Page last updated: 2024-08-23

substance p and sb 223412

substance p has been researched along with sb 223412 in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (25.00)18.2507
2000's7 (58.33)29.6817
2010's2 (16.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Brawner, ME; Elshourbagy, NA; Foley, JJ; Giardina, GA; Griswold, DE; Hay, DW; Martin, LD; Medhurst, AD; Potts, W; Sarau, HM; Schmidt, DB; Webb, EF1
Ames, RS; Brawner, ME; Buckley, PT; Elshourbagy, NA; Feild, JA; Foley, JJ; Giardina, GA; Hay, DW; Luttmann, MA; Nuthulaganti, P; Sarau, HM; Schmidt, DB1
Barré, L; Bennacef, I; Debruyne, D; Dhilly, M; Lasne, MC; Perrio, C; Tymciu, S1
Bissantz, C; Bohnert, C; Hoffmann, T; Malherbe, P; Marcuz, A; Schnider, P1
Griswold, DE; Hay, DW; Martin, LD; Medhurst, AD; Parsons, AA1
Cavagnera, S; Farina, C; Foley, JJ; Giardina, GA; Graziani, D; Grugni, M; Hay, DW; Luttmann, M; Medhurst, AD; Raveglia, LF; Rigolio, R; Sarau, HM; Schmidt, DB; Vecchietti, V1
Angelici, O; Bonanno, G; Carità, F; Clarke, GD; Raiteri, M; Schmid, G; Zaratin, P1
Oh, EJ; Thompson, LP; Weinreich, D1
Anukwu, LU; Canning, BJ; Kajekar, R; Myers, AC; Reynolds, SM1
Goldie, RG; Hay, DW; Myers, AC1
Adolfsson, R; Ahlstedt, I; de Verdier, J; Drmota, T; Engberg, S; Johansson, A; Jussila, R; Kristensson, E; Leffler, A; Lindström, E; Novén, A; Påhlman, I; Sigfridsson, K; Sundqvist, M; von Mentzer, B1
Corboz, MR; Eckel, SP; Rivelli, MA1

Other Studies

12 other study(ies) available for substance p and sb 223412

ArticleYear
Nonpeptide tachykinin receptor antagonists: I. Pharmacological and pharmacokinetic characterization of SB 223412, a novel, potent and selective neurokinin-3 receptor antagonist.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 281, Issue:3

    Topics: Animals; Calcium; CHO Cells; Cricetinae; Dogs; Humans; Mice; Piperidines; Quinolines; Rabbits; Radioligand Assay; Rats; Receptors, Neurokinin-3; Receptors, Tachykinin

1997
Molecular and pharmacological characterization of the murine tachykinin NK(3) receptor.
    European journal of pharmacology, 2001, Feb-16, Volume: 413, Issue:2-3

    Topics: Amino Acid Sequence; Animals; Calcium; Cloning, Molecular; Humans; Mice; Molecular Sequence Data; Neurokinin A; Quinolines; Receptors, Neurokinin-3

2001
Synthesis and biological evaluation of novel fluoro and iodo quinoline carboxamides as potential ligands of NK-3 receptors for in vivo imaging studies.
    Bioorganic & medicinal chemistry, 2004, Aug-15, Volume: 12, Issue:16

    Topics: Fluorine; Iodine; Ligands; Positron-Emission Tomography; Quinolines; Receptors, Neurokinin-3; Tomography, Emission-Computed, Single-Photon

2004
Identification of a crucial amino acid in the helix position 6.51 of human tachykinin neurokinin 1 and 3 receptors contributing to the insurmountable mode of antagonism by dual NK₁/NK₃ antagonists.
    Journal of medicinal chemistry, 2012, Jun-14, Volume: 55, Issue:11

    Topics: Amino Acids; Aminopyridines; Benzeneacetamides; HEK293 Cells; Humans; Inositol Phosphates; Models, Molecular; Mutagenesis, Site-Directed; Mutation; Neurokinin-1 Receptor Antagonists; Protein Structure, Secondary; Radioligand Assay; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Stereoisomerism

2012
In vitro and in vivo characterization of NK3 receptors in the rabbit eye by use of selective non-peptide NK3 receptor antagonists.
    British journal of pharmacology, 1997, Volume: 122, Issue:3

    Topics: Animals; In Vitro Techniques; Iris; Male; Miosis; Muscle Contraction; Muscle, Smooth; Neurokinin B; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Quinolines; Rabbits; Receptors, Neurokinin-3; Substance P

1997
Discovery of a novel class of selective non-peptide antagonists for the human neurokinin-3 receptor. 2. Identification of (S)-N-(1-phenylpropyl)-3-hydroxy-2-phenylquinoline-4-carboxamide (SB 223412).
    Journal of medicinal chemistry, 1999, Mar-25, Volume: 42, Issue:6

    Topics: Animals; Calcium; Cell Line; CHO Cells; Cloning, Molecular; Cricetinae; Humans; In Vitro Techniques; Iris; Mice; Miosis; Motor Activity; Muscle Contraction; Muscle, Smooth; Peptide Fragments; Quinolines; Rabbits; Radioligand Assay; Receptors, Neurokinin-3; Structure-Activity Relationship; Substance P

1999
NK3 receptor blockade prevents hyperalgesia and the associated spinal cord substance P release in monoarthritic rats.
    Neuropharmacology, 2000, Volume: 39, Issue:1

    Topics: Afferent Pathways; Animals; Arthritis, Experimental; Freund's Adjuvant; Hyperalgesia; Inflammation; Male; Pain; Peptide Fragments; Quinolines; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, Neurokinin-3; Spinal Cord; Substance P

2000
Sexually dimorphic regulation of NK-1 receptor-mediated electrophysiological responses in vagal primary afferent neurons.
    Journal of neurophysiology, 2000, Volume: 84, Issue:1

    Topics: Animals; Benzamides; Electrophysiology; Estradiol; Female; Gonadal Steroid Hormones; Guinea Pigs; Male; Membrane Potentials; Neurons, Afferent; Nodose Ganglion; Orchiectomy; Ovariectomy; Piperidines; Pregnancy; Quinolines; Receptors, Neurokinin-1; Serotonin; Sex Characteristics; Substance P; Testosterone

2000
Endogenous neurokinins facilitate synaptic transmission in guinea pig airway parasympathetic ganglia.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2002, Volume: 283, Issue:2

    Topics: Animals; Bronchi; Bronchoconstriction; Electric Stimulation; Excitatory Postsynaptic Potentials; Ganglia, Parasympathetic; Guinea Pigs; Immunohistochemistry; In Vitro Techniques; Male; Neurons; Peptide Fragments; Piperidines; Quinolines; Receptors, Neurokinin-3; Substance P; Synaptic Transmission; Trachea; Vagotomy; Vagus Nerve

2002
A novel role for tachykinin neurokinin-3 receptors in regulation of human bronchial Ganglia neurons.
    American journal of respiratory and critical care medicine, 2005, Feb-01, Volume: 171, Issue:3

    Topics: Acetates; Adult; Bronchi; Capsaicin; Electric Stimulation; Evoked Potentials; Female; Ganglia, Parasympathetic; Humans; Male; Microscopy, Confocal; Middle Aged; Nerve Fibers; Neurons, Afferent; Peptide Fragments; Quinolines; Receptors, Neurokinin-3; Substance P; Synaptic Transmission

2005
Senktide-induced gerbil foot tapping behaviour is blocked by selective tachykinin NK1 and NK3 receptor antagonists.
    European journal of pharmacology, 2007, Dec-22, Volume: 577, Issue:1-3

    Topics: Animals; Autoradiography; Behavior, Animal; Brain; Calcium; CHO Cells; Cloning, Molecular; Cricetinae; Cricetulus; Dose-Response Relationship, Drug; Foot; Gerbillinae; Injections, Intraventricular; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Quinolines; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P

2007
Bronchoconstrictor effect of the tachykinin NK₃-receptor agonists [MePhe⁷]-neurokinin B and senktide in the isolated guinea pig lung.
    Experimental lung research, 2010, Volume: 36, Issue:9

    Topics: Animals; Bronchoconstriction; Bronchoconstrictor Agents; CHO Cells; Cricetinae; Cricetulus; Disease Models, Animal; Guinea Pigs; In Vitro Techniques; Lung; Male; Peptide Fragments; Piperidines; Quinolines; Receptors, Neurokinin-3; Substance P

2010