Page last updated: 2024-08-23

staurosporine and ag-213

staurosporine has been researched along with ag-213 in 19 studies

Research

Studies (19)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's15 (78.95)18.2507
2000's4 (21.05)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chang, CJ; Geahlen, RL1
Chandraratna, RA; Nagpal, S; Thacher, SM; Tsang, KY; Vasudevan, J1
Bayoumy, S; Deckman, IC; Devine, E; Grasberger, B; Ma, HC; Mezzasalma, T; Petrounia, IP; Schalk-Hihi, C; Schubert, C; Springer, BA; Struble, GT; Williams, R; Zeng, L1
Li, LL; Ren, JX; Wei, YQ; Xie, HZ; Yang, L; Yang, SY; Zou, J1
Burroughs, S; Feinstein, MB; Huang, CK; Lau, LF; Pumiglia, KM1
Danaher, M; Fallon, RJ; Saxena, A; Saylors, RL1
Cáceres-Cortés, J; Dumouchel, J; Haddad, P; Hoang, T; Rajotte, D1
Carter, V; Gale, M; Parsons, M1
Chang, NS1
Hoh, E; Kadowaki, T; Kaida, T; Komuro, I; Maemura, K; Nagai, R; Tamemoto, H; Tobe, K; Yamazaki, T; Yazaki, Y1
Finlay, BB; Rosenshine, I; Ruschkowski, S1
Ali, A; Ford-Hutchinson, AW; Nicholson, DW1
Welsh, N1
Bouchelouche, P; De Meyts, P; Ilondo, MM1
Chun, YJ; Koh, WS; Yang, KH1
Buschmann, J; Heinrich, PC; Horn, F; Lottspeich, F; Lütticken, C; Müller-Esterl, W; Roeb, E; Schindler, C; Wegenka, UM; Yuan, J1
Kume, S; Ozaki, Y; Satoh, K; Yatomi, Y1
Ain, R; Seshagiri, PB; Shivaji, S; Uma Devi, K1
Abe, K; Ikebukuro, K; Sode, K; Yagi, YI1

Reviews

2 review(s) available for staurosporine and ag-213

ArticleYear
Protein-tyrosine kinase inhibition: mechanism-based discovery of antitumor agents.
    Journal of natural products, 1992, Volume: 55, Issue:11

    Topics: Animals; Antineoplastic Agents; Drug Screening Assays, Antitumor; Humans; Protein-Tyrosine Kinases

1992
New dermatological agents for the treatment of psoriasis.
    Journal of medicinal chemistry, 2001, Feb-01, Volume: 44, Issue:3

    Topics: Administration, Topical; Anti-Inflammatory Agents; Cholecalciferol; Clinical Trials as Topic; Glucocorticoids; Humans; Immunosuppressive Agents; Ligands; Methotrexate; Psoriasis; Receptors, Cytoplasmic and Nuclear; Receptors, Steroid; Vitamin A

2001

Other Studies

17 other study(ies) available for staurosporine and ag-213

ArticleYear
Protein engineering of the colony-stimulating factor-1 receptor kinase domain for structural studies.
    The Journal of biological chemistry, 2007, Feb-09, Volume: 282, Issue:6

    Topics: Amino Acid Sequence; Animals; Cells, Cultured; Crystallization; Cytoplasm; Humans; Molecular Sequence Data; Mutant Chimeric Proteins; Protein Engineering; Protein Kinase Inhibitors; Protein Structure, Tertiary; Receptor Protein-Tyrosine Kinases; Receptor, Macrophage Colony-Stimulating Factor; Sequence Alignment; Spodoptera

2007
Pharmacophore modeling study based on known spleen tyrosine kinase inhibitors together with virtual screening for identifying novel inhibitors.
    Bioorganic & medicinal chemistry letters, 2009, Apr-01, Volume: 19, Issue:7

    Topics: Computer Simulation; Intracellular Signaling Peptides and Proteins; Models, Molecular; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Small Molecule Libraries; Software; Structure-Activity Relationship; Syk Kinase

2009
Activation of signal transduction in platelets by the tyrosine phosphatase inhibitor pervanadate (vanadyl hydroperoxide).
    The Biochemical journal, 1992, Sep-01, Volume: 286 ( Pt 2)

    Topics: Actins; Adenosine Triphosphate; Alkaloids; Blood Proteins; Blotting, Western; Calcium; Catechols; Cells, Cultured; Electrophoresis, Polyacrylamide Gel; Enzyme Activation; Humans; Nitriles; Phospholipids; Phosphoproteins; Phosphorylation; Platelet Membrane Glycoproteins; Protein Kinase C; Protein Tyrosine Phosphatases; Serotonin; Signal Transduction; Staurosporine; Tetradecanoylphorbol Acetate; Type C Phospholipases; Tyrosine; Tyrphostins; Vanadates

1992
Defective asialoglycoprotein receptor endocytosis mediated by tyrosine kinase inhibitors. Requirement for a tyrosine in the receptor internalization signal.
    The Journal of biological chemistry, 1994, Apr-15, Volume: 269, Issue:15

    Topics: Adenosine Triphosphate; Alkaloids; Asialoglycoprotein Receptor; Carcinoma, Hepatocellular; Catechols; Cell Line; Endocytosis; Genistein; Humans; Isoflavones; Kinetics; Liver Neoplasms; Nitriles; Phosphorylation; Phosphotyrosine; Protein-Tyrosine Kinases; Receptor Protein-Tyrosine Kinases; Receptors, Cell Surface; Signal Transduction; Staurosporine; Transferrin; Tumor Cells, Cultured; Tyrosine; Tyrphostins

1994
Product of the steel locus suppresses apoptosis in hemopoietic cells. Comparison with pathways activated by granulocyte macrophage colony-stimulating factor.
    The Journal of biological chemistry, 1994, Apr-22, Volume: 269, Issue:16

    Topics: Alkaloids; Amiloride; Animals; Apoptosis; Bone Marrow; Bone Marrow Cells; Catechols; Cell Division; Cell Line; Cell Survival; DNA; DNA Damage; Fusion Proteins, bcr-abl; Granulocyte-Macrophage Colony-Stimulating Factor; Hematopoietic Cell Growth Factors; Hematopoietic Stem Cells; Humans; Hydrogen-Ion Concentration; Interleukin-3; Leukemia, Myeloid, Acute; Nitriles; Protein Kinase Inhibitors; Recombinant Proteins; Staurosporine; Stem Cell Factor; Thymidine; Transfection; Tyrphostins

1994
Cell cycle-specific induction of an 89 kDa serine/threonine protein kinase activity in Trypanosoma brucei.
    Journal of cell science, 1994, Volume: 107 ( Pt 7)

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Animals; Catechols; Cell Cycle; Cell Division; Cycloheximide; DNA; Enzyme Induction; Ethers, Cyclic; Flow Cytometry; Genistein; Isoflavones; Isoquinolines; Molecular Weight; Nitriles; Okadaic Acid; Phosphoproteins; Phosphorylation; Phosphotyrosine; Piperazines; Protein Denaturation; Protein Kinase C; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; S Phase; Staurosporine; Trypanosoma brucei brucei; Tyrosine; Tyrphostins

1994
Transforming growth factor-beta 1 induction of novel extracellular matrix proteins that trigger resistance to tumor necrosis factor cytotoxicity in murine L929 fibroblasts.
    The Journal of biological chemistry, 1995, Mar-31, Volume: 270, Issue:13

    Topics: Alkaloids; Animals; Catechols; Cell Survival; Dose-Response Relationship, Drug; Extracellular Matrix Proteins; Fibroblasts; Genistein; Isoflavones; Kinetics; L Cells; Mice; Nitriles; Phenols; Phosphotyrosine; Protein Kinase Inhibitors; Staurosporine; Transforming Growth Factor beta; Tumor Protein, Translationally-Controlled 1; Tyrosine; Tyrphostins

1995
Mechanical loading activates mitogen-activated protein kinase and S6 peptide kinase in cultured rat cardiac myocytes.
    The Journal of biological chemistry, 1993, Jun-05, Volume: 268, Issue:16

    Topics: Alkaloids; Animals; Animals, Newborn; Calcium-Calmodulin-Dependent Protein Kinases; Catechols; Cells, Cultured; Electrophoresis, Polyacrylamide Gel; Enzyme Activation; Gene Expression; Genes, fos; Genistein; Isoflavones; Kinetics; Myelin Basic Protein; Myocardium; Nitriles; Protein Kinase C; Protein Kinases; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Rats; Rats, Wistar; Ribosomal Protein S6 Kinases; Staurosporine; Tetradecanoylphorbol Acetate; Tyrphostins

1993
Inhibitors of cytoskeletal function and signal transduction to study bacterial invasion.
    Methods in enzymology, 1994, Volume: 236

    Topics: Actin Cytoskeleton; Alkaloids; Animals; Bacteria; Catechols; Chelating Agents; Cytochalasins; Cytoskeleton; Genistein; Isoflavones; Nitriles; Nocodazole; Protein Kinase Inhibitors; Signal Transduction; Staurosporine; Tyrphostins; Vinblastine; Vincristine

1994
Activation of protein kinase C down-regulates leukotriene C4 synthase activity and attenuates cysteinyl leukotriene production in an eosinophilic substrain of HL-60 cells.
    Journal of immunology (Baltimore, Md. : 1950), 1994, Jul-15, Volume: 153, Issue:2

    Topics: Alkaloids; Calcimycin; Cysteine; Down-Regulation; Eosinophils; Glutathione Transferase; Humans; Leukemia, Promyelocytic, Acute; Leukotrienes; Nitriles; Phenols; Prostaglandins; Protein Kinase C; Staurosporine; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured; Tyrphostins

1994
A role for tyrosine kinase activation in interleukin-1 beta induced nitric oxide production in the insulin producing cell line RINm-5F.
    Bioscience reports, 1994, Volume: 14, Issue:1

    Topics: Alkaloids; Animals; Catechols; Cell Line; Cyclosporine; Enzyme Activation; Genistein; Insulin; Interleukin-1; Isoflavones; Nitric Oxide; Nitriles; Protein-Tyrosine Kinases; Rats; Staurosporine; Tetradecanoylphorbol Acetate; Tyrphostins

1994
Human growth hormone increases cytosolic free calcium in cultured human IM-9 lymphocytes: a novel mechanism of growth hormone transmembrane signalling.
    Biochemical and biophysical research communications, 1994, Jul-15, Volume: 202, Issue:1

    Topics: Alkaloids; Benzoquinones; Calcium; Catechols; Cell Line; Cell Membrane; Cyclic AMP; Cytosol; Dose-Response Relationship, Drug; Growth Hormone; Humans; Inositol 1,4,5-Trisphosphate; Insulin; Insulin-Like Growth Factor I; Kinetics; Lactams, Macrocyclic; Lymphocytes; Nitriles; Protein-Tyrosine Kinases; Quinones; Rifabutin; Signal Transduction; Staurosporine; Tyrphostins

1994
Suppression of TCDD-induced cytochrome P450 IA1 activity by staurosporine in mouse primary hepatocyte cultures and hepatoma cells.
    Biochemistry and molecular biology international, 1994, Volume: 32, Issue:6

    Topics: Alkaloids; Animals; Blotting, Western; Catechols; Cells, Cultured; Cytochrome P-450 CYP1A1; Cytochrome P-450 Enzyme System; Dose-Response Relationship, Drug; Female; Gene Expression Regulation, Enzymologic; Liver; Liver Neoplasms, Experimental; Mice; Mice, Inbred BALB C; Nitriles; Oxidoreductases; Polychlorinated Dibenzodioxins; Protein-Tyrosine Kinases; Signal Transduction; Staurosporine; Tumor Cells, Cultured; Tyrphostins

1994
The interleukin-6-activated acute-phase response factor is antigenically and functionally related to members of the signal transducer and activator of transcription (STAT) family.
    Molecular and cellular biology, 1994, Volume: 14, Issue:5

    Topics: 3T3 Cells; Alkaloids; Amino Acid Sequence; Animals; Base Sequence; Carcinoma, Hepatocellular; Catechols; Cell Line; Cytokines; DNA-Binding Proteins; Genistein; Growth Inhibitors; Humans; Immune Sera; Interferon-gamma; Interleukin-11; Interleukin-6; Isoflavones; Kinetics; Leukemia Inhibitory Factor; Liver Neoplasms; Lymphokines; Mice; Molecular Sequence Data; Nerve Growth Factors; Nerve Tissue Proteins; Nitriles; Oligodeoxyribonucleotides; Oncostatin M; Peptides; Protein Kinase Inhibitors; Rats; Recombinant Proteins; Signal Transduction; Sphingosine; STAT3 Transcription Factor; Staurosporine; Trans-Activators; Transcription Factors; Tumor Cells, Cultured; Tyrphostins

1994
Synthesis of phosphatidylinositol 3,4-bisphosphate is regulated by protein-tyrosine phosphorylation but the p85 alpha subunit of phosphatidylinositol 3-kinase may not be a target for tyrosine kinases in thrombin-stimulated human platelets.
    Biochimica et biophysica acta, 1994, Jun-02, Volume: 1212, Issue:3

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Blood Platelets; Catechols; Enzyme Activation; Humans; Isoquinolines; Nitriles; Phosphatidylinositol 3-Kinases; Phosphatidylinositol Phosphates; Phosphorylation; Phosphotransferases (Alcohol Group Acceptor); Piperazines; Protein Kinase C; Protein-Tyrosine Kinases; Staurosporine; Tetradecanoylphorbol Acetate; Thrombin; Tyrphostins

1994
Pentoxifylline-stimulated capacitation and acrosome reaction in hamster spermatozoa: involvement of intracellular signalling molecules.
    Molecular human reproduction, 1999, Volume: 5, Issue:7

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Acrosome Reaction; Animals; Aristolochic Acids; Cricetinae; Cyclic AMP; Enzyme Inhibitors; Kinetics; Male; Mesocricetus; Models, Biological; Pentoxifylline; Phenanthrenes; Phospholipases A; Phospholipases A2; Protein Kinase Inhibitors; Protein Kinases; Signal Transduction; Sperm Capacitation; Sperm Motility; Spermatozoa; Staurosporine; Tyrphostins

1999
Kinetic mechanism and inhibitor characterization of WNK1 kinase.
    Biochemistry, 2009, Nov-03, Volume: 48, Issue:43

    Topics: Electrophoretic Mobility Shift Assay; Enzyme Inhibitors; Humans; Inhibitory Concentration 50; Intracellular Signaling Peptides and Proteins; Kinetics; Minor Histocompatibility Antigens; Protein Serine-Threonine Kinases; Pyrazoles; Pyrimidines; Staurosporine; Tyrphostins; WNK Lysine-Deficient Protein Kinase 1

2009