staurosporine has been researched along with serine in 57 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 18 (31.58) | 18.2507 |
2000's | 34 (59.65) | 29.6817 |
2010's | 5 (8.77) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Feinstein, R; Hemi, R; Kanety, H; Karasik, A; Papa, MZ | 1 |
Ali, H; DuBose, RA; Haribabu, B; Richardson, RM; Snyderman, R; Tomhave, ED | 1 |
Banerjee, AK; Das, T; Schneider-Schaulies, S; Schuster, A | 1 |
Terrian, DM; Ways, DK | 1 |
Chang, ZF; Hsue, NC; Huang, DY | 1 |
Jost, E; Leukel, M | 1 |
Agnew, WS; Bendahhou, S; Cummins, TR; Potts, JF; Tong, J | 1 |
Londos, C; Rondinone, CM; Smith, UP; Zarnowski, MJ | 1 |
Badiani, K; Byers, DM; Cook, HW; Ridgway, ND | 1 |
Brown, S; Garcia, DE; Hille, B; Mackie, K | 1 |
Bassini, A; Bertolaso, L; Capitani, S; Gibellini, D; La Placa, M; Milani, D; Pierpaoli, S; Zauli, G | 1 |
Spurney, RF | 1 |
Adachi, K; Hirata, Y; Kiuchi, K | 1 |
Kodama, H; Sagara, Y; Spirito, A; Sugahara, K; Zhang, J; Zhang, M | 1 |
Anderson, HJ; James, WM; Ray, JM; Roberge, M; Sauvé, DM | 1 |
Hamaoka, T; Kosugi, A; Miki, T; Mori, Y; Ogata, M; Oh-hora, M; Okuyama, A; Sawada, M; Takada, T; Uchida, Y | 1 |
Brender, C; Brockdorff, J; Christensen, ST; Engel, AM; Geisler, C; Kaltoft, K; Leick, V; Nielsen, M; Odum, N; Rygaard, J; Skov, S; Svejgaard, A; Woetmann, A | 1 |
Blau, N; Leimbacher, W; Scherer-Oppliger, T; Thöny, B | 1 |
Gales, J; Graves, PR; O'Connor, PM; Piwnica-Worms, H; Sausville, EA; Schwarz, JK; Yu, L | 1 |
Kilpatrick, LE; Korchak, HM; Rossi, MW; Song, YH | 1 |
Ivanov, KI; Mäkinen, K; Merits, A; Puustinen, P; Saarma, M | 1 |
Bazzoni, G; Bontrager, AL; Chen, LB; Hemler, ME; Kraeft, SK; Stipp, CS; Zhang, XA | 1 |
Anguissola, S; Comoglio, PM; Giordano, S; Gual, P; Parker, PJ | 1 |
Beauchemin, N; Fournès, B; Létourneau, S; Sadekova, S; Turbide, C | 1 |
Feldman, RD; Ferguson, SS; Kelvin, DJ; Litchfield, DW; Tan, CM | 1 |
Andjelkovic, M; Brazil, DP; Fabbro, D; Ferrari, S; Hemmings, BA; Hill, MM | 1 |
Akaike, A; Honda, K; Kihara, T; Nakamizo, T; Sawada, H; Shibasaki, H; Shimohama, S | 1 |
Bijur, GN; Jope, RS | 1 |
Correia, MA; Maltby, D; Medzihradszky, KF; Wang, X | 1 |
Chang, NS | 1 |
Arai, H; Fijimoto, M; Nagasaka, Y; Nakamura, K | 1 |
Ellory, JC; Gibson, JS; Kiessling, K; Roberts, N | 1 |
Hodgkinson, CP; Sale, EM; Sale, GJ | 1 |
Deng, X; Gao, F; Jin, Z; Mai, H; May, WS | 1 |
Chen, J; Chen, Q; Gu, L; Zhang, H | 1 |
Mariner, DJ; Reynolds, AB; Xia, X | 1 |
Bloom, DA; Jaiswal, AK | 1 |
Ansari, A; Dorovkov, MV; Ryazanov, AG; Ryazanova, LV | 1 |
Bertorello, AM; Delamere, NA; Khundmiri, SJ; Lederer, ED | 1 |
Cushman, SW; Kondapaka, SB; Sausville, EA; Yver, DR; Zarnowski, M | 1 |
Stern, DF; Tsvetkov, L | 1 |
Min, W; Storz, P; Zhang, W; Zheng, S | 1 |
Chang, NS; Doherty, J; Ensign, A; Hong, Q; Hsu, LJ; Schultz, L | 1 |
Cai, SQ; Hernandez, L; Park, KH; Sesti, F; Wang, Y | 1 |
Bhanumathy, C; Joseph, SK; Khan, MT; Wagner, L; Yule, DI | 1 |
Amann, K; Artunc, F; Grahammer, F; Huang, DY; Hussain, A; Kandolf, R; Klingel, K; Kuhl, D; Lang, F; Vallon, V; Wyatt, AW | 1 |
Doi, J; Katoh, Y; Lin, XZ; Min, L; Miyauchi, A; Muraoka, M; Nakamura, H; Okamoto, M; Satoh, T; Takemori, H; Tamura, M; Tsuchiya, Y; Witters, LA | 1 |
Srivastava, A; Wu, J; Zhao, W; Zhong, L | 1 |
Cribbs, JT; Strack, S | 1 |
Furukawa, Y; Futaki, K; Kano, Y; Kikuchi, J; Odgerel, T; Shimizu, R; Wada, T | 1 |
Fanucchi, S; Veale, RB | 1 |
Ayilavarapu, S; Hasturk, H; Ito, K; Iwata, T; Kantarci, A; Omori, K; Van Dyke, TE; Yagi, M | 1 |
Arrigoni, G; Inagaki, K; Martinez, HM; Pinna, LA; Shimasaki, S; Tibaldi, E | 1 |
Kaliyaperumal, S; Patrick, SM; Williams, KJ | 1 |
Appelqvist, H; Brown, AJ; Garner, B; Kågedal, K; Nilsson, C; Ollinger, K | 1 |
Li, R; Reiser, G | 1 |
Agerman, K; Eckersley, S; Gu, GJ; Kamali-Moghaddam, M; Kvist, AJ; Landegren, U; Lund, H; Milner, R; Nilsson, LN; Sunnemark, D; Wu, D | 1 |
57 other study(ies) available for staurosporine and serine
Article | Year |
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Tumor necrosis factor alpha-induced phosphorylation of insulin receptor substrate-1 (IRS-1). Possible mechanism for suppression of insulin-stimulated tyrosine phosphorylation of IRS-1.
Topics: Alkaloids; Animals; Enzyme Inhibitors; Humans; Insulin; Insulin Receptor Substrate Proteins; Insulin Resistance; Mice; Phosphatidylinositol 3-Kinases; Phosphoproteins; Phosphorylation; Phosphotransferases (Alcohol Group Acceptor); Protein Kinase C; Protein Tyrosine Phosphatases; Rats; Receptor, Insulin; Serine; Staurosporine; Threonine; Tumor Cells, Cultured; Tumor Necrosis Factor-alpha; Tyrosine | 1995 |
Regulation of human interleukin-8 receptor A: identification of a phosphorylation site involved in modulating receptor functions.
Topics: Alkaloids; Amino Acid Sequence; Animals; Antigens, CD; Binding Sites; DNA, Complementary; Epitopes; Humans; Interleukin-8; Molecular Sequence Data; Mutation; Phosphorylation; Precipitin Tests; Protein Kinase C; Rats; Receptors, Interleukin; Receptors, Interleukin-8A; Serine; Staurosporine; Tetradecanoylphorbol Acetate; Threonine; Tumor Cells, Cultured; Up-Regulation | 1995 |
Involvement of cellular casein kinase II in the phosphorylation of measles virus P protein: identification of phosphorylation sites.
Topics: Alkaloids; Amino Acid Sequence; Animals; Base Sequence; Blotting, Western; Casein Kinase II; Cell Line; Cloning, Molecular; Cricetinae; DNA Primers; Electrophoresis, Polyacrylamide Gel; Escherichia coli; Genes, Viral; Histidine; Kidney; Measles virus; Molecular Sequence Data; Phosphoproteins; Phosphorylation; Polymerase Chain Reaction; Protein Kinase C; Protein Serine-Threonine Kinases; Recombinant Proteins; Restriction Mapping; Sequence Tagged Sites; Serine; Staurosporine; Viral Proteins | 1995 |
Persistent enhancement of sustained calcium-dependent glutamate release by phorbol esters: role of calmodulin-independent serine/threonine phosphorylation and actin disassembly.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Actins; Alkaloids; Animals; Barium; Calcium; Calcium-Calmodulin-Dependent Protein Kinases; Calmodulin; Cytochalasin D; Ethers, Cyclic; Glutamates; Guinea Pigs; Hippocampus; Isoquinolines; Male; Okadaic Acid; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphorylation; Phosphotransferases; Piperazines; Protein Kinase C; Serine; Sphingosine; Staurosporine; Subcellular Fractions; Sulfonamides; Synaptosomes; Threonine | 1995 |
Differential phosphorylation of human thymidine kinase in proliferating and M phase-arrested human cells.
Topics: Alkaloids; Cell Division; Cells, Cultured; Cyanogen Bromide; HeLa Cells; Humans; Hydrolysis; Immune Sera; Mitosis; Nocodazole; Phosphorylation; Protein Kinase C; Serine; Staurosporine; Thymidine Kinase | 1994 |
Two conserved serines in the nuclear localization signal flanking region are involved in the nuclear targeting of human lamin A.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acid Phosphatase; Alkaline Phosphatase; Alkaloids; Amino Acid Sequence; Animals; Biological Transport; Cell Nucleus; Chick Embryo; Consensus Sequence; Enzyme Inhibitors; Humans; Isoquinolines; Kinetics; Lamin Type A; Lamins; Molecular Sequence Data; Nuclear Proteins; Phosphorylation; Piperazines; Protein Kinase C; Protein Processing, Post-Translational; Protein Sorting Signals; Serine; Staurosporine | 1995 |
Serine-1321-independent regulation of the mu 1 adult skeletal muscle Na+ channel by protein kinase C.
Topics: Adult; Alkaloids; Amino Acid Sequence; Base Sequence; Cell Line; Consensus Sequence; Conserved Sequence; DNA Primers; Enzyme Inhibitors; Ethers, Cyclic; Humans; Ion Channel Gating; Macromolecular Substances; Membrane Potentials; Molecular Sequence Data; Multiple Sclerosis; Muscle, Skeletal; Mutagenesis, Site-Directed; Naphthalenes; Okadaic Acid; Phosphorylation; Polymerase Chain Reaction; Polyradiculoneuropathy; Protein Kinase C; Recombinant Proteins; Serine; Sodium Channels; Staurosporine; Transfection | 1995 |
The inhibitory effect of staurosporine on insulin action is prevented by okadaic acid. Evidence for an important role of serine/threonine phosphorylation in eliciting insulin-like effects.
Topics: Animals; Biological Transport; Enzyme Activation; Enzyme Inhibitors; Glucose; Insulin; Insulin Antagonists; Male; Okadaic Acid; Phosphatidylinositol 3-Kinases; Phosphoprotein Phosphatases; Phosphorylation; Phosphotransferases (Alcohol Group Acceptor); Protein Kinases; Protein Phosphatase 1; Rats; Receptor, Insulin; Serine; Staurosporine; Threonine; Tyrosine | 1996 |
Inhibition of phosphorylation of the oxysterol binding protein by brefeldin A.
Topics: Animals; Brefeldin A; CHO Cells; Cricetinae; Cyclopentanes; Electrophoresis, Polyacrylamide Gel; Enzyme Inhibitors; Fluorescent Antibody Technique, Indirect; Golgi Apparatus; Hydroxycholesterols; Molecular Weight; Okadaic Acid; Phosphorylation; Protein Kinases; Protein Synthesis Inhibitors; Rabbits; Rats; Receptors, Steroid; Serine; Staurosporine | 1998 |
Protein kinase C disrupts cannabinoid actions by phosphorylation of the CB1 cannabinoid receptor.
Topics: Analgesics; Animals; Benzoxazines; Calcium Channel Blockers; Calcium Channels; Cannabinoids; Carcinogens; Cells, Cultured; Enzyme Activation; GTP-Binding Proteins; Hormone Antagonists; Indoles; Maleimides; Morpholines; Mutagenesis; Naphthalenes; omega-Conotoxin GVIA; Peptides; Phorbols; Phosphorylation; Potassium Channels; Potassium Channels, Inwardly Rectifying; Protein Kinase C; Protein Structure, Tertiary; Rats; Receptors, Cannabinoid; Receptors, Drug; Recombinant Fusion Proteins; Serine; Signal Transduction; Somatostatin; Staurosporine; Tetradecanoylphorbol Acetate; Transfection | 1998 |
Extracellular HIV-1 Tat protein induces the rapid Ser133 phosphorylation and activation of CREB transcription factor in both Jurkat lymphoblastoid T cells and primary peripheral blood mononuclear cells.
Topics: Base Sequence; Binding Sites; Calcium-Calmodulin-Dependent Protein Kinases; Cells, Cultured; Chloramphenicol O-Acetyltransferase; Cyclic AMP Response Element-Binding Protein; DNA; Enzyme Inhibitors; Flavonoids; Gene Products, tat; Genes, Reporter; HIV-1; Humans; Jurkat Cells; Leukocytes, Mononuclear; Phosphorylation; Serine; Signal Transduction; Staurosporine; tat Gene Products, Human Immunodeficiency Virus; Transfection | 1998 |
Role of C-terminal serines in desensitization and phosphorylation of the mouse thromboxane receptor.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Amino Acid Sequence; Animals; Drug Interactions; Drug Resistance; Glomerular Mesangium; Inositol Phosphates; Mice; Mice, Transgenic; Models, Molecular; Molecular Sequence Data; Mutagenesis, Site-Directed; Phorbol 12,13-Dibutyrate; Phosphorylation; Precipitin Tests; Protein Kinase C; Receptors, Thromboxane; Recombinant Proteins; Serine; Staurosporine; Thromboxane A2 | 1998 |
Phosphorylation and activation of p70 S6 kinase by manganese in PC12 cells.
Topics: Animals; Anisomycin; Antibodies; Antibody Specificity; Apoptosis; Binding Sites; Calcium-Calmodulin-Dependent Protein Kinases; Camptothecin; Cisplatin; Cycloheximide; DNA Fragmentation; Enzyme Activation; Immunoblotting; JNK Mitogen-Activated Protein Kinases; Manganese; Mitogen-Activated Protein Kinases; PC12 Cells; Phosphorylation; Protein Processing, Post-Translational; Proto-Oncogene Proteins c-bcl-2; Rats; Ribosomal Protein S6 Kinases; Serine; Staurosporine; Threonine | 1998 |
D-cystathionine ketimine and L-cystathionine ketimine enhance superoxide generation by human neutrophils in a different manner.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Arachidonic Acid; Benzoquinones; Cystathionine; Enzyme Inhibitors; Genistein; Humans; Lactams, Macrocyclic; N-Formylmethionine Leucyl-Phenylalanine; Neutrophil Activation; Neutrophils; Phosphorylation; Protein-Tyrosine Kinases; Quinones; Rifabutin; Serine; Staurosporine; Stereoisomerism; Superoxides; Tetradecanoylphorbol Acetate; Tyrosine | 1999 |
Phosphorylation-induced rearrangement of the histone H3 NH2-terminal domain during mitotic chromosome condensation.
Topics: Anaphase; Antibodies, Monoclonal; Breast Neoplasms; Cell Cycle; Chromosomes, Human; Female; Histones; Humans; Interphase; Metaphase; Mitosis; Phosphorylation; Prophase; Protamine Kinase; Serine; Spermine; Staurosporine; Telophase; Tumor Cells, Cultured | 1999 |
Regulation of phosphorylation level and distribution of PTP36, a putative protein tyrosine phosphatase, by cell-substrate adhesion.
Topics: Animals; Base Sequence; Cell Adhesion; DNA Primers; Enzyme Inhibitors; Female; Mice; Phosphorylation; Protein Tyrosine Phosphatases; Protein Tyrosine Phosphatases, Non-Receptor; Rats; Rats, Inbred Lew; Serine; Staurosporine; Substrate Specificity | 1999 |
Inhibition of protein phosphatase 2A induces serine/threonine phosphorylation, subcellular redistribution, and functional inhibition of STAT3.
Topics: Calcineurin Inhibitors; CD4-Positive T-Lymphocytes; Cell Nucleus; Cyclosporine; Cytoplasm; DNA-Binding Proteins; Enzyme Inhibitors; Humans; Marine Toxins; Microscopy, Confocal; Oxazoles; Phosphoprotein Phosphatases; Phosphorylation; Protein Phosphatase 2; Serine; Signal Transduction; STAT3 Transcription Factor; Staurosporine; Threonine; Trans-Activators; Tumor Cells, Cultured | 1999 |
Serine 19 of human 6-pyruvoyltetrahydropterin synthase is phosphorylated by cGMP protein kinase II.
Topics: Alkaloids; Amino Acid Metabolism, Inborn Errors; Amino Acid Sequence; Animals; Carbazoles; Consensus Sequence; COS Cells; Cyclic GMP-Dependent Protein Kinase Type II; Cyclic GMP-Dependent Protein Kinases; Fibroblasts; Humans; Indoles; Mice; Mice, Knockout; Molecular Sequence Data; Mutation; Phosphorus-Oxygen Lyases; Phosphorylation; Protein Serine-Threonine Kinases; Recombinant Proteins; Serine; Skin; Staurosporine | 1999 |
The Chk1 protein kinase and the Cdc25C regulatory pathways are targets of the anticancer agent UCN-01.
Topics: Alkaloids; Antineoplastic Agents; cdc25 Phosphatases; Cell Cycle Proteins; Checkpoint Kinase 1; Checkpoint Kinase 2; Cloning, Molecular; DNA Damage; Dose-Response Relationship, Radiation; G2 Phase; HeLa Cells; Humans; Membrane Proteins; Models, Biological; Phosphorylation; Plasmids; Protein Kinase Inhibitors; Protein Kinases; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Serine; Staurosporine; Time Factors | 2000 |
Serine phosphorylation of p60 tumor necrosis factor receptor by PKC-delta in TNF-alpha-activated neutrophils.
Topics: Acetophenones; Benzopyrans; Down-Regulation; Enzyme Inhibitors; Humans; Isoenzymes; Neutrophil Activation; Neutrophils; Pancreatic Elastase; Phosphorylation; Protein Kinase C; Protein Kinase C-delta; Receptors, Tumor Necrosis Factor; Serine; Signal Transduction; Staurosporine; Tumor Necrosis Factor-alpha | 2000 |
Phosphorylation down-regulates the RNA binding function of the coat protein of potato virus A.
Topics: Binding, Competitive; Cadmium; Calcium; Capsid; Dose-Response Relationship, Drug; Down-Regulation; Electrophoresis, Gel, Two-Dimensional; Electrophoresis, Polyacrylamide Gel; Enzyme Inhibitors; Immunoblotting; Kinetics; Magnesium; Magnetics; Manganese; Nicotiana; Phosphorylation; Plant Viruses; Plants, Toxic; Plasmids; Recombinant Fusion Proteins; RNA; RNA-Binding Proteins; Serine; Staurosporine; Threonine; Tobacco Mosaic Virus; Trypsin; Zinc | 2001 |
Phosphorylation of a conserved integrin alpha 3 QPSXXE motif regulates signaling, motility, and cytoskeletal engagement.
Topics: Alkaloids; Amino Acid Motifs; Amino Acid Sequence; Animals; Antigens, CD; Benzophenanthridines; Cell Adhesion Molecules; Cell Movement; CHO Cells; Conserved Sequence; Cricetinae; Cricetulus; Cyclic AMP-Dependent Protein Kinases; Cytoskeleton; Enzyme Inhibitors; Genistein; Integrin alpha3; Integrins; Kalinin; Mass Spectrometry; Molecular Sequence Data; Mutagenesis; Phenanthridines; Phosphorylation; Protein Kinase C; Protein-Tyrosine Kinases; Serine; Signal Transduction; Staurosporine | 2001 |
Gab1 phosphorylation: a novel mechanism for negative regulation of HGF receptor signaling.
Topics: Adaptor Proteins, Signal Transducing; Animals; Cell Communication; Cells, Cultured; Enzyme Activation; Enzyme Inhibitors; Female; Hepatocyte Growth Factor; Humans; Isoenzymes; Okadaic Acid; Phosphoprotein Phosphatases; Phosphoproteins; Phosphorylation; Protein Kinase C; Protein Kinase C beta; Protein Kinase C-alpha; Proto-Oncogene Proteins c-met; Serine; Signal Transduction; src Homology Domains; Staurosporine; Threonine | 2001 |
The CEACAM1-L Ser503 residue is crucial for inhibition of colon cancer cell tumorigenicity.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Amino Acid Sequence; Animals; Antigens, CD; Antigens, Differentiation; Calcium-Calmodulin-Dependent Protein Kinases; Carcinoembryonic Antigen; Carcinogenicity Tests; Carcinoma; Cell Adhesion Molecules; Colonic Neoplasms; Cyclic AMP; Enzyme Inhibitors; Epithelial Cells; Female; Humans; Mice; Mice, Inbred BALB C; Molecular Sequence Data; Naphthalenes; Point Mutation; Protein Kinase C; Serine; Staurosporine; Tetradecanoylphorbol Acetate; Thionucleotides; Tumor Cells, Cultured | 2001 |
Tyrosine kinase-mediated serine phosphorylation of adenylyl cyclase.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Amino Acid Sequence; Animals; Blotting, Western; Catalytic Domain; Cells, Cultured; Cyclic AMP; Enzyme Activation; Enzyme Inhibitors; Humans; Intracellular Fluid; Isoenzymes; Molecular Sequence Data; Mutagenesis, Site-Directed; Phosphoamino Acids; Phosphorylation; Protein-Tyrosine Kinases; Proto-Oncogene Proteins c-raf; Rats; Serine; Staurosporine; Tyrosine; Up-Regulation; Vanadates | 2001 |
Insulin-stimulated protein kinase B phosphorylation on Ser-473 is independent of its activity and occurs through a staurosporine-insensitive kinase.
Topics: Animals; Cell Line; Enzyme Activation; Insulin; Phosphorylation; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Serine; Signal Transduction; Staurosporine | 2001 |
Nongenomic antiapoptotic signal transduction by estrogen in cultured cortical neurons.
Topics: Alzheimer Disease; Animals; Apoptosis; Cells, Cultured; Cerebral Cortex; Cyclic AMP Response Element-Binding Protein; Enzyme Inhibitors; Estradiol; Estrogen Replacement Therapy; Fetus; Glutamic Acid; Menopause; Nerve Degeneration; Neurons; Neuroprotective Agents; Phosphatidylinositol 3-Kinases; Phosphorylation; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Proto-Oncogene Proteins c-bcl-2; Rats; Rats, Sprague-Dawley; Serine; Signal Transduction; Staurosporine | 2001 |
Proapoptotic stimuli induce nuclear accumulation of glycogen synthase kinase-3 beta.
Topics: Apoptosis Inducing Factor; Calcium-Calmodulin-Dependent Protein Kinases; Cell Nucleus; Cyclin D1; Enzyme Inhibitors; Flavoproteins; Glycogen Synthase Kinase 3; Glycogen Synthase Kinases; Hot Temperature; Humans; Lithium; Membrane Proteins; Phosphorylation; Serine; Staurosporine; Tumor Cells, Cultured; Tyrosine | 2001 |
Phosphorylation of native and heme-modified CYP3A4 by protein kinase C: a mass spectrometric characterization of the phosphorylated peptides.
Topics: Amino Acid Sequence; Amino Acid Substitution; Animals; Chromatography, Liquid; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme System; Cytosol; Enzyme Inhibitors; Heme; Humans; Kinetics; Liver; Mass Spectrometry; Mixed Function Oxygenases; Models, Molecular; Mutagenesis; Okadaic Acid; Peptide Fragments; Phenylalanine; Phosphopeptides; Phosphorylation; Protein Conformation; Protein Kinase C; Protein Structure, Secondary; Rats; Recombinant Proteins; Sequence Deletion; Serine; Staurosporine | 2001 |
The non-ankyrin C terminus of Ikappa Balpha physically interacts with p53 in vivo and dissociates in response to apoptotic stress, hypoxia, DNA damage, and transforming growth factor-beta 1-mediated growth suppression.
Topics: Animals; Ankyrins; Apoptosis; Cell Division; Cell Line; Cell Nucleus; COS Cells; Cytosol; DNA Damage; DNA-Binding Proteins; Dose-Response Relationship, Drug; Down-Regulation; Etoposide; Genes, Dominant; Humans; Hyaluronoglucosaminidase; Hypoxia; I-kappa B Proteins; Liver; Mice; Microscopy, Fluorescence; Mutagenesis, Site-Directed; NF-KappaB Inhibitor alpha; Phosphorylation; Precipitin Tests; Proline; Protein Binding; Protein Structure, Tertiary; Rats; Recombinant Proteins; Serine; Spleen; Staurosporine; Threonine; Time Factors; Transfection; Transforming Growth Factor beta; Transforming Growth Factor beta1; Tumor Cells, Cultured; Tumor Suppressor Protein p53; Ultraviolet Rays | 2002 |
Inhibition of heat-induced phosphorylation of stathmin by the bioflavonoid quercetin.
Topics: Flavonoids; Hot Temperature; Humans; Immunoblotting; Jurkat Cells; Microtubule Proteins; Mitogen-Activated Protein Kinases; Phosphoproteins; Phosphorylation; Quercetin; Serine; Stathmin; Staurosporine | 2002 |
A comparison in normal individuals and sickle cell patients of reduced glutathione precursors and their transport between plasma and red cells.
Topics: Adult; Amino Acid Transport System ASC; Amino Acid Transport System L; Anemia, Sickle Cell; Biological Transport; Carbon Monoxide; Cysteine; Enzyme Inhibitors; Erythrocytes; Female; Glutamic Acid; Glutamine; Glutathione; Glycine; Humans; Male; Middle Aged; Oxygen; Protein Kinase Inhibitors; Protein Kinases; Serine; Staurosporine | 2000 |
Characterization of PDK2 activity against protein kinase B gamma.
Topics: 3-Phosphoinositide-Dependent Protein Kinases; 3T3 Cells; Animals; COS Cells; Enzyme Inhibitors; Humans; Isoenzymes; Mice; Oncogene Proteins; Phosphorylation; Precipitin Tests; Protein Binding; Protein Kinase C; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins c-akt; Serine; Staurosporine; Transfection; Two-Hybrid System Techniques | 2002 |
A functional role for nicotine in Bcl2 phosphorylation and suppression of apoptosis.
Topics: Antineoplastic Agents; Apoptosis; Cell Survival; Drug Resistance, Neoplasm; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Humans; Mitogen-Activated Protein Kinases; Nicotine; Phosphorylation; Proto-Oncogene Proteins c-bcl-2; Serine; Staurosporine; Tumor Cells, Cultured; Type C Phospholipases | 2003 |
Calyculin A-induced actin phosphorylation and depolymerization in renal epithelial cells.
Topics: Actin Cytoskeleton; Adenosine Triphosphate; Animals; Cell Line; Enzyme Inhibitors; Epithelial Cells; Kidney Tubules, Proximal; Marine Toxins; Oxazoles; Phosphoprotein Phosphatases; Phosphorylation; Polymers; Protein Serine-Threonine Kinases; Serine; Staurosporine | 2003 |
Adhesion-associated and PKC-modulated changes in serine/threonine phosphorylation of p120-catenin.
Topics: 3T3 Cells; Amino Acid Sequence; Animals; Catenins; Cell Adhesion; Cell Adhesion Molecules; Cell Membrane Permeability; Conserved Sequence; Delta Catenin; Enzyme Activation; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Humans; Mice; Models, Biological; Molecular Sequence Data; Mutagenesis, Site-Directed; Phosphoamino Acids; Phosphoproteins; Phosphorylation; Protein Kinase C; Serine; Signal Transduction; Species Specificity; Staurosporine; Substrate Specificity; Threonine; Tumor Cells, Cultured | 2003 |
Phosphorylation of Nrf2 at Ser40 by protein kinase C in response to antioxidants leads to the release of Nrf2 from INrf2, but is not required for Nrf2 stabilization/accumulation in the nucleus and transcriptional activation of antioxidant response element
Topics: Antioxidants; Binding Sites; Blotting, Western; Cell Line; Cell Nucleus; DNA-Binding Proteins; Enzyme Inhibitors; Fluorescent Antibody Technique; Gene Expression; Humans; Immunosorbent Techniques; Leucine Zippers; Mutagenesis, Site-Directed; NAD(P)H Dehydrogenase (Quinone); Naphthalenes; NF-E2-Related Factor 2; Phosphorylation; Protein Kinase C; Response Elements; Serine; Staurosporine; Structure-Activity Relationship; Trans-Activators; Transcription, Genetic; Transfection | 2003 |
Characterization of the protein kinase activity of TRPM7/ChaK1, a protein kinase fused to the transient receptor potential ion channel.
Topics: Acetophenones; Benzopyrans; Calcium; Calmodulin; Catalytic Domain; Cations; Chromatography, Gel; Cobalt; DNA; Dose-Response Relationship, Drug; Electrophoresis, Polyacrylamide Gel; Electrophysiology; Enzyme Inhibitors; Escherichia coli; HeLa Cells; Histones; Humans; Ion Channels; Ions; Kinetics; Magnesium; Membrane Proteins; Molecular Sequence Data; Myelin Basic Protein; Phosphoamino Acids; Phosphorylation; Protein Kinases; Protein Serine-Threonine Kinases; Protein Structure, Tertiary; Serine; Staurosporine; Threonine; Time Factors; TRPM Cation Channels; Zinc | 2004 |
Clathrin-mediated endocytosis of Na+,K+-ATPase in response to parathyroid hormone requires ERK-dependent phosphorylation of Ser-11 within the alpha1-subunit.
Topics: Alanine; Animals; Butadienes; Cattle; Cell Membrane; Clathrin; DNA, Complementary; Endocytosis; Endosomes; Kidney; Mitogen-Activated Protein Kinases; Mutation; Nitriles; Opossums; Parathyroid Hormone; Phosphorylation; Precipitin Tests; Protein Kinase C; Protein Structure, Tertiary; Protein Transport; Rats; Serine; Sodium-Potassium-Exchanging ATPase; Staurosporine; Time Factors; Transfection | 2004 |
7-hydroxystaurosporine (UCN-01) inhibition of Akt Thr308 but not Ser473 phosphorylation: a basis for decreased insulin-stimulated glucose transport.
Topics: Adipose Tissue; Animals; Antineoplastic Agents; Biological Transport; Blotting, Western; Cell Membrane; Cytosol; Dose-Response Relationship, Drug; Enzyme Activation; Glucose; Glucose Transporter Type 4; Immunoblotting; Insulin; Male; Microsomes; Monosaccharide Transport Proteins; Muscle Proteins; Phosphorylation; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Rats; Serine; Staurosporine; Subcellular Fractions; Threonine | 2004 |
Phosphorylation of Plk1 at S137 and T210 is inhibited in response to DNA damage.
Topics: Ataxia Telangiectasia Mutated Proteins; Caffeine; CDC2 Protein Kinase; cdc25 Phosphatases; Cell Cycle Proteins; Cell Division; Cell Line, Tumor; Checkpoint Kinase 1; Checkpoint Kinase 2; Cyclin B; DNA Damage; DNA-Binding Proteins; Doxorubicin; Enzyme Activation; G2 Phase; Humans; Mitosis; Nocodazole; Phosphorylation; Polo-Like Kinase 1; Protein Kinases; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Serine; Signal Transduction; Staurosporine; Threonine; Tumor Suppressor Proteins | 2005 |
Protein kinase D specifically mediates apoptosis signal-regulating kinase 1-JNK signaling induced by H2O2 but not tumor necrosis factor.
Topics: 14-3-3 Proteins; Animals; Apoptosis; Blotting, Western; Carbazoles; Cattle; Cysteine; Cytoplasm; Dose-Response Relationship, Drug; Endothelium, Vascular; Humans; Hydrogen Peroxide; Indoles; JNK Mitogen-Activated Protein Kinases; Maleimides; MAP Kinase Kinase Kinase 5; Models, Biological; Naphthalenes; Phosphorylation; Protein Binding; Protein Isoforms; Protein Kinase C; Protein Structure, Tertiary; RNA, Small Interfering; Serine; Signal Transduction; Staurosporine; Time Factors; Transfection; Tumor Necrosis Factor-alpha; Umbilical Veins | 2005 |
WOX1 is essential for tumor necrosis factor-, UV light-, staurosporine-, and p53-mediated cell death, and its tyrosine 33-phosphorylated form binds and stabilizes serine 46-phosphorylated p53.
Topics: Active Transport, Cell Nucleus; Animals; Anisomycin; Cell Line, Tumor; Cell Nucleus; Cytoplasm; Cytosol; DNA, Complementary; Dose-Response Relationship, Drug; Etoposide; Fibroblasts; Genes, Dominant; Humans; Hypoxia; Imidazoles; Immunoprecipitation; Luminescent Proteins; Mice; Microscopy, Fluorescence; Models, Biological; Oxidoreductases; Phosphorylation; Piperazines; Proteasome Endopeptidase Complex; Protein Binding; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Serine; Staurosporine; Time Factors; Tumor Necrosis Factor-alpha; Tumor Suppressor Protein p53; Tumor Suppressor Proteins; Two-Hybrid System Techniques; Tyrosine; U937 Cells; Ultraviolet Rays; WW Domain-Containing Oxidoreductase | 2005 |
MPS-1 is a K+ channel beta-subunit and a serine/threonine kinase.
Topics: Amino Acid Motifs; Animals; Blotting, Western; Caenorhabditis elegans Proteins; CHO Cells; Cloning, Molecular; Cricetinae; Cricetulus; Dose-Response Relationship, Drug; Electric Stimulation; Enzyme Inhibitors; Humans; Immunoprecipitation; Ion Channel Gating; Membrane Potentials; Myelin Basic Protein; Patch-Clamp Techniques; Phosphorylation; Potassium Channels; Probability; Protein Serine-Threonine Kinases; Protein Subunits; Serine; Staurosporine; Time Factors; Transfection | 2005 |
Akt kinase phosphorylation of inositol 1,4,5-trisphosphate receptors.
Topics: Alanine; Amino Acid Motifs; Amino Acid Sequence; Animals; Apoptosis; Calcium; Calcium Channels; Calcium-Transporting ATPases; Caspase 3; Caspases; Cell Line; Chlorocebus aethiops; CHO Cells; Chromones; COS Cells; Cricetinae; Detergents; DNA, Complementary; Enzyme Activation; Glutamic Acid; Humans; Immunoprecipitation; Inositol 1,4,5-Trisphosphate Receptors; Microcirculation; Molecular Sequence Data; Morpholines; Octoxynol; Phosphatidylinositol 3-Kinases; Phosphorylation; Proto-Oncogene Proteins c-akt; Receptors, Cytoplasmic and Nuclear; Sarcoplasmic Reticulum Calcium-Transporting ATPases; Serine; Staurosporine; Time Factors; Transfection | 2006 |
DOCA-induced phosphorylation of glycogen synthase kinase 3beta.
Topics: Animals; Blotting, Western; Cell Line; Densitometry; Desoxycorticosterone; Enzyme Inhibitors; Glycogen Synthase Kinase 3; Humans; Mice; Mice, Knockout; Myocardium; Phosphorylation; Proto-Oncogene Proteins c-akt; Serine; Staurosporine; Time Factors | 2006 |
Silencing the constitutive active transcription factor CREB by the LKB1-SIK signaling cascade.
Topics: Active Transport, Cell Nucleus; Amino Acid Sequence; AMP-Activated Protein Kinases; Animals; Cell Nucleus; Chlorocebus aethiops; COS Cells; Cyclic AMP Response Element-Binding Protein; Cytoplasm; Gene Silencing; HeLa Cells; Humans; Mice; Molecular Sequence Data; Multienzyme Complexes; Phosphorylation; Protein Serine-Threonine Kinases; Rats; Serine; Signal Transduction; Staurosporine; Threonine; Trans-Activators; Transcription Factors; Transcription, Genetic; Tumor Cells, Cultured | 2006 |
Adeno-associated virus 2-mediated gene transfer: role of a cellular serine/threonine protein phosphatase in augmenting transduction efficiency.
Topics: Cell Line; Dependovirus; Gene Expression; Genetic Therapy; Genetic Vectors; Humans; Kidney; Nuclear Proteins; Parvoviridae Infections; Phosphoprotein Phosphatases; Phosphorylation; Serine; Staurosporine; Threonine; Transduction, Genetic; Transgenes | 2007 |
Reversible phosphorylation of Drp1 by cyclic AMP-dependent protein kinase and calcineurin regulates mitochondrial fission and cell death.
Topics: Animals; Apoptosis; Calcineurin; Calcium; Cell Line, Tumor; Chlorocebus aethiops; COS Cells; Cyclic AMP-Dependent Protein Kinases; GTP Phosphohydrolases; Mitochondria; Mitochondrial Proteins; Mutation; Phosphorylation; Rats; Serine; Staurosporine | 2007 |
The FLT3 inhibitor PKC412 exerts differential cell cycle effects on leukemic cells depending on the presence of FLT3 mutations.
Topics: Apoptosis; bcl-Associated Death Protein; CDC2 Protein Kinase; Cell Cycle; Cell Line, Tumor; Cell Proliferation; Cyclin B; Cyclin-Dependent Kinases; fms-Like Tyrosine Kinase 3; Humans; Leukemia, Myeloid, Acute; Mutation; Phosphorylation; Serine; Signal Transduction; Staurosporine; U937 Cells | 2008 |
Role of p53/FAK association and p53Ser46 phosphorylation in staurosporine-mediated apoptosis: wild type versus mutant p53-R175H.
Topics: Amino Acid Substitution; Apoptosis; Caspase 3; Cell Adhesion; Cell Line, Tumor; Cell Nucleus; Drug Resistance, Neoplasm; Enzyme Activation; Enzyme Inhibitors; Fluorescent Antibody Technique, Indirect; Focal Adhesion Kinase 1; Humans; Immunoblotting; Mutation; Phosphorylation; Protein Transport; Serine; Staurosporine; Tumor Suppressor Protein p53 | 2009 |
PDK1 regulates chemotaxis in human neutrophils.
Topics: 3-Phosphoinositide-Dependent Protein Kinases; Aggressive Periodontitis; Blotting, Western; Cells, Cultured; Chemotaxis, Leukocyte; Enzyme Activation; Enzyme Inhibitors; Gene Expression Regulation, Enzymologic; Gene Silencing; Humans; Neutrophils; Phosphatidylinositol 3-Kinases; Phosphorylation; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins c-akt; RNA, Small Interfering; Serine; Signal Transduction; Staurosporine; Superoxides; Temperature; Threonine; Time Factors | 2009 |
Golgi apparatus casein kinase phosphorylates bioactive Ser-6 of bone morphogenetic protein 15 and growth and differentiation factor 9.
Topics: Animals; Bone Morphogenetic Protein 15; Casein Kinases; Catalysis; Electrophoresis, Polyacrylamide Gel; Female; Golgi Apparatus; Growth Differentiation Factor 9; Humans; Kinetics; Mammary Glands, Animal; Mass Spectrometry; Phosphorylation; Rats; Recombinant Proteins; Serine; Staurosporine | 2010 |
Phosphorylated hMSH6: DNA mismatch versus DNA damage recognition.
Topics: Amino Acid Sequence; Animals; Base Pair Mismatch; Cell Line; Cell Line, Tumor; DNA; DNA Damage; DNA Mismatch Repair; DNA-Binding Proteins; Electrophoretic Mobility Shift Assay; HeLa Cells; Humans; Immunoblotting; Mice; Molecular Sequence Data; Mutation; NIH 3T3 Cells; Phosphorylation; Protein Binding; Protein Kinase Inhibitors; Serine; Signal Transduction; Spodoptera; Staurosporine | 2011 |
Attenuation of the lysosomal death pathway by lysosomal cholesterol accumulation.
Topics: Amides; Androstenes; Animals; Autophagy; bcl-X Protein; Cell Death; Cell Survival; CHO Cells; Cholesterol; Cisplatin; Cricetinae; Cricetulus; Cytoprotection; Fibroblasts; HSP70 Heat-Shock Proteins; Humans; Lysosomes; Membrane Glycoproteins; Myeloid Cell Leukemia Sequence 1 Protein; Protective Agents; Protein Transport; Proto-Oncogene Proteins c-bcl-2; Serine; Signal Transduction; Staurosporine | 2011 |
Phosphorylation of Ser45 and Ser59 of αB-crystallin and p38/extracellular regulated kinase activity determine αB-crystallin-mediated protection of rat brain astrocytes from C2-ceramide- and staurosporine-induced cell death.
Topics: alpha-Crystallin B Chain; Animals; Astrocytes; Blotting, Western; Cell Death; Cell Survival; Cells, Cultured; Down-Regulation; Extracellular Signal-Regulated MAP Kinases; JNK Mitogen-Activated Protein Kinases; Neuroprotective Agents; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Rats; Receptor, PAR-2; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Serine; Sphingosine; Staurosporine | 2011 |
Elevated MARK2-dependent phosphorylation of Tau in Alzheimer's disease.
Topics: Aged; Aged, 80 and over; Alzheimer Disease; Animals; Brain; Cell Line, Transformed; Enzyme Inhibitors; Female; Green Fluorescent Proteins; Humans; Male; Mice; Middle Aged; Phosphorylation; Protein Serine-Threonine Kinases; Serine; Staurosporine; tau Proteins; Transfection | 2013 |