Page last updated: 2024-08-23

substance p and sr 142801

substance p has been researched along with sr 142801 in 57 studies

Research

Studies (57)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's27 (47.37)18.2507
2000's26 (45.61)29.6817
2010's4 (7.02)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Barthò, L; Holzer, P; Maggi, CA; Patacchini, R1
Maggi, CA; Zagorodnyuk, V1
Farina, C; Foley, JJ; Giardina, GA; Grugni, M; Hay, DW; Medhurst, AD; Raveglia, LF; Rigolio, R; Sarau, HM; Schmidt, DB; Vassallo, M; Vecchietti, V1
De Giorgio, R; Giuliani, S; Lecci, A; Maggi, CA; Meini, S; Tramontana, M1
Giuliani, S; Maggi, CA1
Inoue, H; Koshihara, Y; Nagata, N1
Marchionni, D; Nisato, D; Roccon, A1
Barnouin, MC; Emonds-Alt, X; Hayar, A; Jung, M; Le Fur, G; Michaud, JC; Mons, G; Soubrié, P; Souilhac, J; Steinberg, R1
Costa, C; Cozzolino, A; Esposito, C; Falciani, M; Filippelli, A; Porta, R; Rossi, F1
Alonso, R; Carayon, P; Fournier, M; Le Fur, G; Petitpretre, G; Soubrié, P1
Hay, DW; Medhurst, AD; Parsons, AA; Roberts, JC1
Hardwick, JC; Mawe, GM; Parsons, RL1
Griswold, DE; Hay, DW; Martin, LD; Medhurst, AD; Parsons, AA1
Fisher, L; Pennefather, JN1
MacNaughton, W; Moore, B; Vanner, S1
Barbot, L; Cellier, E; Couture, R; Regoli, D1
Chahl, LA; Yip, J1
Bornstein, JC; Burcher, E; Johnson, PJ1
Moore, KA; Taylor, GE; Weinreich, D1
Bougault, I; Le Fur, G; Marco, N; Mons, G; Soubrié, P; Steinberg, R; Thirion, A1
Guo, JZ; Otsuka, M; Yoshioka, K1
Furness, JB; Jenkinson, KM; Southwell, BR1
Linden, DR; Seybold, VS1
Buéno, L; Gebhart, GF; Julia, V; Su, X1
Gerard, NP; Nguyen, N; Pasricha, PJ; Saban, MR; Saban, R1
Bredenbröker, D; Fehmann, H; Klüber, D; Lange, A; Wagner, U; Wichert, P1
Calixto, JB; De Lima, TC; Ribeiro, SJ; Teixeira, RM1
Lee, K; Pinnock, RD; Preston, Z; Richardson, PJ; Widdowson, L1
Barbot, L; Couture, R; Toma, N1
Geraghty, DP; Mazzone, SB1
Barthó, L; Benkó, R; Lázár, Z; Lénárd, L; Maggi, CA; Penke, B; Szolcsányi, J; Tóth, G1
Lee, K; Pinnock, RD; Preston, Z; Richardson, PJ1
Advenier, C; Daoui, S; Emonds-Alt, X; Lagente, V; Naline, E1
Crane, LH; Hamlin, GP; Nimmo, AJ; Williams, MJ1
Advenier, C; Beerens, D; Gustin, P; Halloy, D; Moreaux, B; Nemmar, A; Vincke, G1
Jurzak, M; Langlois, X; Leysen, JE; te Riele , P; Wintmolders, C1
Chen, J; Zheng, JH1
Gibbins, IL; Jobling, P; Messenger, JP1
Aggio, A; Carnicelli, V; Ciccocioppo, R; Onori, L; Severi, C; Taddei, G; Tonini, M1
Manning, BP; Mawe, GM1
Jurzak, M; Langlois, X; Leysen, JE; te Riele, P; Wintmolders, C1
Allouard, N; Bert, L; Bougault, I; Le-Fur, G; Rodier, D; Soubrié, P; Steinberg, R1
Glowinski, J; Godeheu, G; Kemel, ML; Pérez, S; Soubrié, P1
Anukwu, LU; Canning, BJ; Kajekar, R; Myers, AC; Reynolds, SM1
Akhtar, R; Brain, SD; Gerard, NP; Grant, AD1
Hirano, K; Kanaide, H; Naito, S; Nishimura, J; Takahashi, R1
Cvetkovic, V; Fellmann, D; Griffond, B; Poncet, F; Risold, PY1
de Francischi, JN; Lisboa, MC; Santos, JM; Tatsuo, MA; Turchetti-Maia, RM1
Bornstein, JC; Johnson, PJ1
De Man, JG; De Schepper, HU; De Winter, BY; Herman, AG; Pelckmans, PA; Seerden, TC1
Bertrand, PP; Bornstein, JC; Monro, RL1
Candenas, ML; Fernández-Sánchez, M; Orea, A; Pintado, CO; Pinto, FM; Ravina, CG; Seda, M1
Appleyard, CB; Morales, M; Santiago, C1
Kruse, CG; McCreary, AC; Wadman, WJ; Werkman, TR1
Boehm, U; de Croft, S; Herbison, AE1
Ballard, TM; Bissantz, C; Bohnert, C; Knoflach, F; Knust, H; Malherbe, P; Marcuz, A; Ratni, H; Spooren, W; Weber, M1
De Lima, TC; Duarte, FS; Duzzioni, M; Leme, LR; Smith, Sde P1

Other Studies

57 other study(ies) available for substance p and sr 142801

ArticleYear
Activity of SR 142801 at peripheral tachykinin receptors.
    European journal of pharmacology, 1995, May-04, Volume: 278, Issue:1

    Topics: Analysis of Variance; Animals; Binding, Competitive; Capsaicin; Cricetinae; Guinea Pigs; Ileum; In Vitro Techniques; Male; Mesocricetus; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Portal Vein; Pulmonary Artery; Rabbits; Rats; Rats, Wistar; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Trachea

1995
Neuronal tachykinin NK2 receptors mediate release of non-adrenergic non-cholinergic inhibitory transmitters in the circular muscle of guinea-pig colon.
    Neuroscience, 1995, Volume: 69, Issue:2

    Topics: Animals; Colon; Guinea Pigs; Male; Membrane Potentials; Peptide Fragments; Piperidines; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P

1995
2-Phenyl-4-quinolinecarboxamides: a novel class of potent and selective non-peptide competitive antagonists for the human neurokinin-3 receptor.
    Journal of medicinal chemistry, 1996, Jun-07, Volume: 39, Issue:12

    Topics: Animals; Binding, Competitive; CHO Cells; Ciliary Body; Cricetinae; Cricetulus; Drug Design; Guinea Pigs; Humans; Muscle Contraction; Peptide Fragments; Piperidines; Quinolines; Rabbits; Receptors, Neurokinin-3; Recombinant Fusion Proteins; Structure-Activity Relationship; Substance P

1996
In vivo evidence for the involvement of tachykinin NK3 receptors in the hexamethonium-resistant inhibitory transmission in the rat colon.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 353, Issue:6

    Topics: Adrenergic Agents; Animals; Colon; Dose-Response Relationship, Drug; Guanethidine; Hexamethonium; Male; Muscle Contraction; Neurokinin A; NG-Nitroarginine Methyl Ester; Nicotinic Antagonists; Peptide Fragments; Piperidines; Rats; Rats, Wistar; Receptors, Neurokinin-3; Receptors, Tachykinin; Substance P

1996
Effect of SR 142801 on nitric oxide-dependent and independent responses to tachykinin NK3 receptor agonists in isolated guinea-pig colon.
    Naunyn-Schmiedeberg's archives of pharmacology, 1995, Volume: 352, Issue:5

    Topics: Animals; Arginine; Colon; Electric Stimulation; Enzyme Inhibitors; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Nitric Oxide; Nitric Oxide Synthase; Nitroarginine; Peptide Fragments; Piperidines; Receptors, Neurokinin-3; Substance P

1995
Effect of the tachykinin receptor antagonists, SR 140333, FK 888, and SR 142801, on capsaicin-induced mouse ear oedema.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 1996, Volume: 45, Issue:6

    Topics: Animals; Binding Sites; Capsaicin; Dipeptides; Disease Models, Animal; Ear Diseases; Edema; Indoles; Injections, Intravenous; Lethal Dose 50; Male; Mice; Piperidines; Quinuclidines; Receptors, Tachykinin; Skin; Stereoisomerism; Structure-Activity Relationship; Substance P

1996
Study of SR 142801, a new potent non-peptide NK3 receptor antagonist on cardiovascular responses in conscious guinea-pig.
    British journal of pharmacology, 1996, Volume: 118, Issue:5

    Topics: Analysis of Variance; Animals; Blood Pressure; Dose-Response Relationship, Drug; Guinea Pigs; Heart Rate; Injections, Intravenous; Male; Neurokinin A; Neurokinin B; Peptide Fragments; Piperidines; Substance P

1996
Electrophysiological, behavioural and biochemical evidence for activation of brain noradrenergic systems following neurokinin NK3 receptor stimulation.
    Neuroscience, 1996, Volume: 74, Issue:2

    Topics: Adrenergic Fibers; Animals; Brain; Dose-Response Relationship, Drug; Gerbillinae; Guinea Pigs; Locus Coeruleus; Microdialysis; Neuropeptides; Norepinephrine; Peptide Fragments; Piperidines; Prazosin; Receptors, Neurokinin-3; Substance P

1996
Transglutaminase-synthesized spermine derivative of substance P recognizes rat portal vein neurokinin-3 receptors.
    Life sciences, 1997, Volume: 60, Issue:6

    Topics: Androstanes; Animals; Benzimidazoles; In Vitro Techniques; Male; Neurokinin A; Peptide Fragments; Physalaemin; Piperidines; Portal Vein; Rats; Rats, Wistar; Receptors, Neurokinin-3; Substance P; Thiorphan; Transglutaminases; Vasoconstriction

1997
Evidence for modulation of dopamine-neuronal function by tachykinin NK3 receptor stimulation in gerbil mesencephalic cell cultures.
    The European journal of neuroscience, 1996, Volume: 8, Issue:4

    Topics: Animals; Calcium; Cells, Cultured; Dopamine; Gerbillinae; Intracellular Membranes; Mesencephalon; Neurons; Peptide Fragments; Piperidines; Receptors, Neurokinin-3; Receptors, Tachykinin; Substance P

1996
Characterization of NK3 receptors in rabbit isolated iris sphincter muscle.
    British journal of pharmacology, 1997, Volume: 120, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Autoradiography; Benzamides; Electric Stimulation; In Vitro Techniques; Iris; Male; Muscle Contraction; Muscle, Smooth; Neurokinin B; Peptide Fragments; Phenoxybenzamine; Piperidines; Rabbits; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P

1997
Tachykinin-induced activation of non-specific cation conductance via NK3 neurokinin receptors in guinea-pig intracardiac neurones.
    The Journal of physiology, 1997, Oct-01, Volume: 504 ( Pt 1)

    Topics: Animals; Barium; Electrophysiology; Female; Guinea Pigs; Heart; In Vitro Techniques; Ion Channels; Male; Membrane Potentials; Neurons; Patch-Clamp Techniques; Piperidines; Receptors, Neurokinin-3; Substance P; Tachykinins; Tetraethylammonium Compounds

1997
In vitro and in vivo characterization of NK3 receptors in the rabbit eye by use of selective non-peptide NK3 receptor antagonists.
    British journal of pharmacology, 1997, Volume: 122, Issue:3

    Topics: Animals; In Vitro Techniques; Iris; Male; Miosis; Muscle Contraction; Muscle, Smooth; Neurokinin B; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Quinolines; Rabbits; Receptors, Neurokinin-3; Substance P

1997
Potencies of agonists acting at tachykinin receptors in the oestrogen-primed rat uterus: effects of peptidase inhibitors.
    European journal of pharmacology, 1997, Sep-24, Volume: 335, Issue:2-3

    Topics: Animals; Dipeptides; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Inhibitors; Estradiol; Female; Muscle, Smooth; Neurokinin A; Peptide Fragments; Piperidines; Protease Inhibitors; Rats; Rats, Sprague-Dawley; Receptors, Tachykinin; Substance P; Tachykinins; Uterine Contraction; Uterus

1997
Cellular pathways mediating tachykinin-evoked secretomotor responses in guinea pig ileum.
    The American journal of physiology, 1997, Volume: 273, Issue:5

    Topics: Animals; Capsaicin; Electric Stimulation; Evoked Potentials; Guinea Pigs; Ileum; In Vitro Techniques; Intestinal Mucosa; Membrane Potentials; Muscle, Smooth; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Neurons; Peptide Fragments; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Substance P; Tachykinins

1997
Cardiovascular and behavioural effects of intracerebroventricularly administered tachykinin NK3 receptor antagonists in the conscious rat.
    British journal of pharmacology, 1997, Volume: 122, Issue:4

    Topics: Animals; Behavior, Animal; Cardiovascular System; Dogs; Indoles; Injections, Intraventricular; Male; Oligopeptides; Peptide Fragments; Piperidines; Rats; Rats, Wistar; Receptors, Neurokinin-3; Substance P

1997
Localization of Fos-like immunoreactivity induced by the NK3 tachykinin receptor agonist, senktide, in the guinea-pig brain.
    British journal of pharmacology, 1997, Volume: 122, Issue:4

    Topics: Animals; Behavior, Animal; Brain; Female; Guinea Pigs; Male; Neurons; Peptide Fragments; Piperidines; Proto-Oncogene Proteins c-fos; Receptors, Neurokinin-3; Substance P; Tyrosine 3-Monooxygenase

1997
Roles of neuronal NK1 and NK3 receptors in synaptic transmission during motility reflexes in the guinea-pig ileum.
    British journal of pharmacology, 1998, Volume: 124, Issue:7

    Topics: Animals; Female; Gastrointestinal Motility; Guinea Pigs; Ileum; In Vitro Techniques; Male; Neurokinin-1 Receptor Antagonists; Neurons; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Substance P; Synaptic Transmission

1998
Serotonin unmasks functional NK-2 receptors in vagal sensory neurones of the guinea-pig.
    The Journal of physiology, 1999, Jan-01, Volume: 514 ( Pt 1)

    Topics: Animals; Benzamides; Cycloheximide; Enzyme Inhibitors; Guinea Pigs; Hydrazines; Imidazoles; Indoles; Male; Membrane Potentials; Neurons, Afferent; Nitric Oxide; Nitric Oxide Donors; Nodose Ganglion; omega-N-Methylarginine; Penicillamine; Piperidines; Protein Synthesis Inhibitors; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Substance P; Tropisetron

1999
Activation of dopaminergic and cholinergic neurotransmission by tachykinin NK3 receptor stimulation: an in vivo microdialysis approach in guinea pig.
    Neuropeptides, 1998, Volume: 32, Issue:5

    Topics: Acetylcholine; Animals; Brain; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Guinea Pigs; Hippocampus; Male; Microdialysis; Nucleus Accumbens; Peptide Fragments; Piperidines; Prefrontal Cortex; Receptors, Neurokinin-3; Substance P; Substantia Nigra; Synaptic Transmission; Time Factors; Ventral Tegmental Area

1998
Effects of a tachykinin NK3 receptor antagonist, SR 142801, studied in isolated neonatal rat spinal cord.
    Neuropeptides, 1998, Volume: 32, Issue:6

    Topics: Animals; Animals, Newborn; Capsaicin; Electrophysiology; Female; In Vitro Techniques; Male; Membrane Potentials; Neurokinin B; Neurons, Afferent; Patch-Clamp Techniques; Peptide Fragments; Piperidines; Rats; Rats, Wistar; Receptors, Neurokinin-3; Spinal Cord; Spinal Nerve Roots; Substance P

1998
Two affinities for a single antagonist at the neuronal NK1 tachykinin receptor: evidence from quantitation of receptor endocytosis.
    British journal of pharmacology, 1999, Volume: 126, Issue:1

    Topics: Animals; Binding, Competitive; Dose-Response Relationship, Drug; Endocytosis; Female; Fluorescence; Guinea Pigs; Ileum; In Vitro Techniques; Male; Microscopy, Confocal; Neurokinin-1 Receptor Antagonists; Neurons; Peptides, Cyclic; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Substance P

1999
Spinal neurokinin3 receptors mediate thermal but not mechanical hyperalgesia via nitric oxide.
    Pain, 1999, Volume: 80, Issue:1-2

    Topics: Animals; Animals, Newborn; Body Temperature; Electric Stimulation; Enzyme Inhibitors; Hot Temperature; Hyperalgesia; Male; Motor Neurons; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Peptide Fragments; Physical Stimulation; Piperidines; Postural Balance; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-3; Spinal Cord; Substance P

1999
Role of neurokinin 3 receptors on responses to colorectal distention in the rat: electrophysiological and behavioral studies.
    Gastroenterology, 1999, Volume: 116, Issue:5

    Topics: Animals; Colon; Electromyography; Gastrointestinal Motility; Injections, Intraperitoneal; Injections, Intraventricular; Male; Muscle Contraction; Pain Measurement; Peptide Fragments; Piperidines; Pressure; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Neurokinin-3; Rectum; Sensory Thresholds; Substance P; Visceral Afferents

1999
Nerve-mediated motility of ileal segments isolated from NK(1) receptor knockout mice.
    The American journal of physiology, 1999, Volume: 277, Issue:6

    Topics: Animals; Benzamides; Dose-Response Relationship, Drug; Gastrointestinal Motility; Ileum; Male; Mice; Mice, Knockout; Neurokinin A; Neurons, Afferent; Nitric Oxide; Organ Culture Techniques; Piperidines; Receptors, Cholinergic; Receptors, Neurokinin-1; Substance P; Synaptic Transmission

1999
Effects of selective tachykinin-receptor antagonists on tachykinin-induced airway mucus secretion in the rat.
    Neuropeptides, 1999, Volume: 33, Issue:1

    Topics: Animals; Benzamides; Male; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Piperidines; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Respiratory Mucosa; Substance P; Tachykinins; Trachea

1999
Tachykinin NK(3)receptor involvement in anxiety.
    Neuropeptides, 1999, Volume: 33, Issue:2

    Topics: Animals; Anxiety; Cerebral Ventricles; Injections, Intraventricular; Male; Maze Learning; Mice; Neurokinin A; Neurokinin B; Peptide Fragments; Piperidines; Receptors, Neurokinin-3; Substance P; Tachykinins

1999
Tachykinins increase [3H]acetylcholine release in mouse striatum through multiple receptor subtypes.
    Neuroscience, 2000, Volume: 95, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Acetylcholine; Alkaloids; Animals; Benzophenanthridines; Choline O-Acetyltransferase; Corpus Striatum; Electrophysiology; Enzyme Inhibitors; Estrenes; Excitatory Amino Acid Antagonists; In Situ Hybridization; Indoles; Interneurons; Membrane Potentials; Mice; Mice, Inbred C57BL; Neurokinin A; Oligopeptides; omega-N-Methylarginine; Peptide Fragments; Phenanthridines; Phosphodiesterase Inhibitors; Piperidines; Pyrrolidinones; Quinoxalines; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; RNA, Messenger; Signal Transduction; Substance P; Tachykinins; Tetrodotoxin; Tritium

2000
SR142801 behaves as a tachykinin NK-3 receptor agonist on a spinal nociceptive reflex in the rat.
    Life sciences, 2000, Volume: 66, Issue:1

    Topics: Analgesics; Animals; Drug Interactions; Indoles; Male; Naloxone; Narcotic Antagonists; Neurokinin-1 Receptor Antagonists; Oligopeptides; Pain Measurement; Peptide Fragments; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Spinal Cord; Substance P

2000
Respiratory actions of tachykinins in the nucleus of the solitary tract: characterization of receptors using selective agonists and antagonists.
    British journal of pharmacology, 2000, Volume: 129, Issue:6

    Topics: Animals; Benzamides; Indoles; Isoindoles; Male; Microinjections; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Piperidines; Rats; Rats, Wistar; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Respiratory Mechanics; Solitary Nucleus; Substance P; Tachykinins; Tidal Volume

2000
Evidence for the involvement of ATP, but not of VIP/PACAP or nitric oxide, in the excitatory effect of capsaicin in the small intestine.
    European journal of pharmacology, 2000, Mar-31, Volume: 392, Issue:3

    Topics: Acetylcholine; Adenosine Triphosphate; Animals; Capsaicin; Enzyme Inhibitors; Guinea Pigs; Ileum; In Vitro Techniques; Intestine, Small; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Neuropeptides; Nitric Oxide; Nitric Oxide Synthase; Nitroarginine; Peptide Fragments; Physalaemin; Piperidines; Pituitary Adenylate Cyclase-Activating Polypeptide; Pyridoxal Phosphate; Receptors, Neurokinin-3; Sincalide; Substance P; Vasoactive Intestinal Peptide

2000
NK-3 receptors are expressed on mouse striatal gamma-aminobutyric acid-ergic interneurones and evoke [(3)H] gamma-aminobutyric acid release.
    Neuroscience letters, 2000, Apr-21, Volume: 284, Issue:1-2

    Topics: Acetylcholine; Animals; gamma-Aminobutyric Acid; In Situ Hybridization; Interneurons; Mice; Mice, Inbred C57BL; Neostriatum; Nitric Oxide; Nitric Oxide Synthase; Peptide Fragments; Piperidines; Protein Precursors; Receptors, Neurokinin-3; RNA, Messenger; Somatostatin; Substance P; Tachykinins

2000
Neurokinin B- and specific tachykinin NK(3) receptor agonists-induced airway hyperresponsiveness in the guinea-pig.
    British journal of pharmacology, 2000, Volume: 130, Issue:1

    Topics: Acetylcholine; Animals; Bronchi; Bronchoconstrictor Agents; Female; Guinea Pigs; Male; Neurokinin B; Peptide Fragments; Piperidines; Receptors, Neurokinin-3; Substance P; Tachykinins; Vasodilator Agents

2000
Hormonal variation of rat uterine contractile responsiveness to selective neurokinin receptor agonists.
    Biology of reproduction, 2000, Volume: 62, Issue:6

    Topics: Animals; Diestrus; Estrogens; Estrus; Female; Metestrus; Neurokinin A; Ovariectomy; Peptide Fragments; Piperidines; Proestrus; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Uterine Contraction

2000
Role of substance P and tachykinin receptor antagonists in citric acid-induced cough in pigs.
    European journal of pharmacology, 2000, Nov-24, Volume: 408, Issue:3

    Topics: Animals; Benzamides; Citric Acid; Cough; Female; Lung; Male; Neurokinin-1 Receptor Antagonists; Piperidines; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Reflex; Substance P; Swine, Miniature

2000
Detailed distribution of Neurokinin 3 receptors in the rat, guinea pig and gerbil brain: a comparative autoradiographic study.
    Neuropharmacology, 2001, Volume: 40, Issue:2

    Topics: Animals; Autoradiography; Brain; Cerebral Cortex; Gerbillinae; Guinea Pigs; Male; Membranes; Peptide Fragments; Piperidines; Radioligand Assay; Rats; Rats, Wistar; Receptors, Neurokinin-3; Species Specificity; Substance P

2001
Differential roles of spinal neurokinin 1/2 receptors in development of persistent spontaneous nociception and hyperalgesia induced by subcutaneous bee venom injection in the conscious rat.
    Neuropeptides, 2001, Volume: 35, Issue:1

    Topics: Analgesics; Animals; Bee Venoms; Consciousness; Disease Models, Animal; Hot Temperature; Hyperalgesia; Injections, Subcutaneous; Neurokinin-1 Receptor Antagonists; Nociceptors; Pain Threshold; Physical Stimulation; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Spinal Cord; Substance P

2001
Differential expression of functionally identified and immunohistochemically identified NK(1) receptors on sympathetic neurons.
    Journal of neurophysiology, 2001, Volume: 85, Issue:5

    Topics: Action Potentials; Animals; Biotin; Coloring Agents; Enzyme Inhibitors; Female; Ganglia, Sympathetic; Guinea Pigs; Image Processing, Computer-Assisted; Immune Sera; Male; Microelectrodes; Nerve Tissue Proteins; Neurons; Patch-Clamp Techniques; Peptide Fragments; Piperidines; Protein Kinase C; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Substance P; Sympathetic Fibers, Postganglionic; Tachykinins

2001
Contribution of NK3 tachykinin receptors to propulsion in the rabbit isolated distal colon.
    Neurogastroenterology and motility, 2001, Volume: 13, Issue:3

    Topics: Animals; Colon; Complement C6; Dose-Response Relationship, Drug; Gastrointestinal Motility; In Vitro Techniques; Male; Peptide Fragments; Piperidines; Quinolines; Rabbits; Receptors, Neurokinin-3; Substance P

2001
Tachykinins mediate slow excitatory postsynaptic transmission in guinea pig sphincter of Oddi ganglia.
    American journal of physiology. Gastrointestinal and liver physiology, 2001, Volume: 281, Issue:2

    Topics: Animals; Calcium; Capsaicin; Culture Techniques; Excitatory Postsynaptic Potentials; Female; Ganglia; Guinea Pigs; Male; Membrane Potentials; Neurokinin-1 Receptor Antagonists; Neurons; Peptide Fragments; Piperidines; Receptors, Neurokinin-3; Receptors, Tachykinin; Sphincter of Oddi; Substance P; Synaptic Transmission; Tachykinins; Tetrodotoxin

2001
Use of the beta-imager for rapid ex vivo autoradiography exemplified with central nervous system penetrating neurokinin 3 antagonists.
    The Journal of pharmacology and experimental therapeutics, 2001, Volume: 299, Issue:2

    Topics: Animals; Autoradiography; Beta Particles; Brain; Central Nervous System; Dose-Response Relationship, Drug; Gerbillinae; Male; Peptide Fragments; Piperidines; Radionuclide Imaging; Receptors, Neurokinin-3; Substance P

2001
Permissive role of neurokinin NK(3) receptors in NK(1) receptor-mediated activation of the locus coeruleus revealed by SR 142801.
    Synapse (New York, N.Y.), 2002, Volume: 43, Issue:1

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Antiemetics; Dose-Response Relationship, Drug; Guinea Pigs; Locus Coeruleus; Male; Neural Pathways; Neurokinin-1 Receptor Antagonists; Neurons; Norepinephrine; Peptide Fragments; Piperidines; Prefrontal Cortex; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Substance P; Tetrazoles

2002
Facilitation by endogenous tachykinins of the NMDA-evoked release of acetylcholine after acute and chronic suppression of dopaminergic transmission in the matrix of the rat striatum.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2002, Mar-01, Volume: 22, Issue:5

    Topics: Acetylcholine; Animals; Benzamides; Corpus Striatum; Dopamine; Dopamine Antagonists; Enzyme Inhibitors; In Vitro Techniques; Male; N-Methylaspartate; Neural Inhibition; Neurons; Oxidopamine; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Tachykinin; Substance P; Synaptic Transmission; Tachykinins; Time Factors

2002
Endogenous neurokinins facilitate synaptic transmission in guinea pig airway parasympathetic ganglia.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2002, Volume: 283, Issue:2

    Topics: Animals; Bronchi; Bronchoconstriction; Electric Stimulation; Excitatory Postsynaptic Potentials; Ganglia, Parasympathetic; Guinea Pigs; Immunohistochemistry; In Vitro Techniques; Male; Neurons; Peptide Fragments; Piperidines; Quinolines; Receptors, Neurokinin-3; Substance P; Synaptic Transmission; Trachea; Vagotomy; Vagus Nerve

2002
Neurokinin B induces oedema formation in mouse lung via tachykinin receptor-independent mechanisms.
    The Journal of physiology, 2002, Sep-15, Volume: 543, Issue:Pt 3

    Topics: Animals; Antipsychotic Agents; Benzamides; Cyclooxygenase Inhibitors; Edema; Enzyme Inhibitors; Extravascular Lung Water; Female; Indomethacin; Mice; Mice, Inbred C57BL; Mice, Knockout; Neurokinin B; Neurokinin-1 Receptor Antagonists; NG-Nitroarginine Methyl Ester; Piperidines; Plasma; Pulmonary Edema; Receptors, Neurokinin-1; Substance P

2002
The mechanisms for tachykinin-induced contractions of the rabbit corpus cavernosum.
    British journal of pharmacology, 2002, Volume: 137, Issue:6

    Topics: Animals; Benzamides; Calcium; Dose-Response Relationship, Drug; Glycopeptides; In Vitro Techniques; Male; Muscle Contraction; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; NG-Nitroarginine Methyl Ester; Penis; Permeability; Piperidines; Quinuclidines; Rabbits; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Tachykinins; Type C Phospholipases

2002
Diencephalic neurons producing melanin-concentrating hormone are influenced by local and multiple extra-hypothalamic tachykininergic projections through the neurokinin 3 receptor.
    Neuroscience, 2003, Volume: 119, Issue:4

    Topics: Animals; Brain; Colchicine; Feeding Behavior; Hypothalamic Hormones; Hypothalamus; Interneurons; Male; Melanins; Neural Pathways; Neurokinin B; Neurokinin-1 Receptor Antagonists; Neurons; Organ Culture Techniques; Peptide Fragments; Piperidines; Pituitary Hormones; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-3; RNA, Messenger; Sexual Behavior; Substance P; Tachykinins

2003
Leukocyte recruitment to peritoneal cavity of rats following formalin injection: role of tachykinin receptors.
    Journal of pharmacological sciences, 2004, Volume: 94, Issue:4

    Topics: Animals; Benzamides; Cell Movement; Dose-Response Relationship, Drug; Female; Formaldehyde; Injections, Intraperitoneal; Leukocytes; Models, Biological; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Peritoneal Cavity; Peritoneal Lavage; Piperidines; Quinuclidines; Rats; Rats, Inbred Strains; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Substance P; Time Factors

2004
Neurokinin-1 and -3 receptor blockade inhibits slow excitatory synaptic transmission in myenteric neurons and reveals slow inhibitory input.
    Neuroscience, 2004, Volume: 126, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Antipsychotic Agents; Excitatory Postsynaptic Potentials; Female; Guinea Pigs; Male; Myenteric Plexus; Neural Inhibition; Neurokinin-1 Receptor Antagonists; Neurons; Peptide Fragments; Phentolamine; Piperazines; Piperidines; Quinuclidines; Reaction Time; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Serotonin 5-HT1 Receptor Antagonists; Serotonin Antagonists; Substance P; Synaptic Transmission

2004
Functional characterisation of tachykinin receptors in the circular muscle layer of the mouse ileum.
    Regulatory peptides, 2005, Sep-15, Volume: 130, Issue:3

    Topics: Action Potentials; Analgesics; Animals; Antipsychotic Agents; Atropine; Electric Stimulation; Ileum; Indoles; Isoindoles; Mice; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Neurons; Nitroarginine; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P

2005
Slow excitatory post-synaptic potentials in myenteric AH neurons of the guinea-pig ileum are reduced by the 5-hydroxytryptamine7 receptor antagonist SB 269970.
    Neuroscience, 2005, Volume: 134, Issue:3

    Topics: Animals; Drug Interactions; Electric Stimulation; Excitatory Postsynaptic Potentials; Female; Granisetron; Guinea Pigs; Ileum; Male; Myenteric Plexus; Neurons; Peptide Fragments; Phenols; Piperidines; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Substance P; Sulfonamides

2005
A role for tachykinins in the regulation of human sperm motility.
    Human reproduction (Oxford, England), 2007, Volume: 22, Issue:6

    Topics: Benzamides; Humans; Immunohistochemistry; Male; Neurokinin A; Neurokinin B; Piperidines; Quinuclidines; Receptors, Tachykinin; Sperm Motility; Spermatozoa; Substance P; Tachykinins

2007
Chronic inflammation alters the contribution of neurokinin receptor subtypes to epithelial function in rat colon.
    Digestive diseases and sciences, 2008, Volume: 53, Issue:1

    Topics: Anesthetics, Local; Animals; Anti-Inflammatory Agents, Non-Steroidal; Antipsychotic Agents; Benzamides; Colitis; Disease Models, Animal; Indomethacin; Intestinal Mucosa; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; Neurotransmitter Agents; Piperidines; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Stereoisomerism; Substance P; Tetrodotoxin; Trinitrobenzenesulfonic Acid

2008
NK3 receptors mediate an increase in firing rate of midbrain dopamine neurons of the rat and the guinea pig.
    Synapse (New York, N.Y.), 2011, Volume: 65, Issue:8

    Topics: Action Potentials; Animals; Antipsychotic Agents; Dopamine; Dopamine Agonists; Electrophysiology; Guinea Pigs; Male; Mesencephalon; Neurons; Organ Culture Techniques; Peptide Fragments; Piperidines; Rats; Rats, Wistar; Receptors, Neurokinin-3; Species Specificity; Substance P

2011
Neurokinin B activates arcuate kisspeptin neurons through multiple tachykinin receptors in the male mouse.
    Endocrinology, 2013, Volume: 154, Issue:8

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Non-Narcotic; Animals; Arcuate Nucleus of Hypothalamus; Dynorphins; Green Fluorescent Proteins; Kisspeptins; Male; Membrane Potentials; Mice; Mice, Transgenic; Neurokinin B; Neurons; Oligopeptides; Patch-Clamp Techniques; Peptide Fragments; Piperidines; Quinolines; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Opioid, kappa; Receptors, Tachykinin; Substance P

2013
Mapping the binding pocket of a novel, high-affinity, slow dissociating tachykinin NK3 receptor antagonist: biochemical and electrophysiological characterization.
    Neuropharmacology, 2014, Volume: 86

    Topics: Amino Acid Sequence; Animals; Antipsychotic Agents; Binding Sites; Carbamates; Central Nervous System Agents; Dopaminergic Neurons; Female; Gerbillinae; Guinea Pigs; HEK293 Cells; Humans; Locomotion; Male; Models, Molecular; Molecular Sequence Data; Mutation; Neurotransmitter Agents; Pars Compacta; Peptide Fragments; Piperidines; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Tissue Culture Techniques

2014
Evidence for involvement of NK₃ receptors in the anxiogenic-like effect of SP6-11(C-terminal), a metabolite of substance P, in rats evaluated in the elevated plus-maze.
    Behavioural brain research, 2016, Apr-15, Volume: 303

    Topics: Animals; Anxiety; Male; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Receptors, Neurokinin-3; Substance P

2016