Page last updated: 2024-09-05

substance p (6-11), pglu(6)- and substance p

substance p (6-11), pglu(6)- has been researched along with substance p in 12 studies

Compound Research Comparison

Studies
(substance p (6-11), pglu(6)-)
Trials
(substance p (6-11), pglu(6)-)
Recent Studies (post-2010)
(substance p (6-11), pglu(6)-)
Studies
(substance p)
Trials
(substance p)
Recent Studies (post-2010) (substance p)
160017,2892772,010
16002300
160085012

Protein Interaction Comparison

ProteinTaxonomysubstance p (6-11), pglu(6)- (IC50)substance p (IC50)
Substance-P receptorRattus norvegicus (Norway rat)0.0005
Substance-K receptorRattus norvegicus (Norway rat)0.2
Substance-K receptorHomo sapiens (human)0.2455
Substance-P receptorHomo sapiens (human)0.0011
Neuromedin-K receptorHomo sapiens (human)0.125
Substance-K receptorMesocricetus auratus (golden hamster)0.148

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-199010 (83.33)18.7374
1990's2 (16.67)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Iwabuchi, Y; Masuhara, T; Sofuku, S1
Chorev, M; Gilon, C; Laufer, R; Selinger, Z; Wormser, U1
Koziołkiewicz, W; Lachowicz, L; Turski, WA1
Chorev, M; Friedman, ZY; Gilon, C; Rubini, E; Selinger, Z; Wormser, U1
Barth, A; Bergmann, J; Hartrodt, B; Jakubke, HD; Lindau, J; Mehlis, B; Neubert, K; Rüger, M1
Chorev, M; Gilon, C; Laufer, R; Selinger, Z1
Chorev, M; Ewenson, A; Gilon, C; Goldin, E; Karmeli, F; Laufer, R; Rachmilewitz, D; Selinger, Z; Silkoff, P1
Lachowicz, L; Turski, WA1
Kubicki, J; Traczyk, WZ1
Cotrait, M; Hospital, M1
de Wied, D; Gaffori, O; Stewart, JM1
Chorev, M; Friedman, ZY; Gilon, C; Laufer, R; Selinger, Z; Wormser, U1

Other Studies

12 other study(ies) available for substance p (6-11), pglu(6)- and substance p

ArticleYear
Sialogogic effects on rat submandibular gland of analogs of the C-terminal hexapeptide of substance P.
    Japanese journal of pharmacology, 1992, Volume: 58, Issue:3

    Topics: Animals; Male; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Inbred Strains; Salivation; Submandibular Gland; Substance P

1992
Proteolytic resistance and biological activity of N-methylated analogs of [pGlu6] substance P6-11.
    Neuropeptides, 1990, Volume: 16, Issue:1

    Topics: Animals; Hypothalamus; In Vitro Techniques; Methylation; Parotid Gland; Peptide Fragments; Peptide Hydrolases; Pyrrolidonecarboxylic Acid; Rats; Substance P

1990
The preliminary evaluation of degradation of substance P(SP) fragment's analogue less than Glu SP6-11 in the subcellular fractions from different areas of rat brain.
    The International journal of biochemistry, 1985, Volume: 17, Issue:10

    Topics: Animals; Biotransformation; Brain; Female; Hydrogen-Ion Concentration; In Vitro Techniques; Oligopeptides; Peptide Fragments; Peptide Hydrolases; Pyrrolidonecarboxylic Acid; Rats; RNA; Subcellular Fractions; Substance P

1985
Desensitization of substance P-induced K+ release in rat parotid.
    European journal of pharmacology, 1985, Nov-19, Volume: 117, Issue:3

    Topics: Animals; Guinea Pigs; Ileum; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Oligopeptides; Parasympatholytics; Parotid Gland; Peptide Fragments; Potassium; Pyrrolidonecarboxylic Acid; Rats; Receptors, Adrenergic, alpha; Stimulation, Chemical; Substance P; Time Factors

1985
[Synthesis of cyclic and non-cyclic tachykinin partial sequences. 2. Synthesis of the homocyclic substance P(6-11) hexapeptide].
    Die Pharmazie, 1985, Volume: 40, Issue:8

    Topics: Amino Acid Sequence; Animals; Cyclization; Guinea Pigs; Ileum; In Vitro Techniques; Muscle Contraction; Oligopeptides; Peptide Fragments; Pyrrolidonecarboxylic Acid; Substance P

1985
[pGlu6,Pro9]SP6-11, a selective agonist for the substance P P-receptor subtype.
    Journal of medicinal chemistry, 1986, Volume: 29, Issue:7

    Topics: Animals; Guinea Pigs; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Neurons; Oligopeptides; Parotid Gland; Peptide Fragments; Potassium; Pyrrolidonecarboxylic Acid; Rats; Receptors, Neurokinin-1; Receptors, Neurotransmitter; Substance P

1986
Effect of substance P on rat gastrointestinal transit.
    Digestive diseases and sciences, 1988, Volume: 33, Issue:1

    Topics: Animals; Gastrointestinal Transit; Hydroxylamines; Male; Oligopeptides; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Substance P

1988
The effects of the main body cations on the peptidase(s) activity against pyroGlu6[125I-Tyr8]SP6-11 in the nuclear and synaptosomal fraction of the cortex and hippocampus of rat brain.
    The International journal of biochemistry, 1987, Volume: 19, Issue:12

    Topics: Animals; Calcium; Cations; Cell Nucleus; Cerebral Cortex; Female; Hippocampus; In Vitro Techniques; Iodine Radioisotopes; Kinetics; Magnesium; Male; Osmolar Concentration; Peptide Fragments; Peptide Hydrolases; Potassium; Pyrrolidonecarboxylic Acid; Rats; Rats, Inbred Strains; Sodium; Substance P; Synaptosomes

1987
The pressor response to substance P and hexapeptide [pGlu6]SP 6--11 injections into the cerebral ventricles in rats.
    Neuropharmacology, 1980, Volume: 19, Issue:7

    Topics: Animals; Blood Pressure; Dose-Response Relationship, Drug; Injections, Intraventricular; Male; Oligopeptides; Peptide Fragments; Propranolol; Pyrrolidonecarboxylic Acid; Rats; Substance P; Synaptic Transmission; Time Factors; Vagotomy

1980
Conformational studies on substance P. C-terminal pentapeptide pGlu-Phe-Phe-Gly-Leu-Met NH2.
    Biochemical and biophysical research communications, 1982, Dec-31, Volume: 109, Issue:4

    Topics: Amino Acid Sequence; Animals; Oligopeptides; Peptide Fragments; Protein Conformation; Pyrrolidonecarboxylic Acid; Structure-Activity Relationship; Substance P

1982
Influence of substance P and fragments on passive avoidance behavior.
    Experientia, 1984, Jan-15, Volume: 40, Issue:1

    Topics: Animals; Avoidance Learning; Dose-Response Relationship, Drug; Mice; Oligopeptides; Peptide Fragments; Pyrrolidonecarboxylic Acid; Substance P

1984
Substance P degrading systems of rat parotid and hypothalamus.
    Biochimica et biophysica acta, 1984, Mar-22, Volume: 798, Issue:1

    Topics: Amino Acid Sequence; Animals; Guinea Pigs; Hypothalamus; Ileum; In Vitro Techniques; Kinetics; Muscle Contraction; Oligopeptides; Parotid Gland; Peptide Fragments; Protease Inhibitors; Pyrrolidonecarboxylic Acid; Rats; Substance P

1984