Page last updated: 2024-08-23

staurosporine and y 27632

staurosporine has been researched along with y 27632 in 14 studies

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (7.14)18.2507
2000's8 (57.14)29.6817
2010's4 (28.57)24.3611
2020's1 (7.14)2.80

Authors

AuthorsStudies
Bonn, S; Bossemeyer, D; Breitenlechner, CB; Engh, RA; Erlbruch, A; Gassel, M; Herrero, S; Lehmann, W1
Bullock, AN; Fedorov, O; Knapp, S; Marsden, B; Müller, S; Pogacic, V; Rellos, P; Schwaller, J; Sundström, M1
Augustin, M; Davies, SP; Gao, Y; Harvey, KJ; Kovelman, R; Patel, UA; Woodward, A1
Feng, J; Isaka, N; Ito, M; Kureishi, Y; Nakano, T; Okinaka, T1
Amano, M; Fukata, Y; Kaibuchi, K; Shimokawa, H1
Brkic-Koric, D; Pfitzer, G; Sonntag-Bensch, D1
Bauer, J; Parekh, N1
Shimoda, LA; Sylvester, JT; Weigand, L1
Chen, S; Dul, E; Hu, E; Khandekar, SS; Kirkpatrick, RB; Lee, D; Scott, GF; Smith, GK; Wright, LL; Yi, T1
Bisschops, R; Cassiman, D; Fevery, J; Laleman, W; Nevens, F; Roskams, T; Severi, T; Van Landeghem, L; Van Pelt, J; Vander Elst, I; Zeegers, M1
Ehrhard, M; Fritzsching, B; Frommhold, D; Koch, L; Poeschl, J; Ruef, P1
Al-Ghabkari, A; MacDonald, JA; Moffat, LD; Sutherland, C; Walsh, MP1
Kim, BJ; Kim, JN1
Kihara, T; Matsumoto, T; Nakahashi, Y; Tachibana, K1

Other Studies

14 other study(ies) available for staurosporine and y 27632

ArticleYear
Structural analysis of protein kinase A mutants with Rho-kinase inhibitor specificity.
    The Journal of biological chemistry, 2006, Aug-25, Volume: 281, Issue:34

    Topics: Animals; Benzamides; Cattle; Cyclic AMP-Dependent Protein Kinases; Erlotinib Hydrochloride; Imatinib Mesylate; Intracellular Signaling Peptides and Proteins; Models, Molecular; Mutagenesis, Site-Directed; Piperazines; Protein Conformation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Pyrimidines; Quinazolines; Recombinant Fusion Proteins; rho-Associated Kinases; Structure-Activity Relationship; Substrate Specificity

2006
A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.
    Proceedings of the National Academy of Sciences of the United States of America, 2007, Dec-18, Volume: 104, Issue:51

    Topics: Amino Acid Sequence; Binding Sites; Clinical Trials as Topic; Drug Evaluation, Preclinical; Enzyme Stability; Humans; Molecular Sequence Data; Phylogeny; Protein Array Analysis; Protein Conformation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases

2007
A broad activity screen in support of a chemogenomic map for kinase signalling research and drug discovery.
    The Biochemical journal, 2013, Apr-15, Volume: 451, Issue:2

    Topics: Aurora Kinases; Cluster Analysis; Drug Design; Drug Discovery; Drug Evaluation, Preclinical; ErbB Receptors; Humans; Intracellular Signaling Peptides and Proteins; MAP Kinase Kinase 4; p38 Mitogen-Activated Protein Kinases; Protein Kinase Inhibitors; Protein Kinases; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Receptors, Vascular Endothelial Growth Factor; Recombinant Proteins; Reproducibility of Results; Signal Transduction; Small Molecule Libraries; Structure-Activity Relationship; Syk Kinase

2013
Regulation of Ca2+-independent smooth muscle contraction by alternative staurosporine-sensitive kinase.
    European journal of pharmacology, 1999, Jul-09, Volume: 376, Issue:3

    Topics: Amides; Animals; Enzyme Inhibitors; Male; Microcystins; Muscle Contraction; Muscle, Smooth, Vascular; Myosin-Light-Chain Kinase; Peptides, Cyclic; Phosphorylation; Pyridines; Rabbits; Rho Factor; Staurosporine; Vasoconstrictor Agents

1999
Purification and in vitro activity of Rho-associated kinase.
    Methods in enzymology, 2000, Volume: 325

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Amides; Animals; Baculoviridae; Catalytic Domain; Cattle; Guanosine 5'-O-(3-Thiotriphosphate); Intracellular Signaling Peptides and Proteins; Protein Serine-Threonine Kinases; Pyridines; Recombinant Fusion Proteins; rho-Associated Kinases; rhoA GTP-Binding Protein; Staurosporine

2000
Thiophosphorylation-induced Ca(2+) sensitization of guinea-pig ileum contractility is not mediated by Rho-associated kinase.
    The Journal of physiology, 2001, Jun-15, Volume: 533, Issue:Pt 3

    Topics: Actin Cytoskeleton; Adenosine Triphosphate; Amides; Animals; Calcium; Carbachol; Drug Synergism; Enzyme Inhibitors; Female; Gastrointestinal Motility; Guanosine 5'-O-(3-Thiotriphosphate); Guinea Pigs; Ileum; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Male; Phosphorylation; Protein Kinase Inhibitors; Protein Kinases; Protein Serine-Threonine Kinases; Pyridines; rho-Associated Kinases; Staurosporine; Sulfhydryl Compounds; Sulfur

2001
Variations in cell signaling pathways for different vasoconstrictor agonists in renal circulation of the rat.
    Kidney international, 2003, Volume: 63, Issue:6

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Amides; Angiotensin II; Animals; Arginine Vasopressin; Blood Pressure; Calcium Channel Blockers; Enzyme Inhibitors; Female; Gallic Acid; Indoles; Nifedipine; Norepinephrine; Pyridines; Rats; Rats, Wistar; Renal Circulation; Signal Transduction; Staurosporine; Vasoconstrictor Agents

2003
Mechanisms of endothelin-1-induced contraction in pulmonary arteries from chronically hypoxic rats.
    American journal of physiology. Lung cellular and molecular physiology, 2006, Volume: 290, Issue:2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Amides; Animals; Azepines; Endothelin-1; Enzyme Inhibitors; Genistein; Hypoxia; Indoles; Intracellular Signaling Peptides and Proteins; Isometric Contraction; Male; Maleimides; Myosin-Light-Chain Kinase; Potassium Chloride; Protein Kinase C; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Pulmonary Artery; Pyridines; Pyrimidines; Rats; Rats, Wistar; rho-Associated Kinases; src-Family Kinases; Staurosporine; Vasoconstriction

2006
Expression, purification, and characterization of an enzymatically active truncated human rho-kinase I (ROCK I) domain expressed in Sf-9 insect cells.
    Protein and peptide letters, 2006, Volume: 13, Issue:4

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Amides; Amino Acid Sequence; Animals; Humans; Inhibitory Concentration 50; Intracellular Signaling Peptides and Proteins; Molecular Sequence Data; Molecular Weight; Protein Serine-Threonine Kinases; Protein Structure, Tertiary; Pyridines; rho-Associated Kinases; Spodoptera; Staurosporine

2006
Both Ca2+ -dependent and -independent pathways are involved in rat hepatic stellate cell contraction and intrahepatic hyperresponsiveness to methoxamine.
    American journal of physiology. Gastrointestinal and liver physiology, 2007, Volume: 292, Issue:2

    Topics: Actomyosin; Amides; Animals; Calcimycin; Calcium; Cell Shape; Cells, Cultured; Diacetyl; Enzyme Inhibitors; Liver; Male; Marine Toxins; Methoxamine; Myocytes, Cardiac; Myocytes, Smooth Muscle; Myosin-Light-Chain Kinase; Oxazoles; Protein Kinase Inhibitors; Pyridines; Rats; Rats, Wistar; Signal Transduction; Staurosporine; Sulfonamides; Vasoconstrictor Agents

2007
Lipid A decreases human erythrocytes deformability by increasing intracellular Ca(2+): effects of verapamil, staurosporine and the rho-kinase inhibitor Y-27632.
    Clinical hemorheology and microcirculation, 2011, Volume: 49, Issue:1-4

    Topics: Adult; Amides; Calcium Channel Blockers; Calcium Signaling; Depression, Chemical; Drug Interactions; Erythrocyte Deformability; Escherichia coli; Humans; In Vitro Techniques; Lipid A; Male; Protein Kinase Inhibitors; Pyridines; rho-Associated Kinases; Shear Strength; Staurosporine; Verapamil

2011
Prostate-apoptosis response-4 phosphorylation in vascular smooth muscle.
    Archives of biochemistry and biophysics, 2013, Jul-01, Volume: 535, Issue:1

    Topics: Amides; Animals; Apoptosis Regulatory Proteins; Arteries; Blotting, Western; Calcium-Calmodulin-Dependent Protein Kinases; Cyclic AMP-Dependent Protein Kinases; Death-Associated Protein Kinases; Immunoprecipitation; Indoles; Male; Maleimides; Microcystins; Muscle Contraction; Muscle, Smooth, Vascular; Octoxynol; Phosphorylation; Protein Binding; Protein Phosphatase 1; Pyridines; Rats; Rats, Sprague-Dawley; Recombinant Proteins; rho-Associated Kinases; Staurosporine; Threonine; Time Factors

2013
The Mechanism of Action of Ghrelin and Motilin in the Pacemaker Potentials of Interstitial Cells of Cajal from the Murine Small Intestine.
    Molecules and cells, 2019, Jun-30, Volume: 42, Issue:6

    Topics: Acetophenones; Amides; Animals; Benzopyrans; Boron Compounds; Calcium; Carbazoles; Gastrointestinal Motility; Ghrelin; Inositol 1,4,5-Trisphosphate Receptors; Interstitial Cells of Cajal; Intestine, Small; Macrocyclic Compounds; Membrane Potentials; Mice; Mice, Inbred ICR; Motilin; Oligopeptides; Oxazoles; Protein Kinase C; Pyridines; Receptors, Ghrelin; rho-Associated Kinases; Signal Transduction; Staurosporine; Thapsigargin

2019
Mechanical stiffness softening and cell adhesion are coordinately regulated by ERM dephosphorylation in KG-1 cells.
    Human cell, 2021, Volume: 34, Issue:6

    Topics: Actins; Amides; Cell Adhesion; Cell Line, Tumor; Cytochalasin D; Cytoskeletal Proteins; Elasticity; Fibronectins; Humans; Leukemia, Myeloid; Leukocytes; Membrane Proteins; Microfilament Proteins; Microvilli; Phorbol Esters; Phosphorylation; Pyridines; Staurosporine

2021