Page last updated: 2024-09-05

substance p, sar(9)-met(o2)(11)- and neurokinin a

substance p, sar(9)-met(o2)(11)- has been researched along with neurokinin a in 59 studies

Compound Research Comparison

Studies
(substance p, sar(9)-met(o2)(11)-)
Trials
(substance p, sar(9)-met(o2)(11)-)
Recent Studies (post-2010)
(substance p, sar(9)-met(o2)(11)-)
Studies
(neurokinin a)
Trials
(neurokinin a)
Recent Studies (post-2010) (neurokinin a)
151061,7653491

Protein Interaction Comparison

ProteinTaxonomysubstance p, sar(9)-met(o2)(11)- (IC50)neurokinin a (IC50)
Substance-K receptorHomo sapiens (human)0.0017
Neuromedin-K receptorHomo sapiens (human)0.045
Substance-K receptorMesocricetus auratus (golden hamster)0.001

Research

Studies (59)

TimeframeStudies, this research(%)All Research%
pre-19901 (1.69)18.7374
1990's45 (76.27)18.2507
2000's13 (22.03)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chrétien, L; Guillemette, G; Regoli, D; Tousignant, C1
Dam, TV; Martinelli, B; Quirion, R1
Kodner, A; Mayer, EA; Regoli, M; Sachs, G; Sun, XP; Supplisson, S1
Constantine, JW; Lebel, WS; Woody, HA1
Couture, R; Drapeau, G; Guimond, C; Laneuville, O; Regoli, D1
Beaujouan, JC; Glowinski, J; Saffroy, M; Torrens, Y1
Ciccocioppo, R; De Caro, G; Massi, M; Panocka, I; Pompei, P1
Besson, G; Drazen, JM; Israel, E; Lilly, CM; Rodger, IW1
Bristow, LJ; Young, L1
Banasiak, D; Burcher, E1
Barnes, PJ; Belvisi, MG; Maggi, CA; Patacchini, R1
Maggi, CA; Santicioli, P; Zagorodnyuk, V1
Giachetti, A; Giuliani, S; Maggi, CA; Meini, S; Patacchini, R; Potier, E; Quartara, L; Sisto, A1
Hill, RG; Longmore, J; Razzaque, Z; Shaw, D1
Daniel, EE; Fox-Threlkeld, JE; Watson, EG1
Betschart, J; Blanchard, JC; Fardin, V; Flamand, O; Ravard, S1
Brugger, F; Evans, RH; Lepre, M; Olpe, HR1
Coge, F; Regoli, D1
Jackson, A; Rupniak, NM1
Ballati, L; Boni, P; Evangelista, S1
Killingsworth, CR; Shore, SA1
Giachetti, A; Maggi, CA; Santicioli, P; Zagorodnyuk, V1
Mak, JC; Meini, S; Rogers, DF; Rohde, JA1
Alberch, J; Arenas, E; Marsal, J; Pérez-Navarro, E1
Barnes, PJ; Hirayama, Y; Lei, YH; Rogers, DF1
Boucher, S; Couture, R; Gitter, BD; Howbert, JJ; Picard, P; Regoli, D1
Boden, PR; Norris, SK; Woodruff, GN1
Håkanson, R; Wang, ZY1
Dalforno, G; Gaviraghi, G; Hagan, RM; Palea, S; Pietra, C; Trist, DG1
Giachetti, A; Giuliani, S; Maggi, CA; Patacchini, R1
Chahl, LA; Johnston, PA1
Bartho, L; Giuliani, S; Maggi, CA; Santicioli, P1
Bertrand, C; Geppetti, P; Graf, PD; Nadel, JA1
Champion, E; Foulon, DM; Jones, TR; Masson, P; Rodger, IW1
Humpel, C; Saria, A1
McKee, KT; Metters, KM; Millar, L; Rodger, IW1
Betschart, J; Blanchard, JC; Garret, C; Grall, I; Piot, O; Ravard, S1
Fox, AJ; Naeem, S; Patel, IA; Urbán, L; Walpole, C1
Bai, T; Knight, D; McKay, K; Schellenberg, RR; Wiggs, B1
Giuliani, S; Lecci, A; Maggi, CA; Tramontana, M1
Brelière, JC; Emonds-Alt, X; Le Fur, G; Vilain, P1
Kondo, A; Ohmura, M; Saito, M1
Evangelista, S; Giachetti, A; Manzini, S; Paoli, S1
Bordin, G; Brunelleschi, S; Colangelo, D; Viano, I1
Ardell, JL; Armour, JA; Hoover, DB; Thompson, GW1
Bianchi, B; Cappugi, P; Danesi, A; Giannotti, B; Ipponi, P; Johansson, O; Matucci, R; Rossi, R1
Lee, K; Pinnock, RD; Preston, Z; Richardson, PJ; Widdowson, L1
Albera, C; Brunelleschi, S; Gagliardi, L; Ghio, P; Lavagno, L; Nicali, R; Pozzi, E; Viano, I1
Crane, LH; Hamlin, GP; Nimmo, AJ; Williams, MJ1
Coupar, IM; Kerr, KP; Thai, B1
Bayguinov, O; Hagen, B; Sanders, KM1
Burcher, E; Holmgren, S; Johansson, A; Liu, L1
Couture, R; Deschamps, K1
Juszczak, M1
Amato, A; Mulè, F; Serio, R1
Boczek-Leszczyk, E; Juszczak, M; Stempniak, B1
Emala, CW; Gallos, G; Goubaeva, F; Mizuta, F; Mizuta, K; Panettieri, RA; Xu, D; Yang, J; Zhu, D1
Bongianni, F; Cinelli, E; Mutolo, D; Pantaleo, T1
Boczek-Leszczyk, E; Juszczak, M1

Other Studies

59 other study(ies) available for substance p, sar(9)-met(o2)(11)- and neurokinin a

ArticleYear
Characterization of NK-1 receptors in guinea pig and rat brain membranes with NK-1 peptides and a non-peptide antagonist.
    Brain research, 1992, Nov-20, Volume: 596, Issue:1-2

    Topics: Amino Acid Sequence; Animals; Biphenyl Compounds; Brain; Guinea Pigs; Membranes; Molecular Sequence Data; Neurokinin A; Neurokinin B; Rats; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Substance P

1992
Autoradiographic distribution of brain neurokinin-1/substance P receptors using a highly selective ligand [3H]-[Sar9,Met(O2)11]-substance P.
    Brain research, 1990, Oct-29, Volume: 531, Issue:1-2

    Topics: Animals; Autoradiography; Brain; Indicators and Reagents; Iodine Radioisotopes; Male; Neurokinin A; Organ Specificity; Rats; Rats, Inbred Strains; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Substance P; Succinimides; Tritium

1990
Neurokinin receptor-mediated regulation of [Ca]i and Ca-sensitive ion channels in mammalian colonic muscle.
    Annals of the New York Academy of Sciences, 1991, Volume: 632

    Topics: Animals; Calcimycin; Calcium; Calcium Channels; Cells, Cultured; Colon; Membrane Potentials; Muscle, Smooth; Neurokinin A; Peptide Fragments; Rabbits; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P

1991
Inhibition of tachykinin-induced hypotension in dogs by CP-96,345, a selective blocker of NK-1 receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1991, Volume: 344, Issue:4

    Topics: Animals; Biphenyl Compounds; Blood Pressure; Decerebrate State; Dogs; Dose-Response Relationship, Drug; Female; Heart Rate; In Vitro Techniques; Isoproterenol; Male; Neurokinin A; Peptide Fragments; Receptors, Neurotransmitter; Receptors, Tachykinin; Stereoisomerism; Substance P; Tachykinins

1991
Characterization of the peripheral action of neurokinins and neurokinin receptor selective agonists on the rat cardiovascular system.
    Naunyn-Schmiedeberg's archives of pharmacology, 1989, Volume: 340, Issue:5

    Topics: Animals; Cardiovascular System; Female; Injections, Intravenous; Male; Neurokinin A; Neurokinin B; Neurons, Afferent; Parasympathetic Nervous System; Peptide Fragments; Prostaglandins; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Substance P; Sympathetic Nervous System; Tachycardia

1989
Involvement of septide-sensitive tachykinin receptors in inositol phospholipid hydrolysis in the rat urinary bladder.
    Peptides, 1995, Volume: 16, Issue:4

    Topics: Amino Acid Sequence; Animals; Benzamides; Hydrolysis; Indoles; Isoindoles; Male; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth; Neurokinin A; Peptide Fragments; Phosphatidylinositols; Piperidines; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Tachykinin; Substance P; Urinary Bladder

1995
Selective agonists at NK3 tachykinin receptors inhibit alcohol intake in Sardinian alcohol-preferring rats.
    Brain research bulletin, 1994, Volume: 33, Issue:1

    Topics: Alcohol Drinking; Amino Acid Sequence; Animals; Drinking Behavior; Eating; Injections, Intraventricular; Male; Molecular Sequence Data; Neurokinin A; Peptide Fragments; Rats; Rats, Wistar; Receptors, Neurokinin-3; Substance P; Water Deprivation

1994
Capsaicin-induced airway obstruction in tracheally perfused guinea pig lungs.
    American journal of respiratory and critical care medicine, 1994, Volume: 149, Issue:5

    Topics: Animals; Benzamides; Bronchoconstriction; Capsaicin; Dose-Response Relationship, Drug; Guinea Pigs; In Vitro Techniques; Male; Methacholine Chloride; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Perfusion; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Trachea

1994
Chromodacryorrhea and repetitive hind paw tapping: models of peripheral and central tachykinin NK1 receptor activation in gerbils.
    European journal of pharmacology, 1994, Mar-03, Volume: 253, Issue:3

    Topics: Animals; Behavior, Animal; Dose-Response Relationship, Drug; Drug Synergism; Gerbillinae; Harderian Gland; Indoles; Injections, Intravenous; Injections, Intraventricular; Isoindoles; Male; Neurokinin A; Peptide Fragments; Piperidines; Receptors, Neurokinin-1; Substance P

1994
Effect of capsaicin on distribution of binding sites for tachykinins and calcitonin gene-related peptide in rat urinary bladder: a quantitative autoradiographic study.
    Peptides, 1994, Volume: 15, Issue:2

    Topics: Animals; Autoradiography; Calcitonin Gene-Related Peptide; Capsaicin; Male; Neurokinin A; Protein Binding; Rats; Rats, Wistar; Receptors, Calcitonin Gene-Related Peptide; Receptors, Tachykinin; Substance P; Tissue Distribution; Urinary Bladder

1994
Facilitatory effects of selective agonists for tachykinin receptors on cholinergic neurotransmission: evidence for species differences.
    British journal of pharmacology, 1994, Volume: 111, Issue:1

    Topics: Adult; Amino Acid Sequence; Animals; Bronchi; Capsaicin; Electric Stimulation; Guinea Pigs; Humans; In Vitro Techniques; Male; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth; Neurokinin A; Parasympathetic Nervous System; Peptide Fragments; Rabbits; Receptors, Tachykinin; Substance P; Sulfones; Synaptic Transmission; Tachykinins

1994
Different Ca2+ influx pathways mediate tachykinin receptor-induced contraction in circular muscle of guinea-pig colon.
    European journal of pharmacology, 1994, Apr-01, Volume: 255, Issue:1-3

    Topics: Action Potentials; Animals; Calcium Channels; Colon; Electrophysiology; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin-1 Receptor Antagonists; Nifedipine; Peptide Fragments; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Tachykinin; Substance P; Sulfones

1994
Comparison of tachykinin NK1 and NK2 receptors in the circular muscle of the guinea-pig ileum and proximal colon.
    British journal of pharmacology, 1994, Volume: 112, Issue:1

    Topics: Animals; Colon; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin-1 Receptor Antagonists; Nifedipine; Peptide Fragments; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Sulfones

1994
Differences in the effects of NK1-receptor antagonists, (+/-)-CP 96,345 and CP 99,994, on agonist-induced responses in guinea-pig trachea.
    British journal of pharmacology, 1994, Volume: 112, Issue:1

    Topics: Animals; Biphenyl Compounds; Guinea Pigs; In Vitro Techniques; Indoles; Isoindoles; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Substance P; Trachea

1994
Tachykinin-mediated increase in motility acts independently of vasoactive intestinal polypeptide release in the canine ileum.
    Canadian journal of physiology and pharmacology, 1994, Volume: 72, Issue:2

    Topics: Animals; Dogs; Female; Gastrointestinal Motility; Ileum; Male; Neurokinin A; Peptide Fragments; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Vasoactive Intestinal Peptide

1994
Differential ability of tachykinin NK-1 and NK-2 agonists to produce scratching and grooming behaviours in mice.
    Brain research, 1994, Jul-18, Volume: 651, Issue:1-2

    Topics: Animals; Behavior, Animal; Brain; Grooming; Male; Mice; Neurokinin A; Peptide Fragments; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P

1994
Physiological and pharmacological characterization of the spinal tachykinin NK2 receptor.
    European journal of pharmacology, 1994, Jun-02, Volume: 258, Issue:1-2

    Topics: Animals; Animals, Newborn; Biphenyl Compounds; Dose-Response Relationship, Drug; Drug Interactions; Ganglia, Spinal; Gerbillinae; Hypnotics and Sedatives; In Vitro Techniques; Indoles; Isoindoles; Neurokinin A; Oligopeptides; Peptide Fragments; Rats; Receptors, Neurokinin-2; Spinal Cord; Substance P; Tetrodotoxin

1994
NK1 and NK2 receptors are similar in man and rabbit.
    Neuropeptides, 1994, Volume: 26, Issue:6

    Topics: Animals; Binding, Competitive; CHO Cells; Cricetinae; Humans; Iodine Radioisotopes; Kinetics; Muscle, Smooth, Vascular; Neurokinin A; Pulmonary Artery; Rabbits; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Recombinant Proteins; Substance P; Transfection; Tritium; Venae Cavae

1994
Non-specific inhibition of dopamine receptor agonist-induced behaviour by the tachykinin NK1 receptor antagonist CP-99,994 in guinea-pigs.
    European journal of pharmacology, 1994, Sep-01, Volume: 262, Issue:1-2

    Topics: Amphetamine; Analysis of Variance; Animals; Behavior, Animal; Dopamine Agonists; Grooming; Guinea Pigs; Haloperidol; Injections, Intraperitoneal; Injections, Subcutaneous; Male; Motor Activity; Neurokinin A; Neurokinin-1 Receptor Antagonists; Oxazines; Piperidines; Receptors, Neurokinin-1; Stereoisomerism; Substance P

1994
Tachykinin NK1 and NK2 receptors mediate the non-cholinergic bronchospastic response to capsaicin and vagal stimulation in guinea-pigs.
    Journal of autonomic pharmacology, 1995, Volume: 15, Issue:1

    Topics: Animals; Biphenyl Compounds; Bronchial Spasm; Capsaicin; Electric Stimulation; Guinea Pigs; Insufflation; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Peptides, Cyclic; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Vagus Nerve

1995
Tachykinin receptors mediating contraction of guinea pig lung strips.
    Regulatory peptides, 1995, May-30, Volume: 57, Issue:2

    Topics: Acetylcholine; Animals; Benzamides; Biphenyl Compounds; Dipeptides; Guinea Pigs; In Vitro Techniques; Lung; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin B; Peptide Fragments; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Tachykinin; Substance P; Trachea

1995
Evidence that tachykinin NK1 and NK2 receptors mediate non-adrenergic non-cholinergic excitation and contraction in the circular muscle of guinea-pig duodenum.
    British journal of pharmacology, 1995, Volume: 115, Issue:2

    Topics: Action Potentials; Adenosine Diphosphate; Animals; Apamin; Arginine; Atropine; Dose-Response Relationship, Drug; Duodenum; Electric Stimulation; Guanethidine; Guinea Pigs; Indomethacin; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin-1 Receptor Antagonists; Neuromuscular Junction; Nifedipine; Nitroarginine; Oligopeptides; Peptide Fragments; Peptides, Cyclic; Physalaemin; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Suramin; Thionucleotides

1995
Tachykinin control of ferret airways: mucus secretion, bronchoconstriction and receptor mapping.
    Neuropeptides, 1993, Volume: 24, Issue:2

    Topics: Animals; Bronchoconstriction; Capsaicin; Ferrets; Male; Methacholine Chloride; Mucus; Muscle, Smooth; Neurokinin A; Neurokinin B; Peptide Fragments; Receptors, Neurotransmitter; Receptors, Tachykinin; Reproducibility of Results; Stimulation, Chemical; Substance P; Tachykinins; Trachea

1993
Selective resistance of tachykinin-responsive cholinergic neurons in the quinolinic acid lesioned neostriatum.
    Brain research, 1993, Feb-19, Volume: 603, Issue:2

    Topics: Acetylcholine; Animals; Dose-Response Relationship, Drug; Glutamates; Glutamic Acid; In Vitro Techniques; Male; Microinjections; Neostriatum; Neurokinin A; Neurons; Peptide Fragments; Potassium Chloride; Quinolinic Acid; Rats; Rats, Sprague-Dawley; Substance P

1993
Effects of two novel tachykinin antagonists, FK224 and FK888, on neurogenic airway plasma exudation, bronchoconstriction and systemic hypotension in guinea-pigs in vivo.
    British journal of pharmacology, 1993, Volume: 108, Issue:3

    Topics: Animals; Blood Pressure; Bronchoconstriction; Capsaicin; Dipeptides; Electric Stimulation; Evans Blue; Exudates and Transudates; Guinea Pigs; Hypotension; Indoles; Male; Neurokinin A; Peptide Fragments; Peptides, Cyclic; Platelet Activating Factor; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Respiratory Mechanics; Smoking; Substance P; Vagus Nerve

1993
Use of non-peptide tachykinin receptor antagonists to substantiate the involvement of NK1 and NK2 receptors in a spinal nociceptive reflex in the rat.
    European journal of pharmacology, 1993, Mar-02, Volume: 232, Issue:2-3

    Topics: Animals; Benzamides; Biphenyl Compounds; Hypnotics and Sedatives; Injections, Spinal; Male; Neurokinin A; Nociceptors; Pain Measurement; Pain Threshold; Peptide Fragments; Piperidines; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Receptors, Tachykinin; Reflex; Spinal Cord; Substance P

1993
Agonists selective for tachykinin NK1 and NK3 receptors excite subpopulations of neurons in the rat medial habenula nucleus in vitro.
    European journal of pharmacology, 1993, Apr-06, Volume: 234, Issue:2-3

    Topics: Animals; Electrophysiology; Extracellular Space; In Vitro Techniques; Male; Neurokinin A; Neurons; Peptide Fragments; Rats; Rats, Wistar; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Substance P; Tachykinins; Thalamic Nuclei

1993
The rabbit iris sphincter contains NK1 and NK3 but not NK2 receptors: a study with selective agonists and antagonists.
    Regulatory peptides, 1993, Apr-08, Volume: 44, Issue:3

    Topics: Animals; Dactinomycin; Female; Iris; Kinetics; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin B; Peptide Fragments; Rabbits; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P

1993
Further studies on the effects of selective neurokinin agonists upon the activation of micturition reflex in rats. Evidence for a dual NK-1 receptor mediated excitatory and inhibitory activity.
    Neuropeptides, 1993, Volume: 24, Issue:5

    Topics: Animals; Dose-Response Relationship, Drug; Injections, Intra-Arterial; Injections, Intraventricular; Male; Neurokinin A; Peptide Fragments; Physalaemin; Rats; Rats, Wistar; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Reflex; Substance P; Urinary Bladder; Urination

1993
In vivo and in vitro activity of SR 48,968, a non-peptide tachykinin NK-2 receptor antagonist.
    Regulatory peptides, 1993, Jul-02, Volume: 46, Issue:1-2

    Topics: Animals; Benzamides; Biphenyl Compounds; Blood Pressure; Muscle Contraction; Muscle, Smooth; Neurokinin A; Peptide Fragments; Piperidines; Rats; Receptors, Neurokinin-2; Saliva; Substance P; Sulfones; Urinary Bladder

1993
Neurokinin-1, -2 and -3 receptors are candidates for a role in the opiate withdrawal response in guinea-pigs.
    Regulatory peptides, 1993, Jul-02, Volume: 46, Issue:1-2

    Topics: Animals; Cerebral Ventricles; Guinea Pigs; Injections, Intraventricular; Motor Activity; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Substance Withdrawal Syndrome

1993
Tachykinin NK-1 and NK-2 receptors in the circular muscle of the guinea-pig proximal colon.
    Regulatory peptides, 1993, Jul-02, Volume: 46, Issue:1-2

    Topics: Animals; Benzamides; Biphenyl Compounds; Colon; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Peptides, Cyclic; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Sulfones; Tetrodotoxin

1993
Capsaicin increases airflow resistance in guinea pigs in vivo by activating both NK2 and NK1 tachykinin receptors.
    The American review of respiratory disease, 1993, Volume: 148, Issue:4 Pt 1

    Topics: Airway Resistance; Animals; Atropine; Benzamides; Biphenyl Compounds; Capsaicin; Dose-Response Relationship, Drug; Drug Interactions; Guinea Pigs; Histamine; Male; Neurokinin A; Peptide Fragments; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P

1993
NK1 and NK2 receptors mediate tachykinin and resiniferatoxin-induced bronchospasm in guinea pigs.
    The American review of respiratory disease, 1993, Volume: 148, Issue:4 Pt 1

    Topics: Animals; Benzamides; Bronchial Spasm; Bronchoconstriction; Diterpenes; Dose-Response Relationship, Drug; Drug Interactions; Guinea Pigs; Male; Neurokinin A; Peptide Fragments; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Tachykinins

1993
Intranigral injection of selective neurokinin-1 and neurokinin-3 but not neurokinin-2 receptor agonists biphasically modulate striatal dopamine metabolism but not striatal preprotachykinin-A mRNA in the rat.
    Neuroscience letters, 1993, Jul-23, Volume: 157, Issue:2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Corpus Striatum; Dopamine; Female; Gene Expression Regulation; Injections; Neurokinin A; Neurokinin B; Peptide Fragments; Protein Precursors; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; RNA, Messenger; Substance P; Substantia Nigra; Tachykinins

1993
Identification of both NK1 and NK2 receptors in guinea-pig airways.
    British journal of pharmacology, 1993, Volume: 110, Issue:2

    Topics: Animals; Benzamides; Chromatography, High Pressure Liquid; Guinea Pigs; In Vitro Techniques; Iodine Radioisotopes; Lung; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Radioligand Assay; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Respiratory System; Substance P; Trachea

1993
Comparative behavioural profile of centrally administered tachykinin NK1, NK2 and NK3 receptor agonists in the guinea-pig.
    British journal of pharmacology, 1995, Volume: 116, Issue:5

    Topics: Animals; Behavior, Animal; Guinea Pigs; Injections, Intraventricular; Male; Motor Activity; Neurokinin A; Peptide Fragments; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P

1995
Receptors mediating tachykinin-evoked depolarisations of neurons in the neonatal rat spinal cord.
    Acta biologica Hungarica, 1996, Volume: 47, Issue:1-4

    Topics: Animals; Animals, Newborn; Biphenyl Compounds; Evoked Potentials; In Vitro Techniques; Indoles; Isoindoles; Neurokinin A; Neurokinin-1 Receptor Antagonists; Neurons; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Spinal Cord; Substance P; Tachykinins

1996
Localization of leukaemia inhibitory factor to airway epithelium and its amplification of contractile responses to tachykinins.
    British journal of pharmacology, 1997, Volume: 120, Issue:5

    Topics: Animals; Capsaicin; Carbachol; Epithelium; Female; Growth Inhibitors; Guinea Pigs; Humans; Immunohistochemistry; In Vitro Techniques; Interleukin-6; Isoproterenol; Leukemia Inhibitory Factor; Lymphokines; Muscle Contraction; Neurokinin A; Substance P; Trachea

1997
Role of tachykinin NK1 and NK2 receptors on colonic motility in anesthetized rats: effect of agonists.
    Canadian journal of physiology and pharmacology, 1997, Volume: 75, Issue:6

    Topics: Anesthesia; Animals; Benzamides; Colon; Gastrointestinal Motility; Male; Neurokinin A; Peptide Fragments; Peptides, Cyclic; Piperidines; Quinuclidines; Rats; Rats, Wistar; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P

1997
Tachykinin-induced contractions of the guinea pig ileum longitudinal smooth muscle: tonic and phasic muscular activities.
    Canadian journal of physiology and pharmacology, 1997, Volume: 75, Issue:6

    Topics: Animals; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Peptide Fragments; Substance P; Tachykinins

1997
Response of isolated human neurogenic bladders to tachykinins.
    Urologia internationalis, 1997, Volume: 59, Issue:4

    Topics: Adolescent; Atropine; Child; Dose-Response Relationship, Drug; Electric Stimulation; Female; Humans; In Vitro Techniques; Male; Meningomyelocele; Muscle Contraction; Neurokinin A; Neurokinin B; Sacrococcygeal Region; Substance P; Tachykinins; Urinary Bladder, Neurogenic

1997
Involvement of tachykinin NK1 receptors in plasma protein extravasation induced by tachykinins in the guinea pig upper airways.
    Neuropeptides, 1997, Volume: 31, Issue:1

    Topics: Animals; Antigens; Blood Proteins; Capsaicin; Dextrans; Dipeptides; Extravasation of Diagnostic and Therapeutic Materials; Fluorescein-5-isothiocyanate; Glycopeptides; Guinea Pigs; Indoles; Male; Nasal Mucosa; Neurokinin A; Neurokinin-1 Receptor Antagonists; Olfactory Receptor Neurons; Peptide Fragments; Peptides, Cyclic; Protease Inhibitors; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Rhinitis; Substance P

1997
Tachykinin receptors are present on human monocytes and play a role in rheumatoid arthritis.
    Journal of chemotherapy (Florence, Italy), 1998, Volume: 10, Issue:2

    Topics: Aged; Arthritis, Rheumatoid; Cell Separation; Female; Humans; Male; Middle Aged; Monocytes; N-Formylmethionine Leucyl-Phenylalanine; Neurokinin A; Neurokinin B; Peptide Fragments; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Superoxides; Tetradecanoylphorbol Acetate

1998
Canine intrinsic cardiac neurons involved in cardiac regulation possess NK1, NK2, and NK3 receptors.
    The American journal of physiology, 1998, Volume: 275, Issue:5

    Topics: Animals; Dogs; Heart; Myocardial Contraction; Neurokinin A; Neurons, Afferent; Peptide Fragments; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P

1998
Characterization of [3H]substance P binding sites in human skin.
    Journal of the European Academy of Dermatology and Venereology : JEADV, 1999, Volume: 12, Issue:1

    Topics: Aged; Binding, Competitive; Female; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Male; Middle Aged; Neurokinin A; Neurokinin B; Peptide Fragments; Radioligand Assay; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Skin; Substance P; Tritium

1999
Tachykinins increase [3H]acetylcholine release in mouse striatum through multiple receptor subtypes.
    Neuroscience, 2000, Volume: 95, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Acetylcholine; Alkaloids; Animals; Benzophenanthridines; Choline O-Acetyltransferase; Corpus Striatum; Electrophysiology; Enzyme Inhibitors; Estrenes; Excitatory Amino Acid Antagonists; In Situ Hybridization; Indoles; Interneurons; Membrane Potentials; Mice; Mice, Inbred C57BL; Neurokinin A; Oligopeptides; omega-N-Methylarginine; Peptide Fragments; Phenanthridines; Phosphodiesterase Inhibitors; Piperidines; Pyrrolidinones; Quinoxalines; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; RNA, Messenger; Signal Transduction; Substance P; Tachykinins; Tetrodotoxin; Tritium

2000
Tachykinin activation of human monocytes from patients with interstitial lung disease, healthy smokers or healthy volunteers.
    Neuropeptides, 2000, Volume: 34, Issue:1

    Topics: Adult; Aged; Cells, Cultured; Female; Humans; Lung Diseases, Interstitial; Male; Middle Aged; Monocytes; Neurokinin A; Peptide Fragments; Pulmonary Fibrosis; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Reference Values; Sarcoidosis; Smoking; Substance P; Superoxides; Tachykinins

2000
Hormonal variation of rat uterine contractile responsiveness to selective neurokinin receptor agonists.
    Biology of reproduction, 2000, Volume: 62, Issue:6

    Topics: Animals; Diestrus; Estrogens; Estrus; Female; Metestrus; Neurokinin A; Ovariectomy; Peptide Fragments; Piperidines; Proestrus; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Uterine Contraction

2000
Tachykinin-induced contraction of the guinea-pig isolated oesophageal mucosa is mediated by NK(2) receptors.
    British journal of pharmacology, 2000, Volume: 131, Issue:7

    Topics: Animals; Benzamides; Captopril; Dose-Response Relationship, Drug; Esophagus; Guinea Pigs; In Vitro Techniques; Mucous Membrane; Muscle Contraction; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Protease Inhibitors; Quinolines; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Tachykinins; Thiorphan

2000
Substance P modulates localized calcium transients and membrane current responses in murine colonic myocytes.
    British journal of pharmacology, 2003, Volume: 138, Issue:7

    Topics: Animals; Calcium Signaling; Colon; Electric Conductivity; Imidazoles; Indoles; Male; Maleimides; Membrane Potentials; Mice; Mice, Inbred BALB C; Microscopy, Confocal; Myocytes, Smooth Muscle; Neurokinin A; Nicardipine; Patch-Clamp Techniques; Peptide Fragments; Peptides; Physalaemin; Receptors, Tachykinin; Ryanodine; Ryanodine Receptor Calcium Release Channel; Second Messenger Systems; Substance P

2003
Characterization of receptors for two Xenopus gastrointestinal tachykinin peptides in their species of origin.
    Naunyn-Schmiedeberg's archives of pharmacology, 2004, Volume: 370, Issue:1

    Topics: Animals; Binding Sites; Cardia; Dose-Response Relationship, Drug; Eledoisin; Female; Indoles; Intercellular Signaling Peptides and Proteins; Intestine, Small; Iodine Radioisotopes; Isoindoles; Kassinin; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Peptide Fragments; Physalaemin; Receptors, Tachykinin; Species Specificity; Substance P; Xenopus

2004
The ventral tegmental area as a putative target for tachykinins in cardiovascular regulation.
    British journal of pharmacology, 2005, Volume: 145, Issue:6

    Topics: Acetates; Adrenergic beta-Antagonists; Animals; Atenolol; Behavior, Animal; Benzamides; Benzazepines; Blood Pressure; Dopamine D2 Receptor Antagonists; Glutamic Acid; Heart Rate; Indoles; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Quinolines; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Ventral Tegmental Area

2005
Vasopressin release from the rat hypothalamo-neurohypophysial system: effects of tachykinin NK-1 and NK-2 receptors agonists and antagonists.
    Neuro endocrinology letters, 2005, Volume: 26, Issue:4

    Topics: Animals; Hypothalamo-Hypophyseal System; In Vitro Techniques; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; Neurotransmitter Agents; Peptide Fragments; Rats; Rats, Wistar; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Vasopressins

2005
Role for NK(1) and NK(2) receptors in the motor activity in mouse colon.
    European journal of pharmacology, 2007, Sep-10, Volume: 570, Issue:1-3

    Topics: Animals; Atropine; Colon; Electric Stimulation; Mice; Mice, Inbred C57BL; Muscarinic Antagonists; Muscle Contraction; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Sodium Channel Blockers; Substance P; Tetrodotoxin

2007
Effect of melatonin on the vasopressin secretion as influenced by tachykinin NK-1 receptor agonist and antagonist: in vivo and in vitro studies.
    Journal of physiology and pharmacology : an official journal of the Polish Physiological Society, 2007, Volume: 58, Issue:4

    Topics: Analysis of Variance; Animals; Hypothalamo-Hypophyseal System; In Vitro Techniques; Male; Melatonin; Neurokinin A; Neurokinin-1 Receptor Antagonists; Neurotransmitter Agents; Peptide Fragments; Radioimmunoassay; Rats; Rats, Wistar; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Vasopressins

2007
Expression and coupling of neurokinin receptor subtypes to inositol phosphate and calcium signaling pathways in human airway smooth muscle cells.
    American journal of physiology. Lung cellular and molecular physiology, 2008, Volume: 294, Issue:3

    Topics: Boron Compounds; Calcium Signaling; Humans; Imidazoles; Inositol 1,4,5-Trisphosphate; Muscle, Smooth; Neurokinin A; Peptide Fragments; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; RNA, Messenger; Substance P; Trachea

2008
Neurokinin receptor modulation of respiratory activity in the rabbit.
    The European journal of neuroscience, 2008, Volume: 27, Issue:12

    Topics: Animals; Exhalation; Inhalation; Male; Medulla Oblongata; Microinjections; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Phrenic Nerve; Piperidines; Rabbits; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Substance P; Vagotomy

2008
Oxytocin release from the rat neurohypophysis into the blood: effects of tachykinin NK-1 and NK-2 receptors agonists and antagonists.
    Journal of physiology and pharmacology : an official journal of the Polish Physiological Society, 2008, Volume: 59, Issue:3

    Topics: Analysis of Variance; Animals; Injections, Intraventricular; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; Oxytocin; Peptide Fragments; Pituitary Gland, Posterior; Radioimmunoassay; Rats; Rats, Wistar; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P

2008