sr141716 has been researched along with am 630 in 29 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 1 (3.45) | 18.2507 |
| 2000's | 6 (20.69) | 29.6817 |
| 2010's | 20 (68.97) | 24.3611 |
| 2020's | 2 (6.90) | 2.80 |
| Authors | Studies |
|---|---|
| Allarà, M; Benetti, V; Cascio, MG; Di Marzo, V; Ferrarini, PL; Ghelardini, C; Manera, C; Martinelli, A; Saccomanni, G; Tuccinardi, T; Vivoli, E | 1 |
| Bolognini, D; Cascio, MG; Cicione, L; Corelli, F; De Chiaro, M; De Rosa, M; Di Marzo, V; Guida, F; Ligresti, A; Luongo, L; Maione, S; Marini, P; Mugnaini, C; Pasquini, S; Pertwee, R; Semeraro, T | 1 |
| Brogi, S; Corelli, F; Di Marzo, V; Ligresti, A; Mugnaini, C; Pasquini, S; Tafi, A | 1 |
| Abate, M; Arena, C; Bertini, S; Bifulco, M; Chicca, A; Ciaglia, E; Digiacomo, M; Gado, F; Gertsch, J; Lapillo, M; Macchia, M; Manera, C; Poli, G; Tuccinardi, T | 1 |
| Cheng, J; McCorvy, JD; Tan, L; Yan, W | 1 |
| Bánki, L; Deli, MA; Dvorácskó, S; Horváth, G; Kékesi, G; Keresztes, A; Macedonio, G; Mollica, A; Pieretti, S; Stefanucci, A; Tömböly, C; Tuboly, G; Walter, FR; Zádor, F | 1 |
| Harris, D; Kendall, DA; Randall, MD | 1 |
| Bottrill, FE; Ford, WR; Hiley, CR; Ho, WS; White, R | 1 |
| Amato, A; Baldassano, S; Mulè, F; Serio, R | 2 |
| Baldassano, S; Mule', F; Serio, R | 1 |
| Järbe, TU; Li, C; Makriyannis, A; Vadivel, SK | 1 |
| Calignano, A; Clapper, JR; Duranti, A; Guijarro, A; Hohmann, AG; Mor, M; Moreno-Sanz, G; Piomelli, D; Russo, R; Sanchini, S; Sciolino, NR; Spradley, JM; Tarzia, G; Tontini, A; Vacondio, F | 1 |
| Alhouayek, M; Cani, PD; Delzenne, NM; Lambert, DM; Muccioli, GG | 1 |
| Liao, YS; Wang, P; Wu, J; Zhang, H | 1 |
| Hegde, VL; Lombard, C; Nagarkatti, M; Nagarkatti, PS | 1 |
| Atchison, DK; García, NH; Juncos, LI; Silva, GB | 1 |
| Abdullah, RA; Imhof, E; Lichtman, AH; Limebeer, CL; Parker, LA; Rock, EM; Wang, K | 1 |
| Cruz, JS; De Carvalho, CR; Pamplona, FA; Takahashi, RN | 1 |
| Feng, R; Milcarek, CA; Xie, XQ | 1 |
| Degrace, P; Demizieux, L; Gresti, J; Muller, T; Troy-Fioramonti, S; Vergès, B | 1 |
| Ding, X; Dong, X; Song, C; Wu, X; Zheng, L | 1 |
| Gao, F; Ji, M; Li, F; Li, Q; Miao, Y; Qian, WJ; Sun, XH; Wang, SY; Wang, Z; Yang, W | 1 |
| Bellocchio, L; Bindila, L; Busquets-Garcia, A; Cutando, L; Gomis-González, M; Lutz, B; Maldonado, R; Marsicano, G; Ortega-Alvaro, A; Ozaita, A; Remmers, F; Ruehle, S; Srivastava, RK | 1 |
| Antoniou, K; Delis, F; Goldberg, SR; Justinova, Z; Nomikos, GG; Polissidis, A; Poulia, N | 1 |
| Bramanti, P; Giacoppo, S; Grassi, G; Gugliandolo, A; Mazzon, E; Pollastro, F; Trubiani, O | 1 |
| Cha, HJ; Gu, SM; Han, KM; Kim, HS; Kim, YH; Lee, HJ; Lee, TH; Park, HK; Shin, J; Song, YJ; Yun, J | 1 |
| Beier, JP; Karthaus, N; Kim, BS; Ruhl, T | 1 |
| Akdis, C; Akdis, M; Angelina, A; López-Abente, J; Martín-Fontecha, M; Nombela, I; Palomares, O; Pérez-Diego, M; Rückert, B | 1 |
1 review(s) available for sr141716 and am 630
| Article | Year |
|---|---|
Biased Ligands of G Protein-Coupled Receptors (GPCRs): Structure-Functional Selectivity Relationships (SFSRs) and Therapeutic Potential.
Topics: Animals; Drug Discovery; Humans; Ligands; Receptors, G-Protein-Coupled; Signal Transduction; Structure-Activity Relationship | 2018 |
28 other study(ies) available for sr141716 and am 630
| Article | Year |
|---|---|
New 1,8-naphthyridine and quinoline derivatives as CB2 selective agonists.
Topics: Animals; Cell Line; Humans; Mice; Naphthyridines; Pain Measurement; Quinolines; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2 | 2007 |
Investigations on the 4-quinolone-3-carboxylic acid motif. 3. Synthesis, structure-affinity relationships, and pharmacological characterization of 6-substituted 4-quinolone-3-carboxamides as highly selective cannabinoid-2 receptor ligands.
Topics: Amides; Analgesics; Animals; CHO Cells; Cricetinae; Cricetulus; Drug Inverse Agonism; Humans; Ligands; Mice; Pain Measurement; Quinolones; Radioligand Assay; Receptor, Cannabinoid, CB2; Stereoisomerism; Structure-Activity Relationship | 2010 |
Three-dimensional quantitative structure-selectivity relationships analysis guided rational design of a highly selective ligand for the cannabinoid receptor 2.
Topics: Computer Simulation; Drug Design; Humans; Ligands; Models, Molecular; Molecular Structure; Quantitative Structure-Activity Relationship; Quinolones; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Recombinant Proteins; Stereoisomerism | 2011 |
Polypharmacological profile of 1,2-dihydro-2-oxo-pyridine-3-carboxamides in the endocannabinoid system.
Topics: Dose-Response Relationship, Drug; Endocannabinoids; Humans; Molecular Docking Simulation; Molecular Structure; Pyridines; Receptors, Cannabinoid; Structure-Activity Relationship; Tumor Cells, Cultured; U937 Cells | 2018 |
Preparation of bivalent agonists for targeting the mu opioid and cannabinoid receptors.
Topics: Analgesics, Opioid; Animals; Dose-Response Relationship, Drug; Enkephalins; Indoles; Mice; Molecular Structure; Naphthalenes; Oxycodone; Rats; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Receptors, Opioid, mu; Structure-Activity Relationship | 2019 |
Characterization of cannabinoid receptors coupled to vasorelaxation by endothelium-derived hyperpolarizing factor.
Topics: Animals; Benzofurans; Biological Factors; Carbachol; Cyclooxygenase Inhibitors; Endothelium, Vascular; In Vitro Techniques; Indoles; Male; Muscarinic Agonists; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB2; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Vasodilation | 1999 |
Mechanisms of anandamide-induced vasorelaxation in rat isolated coronary arteries.
Topics: Amides; Animals; Arachidonic Acids; Capsaicin; Coronary Vessels; Dose-Response Relationship, Drug; Endocannabinoids; Endothelium, Vascular; Ethanolamines; Gap Junctions; Glycyrrhetinic Acid; In Vitro Techniques; Indoles; Indomethacin; Male; Palmitic Acids; Peptides; Piperidines; Polyunsaturated Alkamides; Potassium Channel Blockers; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB2; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Serotonin; Tetraethylammonium; Vasodilation | 2001 |
Evidence for a modulatory role of cannabinoids on the excitatory NANC neurotransmission in mouse colon.
Topics: Animals; Arachidonic Acids; Benzoxazines; Cannabinoid Receptor Modulators; Cannabinoids; Colon; Dose-Response Relationship, Drug; Electric Stimulation; Endocannabinoids; Enteric Nervous System; Excitatory Postsynaptic Potentials; Gastrointestinal Motility; In Vitro Techniques; Indoles; Inhibitory Postsynaptic Potentials; Mice; Mice, Inbred C57BL; Morpholines; Naphthalenes; Neuromuscular Junction; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Receptors, Tachykinin; Rimonabant; Synaptic Transmission; Tachykinins | 2007 |
Involvement of CB1 and CB2 receptors in the modulation of cholinergic neurotransmission in mouse gastric preparations.
Topics: Animals; Arachidonic Acids; Benzoxazines; Cannabinoid Receptor Modulators; Cannabinoids; Cholinergic Fibers; Electric Stimulation; Endocannabinoids; Excitatory Postsynaptic Potentials; Gastrointestinal Motility; In Vitro Techniques; Indoles; Inhibitory Postsynaptic Potentials; Male; Mice; Mice, Inbred C57BL; Morpholines; Naphthalenes; Neuromuscular Junction; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Receptors, Presynaptic; Rimonabant; Stomach; Synaptic Transmission | 2007 |
Cannabinoid CB(1) receptor activation modulates spontaneous contractile activity in mouse ileal longitudinal muscle.
Topics: Animals; Apamin; Arachidonic Acids; Atropine; Cannabinoid Receptor Modulators; Cannabinoids; Dose-Response Relationship, Drug; Endocannabinoids; Hexamethonium; Ileum; In Vitro Techniques; Indoles; Male; Mice; Mice, Inbred C57BL; Muscle Contraction; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant; Tetrodotoxin | 2008 |
Discriminative stimulus effects of the cannabinoid CB1 receptor antagonist rimonabant in rats.
Topics: Animals; Arachidonic Acids; Avoidance Learning; Camphanes; Discrimination Learning; Discrimination, Psychological; Dose-Response Relationship, Drug; Drinking; Dronabinol; Hallucinogens; Indoles; Injections, Intraperitoneal; Lithium Chloride; Male; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant; Taste | 2008 |
Anandamide suppresses pain initiation through a peripheral endocannabinoid mechanism.
Topics: Amidohydrolases; Animals; Arachidonic Acids; Cannabinoid Receptor Modulators; Cannabinoids; Carrageenan; Chromatography, Liquid; Disease Models, Animal; Drug Administration Routes; Drug Administration Schedule; Endocannabinoids; Enzyme Inhibitors; Escape Reaction; Ethylene Glycols; Feeding Behavior; Formaldehyde; Gene Expression Regulation; Hyperalgesia; Indoles; Male; Mass Spectrometry; Mice; Mice, Inbred C57BL; Mice, Knockout; Monoacylglycerol Lipases; Motor Activity; Oncogene Proteins v-fos; Pain; Pain Measurement; Pain Threshold; Peripheral Nervous System Diseases; Piperidines; Polyunsaturated Alkamides; PPAR alpha; Pyrazoles; Rats; Rats, Sprague-Dawley; Rimonabant; Sciatica; Spinal Cord; Statistics, Nonparametric; Time Factors; Tissue Distribution; Tritium | 2010 |
Increasing endogenous 2-arachidonoylglycerol levels counteracts colitis and related systemic inflammation.
Topics: Animals; Arachidonic Acids; Benzodioxoles; Colitis; Disease Models, Animal; Endocannabinoids; Endotoxemia; Enzyme Inhibitors; Glycerides; Humans; Indoles; Inflammation; Inflammation Mediators; Inflammatory Bowel Diseases; Male; Mice; Mice, Inbred C57BL; Monoacylglycerol Lipases; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant; Trinitrobenzenesulfonic Acid | 2011 |
[Anandamide inhibits the growth of colorectal cancer cells through CB1 and lipid rafts].
Topics: Antineoplastic Agents; Apoptosis; Arachidonic Acids; beta-Cyclodextrins; Caco-2 Cells; Cannabinoid Receptor Modulators; Caspase 3; Cell Proliferation; Dose-Response Relationship, Drug; Endocannabinoids; Humans; Indoles; Membrane Microdomains; Piperidines; Polyunsaturated Alkamides; Proto-Oncogene Proteins c-akt; Pyrazoles; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant | 2011 |
Perinatal exposure to Δ9-tetrahydrocannabinol triggers profound defects in T cell differentiation and function in fetal and postnatal stages of life, including decreased responsiveness to HIV antigens.
Topics: Animals; Apoptosis; Cannabinoid Receptor Agonists; Cannabinoid Receptor Antagonists; Caspases; Dronabinol; Female; Fetus; HIV Antibodies; HIV Antigens; HIV-1; Indoles; Lymphocyte Activation; Lymphopoiesis; Marijuana Smoking; Mice; Mice, Inbred C57BL; Piperidines; Pregnancy; Prenatal Exposure Delayed Effects; Psychotropic Drugs; Pyrazoles; Receptors, Cannabinoid; Rimonabant; T-Lymphocytes; Thymocytes; Thymus Gland | 2011 |
Anandamide inhibits transport-related oxygen consumption in the loop of Henle by activating CB1 receptors.
Topics: Animals; Arachidonic Acids; Benzoxazines; Cannabinoid Receptor Agonists; Cannabinoid Receptor Antagonists; Cannabinoids; Cell Culture Techniques; Endocannabinoids; Indoles; Ion Transport; Loop of Henle; Male; Morpholines; Naphthalenes; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Oxygen Consumption; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Rimonabant | 2013 |
Attenuation of anticipatory nausea in a rat model of contextually elicited conditioned gaping by enhancement of the endocannabinoid system.
Topics: Amidohydrolases; Animals; Anticipation, Psychological; Arachidonic Acids; Brain; Cannabinoid Receptor Antagonists; Carbamates; Endocannabinoids; Enzyme Inhibitors; Glycerides; Indoles; Lithium Chloride; Male; Monoacylglycerol Lipases; Motor Activity; Nausea; Oleic Acids; Piperazines; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant | 2014 |
Endocannabinoids underlie reconsolidation of hedonic memories in Wistar rats.
Topics: Amidohydrolases; Animals; Benzamides; Benzoxazines; Carbamates; Conditioning, Psychological; Cues; Endocannabinoids; Indoles; Male; Memory; Morphine; Morpholines; Naphthalenes; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Recurrence; Rimonabant; Secondary Prevention | 2014 |
Antagonism of cannabinoid receptor 2 pathway suppresses IL-6-induced immunoglobulin IgM secretion.
Topics: Camphanes; Cannabinoids; Cell Line; Cell Proliferation; DNA-Binding Proteins; Humans; Immunoglobulin M; Indoles; Interleukin-6; PAX5 Transcription Factor; Piperidines; Proto-Oncogene Proteins c-bcl-6; Pyrazoles; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant; STAT3 Transcription Factor | 2014 |
Acute activation of cannabinoid receptors by anandamide reduces gastrointestinal motility and improves postprandial glycemia in mice.
Topics: Animals; Arachidonic Acids; Blood Glucose; Endocannabinoids; Gastrointestinal Motility; Gastrointestinal Transit; Hyperglycemia; Indoles; Male; Mice; Mice, Inbred C57BL; Piperidines; Polyunsaturated Alkamides; Postprandial Period; Pyrazoles; Rats; Rats, Wistar; Receptors, Cannabinoid; Reverse Transcriptase Polymerase Chain Reaction; Rimonabant | 2015 |
Effects of Chronic Alcohol Exposure on the Modulation of Ischemia-Induced Glutamate Release via Cannabinoid Receptors in the Dorsal Hippocampus.
Topics: Animals; Arachidonic Acids; Cannabinoids; Dose-Response Relationship, Drug; Ethanol; Glutamic Acid; Hippocampus; Indoles; Infarction, Middle Cerebral Artery; Ischemia; Male; Piperidines; Pyrazoles; Rats; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant | 2015 |
Cannabinoid receptor agonists modulate calcium channels in rat retinal Müller cells.
Topics: Animals; Arachidonic Acids; Benzoxazines; Calcium; Calcium Channels; Cannabinoid Receptor Agonists; Cannabinoid Receptor Antagonists; Cells, Cultured; Dose-Response Relationship, Drug; Endocannabinoids; Ependymoglial Cells; Glycerides; Indoles; Male; Membrane Potentials; Morpholines; Naphthalenes; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant | 2016 |
Peripheral and central CB1 cannabinoid receptors control stress-induced impairment of memory consolidation.
Topics: Animals; Anisomycin; Dopamine beta-Hydroxylase; Electroshock; Hindlimb Suspension; Indoles; Male; Memory Consolidation; Memory Disorders; Mice, Knockout; Neurons; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Rimonabant; Stress, Psychological | 2016 |
Attenuation of Cocaine-Induced Conditioned Place Preference and Motor Activity via Cannabinoid CB2 Receptor Agonism and CB1 Receptor Antagonism in Rats.
Topics: Animals; Cannabinoids; Cocaine; Conditioning, Classical; Indoles; Male; Motor Activity; Piperidines; Pyrazoles; Rats; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant | 2017 |
Cannabinoid CB2 receptors are involved in the protection of RAW264.7 macrophages against the oxidative stress: an in vitro study.
Topics: Animals; bcl-2-Associated X Protein; Cannabinoids; Hydrogen Peroxide; Indoles; Macrophages; Mice; Nitric Oxide Synthase Type II; Oxidative Stress; Piperidines; Poly (ADP-Ribose) Polymerase-1; Proto-Oncogene Proteins c-bcl-2; Pyrazoles; RAW 264.7 Cells; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant; Superoxide Dismutase-1; Tyrosine | 2017 |
A synthetic cannabinoid JWH-210 reduces lymphoid organ weights and T-cell activator levels in mice via CB
Topics: Animals; B7-1 Antigen; Cell Survival; Cytokines; Female; Indoles; Lymphoid Tissue; Male; Mice; Mice, Inbred ICR; Naphthalenes; Organ Size; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB2; Rimonabant; Spleen; T-Lymphocytes; Thymocytes; Tumor Necrosis Factor Receptor Superfamily, Member 7 | 2017 |
The endocannabinoid receptors CB1 and CB2 affect the regenerative potential of adipose tissue MSCs.
Topics: Adipose Tissue; Benzoxazines; Cannabinoids; Cell Differentiation; Cell Self Renewal; Cells, Cultured; Cytokines; Dose-Response Relationship, Drug; Endocannabinoids; Humans; Indoles; Intercellular Signaling Peptides and Proteins; Mesenchymal Stem Cells; Morpholines; Naphthalenes; Primary Cell Culture; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Regeneration; Rimonabant | 2020 |
Cannabinoids induce functional Tregs by promoting tolerogenic DCs via autophagy and metabolic reprograming.
Topics: Anaphylaxis; Animals; Anti-Inflammatory Agents; Autophagy; Cannabinoids; Cells, Cultured; Cellular Reprogramming; Coculture Techniques; Dendritic Cells; Humans; Hypersensitivity; Immune Tolerance; Indoles; Mice; Oxidative Phosphorylation; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant; Signal Transduction; T-Lymphocytes, Regulatory; Th1-Th2 Balance | 2022 |