Page last updated: 2024-08-23

staurosporine and lavendustin a

staurosporine has been researched along with lavendustin a in 19 studies

Research

Studies (19)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's12 (63.16)18.2507
2000's6 (31.58)29.6817
2010's0 (0.00)24.3611
2020's1 (5.26)2.80

Authors

AuthorsStudies
Chang, CJ; Geahlen, RL1
Bullock, AN; Fedorov, O; Knapp, S; Marsden, B; Müller, S; Pogacic, V; Rellos, P; Schwaller, J; Sundström, M1
Chrest, FJ; Gabrielson, EW; Lin, Y1
Toi, M; Umezaza, K1
Chang, NS1
Alam, J; Camhi, S; Choi, AM1
Abe, K; Aoyagi, A; Nishikawa, K; Saito, H1
Bayat-Sarmadi, M; Houdebine, LM1
Cherington, V; Corbley, MJ; Lydon, NB; Roberts, TM; Traxler, PM1
Dluzewski, AR; Garcia, CR1
Goretzki, L; Mueller, BM1
Kramer, RH; Molokanova, E; Savchenko, A; Trivedi, B1
Magga, J; Ruskoaho, H; Taskinen, P; Toth, M; Vuolteenaho, O1
Ardenghi, P; Barros, DM; Izquierdo, I; Izquierdo, LA; Medinam, JH; Mello e Souza, T; Rodrigues, C; Sant'Anna, MK; Vianna, M1
Boxall, AR1
Bödding, M1
Kurihara, K; Moore-Hoon, ML; Nakanishi, N; Turner, RJ1
Jebe, E; Petrunkina, AM; Töpfer-Petersen, E1
Cai, J; Chen, J; Guo, C; Jiang, LL; Li, X; Liu, HB; Pu, W; Wang, L; Wu, D; Yang, A; Yu, F; Zhang, X1

Reviews

1 review(s) available for staurosporine and lavendustin a

ArticleYear
Protein-tyrosine kinase inhibition: mechanism-based discovery of antitumor agents.
    Journal of natural products, 1992, Volume: 55, Issue:11

    Topics: Animals; Antineoplastic Agents; Drug Screening Assays, Antitumor; Humans; Protein-Tyrosine Kinases

1992

Other Studies

18 other study(ies) available for staurosporine and lavendustin a

ArticleYear
A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.
    Proceedings of the National Academy of Sciences of the United States of America, 2007, Dec-18, Volume: 104, Issue:51

    Topics: Amino Acid Sequence; Binding Sites; Clinical Trials as Topic; Drug Evaluation, Preclinical; Enzyme Stability; Humans; Molecular Sequence Data; Phylogeny; Protein Array Analysis; Protein Conformation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases

2007
Reversible G1 arrest of a human lung epithelial cell line by staurosporine.
    Journal of cellular physiology, 1992, Volume: 152, Issue:3

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Cell Division; Cell Line; DNA; Dose-Response Relationship, Drug; G1 Phase; Genistein; Humans; Isoflavones; Isoquinolines; Phenols; Piperazines; Protein Kinase C; Staurosporine; Sulfonamides

1992
[Inhibitors of growth factor functions, possible antineoplastic agents].
    Tanpakushitsu kakusan koso. Protein, nucleic acid, enzyme, 1991, Volume: 36, Issue:7

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Actinomyces; Alkaloids; Animals; Antineoplastic Agents, Phytogenic; Genistein; Isoflavones; Isoquinolines; Mice; Phenols; Phosphatidylinositols; Piperazines; Protein Kinase C; Protein-Tyrosine Kinases; Staurosporine

1991
Transforming growth factor-beta 1 induction of novel extracellular matrix proteins that trigger resistance to tumor necrosis factor cytotoxicity in murine L929 fibroblasts.
    The Journal of biological chemistry, 1995, Mar-31, Volume: 270, Issue:13

    Topics: Alkaloids; Animals; Catechols; Cell Survival; Dose-Response Relationship, Drug; Extracellular Matrix Proteins; Fibroblasts; Genistein; Isoflavones; Kinetics; L Cells; Mice; Nitriles; Phenols; Phosphotyrosine; Protein Kinase Inhibitors; Staurosporine; Transforming Growth Factor beta; Tumor Protein, Translationally-Controlled 1; Tyrosine; Tyrphostins

1995
Identification of a second region upstream of the mouse heme oxygenase-1 gene that functions as a basal level and inducer-dependent transcription enhancer.
    The Journal of biological chemistry, 1995, May-19, Volume: 270, Issue:20

    Topics: Acetylcysteine; Alkaloids; Animals; Base Sequence; Binding Sites; Consensus Sequence; DNA-Binding Proteins; Enhancer Elements, Genetic; Enzyme Induction; Genes; Genistein; Heme Oxygenase (Decyclizing); Isoflavones; L Cells; Mice; Molecular Sequence Data; Mutagenesis, Site-Directed; Naphthalenes; Nuclear Proteins; Phenols; Polycyclic Compounds; Protein Kinase Inhibitors; Rats; Recombinant Fusion Proteins; Repetitive Sequences, Nucleic Acid; Staurosporine; Transcription Factor AP-1; Transcription Factors; Transcription, Genetic; Tumor Cells, Cultured

1995
Characterization of basic fibroblast growth factor-mediated acceleration of axonal branching in cultured rat hippocampal neurons.
    Brain research, 1994, Oct-24, Volume: 661, Issue:1-2

    Topics: Alkaloids; Animals; Antibodies; Axons; Benzoquinones; Cells, Cultured; Dendrites; Dose-Response Relationship, Drug; Embryo, Mammalian; Fibroblast Growth Factor 2; Hippocampus; Humans; Lactams, Macrocyclic; Neurites; Neurons; Phenols; Polysaccharide-Lyases; Protein Kinase C; Protein-Tyrosine Kinases; Quinones; Rats; Rats, Wistar; Recombinant Proteins; Rifabutin; Staurosporine; Tetradecanoylphorbol Acetate; Time Factors

1994
Effect of various protein kinase inhibitors on the induction of milk protein gene expression by prolactin.
    Molecular and cellular endocrinology, 1993, Volume: 92, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenine; Alkaloids; Animals; Cells, Cultured; Epithelial Cells; Epithelium; Female; Gene Expression Regulation; Genistein; Isoflavones; Isoquinolines; Mammary Glands, Animal; Milk Proteins; Phenols; Phenylacetates; Piperazines; Polymyxin B; Pregnancy; Prolactin; Protein Kinase Inhibitors; Quercetin; Rabbits; Sphingosine; Staurosporine; Succinates

1993
A strategy for screening anti-tumor drugs utilizing oncogenes encoded in retroviral vectors.
    International journal of cancer, 1996, Jun-11, Volume: 66, Issue:6

    Topics: 3T3 Cells; Alkaloids; Animals; Antigens, Polyomavirus Transforming; Benzamides; Cell Division; Drug Screening Assays, Antitumor; Enzyme Inhibitors; Ethers, Cyclic; Genes, ras; Genes, src; Genetic Vectors; Hydroquinones; Mice; Okadaic Acid; Oncogenes; Phenols; Protein Kinase C; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-raf; Retroviridae; Signal Transduction; Staurosporine; Styrenes; Sulfones; Thiazoles

1996
Inhibition of invasion and intraerythrocytic development of Plasmodium falciparum by kinase inhibitors.
    Experientia, 1996, Jun-15, Volume: 52, Issue:6

    Topics: Alkaloids; Animals; Antimalarials; Benzylidene Compounds; Cinnamates; Enzyme Inhibitors; Erythrocytes; Ethers, Cyclic; Genistein; Humans; Isoflavones; Nitriles; Okadaic Acid; Phenols; Phosphoric Monoester Hydrolases; Plasmodium falciparum; Protein Kinase Inhibitors; Staurosporine; Tyrphostins

1996
Receptor-mediated endocytosis of urokinase-type plasminogen activator is regulated by cAMP-dependent protein kinase.
    Journal of cell science, 1997, Volume: 110 ( Pt 12)

    Topics: Adenoviruses, Human; Carbazoles; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Endocytosis; Enzyme Inhibitors; Epidermal Growth Factor; Genistein; Humans; Indole Alkaloids; Indoles; Isoflavones; Isoquinolines; Lactoferrin; Low Density Lipoprotein Receptor-Related Protein-1; Maleimides; Melanoma; Naphthalenes; Phenols; Protein Kinase C; Receptors, Immunologic; Signal Transduction; Staurosporine; Sulfonamides; Tumor Cells, Cultured; Urokinase-Type Plasminogen Activator

1997
Modulation of rod photoreceptor cyclic nucleotide-gated channels by tyrosine phosphorylation.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1997, Dec-01, Volume: 17, Issue:23

    Topics: Adenosine Triphosphate; Animals; Cyclic GMP; Enzyme Inhibitors; Eye Proteins; Hydroquinones; Ion Channel Gating; Marine Toxins; Microcystins; Okadaic Acid; Oocytes; Oxazoles; Patch-Clamp Techniques; Peptides, Cyclic; Phenols; Phosphorylation; Protein Processing, Post-Translational; Protein Tyrosine Phosphatases; Rod Cell Outer Segment; Staurosporine; Vanadates; Xenopus laevis

1997
Inhibition of atrial wall stretch-induced cardiac hormone secretion by lavendustin A, a potent tyrosine kinase inhibitor.
    Endocrinology, 1999, Volume: 140, Issue:9

    Topics: Animals; Atrial Function; Atrial Natriuretic Factor; Calcium-Calmodulin-Dependent Protein Kinases; Enzyme Inhibitors; In Vitro Techniques; Male; Myocardium; Myosin-Light-Chain Kinase; Natriuretic Peptide, Brain; Okadaic Acid; Phenols; Physical Stimulation; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Rats; Rats, Sprague-Dawley; Staurosporine

1999
Short- and long-term memory are differentially affected by metabolic inhibitors given into hippocampus and entorhinal cortex.
    Neurobiology of learning and memory, 2000, Volume: 73, Issue:2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Aminoquinolines; Animals; Avoidance Learning; Carbazoles; Entorhinal Cortex; Enzyme Inhibitors; Flavonoids; Guanylate Cyclase; Hippocampus; Indoles; Inhibition, Psychological; Male; Memory; Memory, Short-Term; Phenols; Protein Kinase Inhibitors; Pyrroles; Rats; Rats, Wistar; Sodium Chloride; Staurosporine

2000
GABAergic mIPSCs in rat cerebellar Purkinje cells are modulated by TrkB and mGluR1-mediated stimulation of Src.
    The Journal of physiology, 2000, May-01, Volume: 524 Pt 3

    Topics: Animals; Bicuculline; Brain-Derived Neurotrophic Factor; Enzyme Inhibitors; Evoked Potentials; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; Neural Inhibition; Oligopeptides; Organ Culture Techniques; Phenols; Purkinje Cells; Rats; Receptor, trkB; Receptors, GABA-A; Receptors, Metabotropic Glutamate; Resorcinols; Staurosporine; Synapses; Vanadates

2000
Activation of store-operated Ca2+ entry in RBL cells without the contribution of protein kinases.
    Naunyn-Schmiedeberg's archives of pharmacology, 2001, Volume: 363, Issue:6

    Topics: Animals; Calcium; Enzyme Inhibitors; Leukemia, Basophilic, Acute; Patch-Clamp Techniques; Phenols; Protein Kinase Inhibitors; Protein Kinases; Rats; Staurosporine; Tumor Cells, Cultured

2001
Phosphorylation of the salivary Na(+)-K(+)-2Cl(-) cotransporter.
    American journal of physiology. Cell physiology, 2002, Volume: 282, Issue:4

    Topics: Adenosine Triphosphate; Animals; Carbazoles; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Indole Alkaloids; Indoles; Isoproterenol; Isoquinolines; Maleimides; Marine Toxins; Microcystins; Okadaic Acid; Oxazoles; Parotid Gland; Peptides, Cyclic; Phenols; Phosphorus Radioisotopes; Phosphorylation; Rats; Sodium-Potassium-Chloride Symporters; Solute Carrier Family 12, Member 2; Staurosporine; Sulfonamides; Sympathomimetics; Vanadates

2002
Regulatory and necrotic volume increase in boar spermatozoa.
    Journal of cellular physiology, 2005, Volume: 204, Issue:2

    Topics: Animals; Annexin A5; Cell Size; Chloride Channels; Enzyme Inhibitors; Hypertonic Solutions; Male; Necrosis; Phenols; Phosphoprotein Phosphatases; Phosphorylation; Protein-Tyrosine Kinases; Quinidine; Semen Preservation; Spermatozoa; Staining and Labeling; Staurosporine; Swine; Tamoxifen; Tyrosine; Vanadates

2005
A screening of inhibitors targeting the receptor kinase FERONIA reveals small molecules that enhance plant root immunity.
    Plant biotechnology journal, 2023, Volume: 21, Issue:1

    Topics: Arabidopsis Proteins; Phosphotransferases; Plant Immunity; Plant Roots; Plants; Staurosporine

2023