Page last updated: 2024-09-03

substance p, methyl ester- and naloxone

substance p, methyl ester- has been researched along with naloxone in 2 studies

Compound Research Comparison

Studies
(substance p, methyl ester-)
Trials
(substance p, methyl ester-)
Recent Studies (post-2010)
(substance p, methyl ester-)
Studies
(naloxone)
Trials
(naloxone)
Recent Studies (post-2010) (naloxone)
350120,1341,2573,321

Protein Interaction Comparison

ProteinTaxonomysubstance p, methyl ester- (IC50)naloxone (IC50)
Cytochrome P450 2D6Homo sapiens (human)2
Delta-type opioid receptorMus musculus (house mouse)0.043
Delta-type opioid receptorRattus norvegicus (Norway rat)0.0219
Mu-type opioid receptorRattus norvegicus (Norway rat)0.0019
Kappa-type opioid receptorRattus norvegicus (Norway rat)0.0019
Mu-type opioid receptorHomo sapiens (human)0.0397
Delta-type opioid receptorHomo sapiens (human)0.1896
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)0.05
Kappa-type opioid receptorHomo sapiens (human)0.0795
Mu-type opioid receptorMus musculus (house mouse)0.0154
Mu-type opioid receptorCavia porcellus (domestic guinea pig)0.0089
Beta-2 adrenergic receptorCavia porcellus (domestic guinea pig)0.0055

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19901 (50.00)18.7374
1990's1 (50.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Koelbel, CB; Leduc, L; Mayer, EA; Snape, WJ; Vandeventer, G1
Chorev, M; Friedman, ZY; Gilon, C; Laufer, R; Selinger, Z; Wormser, U1

Other Studies

2 other study(ies) available for substance p, methyl ester- and naloxone

ArticleYear
Neurokinin inhibition of cholinergic myenteric neurons in canine antrum.
    The American journal of physiology, 1990, Volume: 258, Issue:1 Pt 1

    Topics: Acetylcholine; Animals; Atropine; Dinoprostone; Dogs; Electric Stimulation; Enkephalin, Methionine; Female; Hexamethonium; Hexamethonium Compounds; In Vitro Techniques; Indomethacin; Male; Muscle, Smooth; Myenteric Plexus; Naloxone; Neurokinin A; Neurons; Nifedipine; Phentolamine; Propranolol; Pyloric Antrum; Substance P; Tetrodotoxin; Vasoactive Intestinal Peptide

1990
Neurokinin B is a preferred agonist for a neuronal substance P receptor and its action is antagonized by enkephalin.
    Proceedings of the National Academy of Sciences of the United States of America, 1985, Volume: 82, Issue:21

    Topics: Animals; Atropine; Enkephalin, Methionine; Guinea Pigs; Ileum; Muscle Contraction; Muscle, Smooth; Naloxone; Nerve Tissue Proteins; Neurokinin A; Neurokinin B; Neurons; Neurotransmitter Agents; Oligopeptides; Peptide Fragments; Receptors, Muscarinic; Receptors, Neurokinin-1; Receptors, Neurotransmitter; Substance P; Substrate Specificity; Tachykinins

1985