Page last updated: 2024-09-02

st 1435 and pregnanolone

st 1435 has been researched along with pregnanolone in 3 studies

Compound Research Comparison

Studies
(st 1435)
Trials
(st 1435)
Recent Studies (post-2010)
(st 1435)
Studies
(pregnanolone)
Trials
(pregnanolone)
Recent Studies (post-2010) (pregnanolone)
9731331,984111666

Protein Interaction Comparison

ProteinTaxonomyst 1435 (IC50)pregnanolone (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.101
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.101
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.101
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.101
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.101
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.101
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.101
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.101
Sodium- and chloride-dependent GABA transporter 1Rattus norvegicus (Norway rat)0.117
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.101
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.101
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.101
Sodium- and chloride-dependent GABA transporter 2Rattus norvegicus (Norway rat)0.117
Sodium- and chloride-dependent GABA transporter 3Rattus norvegicus (Norway rat)0.117
Sodium- and chloride-dependent betaine transporterRattus norvegicus (Norway rat)0.117
Gamma-aminobutyric acid receptor subunit alpha-1Mus musculus (house mouse)0.071
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.101
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.101
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.101
GABA theta subunitRattus norvegicus (Norway rat)0.101
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.101

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (33.33)29.6817
2010's2 (66.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Begliuomini, S; Casarosa, E; Genazzani, AR; Giannini, A; Kumar, N; Lenzi, E; Luisi, M; Merlini, S; Pluchino, N; Sitruk-Ware, R1
Coqueran, B; De Nicola, AF; Delespierre, B; Guennoun, R; Labombarda, F; Liere, P; Liu, A; Lydon, JP; Marchand-Leroux, C; Margaill, I; Mattern, C; O'Malley, BW; Plotkine, M; Schumacher, M; Sitruk-Ware, R; Zhang, S1
El-Etr, M; Fagart, J; Knibb, AR; Kumar, N; Lambert, JJ; Liere, P; Mitchell, SJ; Petit-Topin, I; Rafestin-Oblin, ME; Rame, M; Schumacher, M; Sitruk-Ware, R1

Other Studies

3 other study(ies) available for st 1435 and pregnanolone

ArticleYear
Central modifications of allopregnanolone and beta-endorphin following subcutaneous administration of Nestorone.
    The Journal of steroid biochemistry and molecular biology, 2009, Volume: 116, Issue:1-2

    Topics: Animals; beta-Endorphin; Brain; Contraceptive Agents, Female; Female; Hippocampus; Hypothalamus; Infusions, Subcutaneous; Models, Animal; Neurotransmitter Agents; Norprogesterones; Ovariectomy; Pregnanolone; Rats; Rats, Wistar

2009
Progesterone receptors: a key for neuroprotection in experimental stroke.
    Endocrinology, 2012, Volume: 153, Issue:8

    Topics: Animals; Brain; Male; Mice; Mice, Knockout; Norprogesterones; Pregnanolone; Progesterone; Receptors, Progesterone; Signal Transduction; Stroke

2012
Nestorone® as a Novel Progestin for Nonoral Contraception: Structure-Activity Relationships and Brain Metabolism Studies.
    Endocrinology, 2017, 01-01, Volume: 158, Issue:1

    Topics: Animals; Brain; Contraceptive Agents, Female; HEK293 Cells; Humans; Mice; Norprogesterones; Patch-Clamp Techniques; Pregnanolone; Receptors, Androgen; Receptors, GABA-A; Receptors, Progesterone; Structure-Activity Relationship

2017