Page last updated: 2024-08-23

staurosporine and gsk 1363089

staurosporine has been researched along with gsk 1363089 in 5 studies

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's4 (80.00)24.3611
2020's1 (20.00)2.80

Authors

AuthorsStudies
Ciceri, P; Davis, MI; Herrgard, S; Hocker, M; Hunt, JP; Pallares, G; Treiber, DK; Wodicka, LM; Zarrinkar, PP1
Dewhurst, S; Gelbard, HA; Goodfellow, VS; Loweth, CJ; Marker, DF; Nguyen, T; Polesskaya, O; Pollack, S; Ravula, SB; Sheppard, D; Todd, DE; Wiemann, T; Xu, Y1
Bao, G; Du, B; Gong, P; Li, W; Lv, J; Ma, J; Wang, L; Xu, B; Zhai, X1
Berger, BT; Chaikuad, A; Drápela, S; Knapp, S; Maier, L; Němec, V; Paruch, K; Souček, K1
Dixit, SM; Kulju, KD; Polasky, DA; Ruotolo, BT; Vallejo, DD1

Other Studies

5 other study(ies) available for staurosporine and gsk 1363089

ArticleYear
Comprehensive analysis of kinase inhibitor selectivity.
    Nature biotechnology, 2011, Oct-30, Volume: 29, Issue:11

    Topics: Catalysis; Drug Design; Enzyme Stability; High-Throughput Screening Assays; Humans; Protein Binding; Protein Kinase Inhibitors; Protein Kinases; Proteomics; Signal Transduction; Substrate Specificity

2011
Discovery, synthesis, and characterization of an orally bioavailable, brain penetrant inhibitor of mixed lineage kinase 3.
    Journal of medicinal chemistry, 2013, Oct-24, Volume: 56, Issue:20

    Topics: Administration, Oral; Animals; Area Under Curve; Biological Availability; Blood-Brain Barrier; Brain; Carbazoles; Cells, Cultured; Cognition Disorders; Drug Discovery; HIV Infections; Humans; JNK Mitogen-Activated Protein Kinases; Male; MAP Kinase Kinase Kinases; Mice; Mice, Inbred C57BL; Mitogen-Activated Protein Kinase Kinase Kinase 11; Models, Chemical; Molecular Structure; Monocytes; Phosphorylation; Protein Kinase Inhibitors; Pyridines; Pyrroles; tat Gene Products, Human Immunodeficiency Virus; Tumor Necrosis Factor-alpha

2013
Design, synthesis, biological evaluation and preliminary mechanism study of novel benzothiazole derivatives bearing indole-based moiety as potent antitumor agents.
    European journal of medicinal chemistry, 2015, Volume: 96

    Topics: Antineoplastic Agents; Benzothiazoles; Cell Line, Tumor; Cell Proliferation; Dose-Response Relationship, Drug; Drug Design; Drug Screening Assays, Antitumor; Humans; Indoles; Models, Molecular; Molecular Structure; Quantitative Structure-Activity Relationship

2015
Highly selective inhibitors of protein kinases CLK and HIPK with the furo[3,2-b]pyridine core.
    European journal of medicinal chemistry, 2021, Apr-05, Volume: 215

    Topics: Animals; Carrier Proteins; Crystallography, X-Ray; Furans; Humans; MCF-7 Cells; Mice; Molecular Structure; Protein Binding; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Pyridines; Structure-Activity Relationship

2021
An Algorithm for Building Multi-State Classifiers Based on Collision-Induced Unfolding Data.
    Analytical chemistry, 2019, 08-20, Volume: 91, Issue:16

    Topics: Algorithms; Anilides; Dasatinib; Escherichia coli; High-Throughput Screening Assays; Humans; Imidazoles; Immunoglobulin Isotypes; Models, Molecular; Multiple Myeloma; Protein Kinase Inhibitors; Protein Structure, Secondary; Pyridazines; Quinolines; Recombinant Proteins; Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization; src-Family Kinases; Static Electricity; Staurosporine

2019