Page last updated: 2024-09-02

sr 95531 and piperidines

sr 95531 has been researched along with piperidines in 13 studies

Compound Research Comparison

Studies
(sr 95531)
Trials
(sr 95531)
Recent Studies (post-2010)
(sr 95531)
Studies
(piperidines)
Trials
(piperidines)
Recent Studies (post-2010) (piperidines)
610020940,2355,22114,545

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (7.69)18.2507
2000's5 (38.46)29.6817
2010's6 (46.15)24.3611
2020's1 (7.69)2.80

Authors

AuthorsStudies
Andre, JM; Boulanger, T; Durant, F; Hoffmann, R; Rognan, D; Vercauteren, DP; Wermuth, CG1
Maksay, G; McKernan, R1
Ebert, B; Fjalland, B; Hansen, SL; Kristiansen, U1
Ebert, B; Frølund, B; Jensen, LS; Kehler, J; Krogsgaard-Larsen, P; Liljefors, T; Stensbøl, TB; Storustovu, SI1
Li, P; Longhurst, JC; Tjen-A-Looi, SC1
Jean, A; Lebrun, B; Roux, J; Trouslard, J; Wanaverbecq, N1
Doengi, M; Gaburro, S; Häring, M; Kamprath, K; Lutz, B; Pape, HC; Romo-Parra, H1
Huang, GZ; Woolley, CS1
Arreto, CD; Bourgeais, L; Condes-Lara, M; Jay, T; Noseda, R; Robert, C; Villanueva, L1
Chen, SR; Pan, HL; Zhu, Y1
Crunelli, V; David, F; Lambert, RC; Leresche, N1
Chen, L; Huang, M; Jiang, B; Li, S; Li, Y; Wang, L; Wang, X; Yang, Y; Zhang, X1
Costa-Ferreira, W; Crestani, CC; Gomes-de-Souza, L; Mendonça, MM; Xavier, CH1

Other Studies

13 other study(ies) available for sr 95531 and piperidines

ArticleYear
Structure and molecular modeling of GABAA receptor antagonists.
    Journal of medicinal chemistry, 1992, May-29, Volume: 35, Issue:11

    Topics: Alkaloids; Androstanes; Azasteroids; Azepines; Bicuculline; Crystallization; Dibenzazepines; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Heterocyclic Compounds, 4 or More Rings; Heterocyclic Compounds, Bridged-Ring; Isoxazoles; Lactones; Models, Molecular; Molecular Conformation; Molecular Structure; Piperidines; Pyridazines; Receptors, GABA-A; Structure-Activity Relationship; Tubocurarine; X-Ray Diffraction

1992
Entropy as the predominant driving force of binding to human recombinant alpha(x)beta(3)gamma(2) GABA(A) receptors.
    European journal of pharmacology, 2001, Jan-05, Volume: 411, Issue:1-2

    Topics: Animals; Binding, Competitive; Dose-Response Relationship, Drug; Entropy; GABA Agonists; GABA Antagonists; Humans; Isoxazoles; L Cells; Membranes; Mice; Muscimol; Piperidines; Pyridazines; Receptors, GABA-A; Recombinant Proteins; Temperature; Tritium

2001
Effects of GABA(A) receptor partial agonists in primary cultures of cerebellar granule neurons and cerebral cortical neurons reflect different receptor subunit compositions.
    British journal of pharmacology, 2001, Volume: 133, Issue:4

    Topics: Animals; Bicuculline; Cells, Cultured; Cerebellum; Cerebral Cortex; Electrophysiology; GABA Agonists; GABA-A Receptor Agonists; Isonicotinic Acids; Isoxazoles; Mice; Neurons; Oocytes; Patch-Clamp Techniques; Piperidines; Pyridazines; Receptors, GABA-A; Xenopus laevis

2001
4-aryl-5-(4-piperidyl)-3-isoxazolol GABAA antagonists: synthesis, pharmacology, and structure-activity relationships.
    Journal of medicinal chemistry, 2007, Apr-19, Volume: 50, Issue:8

    Topics: Animals; Female; GABA-A Receptor Antagonists; Humans; In Vitro Techniques; Isoxazoles; Models, Molecular; Molecular Conformation; Oocytes; Patch-Clamp Techniques; Piperidines; Pyridazines; Structure-Activity Relationship; Xenopus

2007
Processing cardiovascular information in the vlPAG during electroacupuncture in rats: roles of endocannabinoids and GABA.
    Journal of applied physiology (Bethesda, Md. : 1985), 2009, Volume: 106, Issue:6

    Topics: Animals; Benzamides; Cannabinoid Receptor Modulators; Carbamates; Drug Antagonism; Electroacupuncture; Endocannabinoids; gamma-Aminobutyric Acid; Hemodynamics; Male; Periaqueductal Gray; Piperidines; Pyrazoles; Pyridazines; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Reflex; Stomach; Sympathetic Nervous System

2009
Depolarization-induced release of endocannabinoids by murine dorsal motor nucleus of the vagus nerve neurons differentially regulates inhibitory and excitatory neurotransmission.
    Neuropharmacology, 2009, Volume: 56, Issue:8

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Arachidonic Acids; Benzoxazines; Brain Stem; Calcium Signaling; Cannabinoid Receptor Modulators; Capsaicin; Efferent Pathways; Endocannabinoids; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamic Acid; Inhibitory Postsynaptic Potentials; Kynurenic Acid; Male; Mice; Mice, Inbred C57BL; Morpholines; Naphthalenes; Neurons; Piperidines; Pyrazoles; Pyridazines; Receptor, Cannabinoid, CB1; Receptors, Presynaptic; Rimonabant; Tetrodotoxin; Vagus Nerve

2009
Short-term adaptation of conditioned fear responses through endocannabinoid signaling in the central amygdala.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2011, Volume: 36, Issue:3

    Topics: Action Potentials; Adaptation, Psychological; Amygdala; Animals; Behavior, Animal; Cannabinoid Receptor Modulators; Conditioning, Psychological; Electric Stimulation; Endocannabinoids; Excitatory Amino Acid Antagonists; Extinction, Psychological; Fear; GABA Antagonists; Gene Expression Regulation; In Vitro Techniques; Male; Maze Learning; Mice; Mice, Inbred C57BL; Mice, Knockout; Phosphinic Acids; Piperidines; Propanolamines; Pyrazoles; Pyridazines; Quinoxalines; Receptor, Cannabinoid, CB1; Sensory Receptor Cells; Signal Transduction; Time Factors; Valine

2011
Estradiol acutely suppresses inhibition in the hippocampus through a sex-specific endocannabinoid and mGluR-dependent mechanism.
    Neuron, 2012, Jun-07, Volume: 74, Issue:5

    Topics: Animals; Benzodioxoles; Benzoxazines; Biophysics; CA1 Region, Hippocampal; Cannabinoid Receptor Modulators; Castration; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Endocannabinoids; Enzyme Inhibitors; Estradiol; Estrogens; Excitatory Amino Acid Agents; Female; GABA Antagonists; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Lactones; Male; Morpholines; NAD; Naphthalenes; Neural Inhibition; Neurons; Orlistat; Patch-Clamp Techniques; Phenols; Piperidines; Pyrazoles; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate

2012
Paraventricular hypothalamic regulation of trigeminovascular mechanisms involved in headaches.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2013, May-15, Volume: 33, Issue:20

    Topics: Action Potentials; Animals; Biotin; Corticosterone; Dextrans; Disease Models, Animal; GABA Antagonists; GABA-A Receptor Agonists; Male; Muscimol; Neural Pathways; Neurons; Paraventricular Hypothalamic Nucleus; Physical Stimulation; Piperidines; Pituitary Adenylate Cyclase-Activating Polypeptide; Pyridazines; Rats; Rats, Sprague-Dawley; Serotonin Receptor Agonists; Stilbamidines; Stress, Psychological; Trigeminal Nuclei; Tryptamines

2013
Muscarinic receptor subtypes differentially control synaptic input and excitability of cerebellum-projecting medial vestibular nucleus neurons.
    Journal of neurochemistry, 2016, Volume: 137, Issue:2

    Topics: Alkenes; Animals; Bicuculline; Cerebellum; Cholinergic Agents; Drug Interactions; Excitatory Postsynaptic Potentials; GABA-A Receptor Antagonists; Gene Expression Regulation; Male; Neurons; Patch-Clamp Techniques; Phosphopyruvate Hydratase; Piperidines; Pirenzepine; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Synaptic Transmission; Vestibular Nuclei

2016
Dynamic Analysis of the Conditional Oscillator Underlying Slow Waves in Thalamocortical Neurons.
    Frontiers in neural circuits, 2016, Volume: 10

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Benzamides; Calcium; Calcium Channel Blockers; Cats; Cerebral Cortex; Electric Stimulation; Excitatory Amino Acid Antagonists; GABA Antagonists; Geniculate Bodies; In Vitro Techniques; Membrane Potentials; Models, Neurological; Neurons; Nonlinear Dynamics; Organophosphorus Compounds; Patch-Clamp Techniques; Piperidines; Pyridazines

2016
Inhibition of Cdk5 rejuvenates inhibitory circuits and restores experience-dependent plasticity in adult visual cortex.
    Neuropharmacology, 2018, Volume: 128

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Cyclin-Dependent Kinase 5; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; GABA Antagonists; Inhibitory Postsynaptic Potentials; Male; Mice; Mice, Inbred C57BL; N-Methylaspartate; Neuronal Plasticity; Neurons; Phosphopyruvate Hydratase; Piperidines; Pyridazines; Sensory Deprivation; Visual Cortex; Visual Pathways

2018
Lateral hypothalamus involvement in control of stress response by bed nucleus of the stria terminalis endocannabinoid neurotransmission in male rats.
    Scientific reports, 2021, 08-09, Volume: 11, Issue:1

    Topics: Animals; Cannabinoid Receptor Antagonists; Endocannabinoids; GABA Antagonists; GABAergic Neurons; Heart Rate; Hypothalamic Area, Lateral; Male; Models, Neurological; Piperidines; Psychological Distress; Pyrazoles; Pyridazines; Rats; Rats, Wistar; Septal Nuclei; Stress, Psychological; Synaptic Transmission; Tachycardia

2021