro-obsessive" antipsychotic treatment in patients with schizophrenia.
    Journal of psychiatry & neuroscience : JPN, 2015, Volume: 40, Issue:2

    Topics: Adult; Amisulpride; Antipsychotic Agents; Aripiprazole; Benzodiazepines; Brain Mapping; Clozapine; Executive Function; Female; Humans; Inhibition, Psychological; Magnetic Resonance Imaging; Male; Neuropsychological Tests; Obsessive Behavior; Olanzapine; Piperazines; Prefrontal Cortex; Psychiatric Status Rating Scales; Psychomotor Performance; Quinolones; Schizophrenia; Sulpiride

2015
Clozapine augmentation with amisulpride.
    Journal of psychiatry & neuroscience : JPN, 2014, Volume: 39, Issue:6

    Topics: Adult; Amisulpride; Antipsychotic Agents; Clozapine; Drug Synergism; Humans; Male; Schizophrenia; Sulpiride

2014
Skating on thin ice: pragmatic prescribing for medication refractory schizophrenia.
    BMC psychiatry, 2015, Jul-25, Volume: 15

    Topics: Adult; Amisulpride; Antipsychotic Agents; Benzodiazepines; Clozapine; Drug Prescriptions; Drug Therapy, Combination; Female; Humans; Male; Middle Aged; Olanzapine; Quetiapine Fumarate; Schizophrenia; Schizophrenic Psychology; Sulpiride; Valproic Acid

2015
Adjunctive ondansetron in schizophrenia--A pilot study.
    Asian journal of psychiatry, 2016, Volume: 19

    Topics: Adult; Amisulpride; Antipsychotic Agents; Clozapine; Drug Therapy, Combination; Feasibility Studies; Humans; Ondansetron; Pilot Projects; Schizophrenia; Sulpiride; Treatment Outcome

2016
Antipsychotic Drugs Differentially Affect mRNA Expression of Genes Encoding the Neuregulin 1-Downstream ErbB4-PI3K Pathway.
    Pharmacology, 2016, Volume: 98, Issue:1-2

    Topics: Amisulpride; Antipsychotic Agents; Benzodiazepines; Cell Line, Tumor; Cell Survival; Clozapine; Gene Expression Regulation; Haloperidol; Humans; Neuregulin-1; Olanzapine; Phosphatidylinositol 3-Kinases; Quetiapine Fumarate; Receptor, ErbB-4; RNA, Messenger; Schizophrenia; Sulpiride

2016
Metformin-induced acute dystonia in a schizophrenic patient treated with sulpiride and clozapine.
    Psychiatry and clinical neurosciences, 2016, Volume: 70, Issue:8

    Topics: Antipsychotic Agents; Clozapine; Drug Interactions; Drug Therapy, Combination; Dystonia; Female; Humans; Hypoglycemic Agents; Metabolic Syndrome; Metformin; Middle Aged; Schizophrenia; Sulpiride

2016
Level of serum thioredoxin and correlation with neurocognitive functions in patients with schizophrenia using clozapine and other atypical antipsychotics.
    Psychiatry research, 2017, Volume: 247

    Topics: Adult; Amisulpride; Antipsychotic Agents; Benzodiazepines; Clozapine; Cognition; Female; Humans; Male; Middle Aged; Neuropsychological Tests; Olanzapine; Psychotic Disorders; Risperidone; Schizophrenia; Sulpiride; Thioredoxins; Young Adult

2017
Time to Discontinuation of Second-Generation Antipsychotics Versus Haloperidol and Sulpiride in People With Schizophrenia: A Naturalistic, Comparative Study.
    Journal of clinical psychopharmacology, 2017, Volume: 37, Issue:1

    Topics: Adult; Antipsychotic Agents; Clozapine; Female; Haloperidol; Humans; Male; Medication Adherence; Retrospective Studies; Schizophrenia; Sulpiride; Taiwan; Time Factors; Young Adult

2017
Measurement of Clozapine, Norclozapine, and Amisulpride in Plasma and in Oral Fluid Obtained Using 2 Different Sampling Systems.
    Therapeutic drug monitoring, 2017, Volume: 39, Issue:2

    Topics: Adult; Aged; Amisulpride; Antipsychotic Agents; Body Fluids; Chromatography, Liquid; Clozapine; Drug Monitoring; Female; Humans; Male; Middle Aged; Mouth; Plasma; Sulpiride; Tandem Mass Spectrometry; Young Adult

2017
The role of sulpiride in attenuating the cardiac, renal, and immune disruptions in rats receiving clozapine: mRNA expression pattern of the genes encoding Kim-1, TIMP-1, and CYP isoforms.
    Environmental science and pollution research international, 2020, Volume: 27, Issue:20

    Topics: Animals; Clozapine; Cytochrome P-450 Enzyme System; Male; Protein Isoforms; Rats; RNA, Messenger; Sulpiride; Tissue Inhibitor of Metalloproteinase-1

2020
Identification and Quantification of Antipsychotics in Blood Samples by LC-MS-MS: Case Reports and Data from Three Years of Routine Analysis.
    Journal of analytical toxicology, 2020, Dec-12, Volume: 44, Issue:8

    Topics: Adult; Amisulpride; Antipsychotic Agents; Aripiprazole; Benzodiazepines; Chromatography, Liquid; Clozapine; Dibenzothiazepines; Female; Forensic Toxicology; Humans; Male; Olanzapine; Paliperidone Palmitate; Piperazines; Quetiapine Fumarate; Retrospective Studies; Risperidone; Schizophrenia; Substance Abuse Detection; Suicide; Sulpiride; Tandem Mass Spectrometry; Thiazoles

2020
Clozapine-Induced Hypersalivation Treated with Sulpiride - Is It a Solution?
    Psychiatria Danubina, 2021,Spring, Volume: 33, Issue:Suppl 4

    Topics: Antipsychotic Agents; Clozapine; Humans; Schizophrenia; Sialorrhea; Sulpiride

2021
Letter to the Editor: Rethinking The Cost Of Antipsychotic Treatment: The Average Cost Of The Drugs Used In Turkey In 2020.
    Turk psikiyatri dergisi = Turkish journal of psychiatry, 2022,Summer, Volume: 33, Issue:2

    Topics: Adenosine Monophosphate; Adult; Amisulpride; Antipsychotic Agents; Aripiprazole; Benzodiazepines; Chlorpromazine; Clopenthixol; Clozapine; Flupenthixol; Fluphenazine; Haloperidol; Humans; Olanzapine; Paliperidone Palmitate; Pharmaceutical Preparations; Pimozide; Quetiapine Fumarate; Risperidone; Sulpiride; Trifluoperazine

2022
Environmentally-relevant concentrations of the antipsychotic drugs sulpiride and clozapine induce abnormal dopamine and serotonin signaling in zebrafish brain.
    Scientific reports, 2022, 10-26, Volume: 12, Issue:1

    Topics: Animals; Antipsychotic Agents; Brain; Clozapine; Dopamine; Haloperidol; Monoamine Oxidase; RNA, Messenger; Serotonin; Serotonin Plasma Membrane Transport Proteins; Sulpiride; Zebrafish

2022