Page last updated: 2024-08-26

sr141716 and jd5037

sr141716 has been researched along with jd5037 in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's3 (75.00)24.3611
2020's1 (25.00)2.80

Authors

AuthorsStudies
Berbaum, J; Chorvat, RJ; McElroy, JF; Seriacki, K1
Chorvat, RJ1
Carlson, OD; Cieśla, Ł; Cimbro, R; Doyle, ME; Egan, JM; Ghosh, S; González-Mariscal, I; Krzysik-Walker, SM; Liu, QR; Moaddel, R; O'Connell, JF; Santa-Cruz Calvo, S; Witek, RP1
Cinar, R; Gao, B; Godlewski, G; Gunduz-Cinar, O; Herrerias, A; Iyer, MR; Kunos, G; Lin, Y; Santos-Molina, L; Wood, CM; Zawatsky, CN1

Reviews

1 review(s) available for sr141716 and jd5037

ArticleYear
Peripherally restricted CB1 receptor blockers.
    Bioorganic & medicinal chemistry letters, 2013, Sep-01, Volume: 23, Issue:17

    Topics: Animals; Brain; Cocaine; Drug Discovery; Humans; Liver Diseases; Metabolic Diseases; Morpholines; Obesity; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Rimonabant; Sulfonamides

2013

Other Studies

3 other study(ies) available for sr141716 and jd5037

ArticleYear
JD-5006 and JD-5037: peripherally restricted (PR) cannabinoid-1 receptor blockers related to SLV-319 (Ibipinabant) as metabolic disorder therapeutics devoid of CNS liabilities.
    Bioorganic & medicinal chemistry letters, 2012, Oct-01, Volume: 22, Issue:19

    Topics: Amidines; Brain Diseases, Metabolic; Dose-Response Relationship, Drug; Humans; Molecular Structure; Pyrazoles; Receptor, Cannabinoid, CB1; Recombinant Proteins; Structure-Activity Relationship; Sulfonamides

2012
Human CB1 Receptor Isoforms, present in Hepatocytes and β-cells, are Involved in Regulating Metabolism.
    Scientific reports, 2016, 09-19, Volume: 6

    Topics: Amino Acid Sequence; Animals; Cells, Cultured; CHO Cells; Cricetinae; Cricetulus; Gene Expression Profiling; Glucose; Hepatocytes; Humans; Insulin; Insulin Secretion; Insulin-Secreting Cells; Metabolic Diseases; Piperidines; Protein Isoforms; Pyrazoles; Receptor, Cannabinoid, CB1; Rimonabant; Sequence Homology, Amino Acid; Sulfonamides

2016
Effects of a Peripherally Restricted Hybrid Inhibitor of CB1 Receptors and iNOS on Alcohol Drinking Behavior and Alcohol-Induced Endotoxemia.
    Molecules (Basel, Switzerland), 2021, Aug-22, Volume: 26, Issue:16

    Topics: Alcohol Drinking; Animals; Anxiety; Behavior, Animal; Cannabinoid Receptor Antagonists; Catalepsy; Cyclohexanols; Elevated Plus Maze Test; Endotoxemia; Endotoxins; Ethanol; Gastrointestinal Tract; Hypothermia, Induced; Mice, Inbred C57BL; Nitric Oxide Synthase Type II; Pyrazoles; Receptor, Cannabinoid, CB1; Rimonabant; Stereoisomerism; Sulfonamides

2021