staurosporine has been researched along with chloroquine in 20 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 7 (35.00) | 18.2507 |
2000's | 5 (25.00) | 29.6817 |
2010's | 8 (40.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bhattacharjee, AK; Geyer, JA; Kathcart, AK; Li, Z; Mott, BT; Nichols, DA; Prigge, ST; Waters, NC; Woodard, CL | 1 |
Andersen, C; Breton, G; Bursulaya, B; Chatterjee, A; Gray, N; Harper, J; Henson, K; Johnson, J; Kato, N; Kumar, KA; Le Roch, KG; Marr, F; Mason, D; McNamara, C; Nagle, A; Peters, EC; Plouffe, D; Ramachandran, V; Sakata, T; Schultz, PG; Spooner, M; Tuntland, T; Ward, GE; Winzeler, EA; Zhou, Y | 1 |
García-Mera, X; González-Díaz, H; Prado-Prado, FJ | 1 |
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ | 1 |
Barnes, SW; Bonamy, GM; Bopp, SE; Borboa, R; Bright, AT; Chatterjee, A; Che, J; Cohen, S; Dharia, NV; Diagana, TT; Fidock, DA; Froissard, P; Gagaring, K; Gettayacamin, M; Glynne, RJ; Gordon, P; Groessl, T; Kato, N; Kuhen, KL; Lee, MC; Mazier, D; McNamara, CW; Meister, S; Nagle, A; Nam, TG; Plouffe, DM; Richmond, W; Roland, J; Rottmann, M; Sattabongkot, J; Schultz, PG; Tuntland, T; Walker, JR; Winzeler, EA; Wu, T; Zhou, B; Zhou, Y | 1 |
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ | 1 |
Gut, J; Kumar, V; Rosenthal, PJ | 1 |
Clark, J; Connelly, M; González, MA; Rivas, F | 1 |
Bidlack, JM; Gucker, S | 1 |
Humphries, RK; Kay, RJ; Krystal, G; Mui, AL | 1 |
Engleman, EG; Rajasekar, S; Ruegg, CL; Stein, BS | 1 |
Kan, M; McKeehan, WL; Shi, E; Xu, JM | 1 |
Fleer, A; Mattsson, E; Rollof, J; Van Dijk, H; Van Kessel, K; Verhoef, J | 1 |
Chen, SS; Jiang, MC; Lin, JK | 1 |
Amara, SG; Daniels, GM | 1 |
Gafni, M; Keren, O; Sarne, Y; Shapira, M | 1 |
Corte-Real, S; Daniel-Ribeiro, CT; de Fátima Ferreira-da-Cruz, M; Totino, PR | 1 |
Cortes-Hernandez, DG; Gamette, MJ; Jensen, JB; Porter, H | 1 |
Ali, M; Carter, V; Hunt, J; Hurd, H; Matthews, H; Szor, H; Underhill, A | 1 |
Chain, WJ; Fash, DM; Li, Z; Nakashige, ML; Ramos, JW; Sulzmaier, FJ | 1 |
20 other study(ies) available for staurosporine and chloroquine
Article | Year |
---|---|
A three-dimensional in silico pharmacophore model for inhibition of Plasmodium falciparum cyclin-dependent kinases and discovery of different classes of novel Pfmrk specific inhibitors.
Topics: Adenosine Triphosphate; Animals; Antimalarials; Binding Sites; Cyclin-Dependent Kinases; Databases, Factual; Hydrogen Bonding; Hydrophobic and Hydrophilic Interactions; Models, Molecular; Plasmodium falciparum; Protein Kinases; Protozoan Proteins; Quantitative Structure-Activity Relationship | 2004 |
Gene expression signatures and small-molecule compounds link a protein kinase to Plasmodium falciparum motility.
Topics: Adenine; Animals; Antimalarials; Cell Line; Cell Proliferation; CHO Cells; Cricetinae; Cricetulus; Cyclohexylamines; Drug Evaluation, Preclinical; Enzyme Activation; Gene Expression Regulation, Enzymologic; HeLa Cells; Humans; Life Cycle Stages; Malaria; Male; Mice; Mice, Inbred BALB C; Models, Molecular; Molecular Structure; Molecular Weight; Movement; Oligonucleotide Array Sequence Analysis; Parasitic Sensitivity Tests; Plasmodium falciparum; Protein Kinases; Protozoan Proteins; Recombinant Proteins; Small Molecule Libraries; Stereoisomerism; Structure-Activity Relationship; Tissue Distribution | 2008 |
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics | 2010 |
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics | 2010 |
Imaging of Plasmodium liver stages to drive next-generation antimalarial drug discovery.
Topics: Animals; Antimalarials; Cell Line, Tumor; Drug Discovery; Drug Evaluation, Preclinical; Drug Resistance; Erythrocytes; Humans; Imidazoles; Liver; Malaria; Mice; Mice, Inbred BALB C; Molecular Structure; Piperazines; Plasmodium; Plasmodium berghei; Plasmodium falciparum; Plasmodium yoelii; Polymorphism, Single Nucleotide; Protozoan Proteins; Random Allocation; Small Molecule Libraries; Sporozoites | 2011 |
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests | 2013 |
β-amino-alcohol tethered 4-aminoquinoline-isatin conjugates: synthesis and antimalarial evaluation.
Topics: Amino Alcohols; Aminoquinolines; Antimalarials; Cell Survival; Dose-Response Relationship, Drug; HCT116 Cells; Humans; Isatin; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Structure-Activity Relationship | 2014 |
Antimalarial activity of abietane ferruginol analogues possessing a phthalimide group.
Topics: Abietanes; Animals; Antimalarials; CHO Cells; Cricetinae; Cricetulus; Hep G2 Cells; Humans; Phthalimides; Plant Extracts; Plasmodium falciparum | 2014 |
Protein kinase C activation increases the rate and magnitude of agonist-induced delta-opioid receptor down-regulation in NG108-15 cells.
Topics: Alkaloids; Cell Membrane; Cells, Cultured; Chloroquine; Down-Regulation; Enkephalin, Leucine-2-Alanine; Enzyme Activation; Etorphine; In Vitro Techniques; Naloxone; Narcotics; Neurons; Protein Kinase C; Receptors, Opioid, delta; Staurosporine; Tetradecanoylphorbol Acetate | 1992 |
Ligand-induced phosphorylation of the murine interleukin 3 receptor signals its cleavage.
Topics: Alkaloids; Animals; Blotting, Western; Cell Line; Chloroquine; Genistein; Granulocyte-Macrophage Colony-Stimulating Factor; Interleukin-3; Interleukin-5; Isoflavones; Kinetics; Ligands; Macromolecular Substances; Mice; Molecular Weight; Phosphoprotein Phosphatases; Phosphorylation; Protein Kinase C; Protein-Tyrosine Kinases; Receptors, Interleukin-3; Recombinant Proteins; Staurosporine; Tetradecanoylphorbol Acetate; Transfection | 1992 |
Degradation of CD4 following phorbol-induced internalization in human T lymphocytes. Evidence for distinct endocytic routing of CD4 and CD3.
Topics: Alkaloids; Ammonium Chloride; CD4 Antigens; Chloroquine; Electrophoresis, Polyacrylamide Gel; Enzyme-Linked Immunosorbent Assay; Humans; Monensin; Phorbol 12,13-Dibutyrate; Protein Kinase C; Radioimmunoprecipitation Assay; Staurosporine; T-Lymphocytes | 1992 |
16-kilodalton heparin binding (fibroblast) growth factor type one appears in a stable 40-kilodalton complex after receptor-dependent internalization.
Topics: Alkaloids; Animals; Biotin; Cadaverine; Chloroquine; Cross-Linking Reagents; Electrophoresis, Gel, Two-Dimensional; Electrophoresis, Polyacrylamide Gel; Fibroblast Growth Factors; Heparin; Humans; Liver; Molecular Weight; Precipitin Tests; Rats; Staurosporine; Temperature; Tumor Cells, Cultured | 1991 |
Intracellular pathways involved in tumor necrosis factor-alpha release by human monocytes on stimulation with lipopolysaccharide or staphylococcal peptidoglycan are partly similar.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetophenones; Alkaloids; Antimalarials; Cell Communication; Chloroquine; Dose-Response Relationship, Drug; Enzyme Inhibitors; Escherichia coli; GTP-Binding Proteins; Humans; Isoquinolines; Lipopolysaccharides; Monocytes; Pentoxifylline; Peptidoglycan; Piperazines; Protein Kinase Inhibitors; Protein Kinases; Protein-Tyrosine Kinases; Signal Transduction; Staphylococcus epidermidis; Staurosporine; Sulfonamides; Tumor Necrosis Factor-alpha; Vasodilator Agents | 1996 |
Inhibition of HIV-1 Tat-mediated transactivation by quinacrine and chloroquine.
Topics: Acetophenones; Alkaloids; Antimalarials; Benzoquinones; Cell Line; Cell Survival; Chloroquine; Curcumin; Gene Expression Regulation, Viral; Gene Products, tat; HIV Long Terminal Repeat; HIV-1; Humans; Lactams, Macrocyclic; Quinacrine; Quinones; Rifabutin; Staurosporine; tat Gene Products, Human Immunodeficiency Virus; Transcriptional Activation; Tumor Cells, Cultured; Virus Replication | 1996 |
Regulated trafficking of the human dopamine transporter. Clathrin-mediated internalization and lysosomal degradation in response to phorbol esters.
Topics: Acetylcysteine; Animals; Carrier Proteins; Cell Line; Chloroquine; Clathrin; Colforsin; Cycloheximide; Dogs; Dopamine; Dopamine Plasma Membrane Transport Proteins; Endocytosis; Enzyme Activation; Humans; Kinetics; Lysosomes; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Phorbols; Protein Kinase C; Recombinant Proteins; Staurosporine; Tetradecanoylphorbol Acetate; Transfection | 1999 |
Divers pathways mediate delta-opioid receptor down regulation within the same cell.
Topics: Acetylcysteine; Analgesics, Opioid; Animals; Antirheumatic Agents; Chloroquine; Cysteine Proteinase Inhibitors; Diprenorphine; Down-Regulation; Etorphine; Flavonoids; Genistein; GTP-Binding Proteins; Humans; Kidney; MAP Kinase Signaling System; Narcotic Antagonists; Neuroblastoma; Phosphorylation; Radioligand Assay; Receptors, Opioid, delta; Staurosporine; Teprotide; Transfection; Tritium; Tumor Cells, Cultured | 2001 |
Plasmodium falciparum: erythrocytic stages die by autophagic-like cell death under drug pressure.
Topics: Animals; Antimalarials; Apoptosis; Autophagy; Caspase Inhibitors; Cells, Cultured; Chloroquine; DNA Fragmentation; Erythrocytes; Flow Cytometry; Fluorescent Dyes; Humans; In Situ Nick-End Labeling; Membrane Potentials; Microscopy, Electron, Transmission; Nitric Oxide Donors; Penicillamine; Plasmodium falciparum; Rhodamine 123; Staurosporine | 2008 |
Asexual blood stages of Plasmodium falciparum exhibit signs of secondary necrosis, but not classical apoptosis after exposure to febrile temperature (40 C).
Topics: Animals; Antimalarials; Apoptosis; Caspases; Chloroquine; DNA Fragmentation; DNA, Protozoan; Enzyme Activation; Enzyme Inhibitors; Erythrocytes; Glucose; Humans; Membrane Potential, Mitochondrial; Microscopy, Electron, Transmission; Necrosis; Plasmodium falciparum; Protozoan Proteins; Staurosporine; Temperature | 2008 |
Variation in apoptosis mechanisms employed by malaria parasites: the roles of inducers, dose dependence and parasite stages.
Topics: Apoptosis; Caspases; Chloroquine; Chromatin; DNA Fragmentation; Hydrogen Peroxide; Membrane Potentials; Mitochondria; Mitochondrial Membranes; Phosphatidylserines; Plasmodium falciparum; Staurosporine | 2012 |
Englerin a selectively induces necrosis in human renal cancer cells.
Topics: Antineoplastic Agents; Apoptosis; Autophagy; Calcium; Cell Line, Tumor; Cell Survival; Chloroquine; Cytoplasm; Dose-Response Relationship, Drug; HEK293 Cells; Humans; Kidney Neoplasms; Molecular Structure; Necrosis; Reactive Oxygen Species; Sesquiterpenes, Guaiane; Staurosporine | 2012 |