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substance p, sar(9)-met(o2)(11)- and selegiline

substance p, sar(9)-met(o2)(11)- has been researched along with selegiline in 1 studies

Compound Research Comparison

Studies
(substance p, sar(9)-met(o2)(11)-)
Trials
(substance p, sar(9)-met(o2)(11)-)
Recent Studies (post-2010)
(substance p, sar(9)-met(o2)(11)-)
Studies
(selegiline)
Trials
(selegiline)
Recent Studies (post-2010) (selegiline)
151062,575319394

Protein Interaction Comparison

ProteinTaxonomysubstance p, sar(9)-met(o2)(11)- (IC50)selegiline (IC50)
CholinesteraseHomo sapiens (human)0.0055
Cytochrome P450 3A4Homo sapiens (human)0.0039
Alpha-2A adrenergic receptorHomo sapiens (human)1.798
Alpha-2B adrenergic receptorHomo sapiens (human)0.376
Amine oxidase [flavin-containing] BRattus norvegicus (Norway rat)0.2127
Amine oxidase [flavin-containing] A Rattus norvegicus (Norway rat)0.9046
Amine oxidase [flavin-containing] AHomo sapiens (human)1.4408
Adenosine receptor A1Rattus norvegicus (Norway rat)0.0067
Amine oxidase [flavin-containing] BHomo sapiens (human)0.1001
Type-1 angiotensin II receptorSus scrofa (pig)0.048
Alpha-synucleinHomo sapiens (human)0.27
Amine oxidase [flavin-containing] BBos taurus (cattle)1
Sigma intracellular receptor 2Rattus norvegicus (Norway rat)0.017

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hayashi, S; Kato, A; Mizuno, K; Morita, A; Nakata, E; Ohashi, K; Yamamura, K1

Other Studies

1 other study(ies) available for substance p, sar(9)-met(o2)(11)- and selegiline

ArticleYear
Discovery of {1-[4-(2-{hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin-1-yl]cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: de
    Bioorganic & medicinal chemistry, 2010, Nov-01, Volume: 18, Issue:21

    Topics: Analgesics; Animals; Benzimidazoles; Drug Design; Drug Evaluation, Preclinical; Humans; Microsomes, Liver; Neuralgia; Nociceptin Receptor; Pyrroles; Rats; Receptors, Opioid; Structure-Activity Relationship

2010