Page last updated: 2024-09-05

substance p, sar(9)-met(o2)(11)- and cp 99994

substance p, sar(9)-met(o2)(11)- has been researched along with cp 99994 in 13 studies

Compound Research Comparison

Studies
(substance p, sar(9)-met(o2)(11)-)
Trials
(substance p, sar(9)-met(o2)(11)-)
Recent Studies (post-2010)
(substance p, sar(9)-met(o2)(11)-)
Studies
(cp 99994)
Trials
(cp 99994)
Recent Studies (post-2010) (cp 99994)
15106231219

Protein Interaction Comparison

ProteinTaxonomysubstance p, sar(9)-met(o2)(11)- (IC50)cp 99994 (IC50)
Glutamate receptor 1Rattus norvegicus (Norway rat)0.0006
Glutamate receptor 2Rattus norvegicus (Norway rat)0.0006
Glutamate receptor 3Rattus norvegicus (Norway rat)0.0006
Glutamate receptor 4Rattus norvegicus (Norway rat)0.0006
Substance-P receptorHomo sapiens (human)0.0004

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's11 (84.62)18.2507
2000's2 (15.38)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Besson, G; Drazen, JM; Israel, E; Lilly, CM; Rodger, IW1
Bristow, LJ; Young, L1
Hill, RG; Longmore, J; Razzaque, Z; Shaw, D1
Jackson, A; Rupniak, NM1
Killingsworth, CR; Shore, SA1
Champion, E; Foulon, DM; Jones, TR; Masson, P; Rodger, IW1
McKee, KT; Metters, KM; Millar, L; Rodger, IW1
Chrétien, L; Gobeil, F; Jukic, D; Nguyen, QT; Nguyen-Le, XK; Regoli, D1
Lieberman, DN; Mody, I1
Bornstein, JC; Burcher, E; Johnson, PJ1
Khawaja, AM; Liu, Y; Rogers, DF1
Fong, AY; Potts, JT1
Bongianni, F; Cinelli, E; Mutolo, D; Pantaleo, T1

Other Studies

13 other study(ies) available for substance p, sar(9)-met(o2)(11)- and cp 99994

ArticleYear
Capsaicin-induced airway obstruction in tracheally perfused guinea pig lungs.
    American journal of respiratory and critical care medicine, 1994, Volume: 149, Issue:5

    Topics: Animals; Benzamides; Bronchoconstriction; Capsaicin; Dose-Response Relationship, Drug; Guinea Pigs; In Vitro Techniques; Male; Methacholine Chloride; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Perfusion; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Trachea

1994
Chromodacryorrhea and repetitive hind paw tapping: models of peripheral and central tachykinin NK1 receptor activation in gerbils.
    European journal of pharmacology, 1994, Mar-03, Volume: 253, Issue:3

    Topics: Animals; Behavior, Animal; Dose-Response Relationship, Drug; Drug Synergism; Gerbillinae; Harderian Gland; Indoles; Injections, Intravenous; Injections, Intraventricular; Isoindoles; Male; Neurokinin A; Peptide Fragments; Piperidines; Receptors, Neurokinin-1; Substance P

1994
Differences in the effects of NK1-receptor antagonists, (+/-)-CP 96,345 and CP 99,994, on agonist-induced responses in guinea-pig trachea.
    British journal of pharmacology, 1994, Volume: 112, Issue:1

    Topics: Animals; Biphenyl Compounds; Guinea Pigs; In Vitro Techniques; Indoles; Isoindoles; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Substance P; Trachea

1994
Non-specific inhibition of dopamine receptor agonist-induced behaviour by the tachykinin NK1 receptor antagonist CP-99,994 in guinea-pigs.
    European journal of pharmacology, 1994, Sep-01, Volume: 262, Issue:1-2

    Topics: Amphetamine; Analysis of Variance; Animals; Behavior, Animal; Dopamine Agonists; Grooming; Guinea Pigs; Haloperidol; Injections, Intraperitoneal; Injections, Subcutaneous; Male; Motor Activity; Neurokinin A; Neurokinin-1 Receptor Antagonists; Oxazines; Piperidines; Receptors, Neurokinin-1; Stereoisomerism; Substance P

1994
Tachykinin receptors mediating contraction of guinea pig lung strips.
    Regulatory peptides, 1995, May-30, Volume: 57, Issue:2

    Topics: Acetylcholine; Animals; Benzamides; Biphenyl Compounds; Dipeptides; Guinea Pigs; In Vitro Techniques; Lung; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin B; Peptide Fragments; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Tachykinin; Substance P; Trachea

1995
NK1 and NK2 receptors mediate tachykinin and resiniferatoxin-induced bronchospasm in guinea pigs.
    The American review of respiratory disease, 1993, Volume: 148, Issue:4 Pt 1

    Topics: Animals; Benzamides; Bronchial Spasm; Bronchoconstriction; Diterpenes; Dose-Response Relationship, Drug; Drug Interactions; Guinea Pigs; Male; Neurokinin A; Peptide Fragments; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Tachykinins

1993
Identification of both NK1 and NK2 receptors in guinea-pig airways.
    British journal of pharmacology, 1993, Volume: 110, Issue:2

    Topics: Animals; Benzamides; Chromatography, High Pressure Liquid; Guinea Pigs; In Vitro Techniques; Iodine Radioisotopes; Lung; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Radioligand Assay; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Respiratory System; Substance P; Trachea

1993
Neurokinin receptors in the guinea pig ileum.
    Pharmacology, 1996, Volume: 52, Issue:1

    Topics: Acetylcholine; Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzamides; Biphenyl Compounds; Guinea Pigs; Ileum; Male; Myenteric Plexus; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Radioligand Assay; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Stereoisomerism; Structure-Activity Relationship; Substance P

1996
Substance P enhances NMDA channel function in hippocampal dentate gyrus granule cells.
    Journal of neurophysiology, 1998, Volume: 80, Issue:1

    Topics: Animals; Cells, Cultured; Dentate Gyrus; Ion Channel Gating; Male; Neurokinin-1 Receptor Antagonists; Neurons; Patch-Clamp Techniques; Piperidines; Rats; Rats, Wistar; Reaction Time; Receptors, N-Methyl-D-Aspartate; Receptors, Neurokinin-1; Substance P

1998
Roles of neuronal NK1 and NK3 receptors in synaptic transmission during motility reflexes in the guinea-pig ileum.
    British journal of pharmacology, 1998, Volume: 124, Issue:7

    Topics: Animals; Female; Gastrointestinal Motility; Guinea Pigs; Ileum; In Vitro Techniques; Male; Neurokinin-1 Receptor Antagonists; Neurons; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Substance P; Synaptic Transmission

1998
Effect of non-peptide tachykinin NK(1) receptor antagonists on non-adrenergic, non-cholinergic neurogenic mucus secretion in ferret trachea.
    European journal of pharmacology, 1999, Nov-19, Volume: 384, Issue:2-3

    Topics: Acetylcholine; Animals; Binding, Competitive; Dose-Response Relationship, Drug; Ferrets; In Vitro Techniques; Iodine Radioisotopes; Male; Membranes; Mucus; Neurokinin-1 Receptor Antagonists; Peptides, Cyclic; Piperidines; Quinolines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Trachea

1999
Neurokinin-1 receptor activation in Botzinger complex evokes bradypnoea.
    The Journal of physiology, 2006, Sep-15, Volume: 575, Issue:Pt 3

    Topics: Animals; Diaphragm; Electric Stimulation; Male; Microinjections; Phrenic Nerve; Piperidines; Rats; Rats, Wistar; Receptors, Neurokinin-1; Reflex; Respiratory Center; Respiratory Function Tests; Respiratory Mechanics; Substance P; Vagus Nerve

2006
Neurokinin receptor modulation of respiratory activity in the rabbit.
    The European journal of neuroscience, 2008, Volume: 27, Issue:12

    Topics: Animals; Exhalation; Inhalation; Male; Medulla Oblongata; Microinjections; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Phrenic Nerve; Piperidines; Rabbits; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Substance P; Vagotomy

2008