Page last updated: 2024-08-26

sr141716 and am 404

sr141716 has been researched along with am 404 in 40 studies

Research

Studies (40)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (10.00)18.2507
2000's24 (60.00)29.6817
2010's12 (30.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chung, S; Dangott, LJ; Huang, H; Kier, AB; Landrock, D; Landrock, KK; Li, S; Martin, GG; McIntosh, AL; Schroeder, F1
Beltramo, M; Calignano, A; Lin, SY; Makriyannis, A; Piomelli, D; Stella, N1
Beltramo, M; Calignano, A; La Rana, G; Makriyannis, A; Piomelli, D1
Beltramo, M; Calignano, A; La Rana, G; Lin, SY; Makriyannis, A; Piomelli, D1
Chaytor, AT; Evans, WH; Griffith, TM; Martin, PE; Randall, MD1
Chuang, H; Högestätt, ED; Julius, D; Movahed, P; Zygmunt, PM1
Baker, D; Bisogno, T; Brown, P; Croxford, JL; Di Marzo , V; Fezza, F; Khanolkar, A; Layward, L; Makriyannis, A; Pertwee, RG; Pryce, G1
Bari, M; Del Principe, D; Finazzi-Agrò, A; Giuliani, E; MacCarrone, M; Menichelli, A1
Beltramo, M; Giuffrida, A; Piomelli, D1
Rice, AS1
Boachie-Ansah, G; Grainger, J1
Calignano, A; Cuomo, V; Duranti, A; Fegley, D; Gaetani, S; Giustino, A; Kathuria, S; La Rana, G; Mor, M; Palmery, M; Piomelli, D; Tarzia, G; Tattoli, M; Tontini, A; Valiño, F1
de Miguel, R; De Petrocellis, L; Di Marzo, V; Fernández-Ruiz, J; Lastres-Becker, I; Makriyannis, A1
Feuerstein, TJ; Klar, M; Rominger, A; Steffens, M; Szabo, B; Zentner, J1
Dougalis, A; Lees, G1
Gerdeman, GL; Lovinger, DM; Ronesi, J1
Mendiguren, A; Pineda, J1
Bátkai, S; Bukoski, RD; Harvey-White, J; Kunos, G; Liu, J; Mackie, K; Offertáler, L; Osei-Hyiaman, D; Pacher, P; Radaeva, S; Rudd, MA1
Adrian, R; Baratta, J; Giuffrida, A; Piomelli, D; Solbrig, MV1
Bortolato, M; Calignano, A; Campolongo, P; Cuomo, V; Frau, R; Gessa, GL; La Rana, G; Mangieri, RA; Piomelli, D; Russo, R; Scattoni, ML; Trezza, V1
Cowan, A; Ding, Z; Rawls, SM1
Cheer, JF; Wassum, KM; Wightman, RM1
de Novellis, V; Di Marzo, V; Giordano, C; Maione, S; Mangoni, GS; Marabese, I; Palazzo, E; Petrosino, S; Rossi, F; Vita, D1
Herradón, E; López-Miranda, V; Martín, MI1
Bilbao, A; Fernandez-Espejo, E; Ferrer, B; Gorriti, MA; Martín, AB; Moratalla, R; Navarro, M; Rodriguez de Fonseca, F1
Nomikos, GG; Panagis, G; Stamatopoulou, F; Vlachou, S1
Bitencourt, RM; Pamplona, FA; Takahashi, RN3
Davis, MI; Lovinger, DM; Sheinin, A; Talani, G1
Baufreton, J; Manuel, I; Morera-Herreras, T; Rodriguez-Puertas, R; Ruiz-Ortega, JA; Taupignon, A; Ugedo, L1
Alger, BE; Kim, J1
Deadwyler, SA; Hampson, RE; Miller, F; Palchik, G1
Alen, F; Gómez, R; Orio, L; Pavón, FJ; Reyes-Cabello, C; Rivera, P; Rodríguez de Fonseca, F; Serrano, A1
Abou-El-Ela, SH; El-Wakeil, AF; Zaitone, SA1
Bajaj, S; Bergman, J; Makriyannis, A; Nikas, SP; Paronis, CA; Thakur, GA; Vemuri, VK1
Abílio, VC; Almeida, V; Calzavara, MB; Crippa, JA; Hallak, JE; Levin, R; Peres, FF; Suiama, MA; Zuardi, AW1
di Marzo, V; Llorente-Berzal, A; Micale, V; Terzian, AL; Viveros, MP; Wotjak, CT1
Goldberg, SR; Justinova, Z; Makriyannis, A; Redhi, GH; Scherma, M; Schindler, CW; Vadivel, SK1
Drago, F; Eder, M; Jurik, A; Marsch, R; Micale, V; Pamplona, FA; Stepan, J; Wotjak, CT1

Reviews

2 review(s) available for sr141716 and am 404

ArticleYear
Mechanisms of endocannabinoid inactivation: biochemistry and pharmacology.
    The Journal of pharmacology and experimental therapeutics, 2001, Volume: 298, Issue:1

    Topics: Amidohydrolases; Arachidonic Acid; Arachidonic Acids; Biological Transport; Brain; Cannabinoid Receptor Modulators; Cannabinoids; Endocannabinoids; Glycerides; Piperidines; Pyrazoles; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Structure-Activity Relationship

2001
Cannabinoids and pain.
    Current opinion in investigational drugs (London, England : 2000), 2001, Volume: 2, Issue:3

    Topics: Amides; Amidohydrolases; Analgesics; Animals; Arachidonic Acids; Benzoxazines; Brain; Camphanes; Cannabinoid Receptor Modulators; Cannabinoids; Cell Membrane; Clinical Trials as Topic; Disease Models, Animal; Drug Design; Drug Interactions; Endocannabinoids; Enzyme Inhibitors; Ethanolamines; Glycerides; Humans; Injections, Spinal; Molecular Structure; Morpholines; Naphthalenes; Pain; Palmitates; Palmitic Acids; Piperidines; Plant Extracts; Polyunsaturated Alkamides; Pyrazoles; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Spinal Cord

2001

Other Studies

38 other study(ies) available for sr141716 and am 404

ArticleYear
FABP1: A Novel Hepatic Endocannabinoid and Cannabinoid Binding Protein.
    Biochemistry, 2016, 09-20, Volume: 55, Issue:37

    Topics: Animals; Endocannabinoids; Fatty Acid-Binding Proteins; Female; Fluorescent Dyes; Humans; Liver; Male; Mice; Mice, Inbred C57BL; Receptors, Cannabinoid

2016
Functional role of high-affinity anandamide transport, as revealed by selective inhibition.
    Science (New York, N.Y.), 1997, Aug-22, Volume: 277, Issue:5329

    Topics: Analgesics; Animals; Arachidonic Acids; Astrocytes; Benzoxazines; Biological Transport; Bromcresol Green; Cannabinoids; Cells, Cultured; Colforsin; Cyclic AMP; Endocannabinoids; Male; Mice; Morpholines; Naphthalenes; Neurons; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Receptors, Cannabinoid; Receptors, Drug; Rimonabant

1997
Potentiation of anandamide hypotension by the transport inhibitor, AM404.
    European journal of pharmacology, 1997, Oct-15, Volume: 337, Issue:1

    Topics: Animals; Arachidonic Acids; Blood Pressure; Cannabinoids; Depression, Chemical; Dose-Response Relationship, Drug; Drug Synergism; Endocannabinoids; Guinea Pigs; Male; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptors, Drug; Rimonabant; Time Factors

1997
Inhibition of intestinal motility by anandamide, an endogenous cannabinoid.
    European journal of pharmacology, 1997, Dec-11, Volume: 340, Issue:2-3

    Topics: Animals; Arachidonic Acids; Cannabinoids; Cell Membrane; Endocannabinoids; Gastrointestinal Motility; Male; Mice; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptors, Cannabinoid; Receptors, Drug; Rimonabant

1997
The endothelial component of cannabinoid-induced relaxation in rabbit mesenteric artery depends on gap junctional communication.
    The Journal of physiology, 1999, Oct-15, Volume: 520 Pt 2

    Topics: Acetylcholine; Animals; Arachidonic Acids; Benzofurans; Cannabinoid Receptor Modulators; Cannabinoids; COS Cells; Endocannabinoids; Gap Junctions; Glycyrrhetinic Acid; Indomethacin; Isoquinolines; Male; Mesenteric Artery, Superior; Muscle Relaxation; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Phenylephrine; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rabbits; Receptors, Cannabinoid; Receptors, Drug; Rimonabant

1999
The anandamide transport inhibitor AM404 activates vanilloid receptors.
    European journal of pharmacology, 2000, May-12, Volume: 396, Issue:1

    Topics: Animals; Arachidonic Acids; Calcitonin Gene-Related Peptide; Cannabinoids; Capsaicin; Endocannabinoids; Female; Hepatic Artery; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Oocytes; Patch-Clamp Techniques; Peptide Fragments; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Receptors, Drug; Rimonabant; Vasodilation; Xenopus

2000
Endocannabinoids control spasticity in a multiple sclerosis model.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 2001, Volume: 15, Issue:2

    Topics: Amides; Animals; Arachidonic Acids; Brain; Cannabinoid Receptor Modulators; Cannabinoids; Disease Models, Animal; Encephalomyelitis, Autoimmune, Experimental; Endocannabinoids; Ethanolamines; Glycerides; Humans; Mice; Mice, Inbred Strains; Multiple Sclerosis; Palmitic Acids; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Spasm; Spinal Cord

2001
Human platelets bind and degrade 2-arachidonoylglycerol, which activates these cells through a cannabinoid receptor.
    European journal of biochemistry, 2001, Volume: 268, Issue:3

    Topics: Adenosine Diphosphate; Amidohydrolases; Arachidonic Acids; Aspirin; Biological Transport; Blood Platelets; Calcium Channel Blockers; Camphanes; Cannabinoid Receptor Modulators; Collagen; Cyclic AMP; Endocannabinoids; Glycerides; Humans; Hydrolysis; Inositol 1,4,5-Trisphosphate; Kinetics; Piperidines; Platelet Activation; Polyunsaturated Alkamides; Pyrazoles; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Serotonin; Time Factors

2001
Anandamide-induced relaxation of sheep coronary arteries: the role of the vascular endothelium, arachidonic acid metabolites and potassium channels.
    British journal of pharmacology, 2001, Volume: 134, Issue:5

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; 4-Aminopyridine; Animals; Apamin; Arachidonic Acid; Arachidonic Acids; Barium; Calcium Channel Blockers; Cannabinoid Receptor Modulators; Cannabinoids; Capsaicin; Coronary Vessels; Cytochrome P-450 Enzyme Inhibitors; Dose-Response Relationship, Drug; Endocannabinoids; Endothelium, Vascular; Enzyme Inhibitors; Fatty Acids, Unsaturated; Glyburide; In Vitro Techniques; Indomethacin; Miconazole; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Peptides; Phenylmethylsulfonyl Fluoride; Piperidines; Polyunsaturated Alkamides; Potassium; Potassium Channel Blockers; Potassium Channels; Pyrazoles; Receptors, Drug; Rimonabant; Sheep; Tetraethylammonium; Vasoconstrictor Agents; Vasodilation

2001
Modulation of anxiety through blockade of anandamide hydrolysis.
    Nature medicine, 2003, Volume: 9, Issue:1

    Topics: Amidohydrolases; Animals; Anti-Anxiety Agents; Anxiety; Arachidonic Acids; Behavior, Animal; Cannabinoids; Cells, Cultured; Dose-Response Relationship, Drug; Endocannabinoids; Humans; Molecular Structure; Neurons; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Radioligand Assay; Rats; Rats, Wistar; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Vocalization, Animal

2003
Compounds acting at the endocannabinoid and/or endovanilloid systems reduce hyperkinesia in a rat model of Huntington's disease.
    Journal of neurochemistry, 2003, Volume: 84, Issue:5

    Topics: 3,4-Dihydroxyphenylacetic Acid; Amino Acids, Neutral; Animals; Arachidonic Acids; Basal Ganglia; Cannabinoid Receptor Modulators; Capsaicin; Corpus Striatum; Cyclohexanols; Disease Models, Animal; Dopamine; Endocannabinoids; gamma-Aminobutyric Acid; Huntington Disease; Hyperkinesis; Male; Motor Activity; Nitro Compounds; Palmitates; Piperidines; Propionates; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptors, Cannabinoid; Receptors, Drug; Rimonabant

2003
Modulation of electrically evoked acetylcholine release through cannabinoid CB1 receptors: evidence for an endocannabinoid tone in the human neocortex.
    Neuroscience, 2003, Volume: 120, Issue:2

    Topics: Acetylcholine; Adolescent; Adult; Animals; Arachidonic Acids; Benzoxazines; Binding, Competitive; Brain Chemistry; Calcium Channel Blockers; Cannabinoid Receptor Modulators; Child; Choline; Dose-Response Relationship, Drug; Dronabinol; Electric Stimulation; Endocannabinoids; Hemicholinium 3; Humans; Mice; Middle Aged; Morpholines; Naphthalenes; Neocortex; Nootropic Agents; Piperidines; Pyrazoles; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Tritium

2003
Differential effects of the sleep-inducing lipid oleamide and cannabinoids on the induction of long-term potentiation in the CA1 neurons of the rat hippocampus in vitro.
    Brain research, 2004, Jan-30, Volume: 997, Issue:1

    Topics: Amidohydrolases; Analysis of Variance; Animals; Animals, Newborn; Arachidonic Acids; Benzoxazines; Cannabinoids; Capsaicin; Drug Interactions; Electric Stimulation; Electrophysiology; Endocannabinoids; Excitatory Postsynaptic Potentials; Hippocampus; Hypnotics and Sedatives; In Vitro Techniques; Long-Term Potentiation; Male; Morpholines; Naphthalenes; Neurons; Oleic Acids; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rimonabant; Sleep

2004
Disruption of endocannabinoid release and striatal long-term depression by postsynaptic blockade of endocannabinoid membrane transport.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2004, Feb-18, Volume: 24, Issue:7

    Topics: Animals; Arachidonic Acids; Benzoxazines; Biological Transport; Cannabinoid Receptor Modulators; Cell Membrane; Corpus Striatum; Electric Stimulation; Endocannabinoids; Excitatory Postsynaptic Potentials; Glutamic Acid; In Vitro Techniques; Long-Term Synaptic Depression; Morpholines; Naphthalenes; Neurons; Patch-Clamp Techniques; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptors, Drug; Rimonabant; Synapses

2004
Cannabinoids enhance N-methyl-D-aspartate-induced excitation of locus coeruleus neurons by CB1 receptors in rat brain slices.
    Neuroscience letters, 2004, Jun-03, Volume: 363, Issue:1

    Topics: Action Potentials; Analgesics; Animals; Arachidonic Acids; Benzoxazines; Calcium Channel Blockers; Cannabinoids; Cyclohexanols; Drug Interactions; Electrophysiology; Endocannabinoids; Excitatory Amino Acid Agonists; In Vitro Techniques; Locus Coeruleus; Male; Morpholines; N-Methylaspartate; Naphthalenes; Neurons; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Rimonabant

2004
Endocannabinoids acting at cannabinoid-1 receptors regulate cardiovascular function in hypertension.
    Circulation, 2004, Oct-05, Volume: 110, Issue:14

    Topics: Amidohydrolases; Angiotensin II; Animals; Arachidonic Acids; Benzamides; Benzyl Compounds; Blood Pressure; Camphanes; Carbamates; Dronabinol; Endocannabinoids; Endothelium, Vascular; Hypertension; Male; Models, Cardiovascular; Myocardial Contraction; Myocardium; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Inbred Dahl; Rats, Inbred SHR; Rats, Inbred WKY; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Rimonabant; Up-Regulation; Vascular Resistance; Vasodilation; Ventricular Function, Left

2004
A role for endocannabinoids in viral-induced dyskinetic and convulsive phenomena.
    Experimental neurology, 2005, Volume: 194, Issue:2

    Topics: Animals; Anticonvulsants; Arachidonic Acids; Basal Ganglia; Borna Disease; Cannabinoid Receptor Modulators; Convulsants; Disease Models, Animal; Endocannabinoids; Limbic System; Male; Movement Disorders; Naloxone; Narcotic Antagonists; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Inbred Lew; Receptor, Cannabinoid, CB1; Rimonabant; Seizures

2005
Anxiolytic-like properties of the anandamide transport inhibitor AM404.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2006, Volume: 31, Issue:12

    Topics: Animals; Animals, Newborn; Anti-Anxiety Agents; Anxiety Disorders; Anxiety, Separation; Arachidonic Acids; Behavior, Animal; Brain; Cannabinoid Receptor Modulators; Carrier Proteins; Disease Models, Animal; Endocannabinoids; Male; Maze Learning; Neural Inhibition; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptor, Cannabinoid, CB1; Reflex, Startle; Rimonabant

2006
Role of TRPV1 and cannabinoid CB1 receptors in AM 404-evoked hypothermia in rats.
    Pharmacology, biochemistry, and behavior, 2006, Volume: 83, Issue:4

    Topics: Amidohydrolases; Anilides; Animals; Arachidonic Acids; Body Temperature; Capsaicin; Cinnamates; Endocannabinoids; Hypothermia; Male; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Rimonabant; TRPV Cation Channels

2006
Cannabinoid modulation of electrically evoked pH and oxygen transients in the nucleus accumbens of awake rats.
    Journal of neurochemistry, 2006, Volume: 97, Issue:4

    Topics: Animals; Arachidonic Acids; Benzoxazines; Calcium Channel Blockers; Cannabinoids; Cerebrovascular Circulation; Electric Stimulation; Energy Metabolism; Hydrogen-Ion Concentration; Male; Medial Forebrain Bundle; Morpholines; Naphthalenes; Nucleus Accumbens; Oxygen Consumption; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Rimonabant

2006
Neuropathic pain and the endocannabinoid system in the dorsal raphe: pharmacological treatment and interactions with the serotonergic system.
    The European journal of neuroscience, 2006, Volume: 24, Issue:7

    Topics: Action Potentials; Analysis of Variance; Animals; Arachidonic Acids; Behavior, Animal; Benzoxazines; Cannabinoid Receptor Modulators; Disease Models, Animal; Drug Interactions; Endocannabinoids; Hot Temperature; Hyperalgesia; Male; Microdialysis; Morpholines; Naphthalenes; Neurons; Pain Measurement; Piperidines; Pyrazoles; Raphe Nuclei; Rats; Rats, Wistar; Reaction Time; Rimonabant; Sciatic Neuropathy; Serotonin; Touch

2006
Characterization of the vasorelaxant mechanisms of the endocannabinoid anandamide in rat aorta.
    British journal of pharmacology, 2007, Volume: 152, Issue:5

    Topics: Animals; Aorta, Abdominal; Apamin; Arachidonic Acids; Benzamides; Calcitonin Gene-Related Peptide; Camphanes; Cannabinoid Receptor Modulators; Capsaicin; Carbamates; Charybdotoxin; Dose-Response Relationship, Drug; Endocannabinoids; Endothelium, Vascular; In Vitro Techniques; Indomethacin; Isoindoles; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Peptide Fragments; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant; Sulfonamides; Vasodilation

2007
Expression and function of CB1 receptor in the rat striatum: localization and effects on D1 and D2 dopamine receptor-mediated motor behaviors.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2008, Volume: 33, Issue:7

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Arachidonic Acids; Behavior, Animal; Corpus Striatum; Dopamine Agonists; Enkephalins; Gene Expression Regulation; Grooming; Male; Models, Biological; Motor Activity; Movement; Nerve Tissue Proteins; Neurons; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptors, Dopamine D1; Receptors, Dopamine D2; Rimonabant; Substance P

2008
Enhancement of endocannabinoid neurotransmission through CB1 cannabinoid receptors counteracts the reinforcing and psychostimulant effects of cocaine.
    The international journal of neuropsychopharmacology, 2008, Volume: 11, Issue:7

    Topics: Animals; Arachidonic Acids; Benzoxazines; Cannabinoid Receptor Modulators; Central Nervous System Stimulants; Cocaine; Conditioning, Operant; Endocannabinoids; Male; Morpholines; Motor Activity; Naphthalenes; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Reward; Rimonabant; Self Stimulation; Synaptic Transmission

2008
Short- and long-term effects of cannabinoids on the extinction of contextual fear memory in rats.
    Neurobiology of learning and memory, 2008, Volume: 90, Issue:1

    Topics: Animals; Arachidonic Acids; Benzoxazines; Calcium Channel Blockers; Cannabinoids; Conditioning, Psychological; Extinction, Psychological; Fear; Freezing Reaction, Cataleptic; Male; Memory; Morpholines; Naphthalenes; Piperidines; Pyrazoles; Rats; Rats, Wistar; Rimonabant; Time Factors

2008
Endocannabinoid- and mGluR5-dependent short-term synaptic depression in an isolated neuron/bouton preparation from the hippocampal CA1 region.
    Journal of neurophysiology, 2008, Volume: 100, Issue:2

    Topics: Animals; Animals, Newborn; Arachidonic Acids; Benzoxazines; Cannabinoid Receptor Modulators; Drug Interactions; Endocannabinoids; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Glycerides; Hippocampus; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Methoxyhydroxyphenylglycol; Morpholines; Naphthalenes; Neurons; Patch-Clamp Techniques; Piperidines; Pyrazoles; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Rimonabant; Synapses; Synapsins

2008
Facilitation of contextual fear memory extinction and anti-anxiogenic effects of AM404 and cannabidiol in conditioned rats.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 2008, Volume: 18, Issue:12

    Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Arachidonic Acids; Behavior, Animal; Cannabidiol; Capsaicin; Conditioning, Psychological; Dose-Response Relationship, Drug; Drug Administration Schedule; Extinction, Psychological; Fear; Freezing Reaction, Cataleptic; Injections, Intraventricular; Male; Maze Learning; Piperidines; Pyrazoles; Rats; Rats, Wistar; Rimonabant; TRPV Cation Channels

2008
Regulation of subthalamic neuron activity by endocannabinoids.
    Synapse (New York, N.Y.), 2010, Volume: 64, Issue:9

    Topics: Animals; Arachidonic Acids; Benzamides; Cannabinoid Receptor Modulators; Carbamates; Cerebral Cortex; Dose-Response Relationship, Drug; Dronabinol; Electrophysiology; Endocannabinoids; Globus Pallidus; Immunohistochemistry; Injections, Intraventricular; Male; Microinjections; Neurons; Piperidines; Polyunsaturated Alkamides; Prefrontal Cortex; Pyrazoles; Rats; Rats, Sprague-Dawley; Rimonabant; Subthalamic Nucleus

2010
Reduction in endocannabinoid tone is a homeostatic mechanism for specific inhibitory synapses.
    Nature neuroscience, 2010, Volume: 13, Issue:5

    Topics: Agatoxins; Animals; Arachidonic Acids; Benzamides; Benzoxazines; Biophysics; Calcium; Calcium Channel Blockers; Cannabinoid Receptor Modulators; Carbamates; Conotoxins; Dose-Response Relationship, Drug; Down-Regulation; Drug Interactions; Electric Stimulation; Endocannabinoids; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Glycerides; Hippocampus; Homeostasis; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Morpholines; Naphthalenes; Nerve Net; Neural Inhibition; Neurons; Patch-Clamp Techniques; Piperidines; Polyamines; Polyunsaturated Alkamides; Pyrazoles; Rats; Receptor, Cannabinoid, CB1; Rimonabant; Sodium Channel Blockers; Synapses; Tetrodotoxin

2010
Cannabinoid receptor activation modifies NMDA receptor mediated release of intracellular calcium: implications for endocannabinoid control of hippocampal neural plasticity.
    Neuropharmacology, 2011, Volume: 60, Issue:6

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Arachidonic Acids; Benzamides; Benzoxazines; Calcium; Cannabinoid Receptor Modulators; Carbamates; Endocannabinoids; Glycine; Hippocampus; In Vitro Techniques; Morpholines; Naphthalenes; Neuronal Plasticity; Neurons; Phosphorylation; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptors, N-Methyl-D-Aspartate; Rimonabant; Ryanodine Receptor Calcium Release Channel; Second Messenger Systems

2011
Effects of the anandamide uptake blocker AM404 on food intake depend on feeding status and route of administration.
    Pharmacology, biochemistry, and behavior, 2012, Volume: 101, Issue:1

    Topics: Animals; Arachidonic Acids; Eating; Endocannabinoids; Energy Intake; Feeding Behavior; Food Deprivation; Injections, Intraperitoneal; Injections, Intraventricular; Male; Mice; Mice, Knockout; Nutritional Status; Oxazoles; Piperidines; Polyunsaturated Alkamides; PPAR alpha; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Rimonabant; Satiation; Tyrosine

2012
Inhibition of fatty acid amide hydrolase by URB597 attenuates the anxiolytic-like effect of acetaminophen in the mouse elevated plus-maze test.
    Behavioural pharmacology, 2012, Volume: 23, Issue:4

    Topics: Acetaminophen; Amidohydrolases; Animals; Anti-Anxiety Agents; Anxiety; Arachidonic Acids; Benzamides; Carbamates; Disease Models, Animal; Dose-Response Relationship, Drug; Injections, Intraperitoneal; Male; Maze Learning; Mice; Mice, Inbred BALB C; Motor Activity; Piperidines; Pyrazoles; Rimonabant

2012
Diuretic effects of cannabinoids.
    The Journal of pharmacology and experimental therapeutics, 2013, Volume: 344, Issue:1

    Topics: Adamantane; Animals; Arachidonic Acids; Benzoxazines; Body Temperature; Cannabinoid Receptor Antagonists; Cannabinoids; Cannabinol; Confidence Intervals; Diuresis; Diuretics; Dose-Response Relationship, Drug; Dronabinol; Female; Male; Morpholines; Naphthalenes; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Rimonabant; Water

2013
Corticosteroid-endocannabinoid loop supports decrease of fear-conditioned response in rats.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 2014, Volume: 24, Issue:7

    Topics: Adrenal Cortex Hormones; Animals; Arachidonic Acids; Benzoxazines; Cannabinoid Receptor Modulators; Conditioning, Classical; Dexamethasone; Endocannabinoids; Extinction, Psychological; Fear; Freezing Reaction, Cataleptic; Male; Metyrapone; Mifepristone; Mineralocorticoid Receptor Antagonists; Morpholines; Naphthalenes; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptors, Cannabinoid; Receptors, Glucocorticoid; Rimonabant; Spironolactone

2014
Effects of cannabinoid and vanilloid drugs on positive and negative-like symptoms on an animal model of schizophrenia: the SHR strain.
    Schizophrenia research, 2014, Volume: 153, Issue:1-3

    Topics: Analysis of Variance; Animals; Arachidonic Acids; Benzoxazines; Cannabinoid Receptor Modulators; Capsaicin; Disease Models, Animal; Dose-Response Relationship, Drug; Interpersonal Relations; Male; Morpholines; Motor Activity; Naphthalenes; Piperidines; Pyrazoles; Rats; Rats, Inbred SHR; Rats, Wistar; Rimonabant; Schizophrenia; Schizophrenic Psychology; TRPV Cation Channels

2014
2-AG promotes the expression of conditioned fear via cannabinoid receptor type 1 on GABAergic neurons.
    Psychopharmacology, 2015, Volume: 232, Issue:15

    Topics: Animals; Arachidonic Acids; Cannabinoid Receptor Antagonists; Cannabinoids; Emotions; Endocannabinoids; Fear; GABAergic Neurons; Glycerides; Male; Mice; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptor, Cannabinoid, CB1; Rimonabant

2015
Self-administration of the anandamide transport inhibitor AM404 by squirrel monkeys.
    Psychopharmacology, 2016, Volume: 233, Issue:10

    Topics: Animals; Arachidonic Acids; Benzamides; Cannabinoid Receptor Antagonists; Carbamates; Cocaine; Dose-Response Relationship, Drug; Dronabinol; Drug-Seeking Behavior; Endocannabinoids; Male; Nicotine; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Reinforcement, Psychology; Reward; Rimonabant; Saimiri; Self Administration

2016
Extinction of avoidance behavior by safety learning depends on endocannabinoid signaling in the hippocampus.
    Journal of psychiatric research, 2017, Volume: 90

    Topics: Animals; Arachidonic Acids; Avoidance Learning; Cannabinoid Receptor Antagonists; Early Growth Response Protein 1; Extinction, Psychological; Hippocampus; Inhibition, Psychological; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Rimonabant; Voltage-Sensitive Dye Imaging

2017