Page last updated: 2024-08-26

sr141716 and naloxone

sr141716 has been researched along with naloxone in 55 studies

Research

Studies (55)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's9 (16.36)18.2507
2000's32 (58.18)29.6817
2010's14 (25.45)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Bánki, L; Deli, MA; Dvorácskó, S; Horváth, G; Kékesi, G; Keresztes, A; Macedonio, G; Mollica, A; Pieretti, S; Stefanucci, A; Tömböly, C; Tuboly, G; Walter, FR; Zádor, F1
Le Fur, G; Michaud, JC; Soubrié, P; Terranova, JP1
Brown, RE; Dastur, FN; McGregor, IS; McLellan, RA1
French, ED1
Di Chiara, G; Pontieri, FE; Tanda, G1
Coutts, AA; Pertwee, RG1
Chowen, J; de Fonseca, FR; del Arco, I; Koob, GF; Martin, Y; Navarro, M; Roberts, AJ; Rocío A Carrera, M; Villanúa, MA1
Gallate, JE; McGregor, IS1
Gallate, JE; Mallet, PE; McGregor, IS; Saharov, T1
Corchero, J; Fuentes, JA; Manzanares, J1
Keniston, L; Lu, J; Mao, J; Mayer, DJ; Price, DD1
Kirkham, TC; Williams, CM1
Braida, D; Parolaro, D; Pozzi, M; Sala, M1
Clarke, RW; Harris, J; Jenkins, S; Witton, SK1
Capasso, F; Capasso, R; Di Carlo, G; Izzo, AA; Mascolo, N; Pinto, L1
Caneparo, A; Da Nascimento, S; Le Fur, G; Mas-Nieto, M; Noble, F; Pommier, B; Roques, BP; Tzavara, ET1
Carrera, MR; Chowen, JA; Cossu, G; del Arco, I; Fattore, L; Fratta, W; Gomez, R; Koob, GF; Maldonado, R; Navarro, M; Rodriguez de Fonseca, F; Valverde, O; Villanua, MA1
Braida, D; Cavallini, R; Pozzi, M; Sala, M1
Capasso, F; Capasso, R; Di Marzo, V; Fezza, F; Izzo, AA; Mascolo, N; Pinto, A1
Mukherjee, M; Robertson, K; Rowland, NE1
Pietras, TA; Rowland, NE1
Brunetti, G; Carai, MA; Colombo, G; Gessa, GL; Serra, S; Vacca, G1
De Miguel, R; Fernández, B; Gomez, N; Guaza, C; Ramos, JA; Romero, EM; Sagredo, O; Urigüen, L; Viveros, MP1
Assini, FL; Ramos, GA; Takahashi, RN1
Gallate, JE; Mallet, PE; McGregor, IS1
Cox, ML; Welch, SP1
Niederhoffer, N; Pfitzer, T; Szabo, B1
Borrelli, F; Capasso, F; Capasso, R; Izzo, AA; Mascolo, N1
Cossu, G; Deiana, S; Fadda, P; Fattore, L; Fratta, W; Spano, MS1
Braida, D; Iosuè, S; Pegorini, S; Sala, M1
Cossu, G; Deiana, S; Fadda, P; Fattore, L; Fratta, W; Spano, S1
Maor, Y; Mechoulam, R; Pertwee, RG; Stevenson, LA; Thomas, A1
Amico, MC; Morrone, LA; Palmery, M; Romanelli, L; Tucci, P; Valeri, P1
Adrian, R; Baratta, J; Giuffrida, A; Piomelli, D; Solbrig, MV1
De Vries, TJ; Hogenboom, F; Schoffelmeer, AN; Wardeh, G1
Evenden, J; Ko, T1
Trezza, V; Vanderschuren, LJ1
Canals, M; Milligan, G1
Blundell, JE; Rodgers, RJ; Tallett, AJ1
Inno, J; Kurrikoff, K; Matsui, T; Vasar, E1
Baarendse, PJ; Trezza, V; Vanderschuren, LJ1
Allen, CP; Lang, ST; Leri, F; Manwell, LA; Parker, LA; Satvat, E1
Dimitrov, EL; Petrus, E; Usdin, TB1
Castelli, MP; Ennas, MG; Lecca, S; Luchicchi, A; Melis, M; Muntoni, AL; Pistis, M1
Fadda, P; Fattore, L; Fratta, W; Melis, V; Spano, M1
Hillman, C; Rasmussen, EB1
Lecca, S; Luchicchi, A; Melis, M; Muntoni, AL; Pistis, M1
Craft, RM; Laggart, JD; Tsutsui, KT; Wakley, AA1
Rodgers, RJ; Wright, FL1
Lockie, SH; Oldfield, BJ; Stefanidis, A; Tschöp, MH1
Davies, AJ; Kim, D; Lee, JY; Oh, SB; Park, J; Pickering, AE; Vang, H1
Kang, Y; Kim, D; Lee, GJ; Lee, JY; Lee, PR; Oh, SB; Won, CH1

Other Studies

55 other study(ies) available for sr141716 and naloxone

ArticleYear
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Preparation of bivalent agonists for targeting the mu opioid and cannabinoid receptors.
    European journal of medicinal chemistry, 2019, Sep-15, Volume: 178

    Topics: Analgesics, Opioid; Animals; Dose-Response Relationship, Drug; Enkephalins; Indoles; Mice; Molecular Structure; Naphthalenes; Oxycodone; Rats; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Receptors, Opioid, mu; Structure-Activity Relationship

2019
Inhibition of long-term potentiation in rat hippocampal slices by anandamide and WIN55212-2: reversal by SR141716 A, a selective antagonist of CB1 cannabinoid receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1995, Volume: 352, Issue:5

    Topics: Animals; Arachidonic Acids; Benzoxazines; Cannabinoids; Endocannabinoids; Evoked Potentials; Hippocampus; In Vitro Techniques; Long-Term Potentiation; Male; Morpholines; Naloxone; Naphthalenes; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Receptors, Cannabinoid; Receptors, Drug; Rimonabant

1995
Cannabinoid modulation of rat pup ultrasonic vocalizations.
    European journal of pharmacology, 1996, Oct-10, Volume: 313, Issue:1-2

    Topics: Analysis of Variance; Animals; Animals, Newborn; Behavior, Animal; Benzazepines; Body Temperature; Cannabinoids; Cyclohexanols; Dopamine Antagonists; Dose-Response Relationship, Drug; Flumazenil; GABA Modulators; Hypothermia; Motor Activity; Naloxone; Narcotic Antagonists; Piperidines; Pyrazoles; Rats; Rimonabant; Vocalization, Animal

1996
delta9-Tetrahydrocannabinol excites rat VTA dopamine neurons through activation of cannabinoid CB1 but not opioid receptors.
    Neuroscience letters, 1997, May-02, Volume: 226, Issue:3

    Topics: Animals; Cannabinoids; Dopamine; Dose-Response Relationship, Drug; Dronabinol; Male; Naloxone; Narcotic Antagonists; Neurons; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptors, Cannabinoid; Receptors, Drug; Receptors, Opioid; Rimonabant; Stimulation, Chemical; Ventral Tegmental Area

1997
Cannabinoid and heroin activation of mesolimbic dopamine transmission by a common mu1 opioid receptor mechanism.
    Science (New York, N.Y.), 1997, Jun-27, Volume: 276, Issue:5321

    Topics: Animals; Benzoxazines; Dopamine; Dronabinol; Heroin; Male; Microdialysis; Morpholines; Naloxone; Naphthalenes; Narcotic Antagonists; Nucleus Accumbens; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptors, Cannabinoid; Receptors, Drug; Receptors, Opioid, mu; Rimonabant

1997
Inhibition by cannabinoid receptor agonists of acetylcholine release from the guinea-pig myenteric plexus.
    British journal of pharmacology, 1997, Volume: 121, Issue:8

    Topics: Acetylcholine; Benzoxazines; Child, Preschool; Cyclohexanols; Histamine; Humans; In Vitro Techniques; Male; Morpholines; Myenteric Plexus; Naloxone; Naphthalenes; Norepinephrine; Piperidines; Pyrazoles; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Stereoisomerism

1997
CB1 cannabinoid receptor antagonist-induced opiate withdrawal in morphine-dependent rats.
    Neuroreport, 1998, Oct-26, Volume: 9, Issue:15

    Topics: Animals; Brain Chemistry; Gene Expression; In Situ Hybridization; Male; Morphine Dependence; Naloxone; Narcotic Antagonists; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptors, Cannabinoid; Receptors, Drug; Receptors, Opioid, mu; Rimonabant; RNA, Messenger; Substance Withdrawal Syndrome

1998
The motivation for beer in rats: effects of ritanserin, naloxone and SR 141716.
    Psychopharmacology, 1999, Volume: 142, Issue:3

    Topics: Alcohol Drinking; Animals; Beer; Ethanol; Male; Motivation; Motor Activity; Naloxone; Narcotic Antagonists; Piperidines; Pyrazoles; Rats; Rats, Wistar; Rimonabant; Ritanserin; Serotonin Antagonists

1999
Increased motivation for beer in rats following administration of a cannabinoid CB1 receptor agonist.
    European journal of pharmacology, 1999, Apr-16, Volume: 370, Issue:3

    Topics: Animals; Beer; Cannabinoids; Cyclohexanols; Dose-Response Relationship, Drug; Drinking Behavior; Ethanol; Male; Motor Activity; Naloxone; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptors, Cannabinoid; Receptors, Drug; Receptors, Opioid; Rimonabant; Self Administration; Sucrose

1999
Opioid and cannabinoid receptor-mediated regulation of the increase in adrenocorticotropin hormone and corticosterone plasma concentrations induced by central administration of delta(9)-tetrahydrocannabinol in rats.
    Brain research, 1999, Aug-21, Volume: 839, Issue:1

    Topics: Adrenocorticotropic Hormone; Analysis of Variance; Animals; Corticosterone; Dronabinol; Injections, Intraventricular; Male; Naloxone; Narcotic Antagonists; Piperidines; Pituitary-Adrenal System; Psychotropic Drugs; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptors, Cannabinoid; Receptors, Drug; Receptors, Opioid; Rimonabant

1999
Two distinctive antinociceptive systems in rats with pathological pain.
    Neuroscience letters, 2000, Feb-11, Volume: 280, Issue:1

    Topics: Analgesics, Non-Narcotic; Animals; Cannabinoids; Dizocilpine Maleate; Dronabinol; Drug Tolerance; Hot Temperature; Hyperalgesia; Injections, Spinal; Male; Morphine; Naloxone; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Sciatic Nerve

2000
Synergistic efects of opioid and cannabinoid antagonists on food intake.
    Psychopharmacology, 2001, Jan-01, Volume: 153, Issue:2

    Topics: Animals; Cannabinoid Receptor Modulators; Cannabinoids; Drug Synergism; Eating; Male; Naloxone; Narcotic Antagonists; Piperidines; Pyrazoles; Rats; Rimonabant

2001
Intracerebral self-administration of the cannabinoid receptor agonist CP 55,940 in the rat: interaction with the opioid system.
    European journal of pharmacology, 2001, Feb-16, Volume: 413, Issue:2-3

    Topics: Analgesics; Analgesics, Opioid; Animals; Benzimidazoles; Conditioning, Operant; Cyclohexanols; Heroin; Male; Naloxone; Narcotic Antagonists; Narcotics; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptors, Cannabinoid; Receptors, Drug; Reinforcement Schedule; Rimonabant; Self Administration

2001
Cannabinoidergic and opioidergic inhibition of spinal reflexes in the decerebrated, spinalized rabbit.
    Neuropharmacology, 2001, Volume: 40, Issue:4

    Topics: Animals; Decerebrate State; Dose-Response Relationship, Drug; Dronabinol; Female; Fentanyl; Male; Naloxone; Narcotic Antagonists; Piperidines; Pyrazoles; Rabbits; Receptors, Cannabinoid; Receptors, Drug; Reflex; Rimonabant; Spinal Cord; Spinal Cord Injuries

2001
Effect of vanilloid drugs on gastrointestinal transit in mice.
    British journal of pharmacology, 2001, Volume: 132, Issue:7

    Topics: Alkaloids; Animals; Arachidonic Acids; Benzodioxoles; Capsaicin; Dose-Response Relationship, Drug; Endocannabinoids; Gastrointestinal Transit; Hexamethonium; Male; Mice; Mice, Inbred ICR; Naloxone; NG-Nitroarginine Methyl Ester; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptors, Drug; Rimonabant; Yohimbine

2001
Reduction of opioid dependence by the CB(1) antagonist SR141716A in mice: evaluation of the interest in pharmacotherapy of opioid addiction.
    British journal of pharmacology, 2001, Volume: 132, Issue:8

    Topics: Animals; Brain Chemistry; Cannabinoids; Conditioning, Operant; Dynorphins; Male; Mice; Naloxone; Narcotic Antagonists; Opioid-Related Disorders; Piperidines; Pyrazoles; Radioimmunoassay; Receptors, Cannabinoid; Receptors, Drug; Receptors, Opioid, kappa; Rimonabant; Substance Withdrawal Syndrome; Synapses

2001
Functional interaction between opioid and cannabinoid receptors in drug self-administration.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2001, Jul-15, Volume: 21, Issue:14

    Topics: Animals; Avoidance Learning; Cannabinoids; Caudate Nucleus; Conditioning, Operant; Disease Models, Animal; Heroin; Heroin Dependence; Male; Mice; Morphine; Morphine Dependence; Naloxone; Narcotic Antagonists; Nucleus Accumbens; Piperidines; Putamen; Pyrazoles; Rats; Rats, Wistar; Receptors, Cannabinoid; Receptors, Drug; Receptors, Opioid; Rimonabant; RNA, Messenger; Self Administration; Septum of Brain

2001
Conditioned place preference induced by the cannabinoid agonist CP 55,940: interaction with the opioid system.
    Neuroscience, 2001, Volume: 104, Issue:4

    Topics: Analgesics; Analgesics, Opioid; Animals; Brain; Conditioning, Psychological; Cyclohexanols; Dose-Response Relationship, Drug; Drug Interactions; Heroin; Male; Naloxone; Narcotic Antagonists; Opioid Peptides; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptors, Cannabinoid; Receptors, Drug; Reward; Rimonabant

2001
Inhibitory effect of palmitoylethanolamide on gastrointestinal motility in mice.
    British journal of pharmacology, 2001, Volume: 134, Issue:5

    Topics: Adrenergic alpha-Antagonists; Amides; Animals; Anti-Inflammatory Agents, Non-Steroidal; Camphanes; Croton Oil; Dose-Response Relationship, Drug; Endocannabinoids; Enzyme Inhibitors; Ethanolamines; Gastrointestinal Motility; Gastrointestinal Transit; Hexamethonium; Inflammation; Intestine, Small; Male; Mice; Mice, Inbred ICR; Naloxone; NG-Nitroarginine Methyl Ester; Nicotinic Antagonists; Nitric Oxide Synthase; Palmitic Acids; Phenylmethylsulfonyl Fluoride; Piperidines; Pyrazoles; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Yohimbine

2001
Effects of the cannabinoid receptor antagonist SR 141716, alone and in combination with dexfenfluramine or naloxone, on food intake in rats.
    Psychopharmacology, 2001, Volume: 159, Issue:1

    Topics: Animals; Dexfenfluramine; Dose-Response Relationship, Drug; Drug Combinations; Drug Synergism; Eating; Female; Male; Naloxone; Narcotic Antagonists; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Serotonin Receptor Agonists

2001
Effect of opioid and cannabinoid receptor antagonism on orphanin FQ-induced hyperphagia in rats.
    European journal of pharmacology, 2002, May-10, Volume: 442, Issue:3

    Topics: Animals; Dose-Response Relationship, Drug; Drug Synergism; Eating; Female; Hyperphagia; Male; Naloxone; Narcotic Antagonists; Nociceptin; Opioid Peptides; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptors, Cannabinoid; Receptors, Drug; Rimonabant

2002
Boosting effect of morphine on alcohol drinking is suppressed not only by naloxone but also by the cannabinoid CB1 receptor antagonist, SR 141716.
    European journal of pharmacology, 2002, Jun-07, Volume: 445, Issue:1-2

    Topics: Alcohol Drinking; Animals; Dose-Response Relationship, Drug; Male; Morphine; Naloxone; Piperidines; Pyrazoles; Rats; Receptors, Cannabinoid; Receptors, Drug; Rimonabant

2002
Antinociceptive, behavioural and neuroendocrine effects of CP 55,940 in young rats.
    Brain research. Developmental brain research, 2002, Jun-30, Volume: 136, Issue:2

    Topics: Analgesics; Animals; Behavior, Animal; Cannabinoids; Corticosterone; Cyclohexanols; Dopamine; Dose-Response Relationship, Drug; Drug Interactions; Female; Grooming; Male; Marijuana Abuse; Morphine; Motor Activity; Naloxone; Narcotic Antagonists; Neostriatum; Neurosecretory Systems; Nociceptors; Pain Measurement; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Sex Characteristics

2002
Anxiety does not affect the antinociceptive effect of Delta 9-THC in mice: participation of cannabinoid and opioid receptors.
    Pharmacology, biochemistry, and behavior, 2003, Volume: 75, Issue:4

    Topics: Animals; Anxiety; Cannabinoid Receptor Antagonists; Dose-Response Relationship, Drug; Dronabinol; Male; Mice; Naloxone; Narcotic Antagonists; Pain Measurement; Piperidines; Pyrazoles; Receptors, Cannabinoid; Receptors, Opioid; Rimonabant

2003
Combined low dose treatment with opioid and cannabinoid receptor antagonists synergistically reduces the motivation to consume alcohol in rats.
    Psychopharmacology, 2004, Volume: 173, Issue:1-2

    Topics: Alcohol Drinking; Animals; Cannabinoids; Dose-Response Relationship, Drug; Drug Combinations; Drug Synergism; Male; Motivation; Naloxone; Naltrexone; Narcotic Antagonists; Piperidines; Pyrazoles; Rats; Rats, Wistar; Rimonabant

2004
The antinociceptive effect of Delta9-tetrahydrocannabinol in the arthritic rat.
    European journal of pharmacology, 2004, Jun-16, Volume: 493, Issue:1-3

    Topics: Animals; Arthritis, Experimental; Cannabinoid Receptor Antagonists; Dose-Response Relationship, Drug; Dronabinol; Dynorphins; Enkephalin, Leucine; Enkephalin, Methionine; Freund's Adjuvant; Injections, Intradermal; Injections, Intraperitoneal; Male; Morphine; Mycobacterium; Naloxone; Naltrexone; Narcotic Antagonists; Pain; Pain Measurement; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptors, Opioid; Rimonabant

2004
Central effects of the cannabinoid receptor agonist WIN55212-2 on respiratory and cardiovascular regulation in anaesthetised rats.
    British journal of pharmacology, 2004, Volume: 142, Issue:6

    Topics: Analgesics, Opioid; Anesthesia; Animals; Benzoxazines; Blood Pressure; Cannabinoid Receptor Agonists; Cannabinoid Receptor Antagonists; Cardiovascular Physiological Phenomena; Cisterna Magna; Dose-Response Relationship, Drug; Drug Interactions; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Heart Rate; Injections; Male; Morpholines; Naloxone; Naphthalenes; Norepinephrine; Piperidines; Pyrazoles; Rats; Rats, Wistar; Respiration; Rimonabant; Tidal Volume

2004
Inhibitory effect of the antidepressant St. John's wort (hypericum perforatum) on rat bladder contractility in vitro.
    Urology, 2004, Volume: 64, Issue:1

    Topics: Acetylcholine; Adenosine Triphosphate; Animals; Anthracenes; Antidepressive Agents; Atropine; Bridged Bicyclo Compounds; Capsaicin; Depression; Electric Stimulation; Female; Haloperidol; Hypericum; Kaempferols; Male; Methysergide; Muscle Contraction; Muscle, Smooth; Naloxone; Perylene; Phentolamine; Phloroglucinol; Piperidines; Plant Extracts; Propranolol; Pyrazoles; Quercetin; Rats; Rats, Wistar; Rimonabant; Rutin; Terpenes; Tetrodotoxin; Urinary Bladder; Urinary Incontinence; Verapamil

2004
CB1 receptor agonist and heroin, but not cocaine, reinstate cannabinoid-seeking behaviour in the rat.
    British journal of pharmacology, 2004, Volume: 143, Issue:3

    Topics: Animals; Behavior, Animal; Benzoxazines; Cannabinoids; Cocaine; Extinction, Psychological; Heroin; Male; Morpholines; Naloxone; Naphthalenes; Narcotic Antagonists; Piperidines; Pyrazoles; Rats; Rats, Long-Evans; Receptor, Cannabinoid, CB1; Rimonabant; Self Administration; Time Factors

2004
Delta9-tetrahydrocannabinol-induced conditioned place preference and intracerebroventricular self-administration in rats.
    European journal of pharmacology, 2004, Dec-03, Volume: 506, Issue:1

    Topics: Animals; Conditioning, Operant; Dose-Response Relationship, Drug; Dronabinol; Injections, Intraventricular; Male; Naloxone; Narcotic Antagonists; Piperidines; Psychotropic Drugs; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Rimonabant; Self Administration

2004
Cannabinoid CB(1) antagonist SR 141716A attenuates reinstatement of heroin self-administration in heroin-abstinent rats.
    Neuropharmacology, 2005, Volume: 48, Issue:8

    Topics: Animals; Behavior, Addictive; Benzoxazines; Conditioning, Operant; Cyclohexanols; Drug Interactions; Extinction, Psychological; Heroin; Heroin Dependence; Male; Morpholines; Naloxone; Naphthalenes; Piperidines; Pyrazoles; Rats; Rats, Inbred Strains; Receptor, Cannabinoid, CB1; Rimonabant; Self Administration

2005
Evidence that (-)-7-hydroxy-4'-dimethylheptyl-cannabidiol activates a non-CB(1), non-CB(2), non-TRPV1 target in the mouse vas deferens.
    Neuropharmacology, 2005, Volume: 48, Issue:8

    Topics: Adenosine Triphosphate; Adrenergic alpha-2 Receptor Antagonists; Animals; Benzoxazines; Cannabidiol; Cannabinoid Receptor Agonists; Cannabinoid Receptor Antagonists; Capsaicin; In Vitro Techniques; Isometric Contraction; Male; Mice; Morpholines; Naloxone; Naphthalenes; Phenylephrine; Piperidines; Pyrazoles; Rimonabant; Ruthenium Red; TRPV Cation Channels; Vas Deferens; Yohimbine

2005
Involvement of the cannabinoid CB1 receptor in the opioid inhibition of the response to cholecystokinin and acute withdrawal response.
    Neurotoxicology, 2005, Volume: 26, Issue:5

    Topics: Acute Disease; Adenosine A1 Receptor Antagonists; Analgesics, Opioid; Animals; Benzoxazines; Cholecystokinin; Dose-Response Relationship, Drug; Guinea Pigs; Ileum; In Vitro Techniques; Male; Morpholines; Muscle Contraction; Muscle, Smooth; Naloxone; Naphthalenes; Narcotic Antagonists; Neurons; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Receptors, Opioid, kappa; Receptors, Opioid, mu; Rimonabant; Substance Withdrawal Syndrome; Theophylline

2005
A role for endocannabinoids in viral-induced dyskinetic and convulsive phenomena.
    Experimental neurology, 2005, Volume: 194, Issue:2

    Topics: Animals; Anticonvulsants; Arachidonic Acids; Basal Ganglia; Borna Disease; Cannabinoid Receptor Modulators; Convulsants; Disease Models, Animal; Endocannabinoids; Limbic System; Male; Movement Disorders; Naloxone; Narcotic Antagonists; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Inbred Lew; Receptor, Cannabinoid, CB1; Rimonabant; Seizures

2005
Interactions between CB1 cannabinoid and mu opioid receptors mediating inhibition of neurotransmitter release in rat nucleus accumbens core.
    Neuropharmacology, 2006, Volume: 51, Issue:4

    Topics: Animals; Calcium; Dose-Response Relationship, Drug; Dronabinol; Drug Interactions; Excitatory Amino Acid Antagonists; Male; Morphine; Naloxone; Narcotic Antagonists; Neural Inhibition; Neurotransmitter Agents; Nucleus Accumbens; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptors, Opioid, mu; Rimonabant; Tritium

2006
The effects of anorexic drugs on free-fed rats responding under a second-order FI15-min (FR10:S) schedule for high incentive foods.
    Behavioural pharmacology, 2007, Volume: 18, Issue:1

    Topics: Animals; Appetite; Appetite Depressants; Appetitive Behavior; Body Weight; Dextroamphetamine; Dose-Response Relationship, Drug; Energy Intake; Extinction, Psychological; Feeding Behavior; Fenfluramine; Male; Motivation; Naloxone; Piperidines; Pyrazoles; Rats; Rats, Long-Evans; Reinforcement Schedule; Rimonabant

2007
Bidirectional cannabinoid modulation of social behavior in adolescent rats.
    Psychopharmacology, 2008, Volume: 197, Issue:2

    Topics: Analgesics, Opioid; Animals; Benzamides; Benzoxazines; Cannabinoids; Carbamates; Dopamine; Dopamine Antagonists; Exploratory Behavior; Flupenthixol; Male; Morphine; Morpholines; Motor Activity; Naloxone; Naphthalenes; Narcotic Antagonists; Piperidines; Play and Playthings; Pyrazoles; Rats; Rats, Wistar; Receptors, Dopamine; Reward; Rimonabant; Social Behavior

2008
Constitutive activity of the cannabinoid CB1 receptor regulates the function of co-expressed Mu opioid receptors.
    The Journal of biological chemistry, 2008, Apr-25, Volume: 283, Issue:17

    Topics: Benzoxazines; Cannabinoids; Cell Membrane; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Extracellular Signal-Regulated MAP Kinases; Gene Expression Regulation; Humans; Kinetics; Ligands; Models, Biological; Morpholines; Naloxone; Naphthalenes; Phosphorylation; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Receptors, Opioid, mu; Rimonabant

2008
Endogenous opioids and cannabinoids: system interactions in the regulation of appetite, grooming and scratching.
    Physiology & behavior, 2008, Jun-09, Volume: 94, Issue:3

    Topics: Analgesics, Opioid; Analysis of Variance; Animals; Appetite; Behavior, Animal; Body Weight; Cannabinoids; Eating; Grooming; Locomotion; Naloxone; Narcotic Antagonists; Piperidines; Pyrazoles; Rats; Reaction Time; Rimonabant; Time Factors

2008
Stress-induced analgesia in mice: evidence for interaction between endocannabinoids and cholecystokinin.
    The European journal of neuroscience, 2008, Volume: 27, Issue:8

    Topics: Analgesia; Animals; Brain; Cannabinoid Receptor Modulators; Cholecystokinin; Endocannabinoids; Gene Expression; Gene Expression Regulation; Mice; Mice, Mutant Strains; Naloxone; Narcotic Antagonists; Pain Threshold; Piperidines; Pyrazoles; Receptor, Cholecystokinin B; Receptors, Cannabinoid; Receptors, Opioid; Rimonabant; Spinal Cord; Stress, Psychological

2008
Prosocial effects of nicotine and ethanol in adolescent rats through partially dissociable neurobehavioral mechanisms.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2009, Volume: 34, Issue:12

    Topics: Aging; Animals; Anti-Anxiety Agents; Anxiety; Behavior, Animal; Central Nervous System Depressants; Diazepam; Dopamine Antagonists; Ethanol; Exploratory Behavior; Flupenthixol; Locomotion; Male; Naloxone; Narcotic Antagonists; Nicotine; Nicotinic Agonists; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Rimonabant; Social Behavior

2009
FAAH inhibitor, URB-597, promotes extinction and CB(1) antagonist, SR141716, inhibits extinction of conditioned aversion produced by naloxone-precipitated morphine withdrawal, but not extinction of conditioned preference produced by morphine in rats.
    Pharmacology, biochemistry, and behavior, 2009, Volume: 94, Issue:1

    Topics: Amidohydrolases; Animals; Benzamides; Cannabinoid Receptor Modulators; Carbamates; Choice Behavior; Conditioning, Psychological; Dietary Sucrose; Extinction, Psychological; Female; Injections, Intraperitoneal; Injections, Subcutaneous; Male; Morphine; Morphine Dependence; Naloxone; Narcotic Antagonists; Narcotics; Piperidines; Pyrazoles; Rats; Rats, Long-Evans; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Reinforcement Schedule; Rimonabant; Species Specificity; Substance Withdrawal Syndrome

2009
Tuberoinfundibular peptide of 39 residues (TIP39) signaling modulates acute and tonic nociception.
    Experimental neurology, 2010, Volume: 226, Issue:1

    Topics: Amidohydrolases; Animals; Cannabinoid Receptor Modulators; Formaldehyde; In Situ Hybridization; Injections, Intraventricular; Injections, Spinal; Male; Mice; Mice, Knockout; Naloxone; Narcotic Antagonists; Neuropeptides; Nociceptors; Pain; Pain Measurement; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Receptor, Parathyroid Hormone, Type 2; Rimonabant; RNA, Messenger; Signal Transduction; Stress, Psychological; Synapses; Vesicular Glutamate Transport Protein 2

2010
Effects of drugs of abuse on putative rostromedial tegmental neurons, inhibitory afferents to midbrain dopamine cells.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2011, Volume: 36, Issue:3

    Topics: Action Potentials; Animals; Animals, Newborn; Behavior, Animal; Benzoxazines; Cocaine; Dopamine; Drug Interactions; Electric Stimulation; Excitatory Postsynaptic Potentials; Gene Expression Regulation; Illicit Drugs; In Vitro Techniques; Male; Mecamylamine; Morphine; Morpholines; Naloxone; Naphthalenes; Narcotic Antagonists; Neural Inhibition; Neural Pathways; Neurons; Nicotinic Antagonists; Patch-Clamp Techniques; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Rimonabant; Time Factors; Ventral Tegmental Area

2011
Differential effect of opioid and cannabinoid receptor blockade on heroin-seeking reinstatement and cannabinoid substitution in heroin-abstinent rats.
    British journal of pharmacology, 2011, Volume: 163, Issue:7

    Topics: Analgesics, Opioid; Animals; Behavior, Addictive; Behavior, Animal; Benzoxazines; Cannabinoids; Drug Substitution; Drug Synergism; Heroin; Male; Morpholines; Naloxone; Naphthalenes; Narcotic Antagonists; Piperidines; Pyrazoles; Rats; Receptor, Cannabinoid, CB1; Reinforcement Schedule; Rimonabant; Self Administration

2011
Naloxone and rimonabant reduce the reinforcing properties of exercise in rats.
    Experimental and clinical psychopharmacology, 2011, Volume: 19, Issue:6

    Topics: Animals; Cannabinoids; Extinction, Psychological; Female; Naloxone; Narcotic Antagonists; Physical Conditioning, Animal; Piperidines; Pyrazoles; Rats; Rats, Zucker; Reinforcement, Psychology; Rimonabant

2011
Inhibitory inputs from rostromedial tegmental neurons regulate spontaneous activity of midbrain dopamine cells and their responses to drugs of abuse.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2012, Volume: 37, Issue:5

    Topics: Action Potentials; Analysis of Variance; Animals; Benzoxazines; Cannabinoids; Cocaine; Dopaminergic Neurons; Electric Stimulation; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Male; Morphine; Morpholines; Naloxone; Naphthalenes; Narcotic Antagonists; Narcotics; Neural Inhibition; Neural Pathways; Nicotine; Nicotinic Agonists; Patch-Clamp Techniques; Physical Stimulation; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Rimonabant; Tegmentum Mesencephali; Time Factors; Ventral Tegmental Area

2012
Sex differences in cannabinoid 1 vs. cannabinoid 2 receptor-selective antagonism of antinociception produced by delta9-tetrahydrocannabinol and CP55,940 in the rat.
    The Journal of pharmacology and experimental therapeutics, 2012, Volume: 340, Issue:3

    Topics: Analgesics; Animals; Camphanes; Cyclohexanols; Dose-Response Relationship, Drug; Dronabinol; Female; Male; Morphine; Motor Activity; Naloxone; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant; Sex Characteristics

2012
Low dose naloxone attenuates the pruritic but not anorectic response to rimonabant in male rats.
    Psychopharmacology, 2013, Volume: 226, Issue:2

    Topics: Animals; Appetite; Behavior, Animal; Body Weight; Cannabinoid Receptor Antagonists; Compulsive Behavior; Dose-Response Relationship, Drug; Feeding Behavior; Food; Grooming; Locomotion; Male; Naloxone; Narcotic Antagonists; Piperidines; Pruritus; Pyrazoles; Rats; Rimonabant

2013
Combination cannabinoid and opioid receptor antagonists improves metabolic outcomes in obese mice.
    Molecular and cellular endocrinology, 2015, Dec-05, Volume: 417

    Topics: Animals; Body Composition; Cannabinoid Receptor Antagonists; Drug Therapy, Combination; Glucose; Insulin; Male; Mice; Mice, Obese; Naloxone; Narcotic Antagonists; Obesity; Piperidines; Pyrazoles; Rimonabant; Thermogenesis; Treatment Outcome

2015
Hedonic drinking engages a supraspinal inhibition of thermal nociception in adult rats.
    Pain, 2019, Volume: 160, Issue:5

    Topics: Animals; Cannabinoid Receptor Antagonists; Disease Models, Animal; Dose-Response Relationship, Drug; Drinking Behavior; Freund's Adjuvant; Hot Temperature; Hyperalgesia; Injections, Spinal; Male; Naloxone; Narcotic Antagonists; Pain Threshold; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Reaction Time; Rimonabant; Spinal Cord; Sucrose; Sweetening Agents; Water Deprivation

2019
The analgesic effect of refeeding on acute and chronic inflammatory pain.
    Scientific reports, 2019, 11-14, Volume: 9, Issue:1

    Topics: Acute Pain; Analgesics, Opioid; Animals; Chronic Pain; Disease Models, Animal; Eating; Food Deprivation; Formaldehyde; Freund's Adjuvant; Glucose; Hot Temperature; Hyperalgesia; Inflammation; Injections, Intraperitoneal; Male; Mice; Mice, Inbred C57BL; Naloxone; Narcotic Antagonists; Pain Management; Pain Measurement; Rimonabant

2019