Page last updated: 2024-08-26

sr141716 and gamma-aminobutyric acid

sr141716 has been researched along with gamma-aminobutyric acid in 40 studies

Research

Studies (40)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (10.00)18.2507
2000's29 (72.50)29.6817
2010's7 (17.50)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Brotchie, JM; Crossman, AR; Maneuf, YP; Nash, JE1
Rosenberg, HC; Tersigni, TJ1
Brotchie, JM; Crossman, AR; Maneuf, YP1
Sañudo-Peña, MC; Walker, JM1
Cheer, JF; Kendall, DA; Marsden, CA; Mason, R1
Freund, TF; Hájos, N; Katona, I; Ledent, C; MacKie, K; Mody, I; Naiem, SS1
Nicoll, RA; Wilson, RI1
Freund, TF; Hájos, N; Ledent, C1
Antonelli, T; Bebe, BW; Cassano, T; Cuomo, V; Ferraro, L; Magee, P; O'Connor, WT; Siniscalchi, A; Tanganelli, S; Tomasini, MC1
Siemes, S; Szabo, B; Wallmichrath, I1
Azad, SC; Bisogno, T; Cascio, MG; Di Marzo, V; Hermann, H; Hofmann, C; Lutz, B; Marsicano, G; Rammes, G; Tang, J; Wotjak, CT; Zieglgänsberger, W1
Devoto, P; Ferraro, L; Flore, G; Gessa, GL; Pira, L; Pistis, M; Tanganelli, S1
de Miguel, R; De Petrocellis, L; Di Marzo, V; Fernández-Ruiz, J; Lastres-Becker, I; Makriyannis, A1
Hoffman, AF; Lupica, CR; Riegel, AC1
Azad, SC; Behl, C; Cannich, A; Casanova, E; Cascio, MG; Di Marzo, V; Eder, M; Goodenough, S; Gutiérrez, SO; Hermann, H; López-Rodriguez, ML; Lutz, B; Marsicano, G; Monory, K; Schütz, G; van der Stelt, M; Zieglgänsberger, W1
Duguid, IC; Smart, TG1
Cunha, RA; Köfalvi, A; Ledent, C; Mackie, K; Rodrigues, RJ; Sperlágh, B; Vizi, ES1
Brotchie, JM; Crossman, AR; Di Marzo, V; Fox, SH; Hill, M; Petrosino, S; van der Stelt, M1
Bernardi, G; Calabresi, P; Centonze, D; Maccarrone, M; Prosperetti, C; Rossi, S; Tscherter, A1
Alger, BE; Isokawa, M1
Caillé, S; Parsons, LH1
de Miguel, R; Fernández-Ruiz, J; García-Arencibia, M; González, S; Ramos, JA; Scorticati, C1
Anton, A; Freiman, I; Monyer, H; Szabo, B; Urbanski, MJ1
Battista, N; Bernardi, G; Centonze, D; De Chiara, V; Maccarrone, M; Mercuri, NB; Prosperetti, C; Rossi, S; Usiello, A1
Bertekap, R; Bourin, C; Burris, K; Conway, C; Deng, H; Sit, SY; Xie, K1
Argiolas, A; Castelli, MP; Collu, S; Diaz, G; Ennas, MG; Mackie, K; Melis, MR; Melis, T; Piras, AP; Sanna, F; Succu, S1
Blackbeard, J; Hasnie, F; Lambert, DM; Pheby, T; Rice, AS; Segerdahl, AR; Vandevoorde, S; Wallace, VC1
Ma, YL; Stephens, GJ; Weston, SE; Whalley, BJ1
Davis, MI; Lovinger, DM; Sheinin, A; Talani, G1
Benetti, C; Girlanda, E; Large, CH; Sokal, DM1
Di, S; Franco, A; Maxson, MM; Tasker, JG1
Kovacs, FE; Szabo, B; Urbanski, MJ1
Mendiguren, A; Pineda, J1
Leng, G; Ludwig, M; Menzies, JR1
Alger, BE; Kim, J1
Baur, R; Gertsch, J; Sigel, E1
Glanowska, KM; Moenter, SM1
Biggio, F; Biggio, G; Dazzi, L; Lallai, V; Licheri, V; Lutzu, S; Mostallino, MC; Sanna, E; Secci, PP; Talani, G; Utzeri, C1
Bogdanovic, RM; Jafari, M; Potschka, H; von Rüden, EL; Wotjak, CT1
Banks, ML; Bradshaw, HB; Crowe, MS; Kinsey, SG; Leishman, E; Prather, PL; Wilson, CD1

Other Studies

40 other study(ies) available for sr141716 and gamma-aminobutyric acid

ArticleYear
Activation of the cannabinoid receptor by delta 9-tetrahydrocannabinol reduces gamma-aminobutyric acid uptake in the globus pallidus.
    European journal of pharmacology, 1996, Jul-18, Volume: 308, Issue:2

    Topics: Animals; Dose-Response Relationship, Drug; Dronabinol; gamma-Aminobutyric Acid; Globus Pallidus; Male; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptors, Cannabinoid; Receptors, Drug; Rimonabant

1996
Local pressure application of cannabinoid agonists increases spontaneous activity of rat substantia nigra pars reticulata neurons without affecting response to iontophoretically-applied GABA.
    Brain research, 1996, Sep-16, Volume: 733, Issue:2

    Topics: Action Potentials; Analgesics; Analysis of Variance; Animals; Benzoxazines; Bicuculline; Cannabinoids; Cyclohexanols; gamma-Aminobutyric Acid; Iontophoresis; Male; Morpholines; Naphthalenes; Neurons; Piperidines; Pressure; Pyrazoles; Rats; Rats, Sprague-Dawley; Rimonabant; Substantia Nigra

1996
The cannabinoid receptor agonist WIN 55,212-2 reduces D2, but not D1, dopamine receptor-mediated alleviation of akinesia in the reserpine-treated rat model of Parkinson's disease.
    Experimental neurology, 1997, Volume: 148, Issue:1

    Topics: Animals; Basal Ganglia; Benzazepines; Benzoxazines; Dopamine Agonists; gamma-Aminobutyric Acid; Locomotion; Male; Morpholines; Naphthalenes; Nerve Tissue Proteins; Parkinson Disease, Secondary; Piperidines; Pyrazoles; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Cannabinoid; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Drug; Reserpine; Rimonabant

1997
A novel neurotransmitter system involved in the control of motor behavior by the basal ganglia.
    Annals of the New York Academy of Sciences, 1998, Nov-16, Volume: 860

    Topics: Action Potentials; Analgesics; Animals; Basal Ganglia; Benzoxazines; Bicuculline; Cannabinoids; Cyclohexanols; Dopamine; Dopamine Agonists; Electrophysiology; GABA Antagonists; gamma-Aminobutyric Acid; Morpholines; Motor Neurons; Naphthalenes; Nerve Degeneration; Neurotransmitter Agents; Oxidopamine; Piperidines; Pyrazoles; Quinpirole; Rats; Rimonabant; Sympatholytics; Thalamic Nuclei

1998
Lack of response suppression follows repeated ventral tegmental cannabinoid administration: an in vitro electrophysiological study.
    Neuroscience, 2000, Volume: 99, Issue:4

    Topics: Action Potentials; Animals; Bicuculline; Cannabinoids; Dopamine; Dronabinol; Electrophysiology; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Interneurons; Male; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Reward; Rimonabant; Ventral Tegmental Area

2000
Cannabinoids inhibit hippocampal GABAergic transmission and network oscillations.
    The European journal of neuroscience, 2000, Volume: 12, Issue:9

    Topics: Action Potentials; Analgesics; Animals; Antibodies; Benzoxazines; Cannabinoids; Cyclohexanols; Electrophysiology; Epitopes; gamma-Aminobutyric Acid; Hippocampus; Interneurons; Male; Mice; Mice, Inbred Strains; Mice, Knockout; Microscopy, Electron; Morpholines; Naphthalenes; Neural Inhibition; Neural Pathways; Periodicity; Piperidines; Presynaptic Terminals; Pyramidal Cells; Pyrazoles; Rats; Rats, Wistar; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Synaptic Transmission

2000
Endogenous cannabinoids mediate retrograde signalling at hippocampal synapses.
    Nature, 2001, Mar-29, Volume: 410, Issue:6828

    Topics: Animals; Arachidonic Acids; Benzoxazines; Cannabinoid Receptor Modulators; Cannabinoids; Endocannabinoids; gamma-Aminobutyric Acid; Glycerides; Hippocampus; In Vitro Techniques; Morpholines; Naphthalenes; Neural Inhibition; Piperidines; Pyramidal Cells; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptors, Cannabinoid; Receptors, Drug; Receptors, Metabotropic Glutamate; Rimonabant; Signal Transduction; Synapses; Synaptic Transmission

2001
Novel cannabinoid-sensitive receptor mediates inhibition of glutamatergic synaptic transmission in the hippocampus.
    Neuroscience, 2001, Volume: 106, Issue:1

    Topics: Analgesics; Animals; Benzoxazines; Cannabinoids; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Hippocampus; Interneurons; Mice; Mice, Knockout; Morpholines; Naphthalenes; Neural Inhibition; Piperidines; Pyramidal Cells; Pyrazoles; Receptors, Cannabinoid; Receptors, Drug; Receptors, GABA; Receptors, Glutamate; Rimonabant; Synapses; Synaptic Transmission

2001
Cannabinoid receptor agonist WIN 55,212-2 inhibits rat cortical dialysate gamma-aminobutyric acid levels.
    Journal of neuroscience research, 2001, Oct-15, Volume: 66, Issue:2

    Topics: Animals; Benzoxazines; Dose-Response Relationship, Drug; Drug Interactions; gamma-Aminobutyric Acid; Microdialysis; Morpholines; Naphthalenes; Piperidines; Prefrontal Cortex; Pyrazoles; Rats; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Wakefulness

2001
Inhibition of GABAergic neurotransmission in the ventral tegmental area by cannabinoids.
    The European journal of neuroscience, 2002, Volume: 15, Issue:12

    Topics: Analgesics; Animals; Animals, Newborn; Benzoxazines; Cannabinoids; Drug Interactions; GABA Agonists; gamma-Aminobutyric Acid; Membrane Potentials; Morpholines; Muscimol; Naphthalenes; Neural Inhibition; Neural Pathways; Neurons; Nucleus Accumbens; Organ Culture Techniques; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB2; Receptors, Cannabinoid; Receptors, Drug; Receptors, GABA-A; Rimonabant; Synaptic Transmission; Ventral Tegmental Area

2002
The endogenous cannabinoid system controls extinction of aversive memories.
    Nature, 2002, Aug-01, Volume: 418, Issue:6897

    Topics: Acoustic Stimulation; Amygdala; Animals; Cannabinoid Receptor Modulators; Cannabinoids; Conditioning, Classical; Electrophysiology; Extinction, Psychological; Fear; gamma-Aminobutyric Acid; Gene Deletion; In Vitro Techniques; Male; Memory; Mice; Mice, Inbred C57BL; Mice, Knockout; Neuronal Plasticity; Neurons; Piperidines; Pyrazoles; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Synapses

2002
Delta(9)-tetrahydrocannabinol decreases extracellular GABA and increases extracellular glutamate and dopamine levels in the rat prefrontal cortex: an in vivo microdialysis study.
    Brain research, 2002, Sep-06, Volume: 948, Issue:1-2

    Topics: Animals; Dopamine; Dronabinol; Extracellular Space; gamma-Aminobutyric Acid; Glutamic Acid; Male; Microdialysis; Piperidines; Prefrontal Cortex; Psychotropic Drugs; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptors, Drug; Rimonabant

2002
Compounds acting at the endocannabinoid and/or endovanilloid systems reduce hyperkinesia in a rat model of Huntington's disease.
    Journal of neurochemistry, 2003, Volume: 84, Issue:5

    Topics: 3,4-Dihydroxyphenylacetic Acid; Amino Acids, Neutral; Animals; Arachidonic Acids; Basal Ganglia; Cannabinoid Receptor Modulators; Capsaicin; Corpus Striatum; Cyclohexanols; Disease Models, Animal; Dopamine; Endocannabinoids; gamma-Aminobutyric Acid; Huntington Disease; Hyperkinesis; Male; Motor Activity; Nitro Compounds; Palmitates; Piperidines; Propionates; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptors, Cannabinoid; Receptors, Drug; Rimonabant

2003
Functional localization of cannabinoid receptors and endogenous cannabinoid production in distinct neuron populations of the hippocampus.
    The European journal of neuroscience, 2003, Volume: 18, Issue:3

    Topics: Animals; Benzoxazines; Cannabinoids; Electrophysiology; Excitatory Postsynaptic Potentials; gamma-Aminobutyric Acid; Glutamic Acid; Hippocampus; In Vitro Techniques; Interneurons; Male; Morpholines; Naphthalenes; Neural Inhibition; Neurons; Piperidines; Pyramidal Cells; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Synapses; Tissue Distribution

2003
CB1 cannabinoid receptors and on-demand defense against excitotoxicity.
    Science (New York, N.Y.), 2003, Oct-03, Volume: 302, Issue:5642

    Topics: Animals; Arachidonic Acids; Brain; Brain-Derived Neurotrophic Factor; Cannabinoids; Endocannabinoids; Epilepsy; Excitatory Amino Acid Agonists; Excitatory Postsynaptic Potentials; Furans; gamma-Aminobutyric Acid; Gene Expression Regulation; Genes, Immediate-Early; Glutamic Acid; Glycerides; Hippocampus; In Vitro Techniques; Kainic Acid; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Mice, Transgenic; Mitogen-Activated Protein Kinases; Mutation; Neurons; Neuroprotective Agents; Piperidines; Polyunsaturated Alkamides; Prosencephalon; Pyrazoles; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Signal Transduction

2003
Retrograde activation of presynaptic NMDA receptors enhances GABA release at cerebellar interneuron-Purkinje cell synapses.
    Nature neuroscience, 2004, Volume: 7, Issue:5

    Topics: Animals; Animals, Newborn; Cadmium; Calcium; Cerebellum; Chelating Agents; Dose-Response Relationship, Drug; Drug Interactions; Egtazic Acid; Electric Stimulation; Evoked Potentials; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Immunohistochemistry; In Vitro Techniques; Interneurons; Isoenzymes; Membrane Potentials; N-Methylaspartate; Neural Inhibition; Neuronal Plasticity; Patch-Clamp Techniques; Piperidines; Presynaptic Terminals; Purkinje Cells; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Rimonabant; Ryanodine; Sodium Channel Blockers; Synapses; Synaptic Transmission; Synaptophysin; Tetrodotoxin; Time Factors

2004
Involvement of cannabinoid receptors in the regulation of neurotransmitter release in the rodent striatum: a combined immunochemical and pharmacological analysis.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, Mar-16, Volume: 25, Issue:11

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Benzoxazines; Blotting, Western; Calcium; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Immunohistochemistry; Male; Mice; Mice, Knockout; Morpholines; Naphthalenes; Neurotransmitter Agents; Piperidines; Potassium; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Rimonabant; Synapses; Synaptosomes; Tetrodotoxin; Tritium; Tyrosine 3-Monooxygenase; Vesicular Glutamate Transport Protein 1; Vesicular Glutamate Transport Protein 2

2005
A role for endocannabinoids in the generation of parkinsonism and levodopa-induced dyskinesia in MPTP-lesioned non-human primate models of Parkinson's disease.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 2005, Volume: 19, Issue:9

    Topics: Animals; Arachidonic Acids; Callithrix; Cannabinoid Receptor Modulators; Dyskinesia, Drug-Induced; Endocannabinoids; Female; gamma-Aminobutyric Acid; Glycerides; Levodopa; Male; MPTP Poisoning; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptor, Cannabinoid, CB1; Rimonabant

2005
Abnormal sensitivity to cannabinoid receptor stimulation might contribute to altered gamma-aminobutyric acid transmission in the striatum of R6/2 Huntington's disease mice.
    Biological psychiatry, 2005, Jun-15, Volume: 57, Issue:12

    Topics: Animals; Animals, Newborn; Cannabinoid Receptor Antagonists; Corpus Striatum; Drug Interactions; Electric Stimulation; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Huntington Disease; In Vitro Techniques; Membrane Potentials; Mice; Mice, Transgenic; Neural Inhibition; Neurons; Patch-Clamp Techniques; Piperidines; Pyrazoles; Receptors, Cannabinoid; Rimonabant; Synaptic Transmission; Time Factors

2005
Retrograde endocannabinoid regulation of GABAergic inhibition in the rat dentate gyrus granule cell.
    The Journal of physiology, 2005, Sep-15, Volume: 567, Issue:Pt 3

    Topics: Animals; Benzoxazines; Calcium; Dentate Gyrus; Electrophysiology; Enzyme Inhibitors; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Morpholines; Naphthalenes; Patch-Clamp Techniques; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptors, GABA-A; Rimonabant; Ryanodine; Synaptic Transmission; Thapsigargin

2005
Cannabinoid modulation of opiate reinforcement through the ventral striatopallidal pathway.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2006, Volume: 31, Issue:4

    Topics: Analgesics, Opioid; Animals; Area Under Curve; Behavior, Animal; Cannabinoids; Cocaine; Conditioning, Operant; Corpus Striatum; Dopamine; Drug Administration Routes; Drug Interactions; gamma-Aminobutyric Acid; Male; Microdialysis; Morphine; Neural Pathways; Piperidines; Pyrazoles; Rats; Rats, Wistar; Reinforcement, Psychology; Rimonabant; Self Administration; Time Factors

2006
Effects of rimonabant, a selective cannabinoid CB1 receptor antagonist, in a rat model of Parkinson's disease.
    Brain research, 2006, Feb-16, Volume: 1073-1074

    Topics: Adrenergic Agents; Analysis of Variance; Animals; Autoradiography; Brain; Brain Chemistry; Chromatography, High Pressure Liquid; Disease Models, Animal; Dopamine; Dose-Response Relationship, Drug; Drug Interactions; Electrochemistry; gamma-Aminobutyric Acid; Gene Expression; Glutamic Acid; In Situ Hybridization; Injections, Intraventricular; Male; Motor Activity; Oxidopamine; Parkinson Disease; Piperidines; Protein Binding; Pyrazoles; Rats; Rats, Sprague-Dawley; Reaction Time; Receptor, Cannabinoid, CB1; Rimonabant; RNA, Messenger; Rotarod Performance Test; Superoxide Dismutase; Superoxide Dismutase-1; Tyrosine 3-Monooxygenase

2006
Analysis of the effects of cannabinoids on identified synaptic connections in the caudate-putamen by paired recordings in transgenic mice.
    The Journal of physiology, 2006, Sep-15, Volume: 575, Issue:Pt 3

    Topics: Animals; Benzoxazines; Cannabinoids; Caudate Nucleus; Evoked Potentials; gamma-Aminobutyric Acid; Green Fluorescent Proteins; In Vitro Techniques; Interneurons; Mice; Mice, Transgenic; Morpholines; Naphthalenes; Neural Inhibition; Parvalbumins; Patch-Clamp Techniques; Piperidines; Presynaptic Terminals; Putamen; Pyrazoles; Receptor, Cannabinoid, CB1; Rimonabant; Synapses; Synaptic Transmission

2006
Chronic cocaine sensitizes striatal GABAergic synapses to the stimulation of cannabinoid CB1 receptors.
    The European journal of neuroscience, 2007, Volume: 25, Issue:6

    Topics: Animals; Behavior, Animal; Cocaine; Conditioning, Operant; Corpus Striatum; Dopamine Uptake Inhibitors; Dronabinol; Drug Administration Schedule; Drug Interactions; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; gamma-Aminobutyric Acid; Glutamic Acid; Male; Patch-Clamp Techniques; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Rimonabant; Synapses

2007
Novel inhibitors of fatty acid amide hydrolase.
    Bioorganic & medicinal chemistry letters, 2007, Jun-15, Volume: 17, Issue:12

    Topics: Amidohydrolases; Amines; Analgesics; Animals; Cyclohexanecarboxylic Acids; Dose-Response Relationship, Drug; Enzyme Inhibitors; Gabapentin; gamma-Aminobutyric Acid; Humans; Imidazoles; Mice; Mice, Knockout; Morphine; Pain Measurement; Piperidines; Pyrazoles; Rats; Receptor, Cannabinoid, CB1; Rimonabant

2007
Cannabinoid CB1 receptors in the paraventricular nucleus and central control of penile erection: immunocytochemistry, autoradiography and behavioral studies.
    Neuroscience, 2007, Jun-15, Volume: 147, Issue:1

    Topics: Animals; gamma-Aminobutyric Acid; Glutamic Acid; Immunohistochemistry; Male; Microinjections; Neural Inhibition; Neurotransmitter Agents; Oxytocin; Paraventricular Hypothalamic Nucleus; Penile Erection; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Rimonabant; Sexual Behavior, Animal; Signal Transduction; Tissue Distribution

2007
The effect of the palmitoylethanolamide analogue, palmitoylallylamide (L-29) on pain behaviour in rodent models of neuropathy.
    British journal of pharmacology, 2007, Volume: 151, Issue:7

    Topics: Amides; Amines; Animals; Behavior, Animal; Camphanes; Cyclohexanecarboxylic Acids; Dose-Response Relationship, Drug; Endocannabinoids; Ethanolamines; Gabapentin; gamma-Aminobutyric Acid; Hindlimb; Indoles; Injections, Intraperitoneal; Male; Pain; Pain Measurement; Pain Threshold; Palmitic Acids; Physical Stimulation; Piperidines; PPAR alpha; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant; Sciatic Neuropathy; Temperature; Zalcitabine

2007
The phytocannabinoid Delta(9)-tetrahydrocannabivarin modulates inhibitory neurotransmission in the cerebellum.
    British journal of pharmacology, 2008, Volume: 154, Issue:1

    Topics: Animals; Benzoxazines; Bicuculline; Cannabinoids; Cerebellum; Dronabinol; Electrophysiology; Excitatory Postsynaptic Potentials; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Mice; Morpholines; Naphthalenes; Patch-Clamp Techniques; Piperidines; Purkinje Cells; Pyrazoles; Receptor, Cannabinoid, CB1; Rimonabant; Synapses; Synaptic Transmission

2008
Endocannabinoid- and mGluR5-dependent short-term synaptic depression in an isolated neuron/bouton preparation from the hippocampal CA1 region.
    Journal of neurophysiology, 2008, Volume: 100, Issue:2

    Topics: Animals; Animals, Newborn; Arachidonic Acids; Benzoxazines; Cannabinoid Receptor Modulators; Drug Interactions; Endocannabinoids; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Glycerides; Hippocampus; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Methoxyhydroxyphenylglycol; Morpholines; Naphthalenes; Neurons; Patch-Clamp Techniques; Piperidines; Pyrazoles; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Rimonabant; Synapses; Synapsins

2008
The CB1 receptor antagonist, SR141716A, prevents high-frequency stimulation-induced reduction of feedback inhibition in the rat dentate gyrus following perforant path stimulation in vivo.
    Brain research, 2008, Aug-05, Volume: 1223

    Topics: Animals; Cannabinoid Receptor Modulators; Dentate Gyrus; Electric Stimulation; Excitatory Postsynaptic Potentials; Feedback; gamma-Aminobutyric Acid; Glutamic Acid; Interneurons; Long-Term Potentiation; Male; Neural Inhibition; Perforant Pathway; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptors, GABA; Rimonabant; Synaptic Transmission

2008
Glucocorticoids regulate glutamate and GABA synapse-specific retrograde transmission via divergent nongenomic signaling pathways.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2009, Jan-14, Volume: 29, Issue:2

    Topics: Animals; Arginine; Cannabinoid Receptor Modulators; Cyclic AMP-Dependent Protein Kinases; Dexamethasone; Dronabinol; Electric Stimulation; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Glucocorticoids; Glutamic Acid; GTP-Binding Proteins; Guanosine Diphosphate; Hypothalamus; In Vitro Techniques; Male; Neurons; Nitric Oxide; Nitric Oxide Donors; Patch-Clamp Techniques; Penicillamine; Piperidines; Pyrans; Pyrazoles; Quinoxalines; Rats; Rats, Sprague-Dawley; Rimonabant; Signal Transduction; Synapses; Synaptic Transmission; Thionucleotides; Valine

2009
Depolarizing GABAergic synaptic input triggers endocannabinoid-mediated retrograde synaptic signaling.
    Synapse (New York, N.Y.), 2009, Volume: 63, Issue:8

    Topics: Aniline Compounds; Animals; Animals, Newborn; Arachidonic Acids; Benzamides; Bicuculline; Biophysics; Calcium; Calcium Signaling; Cannabinoid Receptor Antagonists; Cannabinoid Receptor Modulators; Carbamates; Cerebellum; Electric Stimulation; Endocannabinoids; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Fluoresceins; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glycerides; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Lactones; Mice; Muscimol; Orlistat; Patch-Clamp Techniques; Piperidines; Purkinje Cells; Pyrazoles; Quinoxalines; Rimonabant; Signal Transduction; Synapses; Valine

2009
Effect of the CB(1) receptor antagonists rimonabant and AM251 on the firing rate of dorsal raphe nucleus neurons in rat brain slices.
    British journal of pharmacology, 2009, Volume: 158, Issue:6

    Topics: Animals; Arachidonic Acids; Cannabinoid Receptor Modulators; Cannabinoids; Endocannabinoids; gamma-Aminobutyric Acid; Male; Neurons; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Rimonabant; Serotonin

2009
Direct and indirect effects of cannabinoids on in vitro GABA release in the rat arcuate nucleus.
    Journal of neuroendocrinology, 2010, Volume: 22, Issue:6

    Topics: Animals; Arcuate Nucleus of Hypothalamus; Cannabinoids; Chromatography, High Pressure Liquid; gamma-Aminobutyric Acid; Male; Piperidines; Potassium; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Rimonabant

2010
Reduction in endocannabinoid tone is a homeostatic mechanism for specific inhibitory synapses.
    Nature neuroscience, 2010, Volume: 13, Issue:5

    Topics: Agatoxins; Animals; Arachidonic Acids; Benzamides; Benzoxazines; Biophysics; Calcium; Calcium Channel Blockers; Cannabinoid Receptor Modulators; Carbamates; Conotoxins; Dose-Response Relationship, Drug; Down-Regulation; Drug Interactions; Electric Stimulation; Endocannabinoids; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Glycerides; Hippocampus; Homeostasis; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Morpholines; Naphthalenes; Nerve Net; Neural Inhibition; Neurons; Patch-Clamp Techniques; Piperidines; Polyamines; Polyunsaturated Alkamides; Pyrazoles; Rats; Receptor, Cannabinoid, CB1; Rimonabant; Sodium Channel Blockers; Synapses; Tetrodotoxin

2010
The cannabinoid CB1 receptor antagonists rimonabant (SR141716) and AM251 directly potentiate GABA(A) receptors.
    British journal of pharmacology, 2012, Volume: 165, Issue:8

    Topics: Animals; Benzofurans; Dronabinol; gamma-Aminobutyric Acid; Oocytes; Piperidines; Pyrans; Pyrazoles; Receptor, Cannabinoid, CB1; Receptors, GABA-A; Recombinant Proteins; Rimonabant; Xenopus

2012
Endocannabinoids and prostaglandins both contribute to GnRH neuron-GABAergic afferent local feedback circuits.
    Journal of neurophysiology, 2011, Volume: 106, Issue:6

    Topics: Action Potentials; Afferent Pathways; Analysis of Variance; Androgens; Animals; Brain; Cannabinoid Receptor Modulators; Dihydrotestosterone; Drug Interactions; Electric Stimulation; Endocannabinoids; Estradiol; Estrogens; Female; gamma-Aminobutyric Acid; Gonadotropin-Releasing Hormone; Green Fluorescent Proteins; In Vitro Techniques; Male; Mice; Mice, Transgenic; Nerve Net; Neurons; Ovariectomy; Patch-Clamp Techniques; Piperidines; Prostaglandins; Pyrazoles; Rimonabant; Synaptic Transmission

2011
Involvement of the cannabinoid CB1 receptor in modulation of dopamine output in the prefrontal cortex associated with food restriction in rats.
    PloS one, 2014, Volume: 9, Issue:3

    Topics: Animals; Anticipation, Psychological; Diet; Dopamine; Exploratory Behavior; Extracellular Space; Feeding Behavior; gamma-Aminobutyric Acid; Gene Expression Regulation; Ligands; Male; Neurons; Nucleus Accumbens; Piperidines; Prefrontal Cortex; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Rimonabant; Ventral Tegmental Area

2014
Analysis in conditional cannabinoid 1 receptor-knockout mice reveals neuronal subpopulation-specific effects on epileptogenesis in the kindling paradigm.
    Neurobiology of disease, 2015, Volume: 73

    Topics: Anilides; Animals; Bromodeoxyuridine; Calcium-Calmodulin-Dependent Protein Kinase Type 1; Cannabinoid Receptor Antagonists; Cinnamates; Disease Models, Animal; Epilepsy; gamma-Aminobutyric Acid; Gene Expression Regulation; Kindling, Neurologic; Male; Mice; Mice, Knockout; Neurogenesis; Neurons; Piperidines; Prosencephalon; Pyrazoles; Receptor, Cannabinoid, CB1; Rimonabant; TRPV Cation Channels

2015
The monoacylglycerol lipase inhibitor KML29 with gabapentin synergistically produces analgesia in mice.
    British journal of pharmacology, 2017, Volume: 174, Issue:23

    Topics: Amines; Analgesics; Animals; Benzodioxoles; Cyclohexanecarboxylic Acids; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Synergism; Drug Tolerance; Enzyme Inhibitors; Gabapentin; gamma-Aminobutyric Acid; Hyperalgesia; Male; Mice; Mice, Inbred C57BL; Monoacylglycerol Lipases; Neuralgia; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Rimonabant; Signal Transduction

2017