Page last updated: 2024-08-23

staurosporine and rifampin

staurosporine has been researched along with rifampin in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (25.00)29.6817
2010's9 (75.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Langsley, G; Lizundia, R; Ralph, SA; Werling, D1
Franzblau, SG; Guo, S; Kozikowski, AP; Mesecar, AD; Mo, S; Orjala, J; Pegan, SD; Tipparaju, SK; Wan, B1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Bloomer, WD; Kaiser, M; Papadopoulou, MV; Rosenzweig, HS1
Bloomer, WD; Papadopoulou, MV; Rosenzweig, HS1
Ansari, I; Jadhav, H; Patel, H; Pawara, R; Surana, S1
Bermudez, LE; Danelishvili, L; Li, YJ; McGarvey, J1
Dutreix, C; Lorenzo, S; Munarini, F; Roesel, J; Wang, Y1
Dutreix, C; Lorenzo, S; Wang, Y1
Chun, DY; Dutreix, C; Einolf, HJ; Gu, H; He, H; Ouatas, T; Rebello, S; Wang, L1

Trials

2 trial(s) available for staurosporine and rifampin

ArticleYear
Investigation into CYP3A4-mediated drug-drug interactions on midostaurin in healthy volunteers.
    Cancer chemotherapy and pharmacology, 2013, Volume: 72, Issue:6

    Topics: Adult; Antineoplastic Agents; Chromatography, Liquid; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inhibitors; Drug Administration Schedule; Drug Interactions; Enzyme Induction; Enzyme Inhibitors; Female; Humans; Ketoconazole; Male; Midazolam; Middle Aged; Rifampin; Staurosporine; Tandem Mass Spectrometry; Young Adult

2013
Comparison of two endogenous biomarkers of CYP3A4 activity in a drug-drug interaction study between midostaurin and rifampicin.
    European journal of clinical pharmacology, 2014, Volume: 70, Issue:8

    Topics: Adult; Biomarkers; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inducers; Drug Interactions; Female; Humans; Hydrocortisone; Hydroxycholesterols; Male; Middle Aged; Protein Kinase Inhibitors; Rifampin; Staurosporine; Young Adult

2014

Other Studies

10 other study(ies) available for staurosporine and rifampin

ArticleYear
Theileria apicoplast as a target for chemotherapy.
    Antimicrobial agents and chemotherapy, 2009, Volume: 53, Issue:3

    Topics: Animals; Antiprotozoal Agents; Cattle; Drug Delivery Systems; Inhibitory Concentration 50; Models, Biological; Plastids; Theileria; Theileriasis

2009
Natural product leads for drug discovery: isolation, synthesis and biological evaluation of 6-cyano-5-methoxyindolo[2,3-a]carbazole based ligands as antibacterial agents.
    Bioorganic & medicinal chemistry, 2009, Oct-15, Volume: 17, Issue:20

    Topics: Anti-Bacterial Agents; Bacillus anthracis; Biological Products; Carbazoles; Drug Discovery; Drug Evaluation, Preclinical; Ligands; Microbial Sensitivity Tests; Mycobacterium tuberculosis

2009
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
The antitrypanosomal and antitubercular activity of some nitro(triazole/imidazole)-based aromatic amines.
    European journal of medicinal chemistry, 2017, Sep-29, Volume: 138

    Topics: Amines; Antitubercular Agents; Dose-Response Relationship, Drug; Imidazoles; Microbial Sensitivity Tests; Molecular Structure; Mycobacterium tuberculosis; Nitro Compounds; Parasitic Sensitivity Tests; Structure-Activity Relationship; Triazoles; Trypanocidal Agents; Trypanosoma brucei rhodesiense; Trypanosoma cruzi

2017
The antitubercular activity of various nitro(triazole/imidazole)-based compounds.
    Bioorganic & medicinal chemistry, 2017, 11-01, Volume: 25, Issue:21

    Topics: Animals; Antitubercular Agents; Cell Line; Chlorocebus aethiops; Dose-Response Relationship, Drug; Humans; Imidazoles; Macrophages; Mice; Microbial Sensitivity Tests; Molecular Structure; Mycobacterium tuberculosis; Nitro Compounds; Structure-Activity Relationship; Triazoles

2017
Pyridine and nitro-phenyl linked 1,3,4-thiadiazoles as MDR-TB inhibitors.
    European journal of medicinal chemistry, 2019, Apr-01, Volume: 167

    Topics: Animals; Antitubercular Agents; Chlorocebus aethiops; Microbial Sensitivity Tests; Mycobacterium tuberculosis; Nitrophenols; Pyridines; Structure-Activity Relationship; Thiadiazoles; Tuberculosis, Multidrug-Resistant; Vero Cells

2019
Mycobacterium tuberculosis infection causes different levels of apoptosis and necrosis in human macrophages and alveolar epithelial cells.
    Cellular microbiology, 2003, Volume: 5, Issue:9

    Topics: Antibiotics, Antitubercular; Apoptosis; bcl-Associated Death Protein; Carrier Proteins; Cell Line; Enzyme Inhibitors; Epithelial Cells; Gene Expression Regulation; Humans; In Situ Nick-End Labeling; Macrophages; Mycobacterium tuberculosis; Necrosis; Oligonucleotide Array Sequence Analysis; Proto-Oncogene Proteins c-bcl-2; Pulmonary Alveoli; Rifampin; Staurosporine

2003
Simultaneous Physiologically Based Pharmacokinetic (PBPK) Modeling of Parent and Active Metabolites to Investigate Complex CYP3A4 Drug-Drug Interaction Potential: A Case Example of Midostaurin.
    Drug metabolism and disposition: the biological fate of chemicals, 2018, Volume: 46, Issue:2

    Topics: Adult; Biomarkers; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inducers; Cytochrome P-450 CYP3A Inhibitors; Drug Interactions; Female; Humans; Hydroxycholesterols; Ketoconazole; Male; Midazolam; Middle Aged; Models, Biological; Rifampin; Staurosporine; Young Adult

2018