Page last updated: 2024-09-05

substance p, pro(9)- and substance p

substance p, pro(9)- has been researched along with substance p in 17 studies

Compound Research Comparison

Studies
(substance p, pro(9)-)
Trials
(substance p, pro(9)-)
Recent Studies (post-2010)
(substance p, pro(9)-)
Studies
(substance p)
Trials
(substance p)
Recent Studies (post-2010) (substance p)
170017,2892772,010

Protein Interaction Comparison

ProteinTaxonomysubstance p, pro(9)- (IC50)substance p (IC50)
Substance-P receptorRattus norvegicus (Norway rat)0.0005
Substance-K receptorRattus norvegicus (Norway rat)0.2
Substance-K receptorHomo sapiens (human)0.2455
Substance-P receptorHomo sapiens (human)0.0011
Neuromedin-K receptorHomo sapiens (human)0.125
Substance-K receptorMesocricetus auratus (golden hamster)0.148

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's16 (94.12)18.2507
2000's1 (5.88)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chassaing, G; Clodic, G; Karoyan, P; Lavielle, S; Sagan, S1
Beaujouan, JC; Brunissen, A; Carruette, A; Chassaing, G; Garret, C; Glowinski, J; Lavielle, S; Petitet, F; Saffroy, M; Torrens, Y1
Beaujouan, JC; Chassaing, G; Glowinski, J; Lavielle, S; Loeuillet, D; Petitet, F; Saffroy, M; Torrens, Y1
Beaujouan, JC; Besseyre, J; Carruette, A; Chassaing, G; Garret, C; Glowinski, J; Lavielle, S; Petitet, F; Saffroy, M; Torrens, Y1
Cordier, J; Delumeau, JC; Glowinski, J; Petitet, F; Prémont, J1
Beaujouan, JC; Glowinski, J; Saffroy, M; Torrens, Y2
Beaujouan, JC; Glowinski, J; Petitet, F; Saffroy, M; Torrens, Y2
Gunne, LM; Liminga, U1
Brunissen, A; Carruette, A; Chassaing, G; Garret, C; Lavielle, S1
Betschart, J; Blanchard, JC; Fardin, V; Flamand, O; Ravard, S1
Liminga, U1
Betschart, J; Blanchard, JC; Garret, C; Grall, I; Piot, O; Ravard, S1
Desban, M; Gauchy, C; Glowinski, J; Kemel, ML1
Beaujouan, JC; Glowinski, J; Saffroy, M; Tencé, M; Torrens, Y1
Lavielle, S; Sagan, S1

Other Studies

17 other study(ies) available for substance p, pro(9)- and substance p

ArticleYear
Asymmetric synthesis of Boc-N-methyl-p-benzoyl-phenylalanine. Preparation of a photoreactive antagonist of substance P.
    Bioorganic & medicinal chemistry letters, 1998, Jun-02, Volume: 8, Issue:11

    Topics: Alkylation; Animals; Biotin; CHO Cells; Cricetinae; Cyclic AMP; Humans; Molecular Conformation; Neurokinin-1 Receptor Antagonists; Phenylalanine; Photochemistry; Receptors, Neurokinin-2; Structure-Activity Relationship; Substance P

1998
[Pro9]SP and [pGlu6, Pro9]SP(6-11) interact with two different receptors in the guinea-pig ileum as demonstrated with new SP antagonists.
    Neuropeptides, 1992, Volume: 23, Issue:2

    Topics: Amino Acid Sequence; Animals; Brain Chemistry; Duodenum; Guinea Pigs; In Vitro Techniques; Male; Molecular Sequence Data; Muscle Contraction; Neurokinin A; Rabbits; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurotransmitter; Substance P; Synaptosomes

1992
[A new tachykinin receptor revealed by substance P analogues in the guinea pig ileum].
    Comptes rendus de l'Academie des sciences. Serie III, Sciences de la vie, 1992, Mar-26, Volume: 314, Issue:7

    Topics: Animals; Cell Membrane; Duodenum; Guinea Pigs; Ileum; Muscle Contraction; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Tachykinin; Substance P

1992
Further demonstration that [Pro9]-substance P is a potent and selective ligand of NK-1 tachykinin receptors.
    Journal of neurochemistry, 1991, Volume: 56, Issue:3

    Topics: Animals; Autoradiography; Binding Sites; Brain; Kinetics; Ligands; Male; Membranes; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P; Succinimides; Tachykinins; Tissue Distribution

1991
Synergistic regulation of cytosolic Ca2+ concentration in mouse astrocytes by NK1 tachykinin and adenosine agonists.
    Journal of neurochemistry, 1991, Volume: 57, Issue:6

    Topics: 2-Chloroadenosine; 5,8,11,14-Eicosatetraynoic Acid; Adenosine; Animals; Arachidonic Acid; Astrocytes; Calcium; Cells, Cultured; Cytosol; Drug Synergism; Enzyme Activation; Mice; Osmolar Concentration; Protein Kinase C; Receptors, Neurotransmitter; Receptors, Purinergic; Receptors, Tachykinin; Substance P; Tachykinins

1991
Involvement of septide-sensitive tachykinin receptors in inositol phospholipid hydrolysis in the rat urinary bladder.
    Peptides, 1995, Volume: 16, Issue:4

    Topics: Amino Acid Sequence; Animals; Benzamides; Hydrolysis; Indoles; Isoindoles; Male; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth; Neurokinin A; Peptide Fragments; Phosphatidylinositols; Piperidines; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Tachykinin; Substance P; Urinary Bladder

1995
A new selective bioassay for tachykinin NK3 receptors based on inositol monophosphate accumulation in the guinea pig ileum.
    European journal of pharmacology, 1993, Oct-15, Volume: 247, Issue:2

    Topics: Animals; Biphenyl Compounds; Guinea Pigs; Hypnotics and Sedatives; Ileum; In Vitro Techniques; Inositol Phosphates; Male; Muscle, Smooth; Neurokinin A; Peptide Fragments; Phosphatidylinositols; Phospholipids; Receptors, Neurokinin-3; Stimulation, Chemical; Substance P; Tachykinins

1993
Intranigral stimulation of oral movements by [Pro9] substance P, a neurokinin-1 receptor agonist, is enhanced in chronically neuroleptic-treated rats.
    Behavioural brain research, 1993, Oct-21, Volume: 57, Issue:1

    Topics: Animals; Female; Fluphenazine; Mastication; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Substance P; Substantia Nigra; Synaptic Transmission

1993
Differential localization of 3H-[Pro9]SP binding sites in the guinea pig and rat brain.
    Brain research, 1994, Jan-07, Volume: 633, Issue:1-2

    Topics: Animals; Brain; Brain Chemistry; Guinea Pigs; Male; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Substance P; Succinimides

1994
Highly potent substance P antagonists substituted with beta-phenyl- or beta-benzyl-proline at position 10.
    European journal of pharmacology, 1994, Jun-13, Volume: 258, Issue:3

    Topics: Amino Acid Sequence; Animals; Guinea Pigs; Ileum; In Vitro Techniques; Male; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Physalaemin; Pyrrolidonecarboxylic Acid; Rabbits; Rats; Receptors, Neurokinin-1; Structure-Activity Relationship; Substance P

1994
Differential ability of tachykinin NK-1 and NK-2 agonists to produce scratching and grooming behaviours in mice.
    Brain research, 1994, Jul-18, Volume: 651, Issue:1-2

    Topics: Animals; Behavior, Animal; Brain; Grooming; Male; Mice; Neurokinin A; Peptide Fragments; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P

1994
Selective neurokinin NK1 and NK2 receptor agonists infused in the substantia nigra of the rat increase vacuous chewing.
    European journal of pharmacology, 1993, Apr-28, Volume: 235, Issue:2-3

    Topics: Animals; Dose-Response Relationship, Drug; Female; Mastication; Neurokinin A; Peptide Fragments; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Substance P; Substantia Nigra

1993
Comparative behavioural profile of centrally administered tachykinin NK1, NK2 and NK3 receptor agonists in the guinea-pig.
    British journal of pharmacology, 1995, Volume: 116, Issue:5

    Topics: Animals; Behavior, Animal; Guinea Pigs; Injections, Intraventricular; Male; Motor Activity; Neurokinin A; Peptide Fragments; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P

1995
Distinct regulations by septide and the neurokinin-1 tachykinin receptor agonist [pro9]substance P of the N-methyl-D-aspartate-evoked release of dopamine in striosome- and matrix-enriched areas of the rat striatum.
    Neuroscience, 1996, Volume: 73, Issue:4

    Topics: Animals; Corpus Striatum; Dopamine; Extracellular Matrix; Indoles; Isoindoles; Male; N-Methylaspartate; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Tachykinin; Substance P

1996
Substance P(6-11) and natural tachykinins interact with septide-sensitive tachykinin receptors coupled to a phospholipase C in the rat urinary bladder.
    Neuropeptides, 1997, Volume: 31, Issue:3

    Topics: Analgesics; Animals; Benzamides; Binding Sites; Inositol Phosphates; Male; Neurokinin A; Neurokinin B; Neuropeptides; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-2; Receptors, Tachykinin; Substance P; Tachykinins; Tritium; Type C Phospholipases; Urinary Bladder

1997
Functional coupling of the NK1 tachykinin receptor to phospholipase D in chinese hamster ovary cells and astrocytoma cells.
    Journal of neurochemistry, 1998, Volume: 70, Issue:5

    Topics: Animals; Astrocytoma; Calcium; CHO Cells; Cricetinae; Cyclic AMP; Enzyme Activation; Glycerophospholipids; GTP-Binding Proteins; Humans; Myristic Acid; Phosphatidic Acids; Phosphatidylcholines; Phospholipase D; Protein Kinase C; Rats; Receptors, Neurokinin-1; Substance P; Tachykinins; Tumor Cells, Cultured

1998
Internalization of [3H]substance P analogues in NK-1 receptor transfected CHO cells.
    Biochemical and biophysical research communications, 2001, Apr-13, Volume: 282, Issue:4

    Topics: Animals; Arsenicals; CHO Cells; Cricetinae; Endocytosis; Kinetics; Models, Biological; Monensin; Peptide Fragments; Receptors, Neurokinin-1; Substance P; Temperature; Transfection

2001