Page last updated: 2024-08-17

sulfamic acid and estrone

sulfamic acid has been researched along with estrone in 15 studies

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (20.00)18.2507
2000's8 (53.33)29.6817
2010's3 (20.00)24.3611
2020's1 (6.67)2.80

Authors

AuthorsStudies
Howarth, NM; Potter, BV; Purohit, A; Reed, MJ1
Elger, W; Hedden, A; Reddersen, G; Schneider, B; Schwarz, S1
Elger, W; Henkel, H; Richter, M; Schwarz, S; Thieme, I; Undeutsch, B1
Barrow, D; Hejaz, HA; Nicholson, RI; Potter, BV; Purohit, A; Reed, MJ; Woo, LW1
Ahmed, S; James, K; Owen, CP; Patel, CK; Patel, M2
Casini, A; Montero, JL; Scozzafava, A; Supuran, CT; Vullo, D; Winum, JY1
Fujii, T; Iwashita, S; Koizumi, N; Nakagawa, T; Okada, M; Takegawa, S1
Liebl, R; von Angerer, E; Walter, G1
Chander, SK; Potter, BV; Purohit, A; Reed, MJ; Woo, LW1
Hejaz, HA; Leese, MP; Mahon, MF; Newman, SP; Potter, BV; Purohit, A; Reed, MJ1
Potter, BV; Purohit, A; Woo, LW1
Edwards, DR; Wolfenden, R1
Potter, BV; Thomas, MP1
Ali, H; Gémes, N; Mernyák, E; Minorics, R; Paragi, G; Resch, V; Szebeni, GJ; Traj, P; Zupkó, I1

Reviews

1 review(s) available for sulfamic acid and estrone

ArticleYear
Development of steroid sulfatase inhibitors.
    Molecular and cellular endocrinology, 2011, Jul-04, Volume: 340, Issue:2

    Topics: Drug Design; Enzyme Inhibitors; Estrone; Humans; Steryl-Sulfatase; Sulfonic Acids

2011

Other Studies

14 other study(ies) available for sulfamic acid and estrone

ArticleYear
Estrone sulfamates: potent inhibitors of estrone sulfatase with therapeutic potential.
    Journal of medicinal chemistry, 1994, Jan-21, Volume: 37, Issue:2

    Topics: Breast Neoplasms; Cell Division; Drug Screening Assays, Antitumor; Estrone; Humans; Sulfatases; Sulfonic Acids; Tumor Cells, Cultured

1994
Sulfamates of various estrogens are prodrugs with increased systemic and reduced hepatic estrogenicity at oral application.
    The Journal of steroid biochemistry and molecular biology, 1995, Volume: 55, Issue:3-4

    Topics: Administration, Oral; Angiotensin I; Animals; Cholesterol; Cholesterol, HDL; Contraceptives, Oral; Drug Evaluation, Preclinical; Estradiol; Estrogens; Estrone; Ethinyl Estradiol; Female; Follicle Stimulating Hormone; Liver; Luteinizing Hormone; Organ Size; Ovariectomy; Prodrugs; Rats; Rats, Wistar; Sulfonic Acids; Uterus

1995
Synthesis of estrogen sulfamates: compounds with a novel endocrinological profile.
    Steroids, 1996, Volume: 61, Issue:12

    Topics: Estradiol; Estriol; Estrogens; Estrone; Magnetic Resonance Spectroscopy; Sulfonic Acids

1996
Non-steroidal and steroidal sulfamates: new drugs for cancer therapy.
    Molecular and cellular endocrinology, 2001, Jan-22, Volume: 171, Issue:1-2

    Topics: Animals; Antineoplastic Agents; Breast Neoplasms; Coumarins; Enzyme Inhibitors; Estrogens; Estrone; Female; Humans; Kinetics; Oxepins; Rats; Rats, Wistar; Sulfatases; Sulfonamides; Sulfonic Acids; Tumor Cells, Cultured

2001
Novel inhibitors of the enzyme estrone sulfatase (ES).
    Bioorganic & medicinal chemistry letters, 2001, Mar-26, Volume: 11, Issue:6

    Topics: Alkanes; Coumarins; Enzyme Inhibitors; Estrone; Inhibitory Concentration 50; Ketones; Mesylates; Sulfatases; Sulfonamides; Sulfonic Acids

2001
Acid dissociation constant, a potential physicochemical factor in the inhibition of the enzyme estrone sulfatase (ES).
    Bioorganic & medicinal chemistry letters, 2001, Apr-09, Volume: 11, Issue:7

    Topics: Estrogens; Estrone; Inhibitory Concentration 50; Kinetics; Phenols; Structure-Activity Relationship; Sulfatases; Sulfonic Acids

2001
Carbonic anhydrase inhibitors. Inhibition of cytosolic isozymes I and II and transmembrane, tumor-associated isozyme IX with sulfamates including EMATE also acting as steroid sulfatase inhibitors.
    Journal of medicinal chemistry, 2003, May-22, Volume: 46, Issue:11

    Topics: Antigens, Neoplasm; Arylsulfatases; Biomarkers, Tumor; Carbonic Anhydrase I; Carbonic Anhydrase II; Carbonic Anhydrase IX; Carbonic Anhydrases; Cytosol; Enzyme Inhibitors; Estrone; Humans; Membrane Proteins; Neoplasm Proteins; Steryl-Sulfatase; Structure-Activity Relationship; Sulfonic Acids

2003
Development of novel steroid sulfatase inhibitors. I. Synthesis and biological evaluation of biphenyl-4-O-sulfamates.
    The Journal of steroid biochemistry and molecular biology, 2003, Volume: 87, Issue:2-3

    Topics: Animals; Biphenyl Compounds; Breast Neoplasms; Cell Line, Tumor; Enzyme Inhibitors; Estradiol; Estrogen Receptor alpha; Estrone; Female; Humans; Liver; Organ Size; Rats; Rats, Sprague-Dawley; Receptors, Estrogen; Steryl-Sulfatase; Structure-Activity Relationship; Sulfonic Acids; Uterus

2003
2-phenylindole sulfamates: inhibitors of steroid sulfatase with antiproliferative activity in MCF-7 breast cancer cells.
    The Journal of steroid biochemistry and molecular biology, 2004, Volume: 88, Issue:4-5

    Topics: Antineoplastic Agents; Breast Neoplasms; Cell Division; Enzyme Inhibitors; Estrone; Female; Gene Expression Regulation, Neoplastic; Humans; Hydrolysis; Hydrophobic and Hydrophilic Interactions; Inhibitory Concentration 50; Receptors, Estrogen; Steryl-Sulfatase; Structure-Activity Relationship; Sulfonic Acids; Transcriptional Activation

2004
The role of steroid sulphatase in regulating the oestrogenicity of oestrogen sulphamates.
    Biochemical and biophysical research communications, 2004, Sep-10, Volume: 322, Issue:1

    Topics: Animals; Coumarins; Drug Combinations; Estrogens; Estrone; Female; Homeostasis; Organ Size; Ovariectomy; Rats; Rats, Wistar; Steryl-Sulfatase; Sulfonamides; Sulfonic Acids; Uterus

2004
A-ring-substituted estrogen-3-O-sulfamates: potent multitargeted anticancer agents.
    Journal of medicinal chemistry, 2005, Aug-11, Volume: 48, Issue:16

    Topics: Angiogenesis Inhibitors; Animals; Antineoplastic Agents; Cell Line, Tumor; Cell Proliferation; Crystallography, X-Ray; Drug Screening Assays, Antitumor; Estradiol; Estrone; Female; Humans; Mice; Molecular Structure; Steryl-Sulfatase; Structure-Activity Relationship; Sulfonic Acids; Transplantation, Heterologous

2005
Proton-in-flight mechanism for the spontaneous hydrolysis of N-methyl O-phenyl sulfamate: implications for the design of steroid sulfatase inhibitors.
    The Journal of organic chemistry, 2012, May-04, Volume: 77, Issue:9

    Topics: Arylsulfatases; Catalysis; Coumarins; Esters; Estrone; Hydrogen-Ion Concentration; Hydrolysis; Kinetics; Molecular Structure; Steryl-Sulfatase; Sulfonamides; Sulfonic Acids

2012
Discovery and Development of the Aryl O-Sulfamate Pharmacophore for Oncology and Women's Health.
    Journal of medicinal chemistry, 2015, Oct-08, Volume: 58, Issue:19

    Topics: Animals; Antineoplastic Agents; Aromatase Inhibitors; Breast Neoplasms; Drug Discovery; Endometriosis; Estrone; Female; Humans; Male; Molecular Targeted Therapy; Prostatic Neoplasms; Steryl-Sulfatase; Sulfonic Acids; Tubulin Modulators

2015
Investigation of the Antineoplastic Effects of 2-(4-Chlorophenyl)-13α-Estrone Sulfamate against the HPV16-Positive Human Invasive Cervical Carcinoma Cell Line SiHa.
    International journal of molecular sciences, 2023, Apr-01, Volume: 24, Issue:7

    Topics: Antineoplastic Agents; Apoptosis; Cell Line; Cell Line, Tumor; Cell Proliferation; Estrone; Female; Human papillomavirus 16; Humans; Uterine Cervical Neoplasms

2023