Page last updated: 2024-08-23

staurosporine and chloroquine

staurosporine has been researched along with chloroquine in 20 studies

Research

Studies (20)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's7 (35.00)18.2507
2000's5 (25.00)29.6817
2010's8 (40.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bhattacharjee, AK; Geyer, JA; Kathcart, AK; Li, Z; Mott, BT; Nichols, DA; Prigge, ST; Waters, NC; Woodard, CL1
Andersen, C; Breton, G; Bursulaya, B; Chatterjee, A; Gray, N; Harper, J; Henson, K; Johnson, J; Kato, N; Kumar, KA; Le Roch, KG; Marr, F; Mason, D; McNamara, C; Nagle, A; Peters, EC; Plouffe, D; Ramachandran, V; Sakata, T; Schultz, PG; Spooner, M; Tuntland, T; Ward, GE; Winzeler, EA; Zhou, Y1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Barnes, SW; Bonamy, GM; Bopp, SE; Borboa, R; Bright, AT; Chatterjee, A; Che, J; Cohen, S; Dharia, NV; Diagana, TT; Fidock, DA; Froissard, P; Gagaring, K; Gettayacamin, M; Glynne, RJ; Gordon, P; Groessl, T; Kato, N; Kuhen, KL; Lee, MC; Mazier, D; McNamara, CW; Meister, S; Nagle, A; Nam, TG; Plouffe, DM; Richmond, W; Roland, J; Rottmann, M; Sattabongkot, J; Schultz, PG; Tuntland, T; Walker, JR; Winzeler, EA; Wu, T; Zhou, B; Zhou, Y1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Gut, J; Kumar, V; Rosenthal, PJ1
Clark, J; Connelly, M; González, MA; Rivas, F1
Bidlack, JM; Gucker, S1
Humphries, RK; Kay, RJ; Krystal, G; Mui, AL1
Engleman, EG; Rajasekar, S; Ruegg, CL; Stein, BS1
Kan, M; McKeehan, WL; Shi, E; Xu, JM1
Fleer, A; Mattsson, E; Rollof, J; Van Dijk, H; Van Kessel, K; Verhoef, J1
Chen, SS; Jiang, MC; Lin, JK1
Amara, SG; Daniels, GM1
Gafni, M; Keren, O; Sarne, Y; Shapira, M1
Corte-Real, S; Daniel-Ribeiro, CT; de Fátima Ferreira-da-Cruz, M; Totino, PR1
Cortes-Hernandez, DG; Gamette, MJ; Jensen, JB; Porter, H1
Ali, M; Carter, V; Hunt, J; Hurd, H; Matthews, H; Szor, H; Underhill, A1
Chain, WJ; Fash, DM; Li, Z; Nakashige, ML; Ramos, JW; Sulzmaier, FJ1

Other Studies

20 other study(ies) available for staurosporine and chloroquine

ArticleYear
A three-dimensional in silico pharmacophore model for inhibition of Plasmodium falciparum cyclin-dependent kinases and discovery of different classes of novel Pfmrk specific inhibitors.
    Journal of medicinal chemistry, 2004, Oct-21, Volume: 47, Issue:22

    Topics: Adenosine Triphosphate; Animals; Antimalarials; Binding Sites; Cyclin-Dependent Kinases; Databases, Factual; Hydrogen Bonding; Hydrophobic and Hydrophilic Interactions; Models, Molecular; Plasmodium falciparum; Protein Kinases; Protozoan Proteins; Quantitative Structure-Activity Relationship

2004
Gene expression signatures and small-molecule compounds link a protein kinase to Plasmodium falciparum motility.
    Nature chemical biology, 2008, Volume: 4, Issue:6

    Topics: Adenine; Animals; Antimalarials; Cell Line; Cell Proliferation; CHO Cells; Cricetinae; Cricetulus; Cyclohexylamines; Drug Evaluation, Preclinical; Enzyme Activation; Gene Expression Regulation, Enzymologic; HeLa Cells; Humans; Life Cycle Stages; Malaria; Male; Mice; Mice, Inbred BALB C; Models, Molecular; Molecular Structure; Molecular Weight; Movement; Oligonucleotide Array Sequence Analysis; Parasitic Sensitivity Tests; Plasmodium falciparum; Protein Kinases; Protozoan Proteins; Recombinant Proteins; Small Molecule Libraries; Stereoisomerism; Structure-Activity Relationship; Tissue Distribution

2008
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
Imaging of Plasmodium liver stages to drive next-generation antimalarial drug discovery.
    Science (New York, N.Y.), 2011, Dec-09, Volume: 334, Issue:6061

    Topics: Animals; Antimalarials; Cell Line, Tumor; Drug Discovery; Drug Evaluation, Preclinical; Drug Resistance; Erythrocytes; Humans; Imidazoles; Liver; Malaria; Mice; Mice, Inbred BALB C; Molecular Structure; Piperazines; Plasmodium; Plasmodium berghei; Plasmodium falciparum; Plasmodium yoelii; Polymorphism, Single Nucleotide; Protozoan Proteins; Random Allocation; Small Molecule Libraries; Sporozoites

2011
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
β-amino-alcohol tethered 4-aminoquinoline-isatin conjugates: synthesis and antimalarial evaluation.
    European journal of medicinal chemistry, 2014, Sep-12, Volume: 84

    Topics: Amino Alcohols; Aminoquinolines; Antimalarials; Cell Survival; Dose-Response Relationship, Drug; HCT116 Cells; Humans; Isatin; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Structure-Activity Relationship

2014
Antimalarial activity of abietane ferruginol analogues possessing a phthalimide group.
    Bioorganic & medicinal chemistry letters, 2014, Nov-15, Volume: 24, Issue:22

    Topics: Abietanes; Animals; Antimalarials; CHO Cells; Cricetinae; Cricetulus; Hep G2 Cells; Humans; Phthalimides; Plant Extracts; Plasmodium falciparum

2014
Protein kinase C activation increases the rate and magnitude of agonist-induced delta-opioid receptor down-regulation in NG108-15 cells.
    Molecular pharmacology, 1992, Volume: 42, Issue:4

    Topics: Alkaloids; Cell Membrane; Cells, Cultured; Chloroquine; Down-Regulation; Enkephalin, Leucine-2-Alanine; Enzyme Activation; Etorphine; In Vitro Techniques; Naloxone; Narcotics; Neurons; Protein Kinase C; Receptors, Opioid, delta; Staurosporine; Tetradecanoylphorbol Acetate

1992
Ligand-induced phosphorylation of the murine interleukin 3 receptor signals its cleavage.
    Proceedings of the National Academy of Sciences of the United States of America, 1992, Nov-15, Volume: 89, Issue:22

    Topics: Alkaloids; Animals; Blotting, Western; Cell Line; Chloroquine; Genistein; Granulocyte-Macrophage Colony-Stimulating Factor; Interleukin-3; Interleukin-5; Isoflavones; Kinetics; Ligands; Macromolecular Substances; Mice; Molecular Weight; Phosphoprotein Phosphatases; Phosphorylation; Protein Kinase C; Protein-Tyrosine Kinases; Receptors, Interleukin-3; Recombinant Proteins; Staurosporine; Tetradecanoylphorbol Acetate; Transfection

1992
Degradation of CD4 following phorbol-induced internalization in human T lymphocytes. Evidence for distinct endocytic routing of CD4 and CD3.
    The Journal of biological chemistry, 1992, Sep-15, Volume: 267, Issue:26

    Topics: Alkaloids; Ammonium Chloride; CD4 Antigens; Chloroquine; Electrophoresis, Polyacrylamide Gel; Enzyme-Linked Immunosorbent Assay; Humans; Monensin; Phorbol 12,13-Dibutyrate; Protein Kinase C; Radioimmunoprecipitation Assay; Staurosporine; T-Lymphocytes

1992
16-kilodalton heparin binding (fibroblast) growth factor type one appears in a stable 40-kilodalton complex after receptor-dependent internalization.
    The Journal of biological chemistry, 1991, Mar-25, Volume: 266, Issue:9

    Topics: Alkaloids; Animals; Biotin; Cadaverine; Chloroquine; Cross-Linking Reagents; Electrophoresis, Gel, Two-Dimensional; Electrophoresis, Polyacrylamide Gel; Fibroblast Growth Factors; Heparin; Humans; Liver; Molecular Weight; Precipitin Tests; Rats; Staurosporine; Temperature; Tumor Cells, Cultured

1991
Intracellular pathways involved in tumor necrosis factor-alpha release by human monocytes on stimulation with lipopolysaccharide or staphylococcal peptidoglycan are partly similar.
    The Journal of infectious diseases, 1996, Volume: 173, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetophenones; Alkaloids; Antimalarials; Cell Communication; Chloroquine; Dose-Response Relationship, Drug; Enzyme Inhibitors; Escherichia coli; GTP-Binding Proteins; Humans; Isoquinolines; Lipopolysaccharides; Monocytes; Pentoxifylline; Peptidoglycan; Piperazines; Protein Kinase Inhibitors; Protein Kinases; Protein-Tyrosine Kinases; Signal Transduction; Staphylococcus epidermidis; Staurosporine; Sulfonamides; Tumor Necrosis Factor-alpha; Vasodilator Agents

1996
Inhibition of HIV-1 Tat-mediated transactivation by quinacrine and chloroquine.
    Biochemical and biophysical research communications, 1996, Sep-04, Volume: 226, Issue:1

    Topics: Acetophenones; Alkaloids; Antimalarials; Benzoquinones; Cell Line; Cell Survival; Chloroquine; Curcumin; Gene Expression Regulation, Viral; Gene Products, tat; HIV Long Terminal Repeat; HIV-1; Humans; Lactams, Macrocyclic; Quinacrine; Quinones; Rifabutin; Staurosporine; tat Gene Products, Human Immunodeficiency Virus; Transcriptional Activation; Tumor Cells, Cultured; Virus Replication

1996
Regulated trafficking of the human dopamine transporter. Clathrin-mediated internalization and lysosomal degradation in response to phorbol esters.
    The Journal of biological chemistry, 1999, Dec-10, Volume: 274, Issue:50

    Topics: Acetylcysteine; Animals; Carrier Proteins; Cell Line; Chloroquine; Clathrin; Colforsin; Cycloheximide; Dogs; Dopamine; Dopamine Plasma Membrane Transport Proteins; Endocytosis; Enzyme Activation; Humans; Kinetics; Lysosomes; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Phorbols; Protein Kinase C; Recombinant Proteins; Staurosporine; Tetradecanoylphorbol Acetate; Transfection

1999
Divers pathways mediate delta-opioid receptor down regulation within the same cell.
    Brain research. Molecular brain research, 2001, Nov-30, Volume: 96, Issue:1-2

    Topics: Acetylcysteine; Analgesics, Opioid; Animals; Antirheumatic Agents; Chloroquine; Cysteine Proteinase Inhibitors; Diprenorphine; Down-Regulation; Etorphine; Flavonoids; Genistein; GTP-Binding Proteins; Humans; Kidney; MAP Kinase Signaling System; Narcotic Antagonists; Neuroblastoma; Phosphorylation; Radioligand Assay; Receptors, Opioid, delta; Staurosporine; Teprotide; Transfection; Tritium; Tumor Cells, Cultured

2001
Plasmodium falciparum: erythrocytic stages die by autophagic-like cell death under drug pressure.
    Experimental parasitology, 2008, Volume: 118, Issue:4

    Topics: Animals; Antimalarials; Apoptosis; Autophagy; Caspase Inhibitors; Cells, Cultured; Chloroquine; DNA Fragmentation; Erythrocytes; Flow Cytometry; Fluorescent Dyes; Humans; In Situ Nick-End Labeling; Membrane Potentials; Microscopy, Electron, Transmission; Nitric Oxide Donors; Penicillamine; Plasmodium falciparum; Rhodamine 123; Staurosporine

2008
Asexual blood stages of Plasmodium falciparum exhibit signs of secondary necrosis, but not classical apoptosis after exposure to febrile temperature (40 C).
    The Journal of parasitology, 2008, Volume: 94, Issue:2

    Topics: Animals; Antimalarials; Apoptosis; Caspases; Chloroquine; DNA Fragmentation; DNA, Protozoan; Enzyme Activation; Enzyme Inhibitors; Erythrocytes; Glucose; Humans; Membrane Potential, Mitochondrial; Microscopy, Electron, Transmission; Necrosis; Plasmodium falciparum; Protozoan Proteins; Staurosporine; Temperature

2008
Variation in apoptosis mechanisms employed by malaria parasites: the roles of inducers, dose dependence and parasite stages.
    Malaria journal, 2012, Aug-28, Volume: 11

    Topics: Apoptosis; Caspases; Chloroquine; Chromatin; DNA Fragmentation; Hydrogen Peroxide; Membrane Potentials; Mitochondria; Mitochondrial Membranes; Phosphatidylserines; Plasmodium falciparum; Staurosporine

2012
Englerin a selectively induces necrosis in human renal cancer cells.
    PloS one, 2012, Volume: 7, Issue:10

    Topics: Antineoplastic Agents; Apoptosis; Autophagy; Calcium; Cell Line, Tumor; Cell Survival; Chloroquine; Cytoplasm; Dose-Response Relationship, Drug; HEK293 Cells; Humans; Kidney Neoplasms; Molecular Structure; Necrosis; Reactive Oxygen Species; Sesquiterpenes, Guaiane; Staurosporine

2012