staurosporine has been researched along with go 6976 in 38 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 8 (21.05) | 18.2507 |
2000's | 23 (60.53) | 29.6817 |
2010's | 7 (18.42) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Goekjian, P; Jochum, A; Jung, M; Kunick, C; Marshall, B; Meier, R; Saunders, L; Sippl, W; Trapp, J; Verdin, E | 1 |
Giranda, VL; Johnson, EF; Luo, Y; Stewart, KD; Woods, KW | 1 |
Bullock, AN; Fedorov, O; Knapp, S; Marsden, B; Müller, S; Pogacic, V; Rellos, P; Schwaller, J; Sundström, M | 1 |
Augustin, M; Davies, SP; Gao, Y; Harvey, KJ; Kovelman, R; Patel, UA; Woodward, A | 1 |
Dickens, G; Guroff, G; Lavarreda, M; Zheng, WH | 1 |
Houghton, PJ; Luo, W; Sharif, M; Sharif, TR | 1 |
Benussi, L; Bianchetti, A; Binetti, G; Gasparini, L; Govoni, S; Racchi, M; Trabucchi, M | 1 |
Alexander, JS; Kevil, CG; Mire, E; Payne, DK | 1 |
Carter, CA; Chambers, T; Parham, GP | 1 |
Chen, J; Chueh, SC; Guh, JH; Hwang, TL; Teng, CM | 1 |
Sharif, M; Sharif, TR | 1 |
Bheekha-Escura, R; Chance, SR; Langdon, JM; MacDonald, SM; MacGlashan, DW | 1 |
Appleyard, SM; Chavkin, C; Pattillo, A; Rogalski, SL; Terman, GW | 1 |
Kataoka, K; Nakamura, Y; Si, Q | 1 |
Chen, H; Fetscher, C; Heusch, G; Michel, MC; Schäfers, RF; Wambach, G | 1 |
Altura, BM; Altura, BT; Li, W; Zheng, T | 1 |
Barman, SA | 1 |
Zawalich, KC; Zawalich, WS | 1 |
Chen, JS; Song, JG | 1 |
Leung, HW; Leung, KN; Lung, HL; Mak, NK; Tsang, HY; Wong, RN | 1 |
Elia, MG; Greco, S; Marsigliante, S; Muscella, A; Salvatore, P; Storelli, C | 1 |
Blomhoff, HK; Myklebust, JH; Rusten, LS; Smeland, EB; Stokke, T | 1 |
Akita, Y; Gutierrez-Hartmann, A; Manning, N; Pickett, CA | 1 |
Bernhardt, R; Bureik, M; Zeeh, A | 1 |
Chain, BM; Cho, JY; Katz, DR | 1 |
Cunningham, FM; Goode, NT; Greenaway, EC; Sepulveda, MF | 1 |
Honda, Y; Kemmochi, S; Miyamoto, N; Oh, H; Ohashi, H; Ojima, T; Sato, Y; Suganami, E; Suzuma, I; Suzuma, K; Takagi, H; Uemura, A; Watanabe, D | 1 |
Altura, BM; Altura, BT; Li, J; Li, W; Liu, W | 1 |
Carpenter, DO; Hussain, RJ | 1 |
Garvin, JL; Hong, NJ; Ortiz, PA; Silva, GB | 1 |
Amiel, S; Asare-Anane, H; Gray, E; Huang, GC; Jones, PM; Muller, D; Persaud, SJ; Squires, PE | 1 |
Namiki, H; Takahashi, H | 1 |
Borda, E; Orman, B; Sterin-Borda, L; Villarruel, EQ | 1 |
Carlson, M; Lampinen, M; Venge, P | 1 |
Potter, LR; Robinson, JW | 1 |
Chan, E; Heffron, TP; La, H; Lee, HJ; Malek, S; Merchant, M; Pirazzoli, V; Politi, K; Schaefer, G; Settleman, J; Shao, L; Sideris, S; Ubhayakar, S; Yauch, RL; Ye, X | 1 |
Cao, HL; Chi, LT; Li, WZ; Wang, Q; Wang, YZ; Yang, WC | 1 |
Kim, BJ; Kim, JN | 1 |
38 other study(ies) available for staurosporine and go 6976
Article | Year |
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Adenosine mimetics as inhibitors of NAD+-dependent histone deacetylases, from kinase to sirtuin inhibition.
Topics: Acetylation; Adenosine; Binding Sites; Cell Line, Tumor; Histone Deacetylase Inhibitors; Histone Deacetylases; Humans; Models, Molecular; Molecular Mimicry; Protein Kinase Inhibitors; Sirtuins; Structure-Activity Relationship; Tubulin | 2006 |
Pharmacological and functional comparison of the polo-like kinase family: insight into inhibitor and substrate specificity.
Topics: Adenosine Triphosphate; Amino Acid Sequence; Androstadienes; Binding Sites; Cell Cycle Proteins; Humans; Models, Molecular; Molecular Sequence Data; Peptide Library; Polo-Like Kinase 1; Protein Conformation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Pteridines; Substrate Specificity; Wortmannin | 2007 |
A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.
Topics: Amino Acid Sequence; Binding Sites; Clinical Trials as Topic; Drug Evaluation, Preclinical; Enzyme Stability; Humans; Molecular Sequence Data; Phylogeny; Protein Array Analysis; Protein Conformation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases | 2007 |
A broad activity screen in support of a chemogenomic map for kinase signalling research and drug discovery.
Topics: Aurora Kinases; Cluster Analysis; Drug Design; Drug Discovery; Drug Evaluation, Preclinical; ErbB Receptors; Humans; Intracellular Signaling Peptides and Proteins; MAP Kinase Kinase 4; p38 Mitogen-Activated Protein Kinases; Protein Kinase Inhibitors; Protein Kinases; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Receptors, Vascular Endothelial Growth Factor; Recombinant Proteins; Reproducibility of Results; Signal Transduction; Small Molecule Libraries; Structure-Activity Relationship; Syk Kinase | 2013 |
Involvement of protein kinase C in nerve growth factor- and K-252a-stimulated calcium uptake into PC12 cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenosine Triphosphate; Animals; Calcium; Calcium Channel Agonists; Carbazoles; Carcinogens; Enzyme Inhibitors; Indole Alkaloids; Indoles; Isoenzymes; Naphthalenes; Nerve Growth Factors; PC12 Cells; Phorbol Esters; Protein Kinase C; Protein Kinase C-alpha; Rats; Receptors, Nerve Growth Factor; Signal Transduction; Staurosporine; Tetradecanoylphorbol Acetate | 1997 |
CGP 41251 and tamoxifen selectively inhibit mitogen-activated protein kinase activation and c-Fos phosphoprotein induction by substance P in human astrocytoma cells.
Topics: Astrocytoma; Calcium-Calmodulin-Dependent Protein Kinases; Carbazoles; Cyclic AMP Response Element-Binding Protein; Enzyme Activation; Enzyme Inhibitors; Humans; Indoles; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase C; Proto-Oncogene Proteins c-fos; Staurosporine; Substance P; Tamoxifen; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured; Tyrosine | 1997 |
Specific role for protein kinase C alpha in the constitutive and regulated secretion of amyloid precursor protein in human skin fibroblasts.
Topics: Aged; Amyloid beta-Protein Precursor; Biopsy; Blotting, Northern; Blotting, Western; Carbazoles; Cells, Cultured; Female; Fibroblasts; Humans; Indoles; Isoenzymes; Male; Middle Aged; Phorbol 12,13-Dibutyrate; Protein Kinase C; Protein Kinase C-alpha; Skin; Staurosporine | 1998 |
Vascular permeability factor/vascular endothelial cell growth factor-mediated permeability occurs through disorganization of endothelial junctional proteins.
Topics: Androstadienes; Antigens, CD; Cadherins; Calcium-Calmodulin-Dependent Protein Kinases; Carbazoles; Cell Membrane Permeability; Endothelial Growth Factors; Endothelium, Vascular; Enzyme Inhibitors; Flavonoids; Histocytochemistry; Humans; Indoles; Lymphokines; Membrane Proteins; Muscle, Smooth, Vascular; Nitriles; Occludin; Phosphoinositide-3 Kinase Inhibitors; Protein Kinase C; Serum Albumin; Staurosporine; Tyrphostins; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors; Wortmannin | 1998 |
Cytoskeletal reorganization induced by retinoic acid treatment of human endometrial adenocarcinoma (RL95-2) cells is correlated with alterations in protein kinase C-alpha.
Topics: Adenocarcinoma; Antineoplastic Agents; Carbazoles; Cell Differentiation; Cytoskeleton; Enzyme Inhibitors; Female; Humans; Immunohistochemistry; Indoles; Isoenzymes; Maleimides; Phenotype; Protein Kinase C; Protein Kinase C-alpha; Staurosporine; Tretinoin; Tumor Cells, Cultured; Uterine Neoplasms | 1998 |
Cell proliferation in human prostatic smooth muscle cells involves the modulation of protein kinase C isozymes.
Topics: Carbazoles; Cell Division; Culture Media; Enzyme Inhibitors; Humans; Indoles; Isoenzymes; Male; Muscle, Smooth; Prostate; Protein Kinase C; Staurosporine; Subcellular Fractions | 1998 |
A high throughput system for the evaluation of protein kinase C inhibitors based on Elk1 transcriptional activation in human astrocytoma cells.
Topics: Antineoplastic Agents; Astrocytoma; Carbazoles; Cell Division; DNA-Binding Proteins; Drug Screening Assays, Antitumor; Enzyme Inhibitors; ets-Domain Protein Elk-1; Humans; Indoles; Potassium Channels; Protein Kinase C; Proto-Oncogene Proteins; Staurosporine; Transcription Factors; Transcriptional Activation; Tumor Cells, Cultured | 1999 |
Pharmacologic regulation of histamine release by the human recombinant histamine-releasing factor.
Topics: Acetophenones; Antibodies, Anti-Idiotypic; Basophils; Benzopyrans; Biomarkers, Tumor; Calcium-Calmodulin-Dependent Protein Kinases; Carbazoles; Enzyme Inhibitors; Histamine Release; Humans; Immunoglobulin E; Indoles; Lymphokines; Pertussis Toxin; Protein Kinase C; Recombinant Proteins; Staurosporine; Tumor Protein, Translationally-Controlled 1; Virulence Factors, Bordetella | 1999 |
TrkB activation by brain-derived neurotrophic factor inhibits the G protein-gated inward rectifier Kir3 by tyrosine phosphorylation of the channel.
Topics: Amino Acid Sequence; Animals; Brain-Derived Neurotrophic Factor; Carbazoles; DNA, Complementary; Dose-Response Relationship, Drug; Electrophysiology; Enzyme Activation; Enzyme Inhibitors; G Protein-Coupled Inwardly-Rectifying Potassium Channels; Genistein; GTP-Binding Proteins; Indole Alkaloids; Indoles; Lysine; Models, Biological; Molecular Sequence Data; Mutation; Oocytes; Phosphorylation; Potassium Channels; Potassium Channels, Inwardly Rectifying; Precipitin Tests; Receptor, trkB; RNA, Messenger; Staurosporine; Tyrosine; Xenopus | 2000 |
Differential regulation of microglial NO production by protein kinase C inhibitors.
Topics: Animals; Carbazoles; Drug Synergism; Enzyme Induction; Enzyme Inhibitors; Indoles; Isoquinolines; Lipopolysaccharides; Microglia; Nerve Tissue Proteins; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Protein Isoforms; Protein Kinase C; Pyrroles; Rats; Signal Transduction; Staurosporine; Sulfonamides; Tetradecanoylphorbol Acetate | 2001 |
Modulation of noradrenaline-induced microvascular constriction by protein kinase inhibitors.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Blood Vessels; Calcium-Calmodulin-Dependent Protein Kinases; Carbazoles; Dose-Response Relationship, Drug; Enzyme Inhibitors; Flavonoids; Genistein; In Vitro Techniques; Indoles; Kidney; Male; Maleimides; Mesentery; Norepinephrine; Protein Kinase C; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Rats; Rats, Sprague-Dawley; Staurosporine; Tyrphostins; Vasoconstriction | 2001 |
Use of protein kinase C inhibitors results in rapid [Mg(2+)](i) mobilization in primary cultured rat aortic smooth muscle cells: are certain kinase C isoforms natural homeostatic regulators of cystolic free Mg(2+).
Topics: Alkaloids; Animals; Aorta; Benzophenanthridines; Carbazoles; Cells, Cultured; Enzyme Inhibitors; Indoles; Magnesium; Maleimides; Muscle, Smooth, Vascular; Naphthalenes; Phenanthridines; Protein Isoforms; Protein Kinase C; Rats; Staurosporine | 2001 |
Effect of protein kinase C inhibition on hypoxic pulmonary vasoconstriction.
Topics: Animals; Calcium Channel Blockers; Calcium Channels, L-Type; Carbazoles; Dogs; Enzyme Inhibitors; Female; Hypoxia; In Vitro Techniques; Indoles; Male; Naphthalenes; Perfusion; Phorbol Esters; Protein Kinase C; Pulmonary Circulation; Staurosporine; Vascular Resistance; Vasoconstriction | 2001 |
Effects of protein kinase C inhibitors on insulin secretory responses from rodent pancreatic islets.
Topics: Animals; Carbachol; Carbazoles; Cholinergic Agonists; Colforsin; Drug Interactions; Enzyme Activation; Enzyme Inhibitors; Glucose; Indoles; Insulin; Insulin Secretion; Islets of Langerhans; Kinetics; Mice; Potassium; Protein Kinase C; Rats; Rats, Sprague-Dawley; Staurosporine; Tetradecanoylphorbol Acetate | 2001 |
Bradykinin induces protein kinase C-dependent activation of phospholipase D in A-431 cells.
Topics: Acetophenones; Benzopyrans; Bradykinin; Carbazoles; Enzyme Activation; Enzyme Inhibitors; Epidermal Growth Factor; Humans; Immunoblotting; Indoles; Isoenzymes; Kinetics; Maleimides; Phospholipase D; Phospholipids; Protein Kinase C; Staurosporine; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 2001 |
Expression of protein kinase C isoforms in euxanthone-induced differentiation of neuroblastoma cells.
Topics: Animals; Antineoplastic Agents, Phytogenic; Carbazoles; Cell Differentiation; Enzyme Inhibitors; Gene Expression Regulation, Enzymologic; Gene Expression Regulation, Neoplastic; Indoles; Isoenzymes; Mice; Neurites; Neuroblastoma; Protein Kinase C; Rosales; Staurosporine; Xanthenes; Xanthones | 2001 |
Activation of angiotensin II type I receptor promotes protein kinase C translocation and cell proliferation in human cultured breast epithelial cells.
Topics: Analysis of Variance; Angiotensin II; Angiotensin Receptor Antagonists; Biological Transport; Breast; Calcium Signaling; Carbazoles; Cell Division; Enzyme Activation; Enzyme Inhibitors; Epithelial Cells; Estrenes; Female; Humans; Indoles; Isoenzymes; Losartan; Protein Kinase C; Pyrrolidinones; Receptor, Angiotensin, Type 1; Receptors, Angiotensin; Staurosporine; Thapsigargin; Type C Phospholipases | 2002 |
Activation of phosphatidylinositol 3-kinase is important for erythropoietin-induced erythropoiesis from CD34(+) hematopoietic progenitor cells.
Topics: Adult; Antigens, CD34; Antigens, Differentiation; Butadienes; Carbazoles; Cell Cycle; Cell Differentiation; Cell Division; Cells, Cultured; Chromones; Enzyme Activation; Enzyme Inhibitors; Erythroid Precursor Cells; Erythropoiesis; Erythropoietin; Flavonoids; Glycophorins; Hematopoietic Stem Cells; Humans; Indoles; Isoenzymes; Morpholines; Naphthalenes; Nitriles; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Protein Kinase C; Protein Kinase C-alpha; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Recombinant Proteins; Staurosporine; Stem Cell Factor | 2002 |
Role of specific protein kinase C isozymes in mediating epidermal growth factor, thyrotropin-releasing hormone, and phorbol ester regulation of the rat prolactin promoter in GH4/GH4C1 pituitary cells.
Topics: Acetophenones; Animals; Benzopyrans; Calcium; Carbazoles; Cell Line; Enzyme Inhibitors; Epidermal Growth Factor; Gene Expression Regulation; Indoles; Isoenzymes; Maleimides; Naphthalenes; Phorbol Esters; Pituitary Gland; Prolactin; Promoter Regions, Genetic; Protein Kinase C; Protein Kinase C-delta; Protein Kinase C-epsilon; Rats; Staurosporine; Thyrotropin-Releasing Hormone; Transcription, Genetic | 2002 |
Modulation of steroid hydroxylase activity in stably transfected V79MZh11B1 and V79MZh11B2 cells by PKC and PKD inhibitors.
Topics: Acetophenones; Alkaloids; Benzophenanthridines; Benzopyrans; Carbazoles; Cell Line; Cortodoxone; Desoxycorticosterone; Enzyme Inhibitors; Hydroxylation; Indoles; Phenanthridines; Protein Kinase C; Staurosporine; Steroid Hydroxylases; Transfection | 2002 |
Staurosporine induces rapid homotypic intercellular adhesion of U937 cells via multiple kinase activation.
Topics: Acetophenones; Adenosine Triphosphate; Benzopyrans; Calcium-Calmodulin-Dependent Protein Kinases; Carbazoles; CD18 Antigens; Cell Aggregation; Cycloheximide; Cytoskeleton; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Genistein; Humans; Imidazoles; Indoles; Integrin beta1; Isoenzymes; Maleimides; Mitogen-Activated Protein Kinases; Naphthalenes; Phosphorylation; Phosphotransferases; Protein Kinase C; Protein-Tyrosine Kinases; Pyridines; Staurosporine; Temperature; Tetradecanoylphorbol Acetate; Time Factors; Tyrosine; U937 Cells | 2003 |
Protein kinase C (PKC) isotype profile in eosinophils from ponies with sweet itch and role in histamine-induced eosinophil activation.
Topics: Animals; Blotting, Western; Carbazoles; Dermatitis, Allergic Contact; Enzyme Inhibitors; Eosinophils; Histamine; Horse Diseases; Horses; Indoles; Isoenzymes; Lymphocyte Activation; Male; Protein Kinase C; Staurosporine; Superoxides | 2003 |
Transcription factor Ets-1 mediates ischemia- and vascular endothelial growth factor-dependent retinal neovascularization.
Topics: Adenoviridae; Angiopoietin-2; Animals; Blotting, Northern; Blotting, Western; Butadienes; Carbazoles; Cattle; Cell Division; Disease Models, Animal; DNA; Enzyme Inhibitors; Flavonoids; Genes, Dominant; Humans; Hypoxia; Indoles; Maleimides; Mice; Models, Biological; Neovascularization, Pathologic; Neuropilin-1; Nitriles; Phosphorylation; Proto-Oncogene Protein c-ets-1; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-ets; Reperfusion Injury; Retina; RNA, Messenger; Staurosporine; Time Factors; Transcription Factors; Up-Regulation; Vascular Endothelial Growth Factor A | 2004 |
Mechanisms of hydroxyl radical-induced contraction of rat aorta.
Topics: Androstadienes; Animals; Aorta; Calcium; Carbazoles; Cells, Cultured; Cytochrome P-450 Enzyme Inhibitors; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Inhibitors; Ferrous Compounds; Genistein; Hydrogen Peroxide; Hydroxyl Radical; In Vitro Techniques; Indoles; Male; Maleimides; Mitogen-Activated Protein Kinases; Muscle, Smooth, Vascular; Phosphoinositide-3 Kinase Inhibitors; Proadifen; Protein Kinase C; Protein-Tyrosine Kinases; Rats; Rats, Wistar; Staurosporine; Vasoconstriction; Wortmannin | 2004 |
A comparison of the roles of protein kinase C in long-term potentiation in rat hippocampal areas CA1 and CA3.
Topics: Animals; Carbazoles; Carcinogens; Diterpenes; Enzyme Inhibitors; Hippocampus; Indoles; Isoenzymes; Lactams; Long-Term Potentiation; Male; Protein Kinase C; Rats; Rats, Wistar; Sphingosine; Staurosporine | 2005 |
Superoxide stimulates NaCl absorption in the thick ascending limb via activation of protein kinase C.
Topics: Absorption; Animals; Carbazoles; Chlorides; Enzyme Activation; Enzyme Inhibitors; In Vitro Techniques; Indoles; Ion Transport; Isoenzymes; Loop of Henle; Male; Protein Kinase C; Rats; Rats, Sprague-Dawley; Sodium Chloride; Staurosporine; Superoxides | 2006 |
Activation of the extracellular calcium-sensing receptor initiates insulin secretion from human islets of Langerhans: involvement of protein kinases.
Topics: Aniline Compounds; Antibodies, Monoclonal; Benzylamines; Calcium; Calcium-Calmodulin-Dependent Protein Kinases; Carbazoles; Cell Communication; Cell Line; Cells, Cultured; Estrenes; Extracellular Fluid; Flavonoids; Glucose; Humans; Immunohistochemistry; Indoles; Insulin; Insulin Secretion; Insulin-Secreting Cells; Mitogen-Activated Protein Kinases; Phenethylamines; Propylamines; Protein Kinase C; Protein Kinases; Pyrrolidinones; Receptors, Calcium-Sensing; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Staurosporine; Stimulation, Chemical; Sulfonamides; Type C Phospholipases | 2006 |
Mechanism of membrane redistribution of protein kinase C by its ATP-competitive inhibitors.
Topics: Amino Acid Sequence; Amino Acid Substitution; Animals; Binding, Competitive; Carbazoles; Cell Membrane; Chlorocebus aethiops; COS Cells; Diglycerides; Estrenes; HeLa Cells; HL-60 Cells; Humans; Indoles; Maleimides; Membranes; Microscopy, Confocal; Phorbol 12,13-Dibutyrate; Protein Kinase C; Protein Transport; Pyrrolidinones; Staurosporine | 2007 |
Lidocaine-induced apoptosis of gingival fibroblasts: participation of cAMP and PKC activity.
Topics: Apoptosis; Carbazoles; Caspase 3; Cells, Cultured; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Fibroblasts; Gingiva; Humans; In Situ Nick-End Labeling; Isoquinolines; Lidocaine; Protein Kinase C; Protein Kinase Inhibitors; Staurosporine; Sulfonamides | 2011 |
C3b-induced eosinophil degranulation involves PI3-kinases and is inhibited by protein kinase C activity.
Topics: Carbazoles; Cell Degranulation; Complement C3b; Eosinophils; Extracellular Signal-Regulated MAP Kinases; Flavonoids; Humans; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Protein Kinase C; Protein Kinase Inhibitors; Staurosporine | 2011 |
ATP potentiates competitive inhibition of guanylyl cyclase A and B by the staurosporine analog, Gö6976: reciprocal regulation of ATP and GTP binding.
Topics: Adenosine Triphosphate; Binding Sites; Carbazoles; Cell Line; Enzyme Activation; Enzyme Inhibitors; Guanosine Triphosphate; Humans; Protein Binding; Receptors, Atrial Natriuretic Factor; Staurosporine | 2011 |
Noncovalent wild-type-sparing inhibitors of EGFR T790M.
Topics: Acrylamides; Amino Acid Substitution; Animals; Area Under Curve; Base Sequence; Carbazoles; Cell Line, Tumor; Drug Resistance, Neoplasm; ErbB Receptors; Erlotinib Hydrochloride; Humans; Immunoblotting; Lung; Lung Neoplasms; Mice; Mice, Inbred BALB C; Mice, Nude; Mice, Transgenic; Mutation; Protein Kinase Inhibitors; Pyrimidines; Quinazolines; RNA Interference; Staurosporine; Xenograft Model Antitumor Assays | 2013 |
Therapeutic hypercapnia reduces blood-brain barrier damage possibly via protein kinase Cε in rats with lateral fluid percussion injury.
Topics: Animals; Blood Pressure; Blood-Brain Barrier; Brain Edema; Brain Injuries, Traumatic; Carbazoles; Carbon Dioxide; Disease Models, Animal; Heart Rate; Hypercapnia; Male; Neurologic Examination; Oxygen; Protein Kinase C-epsilon; Protein Kinase Inhibitors; Rats; Rats, Sprague-Dawley; Staurosporine; Time Factors; Tomography Scanners, X-Ray Computed | 2019 |
The Mechanism of Action of Ghrelin and Motilin in the Pacemaker Potentials of Interstitial Cells of Cajal from the Murine Small Intestine.
Topics: Acetophenones; Amides; Animals; Benzopyrans; Boron Compounds; Calcium; Carbazoles; Gastrointestinal Motility; Ghrelin; Inositol 1,4,5-Trisphosphate Receptors; Interstitial Cells of Cajal; Intestine, Small; Macrocyclic Compounds; Membrane Potentials; Mice; Mice, Inbred ICR; Motilin; Oligopeptides; Oxazoles; Protein Kinase C; Pyridines; Receptors, Ghrelin; rho-Associated Kinases; Signal Transduction; Staurosporine; Thapsigargin | 2019 |