Page last updated: 2024-09-02

sr 95531 and picrotoxin

sr 95531 has been researched along with picrotoxin in 46 studies

Compound Research Comparison

Studies
(sr 95531)
Trials
(sr 95531)
Recent Studies (post-2010)
(sr 95531)
Studies
(picrotoxin)
Trials
(picrotoxin)
Recent Studies (post-2010) (picrotoxin)
61002094,1356406

Research

Studies (46)

TimeframeStudies, this research(%)All Research%
pre-19902 (4.35)18.7374
1990's10 (21.74)18.2507
2000's22 (47.83)29.6817
2010's11 (23.91)24.3611
2020's1 (2.17)2.80

Authors

AuthorsStudies
Crema, A; De Petris, G; Manzo, L; Onori, L; Rizzi, CA; Tonini, M1
Asaro, D; Pellegrini, G; Pittaluga, A; Raiteri, M1
Bormann, J; Feigenspan, A1
Candura, SM; Coccini, T; Costa, LG; Manzo, L; Tonini, M1
Lukasiewicz, PD; Werblin, FS1
Mody, I; Soltesz, I1
Lukasiewicz, PD; Maple, BR; Werblin, FS1
Feltz, P; Hayar, A; Piguet, P1
Amato, F; Biggio, G; Deserra, T; Motzo, C; Murgia, A; Sanna, E1
Biggio, G; Casula, A; Murgia, A; Sanna, E1
Fischer, KF; Lukasiewicz, PD; Wong, RO1
Paladini, CA; Tepper, JM1
Shen, W; Slaughter, MM1
Bai, D; Jackson, MF; MacDonald, JF; Orser, BA; Pennefather, P; Zhu, G1
Karnup, S; Stelzer, A1
Abaigar, W; Bovill, JG; Laster, MJ; Sonner, JM; Stabernack, C; Xing, Y; Zhang, Y1
Baxi, S; Evans, C; Irnaten, M; Mendelowitz, D; Venkatesan, P; Wang, J; Wang, X1
Grillner, S; Hill, RH; Schmitt, DE1
Bevan, MD; Hallworth, NE1
Endo, T; Isa, T; Obata, K; Yanagawa, Y1
Andersson, A; Asztely, F; Heeroma, JH; McEvoy, AW; Rydenhag, B; Scimemi, A; Strandberg, J; Thom, M; Walker, MC1
Eisenman, LN; Kress, G; Mennerick, S; Zorumski, CF1
Manabe, T; Nakamura, M; Sekino, Y1
Cherubini, E; Marchionni, I; Omrani, A1
Armstrong, WE; Li, C; Tripathi, PK1
Jembrek, MJ; Pericić, D; Strac, DS; Vlainić, J1
Amin, J; Hadley, SH1
Park, JB; Skalska, S; Son, S; Stern, JE1
Ishii, H; Kato, M; Sakuma, Y; Tanaka, N; Yin, C1
Connors, BW; Fanselow, EE; Richardson, KA1
Cox, PJ; Güçlü, B; Mahoney, GK; Pack, AK; Pawson, L; Prestia, LT1
Basson, MD; Kouatli, Y; Marsh, HM; Shiratsuchi, H; Yu, GX1
Berns, M; Kerner, T; Schmidt, M; Seeberg, L; Zacharias, R1
Bracha, V; Carrel, AJ; Parker, KL; Zbarska, S1
Davis, T; Kalmbach, BE; Mauk, MD; Nores, WL; Ohyama, T; Riusech, F1
Aguilar, J; Bautista, W; Delgado-Lezama, R; Loeza-Alcocer, JE1
Burdakov, D; Fugger, L; Jensen, LT; Karnani, MM; Venner, A1
Dizon, MJ; Khodakhah, K1
Carlson, BA; George, AA; Lyons-Warren, AM; Ma, X1
Dretchen, KL; Gillis, RA; Herman, MA; Sahibzada, N; Vicini, S1
Dierkes, PW; Kilb, W; Kolbaev, SN; Luhmann, HJ; Sharopov, S1
Ayling, OG; Harrison, TC; Murphy, TH1
Chesnoy-Marchais, D1
Fleck, MW; Hoerbelt, P; Lindsley, TA1
Bhattarai, JP; Cho, DH; Chun, SW; Han, SK; Park, SJ1
Bae, JY; Bae, YC; Cheong, E; Choi, JW; Feng, J; Ha, GE; Kim, KH; Kim, S; Kim, YS; Koh, W; Kwak, H; Kwon, SW; Lee, CJ; Lee, D; Lee, EH; Lee, H; Lee, J; Lee, JM; Lee, SE; Li, Y; Oh, JE; Park, KD; Park, YM; Shin, JI; Son, T; Song, K; Woo, J; Yoon, BE1

Other Studies

46 other study(ies) available for sr 95531 and picrotoxin

ArticleYear
The role of GABAA receptor function in peristaltic activity of the guinea-pig ileum: a comparative study with bicuculline, SR 95531 and picrotoxinin.
    British journal of pharmacology, 1989, Volume: 97, Issue:2

    Topics: Animals; Bicuculline; Electric Stimulation; GABA Antagonists; Gastrointestinal Motility; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Peristalsis; Picrotoxin; Pyridazines; Receptors, GABA-A; Sesterterpenes

1989
Studies on [3H]GABA and endogenous GABA release in rat cerebral cortex suggest the presence of autoreceptors of the GABAB type.
    European journal of pharmacology, 1987, Nov-24, Volume: 144, Issue:1

    Topics: Animals; Anticonvulsants; Baclofen; Bicuculline; Cerebral Cortex; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Median Eminence; Nipecotic Acids; Picrotoxin; Potassium; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptosomes

1987
Differential pharmacology of GABAA and GABAC receptors on rat retinal bipolar cells.
    European journal of pharmacology, 1994, Dec-15, Volume: 288, Issue:1

    Topics: Animals; Bicuculline; Binding Sites; Cells, Cultured; Chickens; Chloride Channels; Dose-Response Relationship, Drug; Flunitrazepam; GABA Antagonists; GABA-A Receptor Antagonists; Hexachlorocyclohexane; Patch-Clamp Techniques; Pentobarbital; Picrotoxin; Pyridazines; Rats; Rats, Wistar; Receptors, GABA; Receptors, GABA-A; Retina; Sesterterpenes; Signal Transduction

1994
Interaction of the neurotoxic pesticides ivermectin and lindane with the enteric GABAA receptor-ionophore complex in the guinea-pig.
    European journal of pharmacology, 1993, Jun-01, Volume: 248, Issue:1

    Topics: Animals; Chloride Channels; Female; GABA-A Receptor Antagonists; Guinea Pigs; Hexachlorocyclohexane; In Vitro Techniques; Intestine, Small; Isometric Contraction; Ivermectin; Male; Membrane Proteins; Muscle, Smooth; Picrotoxin; Pyridazines; Receptors, GABA-A; Scopolamine; Sesterterpenes; Taurine; Tetrodotoxin

1993
A novel GABA receptor modulates synaptic transmission from bipolar to ganglion and amacrine cells in the tiger salamander retina.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1994, Volume: 14, Issue:3 Pt 1

    Topics: Animals; Calcium; Chlorides; Crotonates; Electrophysiology; GABA-A Receptor Antagonists; Light; Neurotransmitter Agents; Picrotoxin; Pyridazines; Receptors, GABA; Receptors, GABA-A; Retina; Retinal Ganglion Cells; Synaptic Transmission; Urodela

1994
Patch-clamp recordings reveal powerful GABAergic inhibition in dentate hilar neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1994, Volume: 14, Issue:4

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Chlorides; Electrophysiology; GABA-A Receptor Antagonists; Hippocampus; In Vitro Techniques; Kinetics; Male; Membrane Potentials; Neurons; Picrotoxin; Pyridazines; Quinoxalines; Rats; Rats, Wistar; Receptors, GABA-A; Tetrodotoxin; Time Factors

1994
A novel GABA receptor on bipolar cell terminals in the tiger salamander retina.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1994, Volume: 14, Issue:3 Pt 1

    Topics: Animals; Bicuculline; Chlorides; Crotonates; Electrophysiology; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Muscimol; Pentobarbital; Picrotoxin; Pyridazines; Receptors, GABA; Receptors, GABA-A; Retina; Retinal Ganglion Cells; Urodela

1994
GABA-induced responses in electrophysiologically characterized neurons within the rat rostro-ventrolateral medulla in vitro.
    Brain research, 1996, Feb-19, Volume: 709, Issue:2

    Topics: Animals; Baclofen; Bicuculline; Brain Stem; Electrophysiology; GABA Agonists; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Heart Conduction System; In Vitro Techniques; Medulla Oblongata; Neurons; Organophosphorus Compounds; Picrotoxin; Pyridazines; Rats; Rats, Wistar; Synapses

1996
Expression of native GABAA receptors in Xenopus oocytes injected with rat brain synaptosomes.
    Journal of neurochemistry, 1996, Volume: 67, Issue:5

    Topics: Anesthetics; Animals; Brain; Cell Membrane; Chloride Channels; Chlorides; Diazepam; Female; GABA Antagonists; gamma-Aminobutyric Acid; Membrane Potentials; Oocytes; Picrotoxin; Pregnanediones; Pyridazines; Rats; Receptors, GABA-A; Synaptosomes; Xenopus laevis; Zinc Compounds

1996
Differential subunit dependence of the actions of the general anesthetics alphaxalone and etomidate at gamma-aminobutyric acid type A receptors expressed in Xenopus laevis oocytes.
    Molecular pharmacology, 1997, Volume: 51, Issue:3

    Topics: Anesthetics; Animals; Binding Sites; Chlorides; Etomidate; Oocytes; Picrotoxin; Pregnanediones; Pyridazines; Receptors, GABA-A; Recombinant Proteins; Xenopus laevis

1997
Age-dependent and cell class-specific modulation of retinal ganglion cell bursting activity by GABA.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1998, May-15, Volume: 18, Issue:10

    Topics: Aging; Animals; Animals, Newborn; Bicuculline; Electrophysiology; Female; Ferrets; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Glycine; Glycine Agents; Membrane Potentials; Periodicity; Picrotoxin; Pregnancy; Pyridazines; Retinal Ganglion Cells; Strychnine

1998
GABA(A) and GABA(B) antagonists differentially affect the firing pattern of substantia nigra dopaminergic neurons in vivo.
    Synapse (New York, N.Y.), 1999, Jun-01, Volume: 32, Issue:3

    Topics: Action Potentials; Animals; Baclofen; Bicuculline; Dopamine; Electrophysiology; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; Kinetics; Male; Neurons; Phosphinic Acids; Picrotoxin; Propanolamines; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B; Substantia Nigra

1999
Multireceptor GABAergic regulation of synaptic communication in amphibian retina.
    The Journal of physiology, 2001, Jan-01, Volume: 530, Issue:Pt 1

    Topics: Ambystoma; Animals; Cell Communication; Excitatory Postsynaptic Potentials; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Light; Organophosphorus Compounds; Patch-Clamp Techniques; Phosphinic Acids; Picrotoxin; Propanolamines; Pyridazines; Receptors, GABA; Receptors, GABA-A; Receptors, GABA-B; Receptors, Kainic Acid; Retina; Retinal Ganglion Cells; Synapses

2001
Distinct functional and pharmacological properties of tonic and quantal inhibitory postsynaptic currents mediated by gamma-aminobutyric acid(A) receptors in hippocampal neurons.
    Molecular pharmacology, 2001, Volume: 59, Issue:4

    Topics: Animals; Bicuculline; Cells, Cultured; Dose-Response Relationship, Drug; Drug Synergism; Excitatory Postsynaptic Potentials; GABA Antagonists; GABA-A Receptor Antagonists; Hippocampus; Hypnotics and Sedatives; In Vitro Techniques; Mice; Midazolam; Models, Neurological; Neural Inhibition; Neurons; Patch-Clamp Techniques; Picrotoxin; Propofol; Pyridazines; Receptors, GABA-A

2001
Seizure-like activity in the disinhibited CA1 minislice of adult guinea-pigs.
    The Journal of physiology, 2001, May-01, Volume: 532, Issue:Pt 3

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Age Factors; Animals; Bicuculline; Epilepsy; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; Glycine; Guinea Pigs; Hippocampus; Neural Inhibition; Neurons, Afferent; Organ Culture Techniques; Picrotoxin; Pyridazines; Receptors, AMPA; Receptors, GABA-A; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Resorcinols

2001
GABA(A) receptor blockade antagonizes the immobilizing action of propofol but not ketamine or isoflurane in a dose-related manner.
    Anesthesia and analgesia, 2003, Volume: 96, Issue:3

    Topics: Anesthetics, Dissociative; Anesthetics, Inhalation; Anesthetics, Intravenous; Animals; Bicuculline; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; GABA Antagonists; GABA-A Receptor Antagonists; Glycine Agents; Infusions, Intravenous; Injections, Intraperitoneal; Isoflurane; Ketamine; Male; Picrotoxin; Propofol; Pulmonary Alveoli; Pyridazines; Rats; Rats, Sprague-Dawley; Strychnine

2003
Endogenous acetylcholine and nicotine activation enhances GABAergic and glycinergic inputs to cardiac vagal neurons.
    Journal of neurophysiology, 2003, Volume: 89, Issue:5

    Topics: 2-Amino-5-phosphonovalerate; Acetylcholine; Animals; Cholinesterase Inhibitors; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Fluorescent Dyes; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; Glycine Agents; Heart; Neostigmine; Neurons; Nicotine; Nicotinic Agonists; Parasympathetic Nervous System; Picrotoxin; Pyridazines; Rats; Strychnine; Synaptic Transmission; Vagus Nerve

2003
The spinal GABAergic system is a strong modulator of burst frequency in the lamprey locomotor network.
    Journal of neurophysiology, 2004, Volume: 92, Issue:4

    Topics: Algorithms; Animals; Calcium Channel Blockers; Chloride Channels; Electrophysiology; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Lampreys; Locomotion; Models, Neurological; Nerve Net; Phosphinic Acids; Picrotoxin; Potassium Channels, Calcium-Activated; Propanolamines; Pyridazines; Pyridines; Receptors, GABA; Receptors, GABA-B; Receptors, N-Methyl-D-Aspartate; Spinal Cord

2004
Globus pallidus neurons dynamically regulate the activity pattern of subthalamic nucleus neurons through the frequency-dependent activation of postsynaptic GABAA and GABAB receptors.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, Jul-06, Volume: 25, Issue:27

    Topics: 2-Amino-5-phosphonovalerate; Action Potentials; Animals; Evoked Potentials; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Globus Pallidus; Lysine; Male; Mice; Mice, Inbred C57BL; Neural Pathways; Neurons; Parkinson Disease; Patch-Clamp Techniques; Picrotoxin; Pyridazines; Quinoxalines; Receptors, GABA-A; Receptors, GABA-B; Subthalamic Nucleus; Synapses; Tetrodotoxin

2005
Nicotinic acetylcholine receptor subtypes involved in facilitation of GABAergic inhibition in mouse superficial superior colliculus.
    Journal of neurophysiology, 2005, Volume: 94, Issue:6

    Topics: Acetylcholine; Animals; Bicuculline; Bungarotoxins; Cadmium; Conotoxins; Dihydro-beta-Erythroidine; Dimethylphenylpiperazinium Iodide; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Drug Interactions; Electric Stimulation; GABA Antagonists; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Green Fluorescent Proteins; In Vitro Techniques; Isoenzymes; Mecamylamine; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Transgenic; Neural Inhibition; Neural Networks, Computer; Neurons; Nicotinic Agonists; Nicotinic Antagonists; Patch-Clamp Techniques; Picrotoxin; Protein Subunits; Pyridazines; Receptors, Nicotinic; Superior Colliculi

2005
Tonic GABA(A) receptor-mediated currents in human brain.
    The European journal of neuroscience, 2006, Volume: 24, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Cerebral Cortex; Dentate Gyrus; Desoxycorticosterone; Electrophysiology; GABA Antagonists; Humans; Interneurons; Membrane Potentials; Neurons; Picrotoxin; Pyridazines; Receptors, GABA-A

2006
A spontaneous tonic chloride conductance in solitary glutamatergic hippocampal neurons.
    Brain research, 2006, Nov-06, Volume: 1118, Issue:1

    Topics: Animals; Animals, Newborn; Bicuculline; Cells, Cultured; Chloride Channels; GABA Antagonists; Glutamic Acid; Hippocampus; Membrane Potentials; Neural Inhibition; Neurons; Patch-Clamp Techniques; Picrotoxin; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Small-Conductance Calcium-Activated Potassium Channels; Synaptic Transmission

2006
GABAergic interneurons facilitate mossy fiber excitability in the developing hippocampus.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2007, Feb-07, Volume: 27, Issue:6

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Axons; Bicuculline; Cyclopropanes; Enkephalin, Methionine; Excitatory Postsynaptic Potentials; Fluorescent Dyes; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Glycine; Hippocampus; Interneurons; Male; Mice; Mice, Inbred C57BL; Mossy Fibers, Hippocampal; Muscimol; Patch-Clamp Techniques; Picrotoxin; Presynaptic Terminals; Pyridazines; Pyridinium Compounds; Receptors, GABA-A; Synaptic Transmission; Tetrodotoxin

2007
In the developing rat hippocampus a tonic GABAA-mediated conductance selectively enhances the glutamatergic drive of principal cells.
    The Journal of physiology, 2007, Jun-01, Volume: 581, Issue:Pt 2

    Topics: Animals; Animals, Newborn; Electric Stimulation; GABA Antagonists; GABA Plasma Membrane Transport Proteins; GABA Uptake Inhibitors; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Glutamine; Hippocampus; In Vitro Techniques; Interneurons; Membrane Potentials; Neural Inhibition; Neuronal Plasticity; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Oximes; Patch-Clamp Techniques; Picrotoxin; Pyramidal Cells; Pyridazines; Rats; Rats, Wistar; Receptors, GABA-A; Synaptic Transmission; Time Factors

2007
Differences in spike train variability in rat vasopressin and oxytocin neurons and their relationship to synaptic activity.
    The Journal of physiology, 2007, May-15, Volume: 581, Issue:Pt 1

    Topics: Action Potentials; Animals; Excitatory Postsynaptic Potentials; Female; GABA Antagonists; Inhibitory Postsynaptic Potentials; Neurons; Oxytocin; Patch-Clamp Techniques; Picrotoxin; Pyridazines; Rats; Rats, Sprague-Dawley; Supraoptic Nucleus; Synapses; Synaptic Transmission; Vasopressins

2007
Allosteric uncoupling and up-regulation of benzodiazepine and GABA recognition sites following chronic diazepam treatment of HEK 293 cells stably transfected with alpha1beta2gamma2S subunits of GABA (A) receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 2007, Volume: 375, Issue:3

    Topics: Allosteric Regulation; Animals; Benzodiazepines; Binding Sites; Binding, Competitive; Cell Line; Diazepam; Flumazenil; Flunitrazepam; GABA Antagonists; gamma-Aminobutyric Acid; Humans; Muscimol; Picrotoxin; Protein Subunits; Pyridazines; Radioligand Assay; Rats; Receptors, GABA-A; Receptors, GABA-B; Transfection; Up-Regulation

2007
Rat alpha6beta2delta GABAA receptors exhibit two distinct and separable agonist affinities.
    The Journal of physiology, 2007, Jun-15, Volume: 581, Issue:Pt 3

    Topics: Action Potentials; Animals; beta-Alanine; Bicuculline; Crotonates; Desoxycorticosterone; Dose-Response Relationship, Drug; Female; Furosemide; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Imidazoles; Microinjections; Mutation; Neural Inhibition; Neurons; Oocytes; Picrotoxin; Pyridazines; Rats; Receptors, GABA-A; Sesterterpenes; Taurine; Xenopus laevis; Zinc

2007
Dual GABAA receptor-mediated inhibition in rat presympathetic paraventricular nucleus neurons.
    The Journal of physiology, 2007, Jul-15, Volume: 582, Issue:Pt 2

    Topics: Animals; Bicuculline; Electrophysiology; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Inhibitory Postsynaptic Potentials; Isoxazoles; Male; Medulla Oblongata; Neural Inhibition; Neurons; Paraventricular Hypothalamic Nucleus; Patch-Clamp Techniques; Picrotoxin; Pyridazines; Rats; Receptors, GABA-A; Synapses

2007
Activation of A-type gamma-amino butyric acid receptors excites gonadotrophin-releasing hormone neurones isolated from adult rats.
    Journal of neuroendocrinology, 2008, Volume: 20, Issue:5

    Topics: Action Potentials; Age Factors; Animals; Animals, Genetically Modified; Cell Culture Techniques; Cells, Cultured; Electrophysiology; Female; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Gonadotropin-Releasing Hormone; Green Fluorescent Proteins; Male; Neurons; Picrotoxin; Pyridazines; Rats; Receptors, GABA-A; Steroids

2008
Selective, state-dependent activation of somatostatin-expressing inhibitory interneurons in mouse neocortex.
    Journal of neurophysiology, 2008, Volume: 100, Issue:5

    Topics: Action Potentials; Analysis of Variance; Animals; Dose-Response Relationship, Radiation; Electric Stimulation; Excitatory Amino Acid Antagonists; GABA Antagonists; Green Fluorescent Proteins; In Vitro Techniques; Interneurons; Mice; Mice, Transgenic; Muscarine; Neocortex; Nerve Net; Neural Inhibition; Picrotoxin; Pyridazines; Somatostatin

2008
GABAergic/glutamatergic-glial/neuronal interaction contributes to rapid adaptation in pacinian corpuscles.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2009, Mar-04, Volume: 29, Issue:9

    Topics: Action Potentials; Adaptation, Physiological; Animals; Cats; DNA; DNA Primers; Electrophysiology; Female; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Immunohistochemistry; Neuroglia; Neurons; Pacinian Corpuscles; Picrotoxin; Pyridazines; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger

2009
Propofol inhibits pressure-stimulated macrophage phagocytosis via the GABAA receptor and dysregulation of p130cas phosphorylation.
    American journal of physiology. Cell physiology, 2009, Volume: 296, Issue:6

    Topics: Anesthetics, Intravenous; Cell Line; Crk-Associated Substrate Protein; Dose-Response Relationship, Drug; GABA Antagonists; Humans; Macrophages; Phagocytosis; Phosphorylation; Picrotoxin; Pressure; Propofol; Pyridazines; Receptors, GABA-A; RNA Interference; RNA, Small Interfering; Signal Transduction; Stress, Mechanical; Time Factors

2009
Effects of sevoflurane on primary neuronal cultures of embryonic rats.
    European journal of anaesthesiology, 2009, Volume: 26, Issue:7

    Topics: Anesthetics, Inhalation; Animals; Cell Survival; Cells, Cultured; Cerebral Cortex; Dose-Response Relationship, Drug; GABA Antagonists; Methyl Ethers; Neurons; Picrotoxin; Pyridazines; Rats; Rats, Wistar; Receptors, GABA-A; Sevoflurane; Time Factors

2009
Blocking GABAA neurotransmission in the interposed nuclei: effects on conditioned and unconditioned eyeblinks.
    Brain research, 2009, Oct-06, Volume: 1292

    Topics: Animals; Blinking; Cerebellum; Conditioning, Eyelid; Dose-Response Relationship, Drug; GABA Antagonists; GABA-A Receptor Antagonists; Male; Photic Stimulation; Physical Stimulation; Picrotoxin; Psychomotor Performance; Pyridazines; Rabbits; Receptors, GABA-A; Synaptic Transmission; Time Factors; Trigeminal Nuclei

2009
Cerebellar cortex contributions to the expression and timing of conditioned eyelid responses.
    Journal of neurophysiology, 2010, Volume: 103, Issue:4

    Topics: Animals; Cerebellar Cortex; Conditioning, Eyelid; GABA Antagonists; Infusions, Intraventricular; Lidocaine; Male; Models, Animal; Neuronal Plasticity; Picrotoxin; Purkinje Cells; Pyridazines; Rabbits; Reaction Time; Receptors, GABA-A

2010
Pre- and postsynaptic modulation of monosynaptic reflex by GABAA receptors on turtle spinal cord.
    The Journal of physiology, 2010, Jul-15, Volume: 588, Issue:Pt 14

    Topics: Animals; Bicuculline; Furosemide; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Motor Neurons; Picrotoxin; Presynaptic Terminals; Pyridazines; Receptors, GABA-A; Reflex, Monosynaptic; Spinal Cord; Synaptic Potentials; Turtles

2010
Direct and indirect control of orexin/hypocretin neurons by glycine receptors.
    The Journal of physiology, 2011, Feb-01, Volume: 589, Issue:Pt 3

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Aging; Alanine; Animals; Animals, Newborn; Benzothiadiazines; Chloride Channels; Electrophysiological Phenomena; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Glycine; Green Fluorescent Proteins; Hypothalamus; Intracellular Signaling Peptides and Proteins; Membrane Potentials; Mice; Mice, Transgenic; Neurons; Neuropeptides; Orexins; Patch-Clamp Techniques; Picrotoxin; Pyridazines; Receptors, GABA; Receptors, Glutamate; Receptors, Glycine; Strychnine; Synaptic Potentials

2011
The role of interneurons in shaping Purkinje cell responses in the cerebellar cortex.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2011, Jul-20, Volume: 31, Issue:29

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Age Factors; Animals; Animals, Newborn; Central Nervous System Stimulants; Cerebellar Cortex; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; In Vitro Techniques; Interneurons; Myasthenic Syndromes, Congenital; Nerve Net; Neural Inhibition; Patch-Clamp Techniques; Phosphinic Acids; Photic Stimulation; Photolysis; Picrotoxin; Propanolamines; Purkinje Cells; Pyridazines; Rats; Rats, Wistar

2011
A diversity of synaptic filters are created by temporal summation of excitation and inhibition.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2011, Oct-12, Volume: 31, Issue:41

    Topics: Action Potentials; Analysis of Variance; Animals; Axons; Biophysics; Dendrites; Electric Fish; Electric Organ; Electric Stimulation; Female; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Models, Neurological; Movement; Neural Inhibition; Neural Pathways; Neurons; Patch-Clamp Techniques; Picrotoxin; Pyridazines; Synaptic Potentials

2011
Tonic GABAA receptor conductance in medial subnucleus of the tractus solitarius neurons is inhibited by activation of μ-opioid receptors.
    Journal of neurophysiology, 2012, Volume: 107, Issue:3

    Topics: Analgesics, Opioid; Animals; Bicuculline; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; GABA Agonists; GABA Antagonists; GABA-A Receptor Antagonists; Isoxazoles; Male; Mice; Mice, Inbred C57BL; Neurons; Patch-Clamp Techniques; Picrotoxin; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, Opioid, mu; Sodium Channel Blockers; Solitary Nucleus; Tetrodotoxin

2012
Phasic GABAA -receptor activation is required to suppress epileptiform activity in the CA3 region of the immature rat hippocampus.
    Epilepsia, 2012, Volume: 53, Issue:5

    Topics: Action Potentials; Age Factors; Animals; Animals, Newborn; Biophysical Phenomena; CA3 Region, Hippocampal; Convulsants; Electric Stimulation; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Patch-Clamp Techniques; Picrotoxin; Pyridazines; Rats; Rats, Wistar; Receptors, GABA-A; Sodium Channel Blockers; Tetrodotoxin

2012
Distinct cortical circuit mechanisms for complex forelimb movement and motor map topography.
    Neuron, 2012, Apr-26, Volume: 74, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Analysis of Variance; Animals; Bacterial Proteins; Biophysics; Brain Mapping; Central Nervous System Stimulants; Channelrhodopsins; Dizocilpine Maleate; Electric Stimulation; Electromyography; Evoked Potentials, Motor; Excitatory Amino Acid Antagonists; Forelimb; GABA Antagonists; Green Fluorescent Proteins; Light; Luminescent Proteins; Mice; Mice, Transgenic; Motor Cortex; Movement; Nerve Net; Neural Pathways; Optics and Photonics; Picrotoxin; Pyridazines; Reaction Time; Synaptic Transmission; Thy-1 Antigens; Transduction, Genetic; Video Recording; Wakefulness

2012
Bicuculline- and neurosteroid-sensitive tonic chloride current in rat hypoglossal motoneurons and atypical dual effect of SR95531.
    The European journal of neuroscience, 2013, Volume: 37, Issue:3

    Topics: Action Potentials; Animals; Bicuculline; Brain Stem; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Motor Neurons; Picrotoxin; Pregnanolone; Protein Subunits; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, GABA; Receptors, GABA-A

2013
Dopamine directly modulates GABAA receptors.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2015, Feb-25, Volume: 35, Issue:8

    Topics: Amino Acid Sequence; Animals; Bicuculline; Cells, Cultured; Corpus Striatum; Dopamine; Female; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; HEK293 Cells; Humans; Male; Molecular Sequence Data; Mutation; Neurons; Picrotoxin; Protein Binding; Protein Subunits; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Zinc

2015
Activation of synaptic and extrasynaptic glycine receptors by taurine in preoptic hypothalamic neurons.
    Neuroscience letters, 2015, Nov-03, Volume: 608

    Topics: Action Potentials; Animals; Bicuculline; Dose-Response Relationship, Drug; GABA-A Receptor Antagonists; Glycine Agents; In Vitro Techniques; Mice; Neurons; Picrotoxin; Preoptic Area; Pyridazines; Receptors, Glycine; Strychnine; Synapses; Taurine

2015
Astrocytes Control Sensory Acuity via Tonic Inhibition in the Thalamus.
    Neuron, 2020, 11-25, Volume: 108, Issue:4

    Topics: Aldehyde Dehydrogenase 1 Family; Amine Oxidase (Copper-Containing); Animals; Astrocytes; Bestrophins; Female; GABA Antagonists; gamma-Aminobutyric Acid; Immunohistochemistry; Inhibitory Postsynaptic Potentials; Macrolides; Male; Mice; Mice, Knockout; Microscopy, Electron; Neural Inhibition; Neurons; Patch-Clamp Techniques; Picrotoxin; Primary Cell Culture; Pyridazines; Retinal Dehydrogenase; RNA, Small Interfering; Thalamus; Touch Perception

2020