Page last updated: 2024-09-02

sr 95531 and tetrahydrodeoxycorticosterone

sr 95531 has been researched along with tetrahydrodeoxycorticosterone in 5 studies

Compound Research Comparison

Studies
(sr 95531)
Trials
(sr 95531)
Recent Studies (post-2010)
(sr 95531)
Studies
(tetrahydrodeoxycorticosterone)
Trials
(tetrahydrodeoxycorticosterone)
Recent Studies (post-2010) (tetrahydrodeoxycorticosterone)
6100209269533

Protein Interaction Comparison

ProteinTaxonomysr 95531 (IC50)tetrahydrodeoxycorticosterone (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.1503
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.1503
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.1503
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.1503
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.1503
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.1503
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.1503
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.1503
Sodium- and chloride-dependent GABA transporter 1Rattus norvegicus (Norway rat)0.22
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.1503
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.1503
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.1503
Sodium- and chloride-dependent GABA transporter 2Rattus norvegicus (Norway rat)0.22
Sodium- and chloride-dependent GABA transporter 3Rattus norvegicus (Norway rat)0.22
Sodium- and chloride-dependent betaine transporterRattus norvegicus (Norway rat)0.22
Gamma-aminobutyric acid receptor subunit alpha-1Mus musculus (house mouse)0.039
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.1503
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.1503
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.1503
GABA theta subunitRattus norvegicus (Norway rat)0.1503
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.1503

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (40.00)18.2507
2000's2 (40.00)29.6817
2010's1 (20.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Acosta-Burruel, M; Goodnough, DB; Hawkinson, JE; Kimbrough, CL; Wood, PL1
Biggio, G; Concas, A; Marino, G; Minei, R; Mostallino, MC; Pierobon, P; Porcu, P1
Andersson, A; Asztely, F; Heeroma, JH; McEvoy, AW; Rydenhag, B; Scimemi, A; Strandberg, J; Thom, M; Walker, MC1
Amin, J; Hadley, SH1
Bayliss, DA; Chen, X; Kapur, J; Schwartz, LC; Shu, S; Sun, C1

Other Studies

5 other study(ies) available for sr 95531 and tetrahydrodeoxycorticosterone

ArticleYear
Steroid inhibition of [3H]SR 95531 binding to the GABAA recognition site.
    European journal of pharmacology, 1996, May-23, Volume: 304, Issue:1-3

    Topics: Allosteric Regulation; Androstanes; Animals; Azasteroids; Cell Membrane; Cerebral Cortex; Desoxycorticosterone; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Pregnanolone; Pregnenolone; Protein Binding; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, GABA; Steroids

1996
Modulation of gamma-aminobutyric acid (GABA) receptors and the feeding response by neurosteroids in Hydra vulgaris.
    Neuroscience, 1998, Volume: 85, Issue:3

    Topics: Anesthetics; Animals; Anti-Anxiety Agents; Bicuculline; Carbolines; Cerebral Cortex; Chemoreceptor Cells; Clonazepam; Desoxycorticosterone; Diazepam; Feeding Behavior; GABA Antagonists; GABA Modulators; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Glutathione; Hydra; Neurotransmitter Agents; Pregnanolone; Progesterone; Pyridazines; Radioligand Assay; Rats; Receptors, GABA-A; Tritium

1998
Tonic GABA(A) receptor-mediated currents in human brain.
    The European journal of neuroscience, 2006, Volume: 24, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Cerebral Cortex; Dentate Gyrus; Desoxycorticosterone; Electrophysiology; GABA Antagonists; Humans; Interneurons; Membrane Potentials; Neurons; Picrotoxin; Pyridazines; Receptors, GABA-A

2006
Rat alpha6beta2delta GABAA receptors exhibit two distinct and separable agonist affinities.
    The Journal of physiology, 2007, Jun-15, Volume: 581, Issue:Pt 3

    Topics: Action Potentials; Animals; beta-Alanine; Bicuculline; Crotonates; Desoxycorticosterone; Dose-Response Relationship, Drug; Female; Furosemide; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Imidazoles; Microinjections; Mutation; Neural Inhibition; Neurons; Oocytes; Picrotoxin; Pyridazines; Rats; Receptors, GABA-A; Sesterterpenes; Taurine; Xenopus laevis; Zinc

2007
Homeostatic regulation of synaptic excitability: tonic GABA(A) receptor currents replace I(h) in cortical pyramidal neurons of HCN1 knock-out mice.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2010, Feb-17, Volume: 30, Issue:7

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Anti-Anxiety Agents; Bicuculline; Cerebral Cortex; Cyclic Nucleotide-Gated Cation Channels; Desoxycorticosterone; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; GABA Agents; Homeostasis; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Male; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Knockout; Models, Neurological; Patch-Clamp Techniques; Potassium Channels; Protein Subunits; Pyramidal Cells; Pyridazines; Pyrimidines; Receptors, GABA-A; Sodium Channel Blockers; Synapses; Tetrodotoxin; Up-Regulation; Valine

2010