Page last updated: 2024-09-02

st 587 and talipexole

st 587 has been researched along with talipexole in 15 studies

Compound Research Comparison

Studies
(st 587)
Trials
(st 587)
Recent Studies (post-2010)
(st 587)
Studies
(talipexole)
Trials
(talipexole)
Recent Studies (post-2010) (talipexole)
6700426212

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-199013 (86.67)18.7374
1990's2 (13.33)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Batink, H; de Jonge, A; Thoolen, MJ; Timmermans, PB; van Zwieten, PA; Wilffert, B1
Tabrizchi, R; Triggle, CR2
de Jonge, A; Thoolen, MJ; Timmermans, PB; van Zwieten, PA; Wilffert, B1
Eskinder, H; Gross, GJ1
Förstermann, U; Hohlfeld, J; Liebau, S1
De Peyer, JE; Haeusler, G1
Kobinger, W; Pichler, L1
Cooke, JP; Flavahan, NA; Rimele, TJ; Vanhoutte, PM1
Bou, J; Massingham, R1
Kubo, T; Misu, Y; Nagura, J1
Korstanje, C; van Zwieten, PA1
de Jonge, A; Mathy, MJ; Thoolen, MJ; Timmermans, PB; van Zwieten, PA; Wilffert, B1
de Jonge, A; Innemee, HC; Timmermans, PB; van Meel, JC; van Zwieten, PA1
Lues, I; Schümann, HJ1

Other Studies

15 other study(ies) available for st 587 and talipexole

ArticleYear
Quantitative relationships between alpha-adrenergic activity and binding affinity of alpha-adrenoceptor agonists and antagonists.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Blood Pressure; Brain; Cell Membrane; Clonidine; Kinetics; Prazosin; Quinazolines; Rats; Receptors, Adrenergic, alpha; Structure-Activity Relationship; Vasoconstriction

1984
The interrelationship between the effects of captopril and nifedipine on pressor responses elicited by selective alpha-adrenoceptor agonists in the pithed rat preparation.
    Journal of cardiovascular pharmacology, 1992, Volume: 19, Issue:4

    Topics: Adrenergic alpha-Agonists; Animals; Azepines; Blood Pressure; Captopril; Clonidine; Decerebrate State; Imidazoles; Male; Nifedipine; Rats; Rats, Inbred Strains

1992
Effects of staurosporine on the pressor responses to alpha-adrenoceptor agonists in pithed rats: a comparison with nifedipine.
    Pharmacology, 1991, Volume: 43, Issue:3

    Topics: Adrenergic alpha-Agonists; Alkaloids; Animals; Azepines; Blood Pressure; Clonidine; Decerebrate State; Imidazoles; Male; Muscle, Smooth, Vascular; Nifedipine; Protein Kinase C; Rats; Rats, Inbred Strains; Staurosporine

1991
Calcium dependency of vasoconstriction mediated by alpha 1- and alpha 2-adrenoceptors.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Azepines; Blood Pressure; Calcium; Calcium Channel Blockers; Clonidine; Imidazoles; Ion Channels; Nifedipine; Rats; Receptors, Adrenergic, alpha; Regional Blood Flow; Structure-Activity Relationship; Vasoconstriction

1985
Sensitivity of alpha-adrenoceptor agonists to the calcium channel activator, Bay K 8644, in canine saphenous vein.
    Pharmacology, 1987, Volume: 35, Issue:5

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenergic alpha-Agonists; Animals; Azepines; Clonidine; Dogs; Female; In Vitro Techniques; Ion Channels; Male; Muscle, Smooth, Vascular; Saphenous Vein

1987
The inhibition of alpha 1-adrenoceptor-mediated contractions of rabbit pulmonary artery by Ca2+-withdrawal, pertussis toxin and N-ethylmaleimide is dependent on agonist intrinsic efficacy.
    Naunyn-Schmiedeberg's archives of pharmacology, 1989, Volume: 339, Issue:5

    Topics: Adrenergic alpha-Agonists; Animals; Azepines; Calcium; Calcium Channel Blockers; Clonidine; Ethylmaleimide; Female; Gallic Acid; In Vitro Techniques; Male; Methoxamine; Muscle Contraction; Muscle, Smooth, Vascular; Pertussis Toxin; Phenylephrine; Pulmonary Artery; Rabbits; Receptors, Adrenergic, alpha; Virulence Factors, Bordetella

1989
Electrical membrane events in response to alpha-adrenoceptor stimulation.
    Clinical science (London, England : 1979), 1985, Volume: 68 Suppl 10

    Topics: Adrenergic alpha-Agonists; Animals; Azepines; Calcium; Cell Membrane; Clonidine; Female; Male; Membrane Potentials; Methoxamine; Muscle Contraction; Muscle, Smooth, Vascular; Potassium; Pulmonary Artery; Rabbits; Receptors, Adrenergic, alpha; Stimulation, Chemical; Strychnine

1985
Alpha 2-adrenoceptor blocking properties of the alpha 1-selective agonist 2-(2-chloro-5-trifluoromethylphenylimino)imidazolidine (St 587).
    Arzneimittel-Forschung, 1985, Volume: 35, Issue:1A

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Behavior, Animal; Clonidine; Dogs; Drug Interactions; Electric Stimulation; Exploratory Behavior; Female; Heart Rate; Male; Mice; Prazosin; Pressoreceptors; Rats; Spinal Cord; Vagotomy

1985
Nimodipine and inhibition of alpha adrenergic activation of the isolated canine saphenous vein.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 234, Issue:3

    Topics: Adrenergic alpha-Agonists; Animals; Azepines; Calcium Channel Blockers; Clonidine; Dogs; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Male; Nicotinic Acids; Nimodipine; Potassium; Receptors, Adrenergic, alpha; Saphenous Vein; Tyramine; Vasoconstriction

1985
Effect of diltiazem upon contractile responses to phenylephrine, cirazoline, Sgd 101/75, St 587 and B-HT 920 in rabbit aorta and dog saphenous vein preparations.
    European journal of pharmacology, 1986, Mar-04, Volume: 121, Issue:3

    Topics: Adrenergic alpha-Agonists; Animals; Aorta, Thoracic; Azepines; Benzazepines; Clonidine; Diltiazem; Dogs; Drug Interactions; Female; Imidazoles; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Phenylephrine; Rabbits; Saphenous Vein

1986
Pharmacological characterization of spinal alpha adrenoceptors related to blood pressure control in rats.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 240, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Azepines; Blood Pressure; Brain Stem; Clonidine; Dopamine; Guanabenz; Hydroxydopamines; Injections, Spinal; Male; Norepinephrine; Oxidopamine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Spinal Cord; Yohimbine

1987
Characterization of alpha-adrenoreceptor mediated reduction of flow in a saline-perfused constant pressure model of rat perfused hindquarters.
    Journal of autonomic pharmacology, 1987, Volume: 7, Issue:1

    Topics: Acid-Base Equilibrium; Adrenergic alpha-Agonists; Angiotensin II; Animals; Azepines; Blood Pressure; Calcium; Clonidine; Dinoprost; Gallopamil; Hindlimb; Male; Perfusion; Potassium Chloride; Prostaglandins F; Rats; Receptors, Adrenergic, alpha; Regional Blood Flow; Reserpine

1987
Effects of the irreversible alpha-adrenoceptor antagonists phenoxybenzamine and benextramine on the effectiveness of nifedipine in inhibiting alpha 1- and alpha 2-adrenoceptor mediated vasoconstriction in pithed rats.
    Naunyn-Schmiedeberg's archives of pharmacology, 1985, Volume: 329, Issue:4

    Topics: Animals; Azepines; Clonidine; Cystamine; Decerebrate State; Diastole; Dose-Response Relationship, Drug; Imidazoles; Male; Nifedipine; Phenoxybenzamine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Vasoconstriction

1985
Differential effects of selective alpha 1- and alpha 2-adrenoceptor agonists on intraocular pressure in the conscious rabbit.
    Documenta ophthalmologica. Advances in ophthalmology, 1982, Jan-29, Volume: 52, Issue:3-4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Clonidine; Female; Intraocular Pressure; Male; Phenylephrine; Procaine; Pupil; Yohimbine

1982
Effect of removing the endothelial cells on the reactivity of rat aortic segments to different alpha-adrenoceptor agonists.
    Naunyn-Schmiedeberg's archives of pharmacology, 1984, Volume: 328, Issue:2

    Topics: Adrenergic alpha-Agonists; Animals; Aorta, Thoracic; Azepines; Clonidine; Endothelium; Imidazoles; In Vitro Techniques; Male; Methoxamine; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Rats; Rats, Inbred Strains; Xylazine; Yohimbine

1984