Page last updated: 2024-09-02

st 587 and phenylephrine

st 587 has been researched along with phenylephrine in 15 studies

Compound Research Comparison

Studies
(st 587)
Trials
(st 587)
Recent Studies (post-2010)
(st 587)
Studies
(phenylephrine)
Trials
(phenylephrine)
Recent Studies (post-2010) (phenylephrine)
670013,7978572,083

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-199010 (66.67)18.7374
1990's5 (33.33)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Batink, H; de Jonge, A; Thoolen, MJ; Timmermans, PB; van Zwieten, PA; Wilffert, B1
Esbenshade, TA; Han, C; Hollinger, S; Minneman, KP; Theroux, TL1
Armah, BI; Göthert, M; Molderings, GJ1
Förstermann, U; Hohlfeld, J; Liebau, S1
Badia, A; Sallés, J1
Harsing, LG; Somogyi, GT; Vizi, ES; Zimanyi, I1
Bou, J; Massingham, R1
Chiu, AT; McCall, DE; Thoolen, MJ; Timmermans, PB1
Geiger, G; Grimes, D; Heaslip, RJ; Henry, DE; Lee, DK; Rimele, TJ1
Cooke, JP; Flavahan, NA; Rimele, TJ; Vanhoutte, PM1
de Jonge, A; Innemee, HC; Timmermans, PB; van Meel, JC; van Zwieten, PA1
de Jonge, A; Kalkman, HO; Mathy, MJ; Thoolen, MJ; Timmermans, PB; van Meel, JC; van Zwieten, PA; Wilffert, B1
Faber, JE; Tateishi, J1
Giraldo, J; Tabernero, A; Vila, E1
Hasegawa, Y; Ono, H; Wada, T1

Other Studies

15 other study(ies) available for st 587 and phenylephrine

ArticleYear
Quantitative relationships between alpha-adrenergic activity and binding affinity of alpha-adrenoceptor agonists and antagonists.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Blood Pressure; Brain; Cell Membrane; Clonidine; Kinetics; Prazosin; Quinazolines; Rats; Receptors, Adrenergic, alpha; Structure-Activity Relationship; Vasoconstriction

1984
Selectivity of agonists for cloned alpha 1-adrenergic receptor subtypes.
    Molecular pharmacology, 1994, Volume: 46, Issue:5

    Topics: Adrenergic alpha-1 Receptor Agonists; Animals; Binding, Competitive; Catecholamines; Cattle; Cell Line; Cloning, Molecular; Cricetinae; Humans; Imidazoles; Inositol Phosphates; Phenethylamines; Phenoxybenzamine; Radioligand Assay; Rats; Receptors, Adrenergic, alpha-1; Recombinant Proteins; Tetralones

1994
Effect of temperature on alpha 2- and alpha 1-adrenoceptor-mediated responses in the pithed rat and in the rat vena cava.
    Journal of autonomic pharmacology, 1990, Volume: 10, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Animals; Clonidine; Cold Temperature; Dose-Response Relationship, Drug; Imidazoles; Male; Norepinephrine; Phenylephrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Neurotransmitter; Temperature; Tritium; Tyramine; Vena Cava, Inferior

1990
The inhibition of alpha 1-adrenoceptor-mediated contractions of rabbit pulmonary artery by Ca2+-withdrawal, pertussis toxin and N-ethylmaleimide is dependent on agonist intrinsic efficacy.
    Naunyn-Schmiedeberg's archives of pharmacology, 1989, Volume: 339, Issue:5

    Topics: Adrenergic alpha-Agonists; Animals; Azepines; Calcium; Calcium Channel Blockers; Clonidine; Ethylmaleimide; Female; Gallic Acid; In Vitro Techniques; Male; Methoxamine; Muscle Contraction; Muscle, Smooth, Vascular; Pertussis Toxin; Phenylephrine; Pulmonary Artery; Rabbits; Receptors, Adrenergic, alpha; Virulence Factors, Bordetella

1989
Effects of St-587 on the alpha-adrenoceptors in the bisected rat vas deferens.
    The Journal of pharmacy and pharmacology, 1989, Volume: 41, Issue:9

    Topics: Animals; Clonidine; Electric Stimulation; Epididymis; In Vitro Techniques; Male; Muscle, Smooth; Phenylephrine; Prazosin; Prostate; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Vas Deferens; Yohimbine

1989
Release of [3H]noradrenaline by alpha 1-adrenoceptor agonists.
    Neurochemical research, 1986, Volume: 11, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Clonidine; Cocaine; In Vitro Techniques; Male; Mice; Norepinephrine; Phenylephrine; Temperature; Vas Deferens

1986
Effect of diltiazem upon contractile responses to phenylephrine, cirazoline, Sgd 101/75, St 587 and B-HT 920 in rabbit aorta and dog saphenous vein preparations.
    European journal of pharmacology, 1986, Mar-04, Volume: 121, Issue:3

    Topics: Adrenergic alpha-Agonists; Animals; Aorta, Thoracic; Azepines; Benzazepines; Clonidine; Diltiazem; Dogs; Drug Interactions; Female; Imidazoles; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Phenylephrine; Rabbits; Saphenous Vein

1986
Ca++ utilization in the constriction of rat aorta to full and partial alpha-1 adrenoceptor agonists.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 238, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Aorta; Calcium; Clonidine; Dose-Response Relationship, Drug; Ethanolamines; Imidazoles; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phenylephrine; Potassium; Rats; Rats, Inbred Strains; Tetrahydronaphthalenes

1986
Tissue-dependent alpha adrenoceptor activity of buspirone and related compounds.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:3

    Topics: Animals; Buspirone; Cerebral Cortex; Clonidine; Guinea Pigs; Male; Norepinephrine; Phenylephrine; Prazosin; Pyrimidines; Rabbits; Rats; Receptors, Adrenergic, alpha; Vas Deferens

1987
Characterization of postjunctional alpha-1 and alpha-2 adrenoceptors activated by exogenous or nerve-released norepinephrine in the canine saphenous vein.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 230, Issue:3

    Topics: Animals; Clonidine; Dogs; Dose-Response Relationship, Drug; Electric Stimulation; Female; Imidazoles; Male; Methoxamine; Norepinephrine; Phenoxybenzamine; Phenylephrine; Prazosin; Receptors, Adrenergic, alpha; Saphenous Vein; Sympathetic Nervous System; Tyramine; Yohimbine

1984
Differential effects of selective alpha 1- and alpha 2-adrenoceptor agonists on intraocular pressure in the conscious rabbit.
    Documenta ophthalmologica. Advances in ophthalmology, 1982, Jan-29, Volume: 52, Issue:3-4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Clonidine; Female; Intraocular Pressure; Male; Phenylephrine; Procaine; Pupil; Yohimbine

1982
Differential effect of calcium entry blockers on alpha 1-adrenoceptor-mediated vasoconstriction in vivo.
    Naunyn-Schmiedeberg's archives of pharmacology, 1983, Volume: 324, Issue:4

    Topics: Adrenergic alpha-Agonists; Animals; Blood Pressure; Calcium Channel Blockers; Catecholamines; Clonidine; Ethanolamines; Imidazoles; Imidazolines; Male; Methoxamine; Nifedipine; Phenylephrine; Rats; Rats, Inbred Strains; Vasoconstriction; Verapamil

1983
ATP-sensitive K+ channels mediate alpha 2D-adrenergic receptor contraction of arteriolar smooth muscle and reversal of contraction by hypoxia.
    Circulation research, 1995, Volume: 76, Issue:1

    Topics: Adenosine Triphosphate; Animals; Brimonidine Tartrate; Cell Hypoxia; Clonidine; Glyburide; In Vitro Techniques; Muscle, Smooth, Vascular; Nitroprusside; Phenylephrine; Potassium Channels; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Vasoconstriction

1995
Effect of NG-nitro-L-arginine methylester (L-NAME) on functional and biochemical alpha 1-adrenoceptor-mediated responses in rat blood vessels.
    British journal of pharmacology, 1996, Volume: 117, Issue:4

    Topics: Adrenergic alpha-Agonists; Animals; Arginine; Arteries; Clonidine; In Vitro Techniques; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Phenoxybenzamine; Phenylephrine; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Tail; Vasoconstriction

1996
Characterization of alpha1-adrenoceptor subtypes in facilitation of rat spinal motoneuron activity.
    European journal of pharmacology, 1997, Dec-04, Volume: 340, Issue:1

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Bridged-Ring Compounds; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Electric Stimulation; Epinephrine; Male; Methoxamine; Motor Neurons; Norepinephrine; Oxazines; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Spinal Cord

1997